Page last updated: 2024-09-03

cgp 42112a and pk 11195

cgp 42112a has been researched along with pk 11195 in 2 studies

Compound Research Comparison

Studies
(cgp 42112a)
Trials
(cgp 42112a)
Recent Studies (post-2010)
(cgp 42112a)
Studies
(pk 11195)
Trials
(pk 11195)
Recent Studies (post-2010) (pk 11195)
2330351,06311259

Protein Interaction Comparison

ProteinTaxonomycgp 42112a (IC50)pk 11195 (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.005
Translocator proteinRattus norvegicus (Norway rat)0.003
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.005
Translocator proteinHomo sapiens (human)0.1645
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.005
Nuclear receptor subfamily 1 group I member 3 Homo sapiens (human)0.39
GABA theta subunitRattus norvegicus (Norway rat)0.005
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.005

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Jarrott, B; Lawrence, AJ; Roulston, CL; Widdop, RE2

Other Studies

2 other study(ies) available for cgp 42112a and pk 11195

ArticleYear
Non-angiotensin II [(125)I] CGP42112 binding is a sensitive marker of neuronal injury in brainstem following unilateral nodose ganglionectomy: comparison with markers for activated microglia.
    Neuroscience, 2004, Volume: 127, Issue:3

    Topics: Angiotensin II; Animals; Autoradiography; Biomarkers; Brain Stem; Ganglionectomy; Glial Fibrillary Acidic Protein; Gliosis; Iodine Radioisotopes; Isoquinolines; Male; Microglia; Nodose Ganglion; Oligopeptides; Rats; Rats, Inbred WKY; Tritium; Vasoconstrictor Agents

2004
Minocycline treatment attenuates microglia activation and non-angiotensin II [125I] CGP42112 binding in brainstem following nodose ganglionectomy.
    Neuroscience, 2005, Volume: 135, Issue:4

    Topics: Animals; Anti-Bacterial Agents; Antineoplastic Agents; Autoradiography; Brain Stem; Ganglionectomy; Immunohistochemistry; Isoquinolines; Male; Microglia; Minocycline; Nodose Ganglion; Oligopeptides; Rats; Rats, Wistar; Receptor, Angiotensin, Type 2

2005