Page last updated: 2024-09-03

cgp 42112a and cyclic gmp

cgp 42112a has been researched along with cyclic gmp in 12 studies

Compound Research Comparison

Studies
(cgp 42112a)
Trials
(cgp 42112a)
Recent Studies (post-2010)
(cgp 42112a)
Studies
(cyclic gmp)
Trials
(cyclic gmp)
Recent Studies (post-2010) (cyclic gmp)
23303522,3463334,062

Protein Interaction Comparison

ProteinTaxonomycgp 42112a (IC50)cyclic gmp (IC50)
Phosphodiesterase Bos taurus (cattle)0.1
cGMP-inhibited 3',5'-cyclic phosphodiesterase BHomo sapiens (human)2.4
cGMP-inhibited 3',5'-cyclic phosphodiesterase AHomo sapiens (human)2.4

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (50.00)18.2507
2000's4 (33.33)29.6817
2010's2 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bottari, SP; Brechler, V; De Gasparo, M; Levens, NR1
Bottari, SP; Buisson, B; de Gasparo, M; Gallo-Payet, N; Laflamme, L; Payet, MD1
Heitsch, H; Linz, W; Schölkens, BA; Wagner, A; Wiemer, G1
Raizada, MK; Richards, EM; Sumners, C; Tang, W1
Bottari, SP; Brechler, V; de Gasparo, M; Jones, PW; Levens, NR1
Carey, RM; Guerrant, RL; Jin, XH; Siragy, HM; Wang, ZQ1
Ishii, K; Isobe, K; Kawakami, Y; Nakai, T; Nanmoku, T; Takekoshi, K1
Ishii, K; Isobe, K; Kawakami, Y; Nakai, T; Takekoshi, K1
Hakam, AC; Hussain, T2
Asghar, M; Hussain, T; Sabuhi, R1
Chen, C; Han, Y; He, D; Hopfer, U; Jose, PA; Ren, H; Yang, J; Zeng, C; Zhou, L1

Other Studies

12 other study(ies) available for cgp 42112a and cyclic gmp

ArticleYear
Angiotensin AT2 receptor mediated inhibition of particulate guanylate cyclase: a link with protein tyrosine phosphatase stimulation?
    Receptors & channels, 1994, Volume: 2, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-GMP Phosphodiesterases; Angiotensin II; Animals; Aorta; Arsenicals; Atrial Natriuretic Factor; Cell Membrane; Cells, Cultured; Cyclic GMP; GTP-Binding Proteins; Guanylate Cyclase; Muscle, Smooth, Vascular; Oligopeptides; PC12 Cells; Protein Tyrosine Phosphatases; Rats; Receptors, Angiotensin; Vanadates

1994
A G protein is involved in the angiotensin AT2 receptor inhibition of the T-type calcium current in non-differentiated NG108-15 cells.
    The Journal of biological chemistry, 1995, Jan-27, Volume: 270, Issue:4

    Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Calcium Channels; Cyclic GMP; Glioma; GTP-Binding Proteins; Hybrid Cells; Kinetics; Membrane Potentials; Neuroblastoma; Oligopeptides; Patch-Clamp Techniques; Receptors, Angiotensin; Time Factors

1995
The possible role of angiotensin II subtype AT2 receptors in endothelial cells and isolated ischemic rat hearts.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1993, Volume: 11, Issue:5

    Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Arginine; Bradykinin; Cattle; Cells, Cultured; Cyclic GMP; Endothelium, Vascular; Female; In Vitro Techniques; Male; Myocardial Ischemia; Nitric Oxide; Nitroarginine; Oligopeptides; Rats; Rats, Wistar; Receptors, Angiotensin

1993
Angiotensin II type 2 receptor expression in neuronal cultures from spontaneously hypertensive rat brain.
    Regulatory peptides, 1993, Mar-19, Volume: 44, Issue:2

    Topics: Angiotensin II; Animals; Brain Stem; Cells, Cultured; Cyclic GMP; Hypertension; Hypothalamus; Neurons; Oligopeptides; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Angiotensin; Tumor Cells, Cultured

1993
Agonistic and antagonistic properties of angiotensin analogs at the AT2 receptor in PC12W cells.
    Regulatory peptides, 1993, Mar-19, Volume: 44, Issue:2

    Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Binding, Competitive; Biphenyl Compounds; Cyclic GMP; Imidazoles; Losartan; Oligopeptides; PC12 Cells; Pyridines; Rats; Receptors, Angiotensin; Tetrazoles

1993
Regulation of jejunal sodium and water absorption by angiotensin subtype receptors.
    The American journal of physiology, 1998, Volume: 275, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Cyclic AMP; Cyclic GMP; Diet, Sodium-Restricted; Dinoprostone; Dose-Response Relationship, Drug; Guanethidine; Homeostasis; Imidazoles; Intestinal Absorption; Intestinal Mucosa; Jejunum; Kinetics; Losartan; Male; Mesenteric Arteries; Oligopeptides; Prazosin; Pyridines; Rats; Rats, Wistar; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Time Factors; Water

1998
Angiotensin-II subtype 2 receptor agonist (CGP-42112) inhibits catecholamine biosynthesis in cultured porcine adrenal medullary chromaffin cells.
    Biochemical and biophysical research communications, 2000, Jun-07, Volume: 272, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenal Medulla; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Benzimidazoles; Binding, Competitive; Biphenyl Compounds; Catecholamines; Cells, Cultured; Chromaffin Cells; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Induction; Imidazoles; Oligopeptides; Pyridines; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; RNA, Messenger; Swine; Tetrazoles; Tyrosine 3-Monooxygenase

2000
Activation of angiotensin II subtype 2 receptor induces catecholamine release in an extracellular Ca(2+)-dependent manner through a decrease of cyclic guanosine 3',5'-monophosphate production in cultured porcine adrenal medullary chromaffin Cells.
    Endocrinology, 2001, Volume: 142, Issue:7

    Topics: Adrenal Medulla; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Benzimidazoles; Biphenyl Compounds; Calcium; Catecholamines; Cells, Cultured; Chromaffin Cells; Cyclic GMP; Extracellular Space; Imidazoles; Inositol 1,4,5-Trisphosphate; Intracellular Membranes; Oligopeptides; Pyridines; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Swine; Tetrazoles; Virulence Factors, Bordetella

2001
Angiotensin II AT2 receptors inhibit proximal tubular Na+-K+-ATPase activity via a NO/cGMP-dependent pathway.
    American journal of physiology. Renal physiology, 2006, Volume: 290, Issue:6

    Topics: Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Angiotensin II Type 2 Receptor Blockers; Animals; Cyclic GMP; Diuresis; Enzyme Inhibitors; Glomerular Filtration Rate; Kidney Tubules, Proximal; Male; Natriuresis; Nitrates; Nitric Oxide; Nitrites; Oligopeptides; Rats; Rats, Sprague-Dawley; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Sodium-Potassium-Exchanging ATPase

2006
Angiotensin II type 2 receptor agonist directly inhibits proximal tubule sodium pump activity in obese but not in lean Zucker rats.
    Hypertension (Dallas, Tex. : 1979), 2006, Volume: 47, Issue:6

    Topics: Animals; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Imidazoles; Kidney Tubules, Proximal; Male; Nitrates; Nitrites; Obesity; Oligopeptides; Phosphorylation; Pyridines; Rats; Rats, Zucker; Receptor, Angiotensin, Type 2; Sodium-Potassium-Exchanging ATPase; Thinness

2006
Inhibition of NAD(P)H oxidase potentiates AT2 receptor agonist-induced natriuresis in Sprague-Dawley rats.
    American journal of physiology. Renal physiology, 2010, Volume: 299, Issue:4

    Topics: Acetophenones; Angiotensin II Type 1 Receptor Blockers; Animals; Benzimidazoles; Biphenyl Compounds; Blood Pressure; Cyclic GMP; Glomerular Filtration Rate; Homeostasis; Male; NADPH Oxidases; Natriuresis; Nitric Oxide; Oligopeptides; Rats; Rats, Sprague-Dawley; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Sodium; Tetrazoles

2010
Angiotensin II AT(2) receptor decreases AT(1) receptor expression and function via nitric oxide/cGMP/Sp1 in renal proximal tubule cells from Wistar-Kyoto rats.
    Journal of hypertension, 2012, Volume: 30, Issue:6

    Topics: Animals; Base Sequence; Cell Line, Transformed; Cyclic GMP; DNA Primers; Electrophoretic Mobility Shift Assay; Kidney Tubules, Proximal; Microscopy, Confocal; Nitric Oxide; Oligopeptides; Rats; Rats, Inbred WKY; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Reverse Transcriptase Polymerase Chain Reaction; Sodium-Potassium-Exchanging ATPase; Sp1 Transcription Factor

2012