Page last updated: 2024-09-02

cgp 39551 and donepezil

cgp 39551 has been researched along with donepezil in 1 studies

Compound Research Comparison

Studies
(cgp 39551)
Trials
(cgp 39551)
Recent Studies (post-2010)
(cgp 39551)
Studies
(donepezil)
Trials
(donepezil)
Recent Studies (post-2010) (donepezil)
75043,1935571,594

Protein Interaction Comparison

ProteinTaxonomycgp 39551 (IC50)donepezil (IC50)
AcetylcholinesteraseElectrophorus electricus (electric eel)0.4231
AcetylcholinesteraseTetronarce californica (Pacific electric ray)0.0265
Amyloid-beta precursor proteinHomo sapiens (human)0.022
CholinesteraseHomo sapiens (human)4.5742
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)7.42
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)5
Amine oxidase [flavin-containing] A Rattus norvegicus (Norway rat)7.4
AcetylcholinesteraseMus musculus (house mouse)1.5489
AcetylcholinesteraseHomo sapiens (human)0.3257
Acetylcholinesterase Bos taurus (cattle)0.1644
Choline O-acetyltransferase Rattus norvegicus (Norway rat)0.0053
AcetylcholinesteraseRattus norvegicus (Norway rat)0.0182
Beta-secretase 1Homo sapiens (human)0.8666
CholinesteraseEquus caballus (horse)3.7325
CholinesteraseMus musculus (house mouse)1.992
Acetylcholine receptor subunit epsilonHomo sapiens (human)0.0324
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.7844
Acyl-CoA:cholesterol acyltransferase Oryctolagus cuniculus (rabbit)0.008
Carboxylic ester hydrolase Rattus norvegicus (Norway rat)4.715
Carboxylic ester hydrolase Equus caballus (horse)4.5551
Histamine H3 receptorHomo sapiens (human)0.35

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ivanov, VB; Schilström, B; Svensson, TH; Wiker, C1

Other Studies

1 other study(ies) available for cgp 39551 and donepezil

ArticleYear
Galantamine enhances dopaminergic neurotransmission in vivo via allosteric potentiation of nicotinic acetylcholine receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2007, Volume: 32, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Analysis of Variance; Animals; Cholinesterase Inhibitors; Donepezil; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Galantamine; Indans; Male; Mecamylamine; Microdialysis; Neurons; Nicotinic Antagonists; Piperidines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Synaptic Transmission; Ventral Tegmental Area

2007