Page last updated: 2024-09-03

cgp 42112a and phentolamine

cgp 42112a has been researched along with phentolamine in 1 studies

Compound Research Comparison

Studies
(cgp 42112a)
Trials
(cgp 42112a)
Recent Studies (post-2010)
(cgp 42112a)
Studies
(phentolamine)
Trials
(phentolamine)
Recent Studies (post-2010) (phentolamine)
2330359,141270265

Protein Interaction Comparison

ProteinTaxonomycgp 42112a (IC50)phentolamine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.396
Alpha-2A adrenergic receptorHomo sapiens (human)0.006
Cytochrome P450 2D6Homo sapiens (human)10
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0316
Alpha-2B adrenergic receptorHomo sapiens (human)0.018
Alpha-2C adrenergic receptorHomo sapiens (human)0.11
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0492
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.0316
Alpha-1D adrenergic receptorHomo sapiens (human)0.0173
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.359
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.396
Alpha-1A adrenergic receptorHomo sapiens (human)0.0011
Alpha-1B adrenergic receptorHomo sapiens (human)0.0108
5-hydroxytryptamine receptor 2BHomo sapiens (human)3.807
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0316
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.5495

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Buikema, H; Morshuis, WJ; Nickenig, G; Plokker, HW; van de Wal, RM; van der Harst, P; van Gilst, WH; van Veldhuisen, DJ; Voors, AA; Wagenaar, LJ; Wassmann, S1

Other Studies

1 other study(ies) available for cgp 42112a and phentolamine

ArticleYear
Angiotensin II type 2 receptor vasoactivity in internal mammary arteries of patients with coronary artery disease.
    Journal of cardiovascular pharmacology, 2007, Volume: 50, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Benzimidazoles; Biphenyl Compounds; Coronary Artery Disease; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Male; Mammary Arteries; Middle Aged; Oligopeptides; Phentolamine; Phenylephrine; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Sodium Nitrite; Tetrazoles; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2007