Page last updated: 2024-09-03

cgp 42112a and dinoprostone

cgp 42112a has been researched along with dinoprostone in 7 studies

Compound Research Comparison

Studies
(cgp 42112a)
Trials
(cgp 42112a)
Recent Studies (post-2010)
(cgp 42112a)
Studies
(dinoprostone)
Trials
(dinoprostone)
Recent Studies (post-2010) (dinoprostone)
23303529,1051,3466,357

Protein Interaction Comparison

ProteinTaxonomycgp 42112a (IC50)dinoprostone (IC50)
Prostaglandin E2 receptor EP1 subtypeHomo sapiens (human)0.0155
Prostaglandin E2 receptor EP4 subtypeHomo sapiens (human)0.0031
Prostaglandin E2 receptor EP4 subtypeRattus norvegicus (Norway rat)0.0021
Prostaglandin E2 receptor EP3 subtypeHomo sapiens (human)0.002
Prostaglandin E2 receptor EP2 subtypeHomo sapiens (human)0.0087
Prostacyclin receptorHomo sapiens (human)0.26
Prostaglandin E2 receptor EP2 subtypeRattus norvegicus (Norway rat)0.0052

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (57.14)18.2507
2000's3 (42.86)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chappell, MC; Diz, DI; Ferrario, CM; Jaiswal, N; Khosla, MC1
Egidy, G; Friedman, J; Saavedra, JM; Viswanathan, M; Wahl, LM1
Bottari, SP; Bourmeyster, N; Chambaz, EM; Defaye, G; Liakos, P1
Carey, RM; Guerrant, RL; Jin, XH; Siragy, HM; Wang, ZQ1
Sakata, Y; Wada, M; Watanabe, T1
Kim, MP; Wahl, LM; Zhou, M1
Duvetorp, A; Ewert, S; Fandriks, L; Holm, M; Johansson, B; Sjoberg, T1

Other Studies

7 other study(ies) available for cgp 42112a and dinoprostone

ArticleYear
Stimulation of endothelial cell prostaglandin production by angiotensin peptides. Characterization of receptors.
    Hypertension (Dallas, Tex. : 1979), 1992, Volume: 19, Issue:2 Suppl

    Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Cells, Cultured; Dinoprostone; Endothelium, Vascular; Epoprostenol; Imidazoles; Losartan; Oligopeptides; Prostaglandins; Pyridines; Receptors, Angiotensin; Tetrazoles

1992
CGP-42112 partially activates human monocytes and reduces their stimulation by lipopolysaccharides.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 1

    Topics: Animals; Binding, Competitive; Cell Adhesion; Cells, Cultured; Collagenases; Culture Media, Serum-Free; Cytokines; Dinoprostone; Humans; Interleukin-1; Interleukin-10; Interleukin-6; Lipopolysaccharides; Matrix Metalloproteinase 9; Monocytes; Oligopeptides; Rats; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Tumor Necrosis Factor-alpha

1997
ANG II AT1 and AT2 receptors both inhibit bFGF-induced proliferation of bovine adrenocortical cells.
    The American journal of physiology, 1997, Volume: 273, Issue:4

    Topics: Adrenal Cortex; Angiotensin II; Animals; Cattle; Cell Cycle; Cell Division; Cells, Cultured; Cyclin D1; Dinoprostone; Fibroblast Growth Factor 2; G1 Phase; Imidazoles; Indomethacin; Oligopeptides; Prostaglandin D2; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin

1997
Regulation of jejunal sodium and water absorption by angiotensin subtype receptors.
    The American journal of physiology, 1998, Volume: 275, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Cyclic AMP; Cyclic GMP; Diet, Sodium-Restricted; Dinoprostone; Dose-Response Relationship, Drug; Guanethidine; Homeostasis; Imidazoles; Intestinal Absorption; Intestinal Mucosa; Jejunum; Kinetics; Losartan; Male; Mesenteric Arteries; Oligopeptides; Prazosin; Pyridines; Rats; Rats, Wistar; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Time Factors; Water

1998
Angiotensin AT1 receptors in the preoptic area negatively modulate the cardiovascular and ACTH responses induced in rats by intrapreoptic injection of prostaglandin E2.
    Brain research, 2000, Jan-03, Volume: 852, Issue:1

    Topics: Adrenocorticotropic Hormone; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Blood Pressure; Cardiovascular System; Dinoprostone; Injections; Losartan; Male; Oligopeptides; Preoptic Area; Rats; Rats, Wistar; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin

2000
Angiotensin II increases human monocyte matrix metalloproteinase-1 through the AT2 receptor and prostaglandin E2: implications for atherosclerotic plaque rupture.
    Journal of leukocyte biology, 2005, Volume: 78, Issue:1

    Topics: Angiotensin II; Angiotensin II Type 2 Receptor Blockers; Angiotensin-Converting Enzyme Inhibitors; Anti-Inflammatory Agents; Cells, Cultured; Coronary Artery Disease; Dinoprostone; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Hypertension; Imidazoles; Matrix Metalloproteinase 1; Monocytes; Myocardial Infarction; Oligopeptides; Phosphoprotein Phosphatases; Pyridines; Receptor, Angiotensin, Type 2; Time Factors; Tumor Necrosis Factor-alpha; Up-Regulation

2005
Dynamic expression of the angiotensin II type 2 receptor and duodenal mucosal alkaline secretion in the Sprague-Dawley rat.
    Experimental physiology, 2006, Volume: 91, Issue:1

    Topics: Angiotensin II; Animals; Dinoprostone; Duodenum; Intestinal Mucosa; Male; Oligopeptides; Rats; Rats, Sprague-Dawley; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; RNA, Messenger

2006