Page last updated: 2024-09-02

cgp 39551 and cycloserine

cgp 39551 has been researched along with cycloserine in 3 studies

Compound Research Comparison

Studies
(cgp 39551)
Trials
(cgp 39551)
Recent Studies (post-2010)
(cgp 39551)
Studies
(cycloserine)
Trials
(cycloserine)
Recent Studies (post-2010) (cycloserine)
75042,583192482

Protein Interaction Comparison

ProteinTaxonomycgp 39551 (IC50)cycloserine (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)4.835
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)2.3
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)2.3
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)2.3
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)2.3
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)2.3
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)2.3

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kretschmer, BD; Schmidt, WJ; Volz, L; Volz, TL; Zadow, B1
Millan, MJ; Seguin, L1
Danysz, W; Karcz-Kubicha, M; Wedzony, K; Zajaczkowski, W1

Other Studies

3 other study(ies) available for cgp 39551 and cycloserine

ArticleYear
The contribution of the different binding sites of the N-methyl-D-aspartate (NMDA) receptor to the expression of behavior.
    Journal of neural transmission. General section, 1992, Volume: 87, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Behavior, Animal; Binding Sites; Catalepsy; Cycloserine; Dizocilpine Maleate; Haloperidol; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate

1992
Chemically-diverse ligands at the glycine B site coupled to N-methyl-D-aspartate (NMDA) receptors selectively block the late phase of formalin-induced pain in mice.
    Neuroscience letters, 1994, Aug-29, Volume: 178, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Acetates; Acetic Acid; Animals; Anticonvulsants; Cycloserine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Formaldehyde; Indoles; Ligands; Male; Mice; Mice, Inbred Strains; Motor Activity; Pain; Propionates; Pyrrolidinones; Quinolones; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate

1994
NMDA receptor antagonists acting at the glycineB site in rat models for antipsychotic-like activity.
    Journal of neural transmission (Vienna, Austria : 1996), 1999, Volume: 106, Issue:11-12

    Topics: 2-Amino-5-phosphonovalerate; Amphetamine; Animals; Antimetabolites; Antipsychotic Agents; Binding Sites; Cycloleucine; Cycloserine; Disease Models, Animal; Dopamine Agents; Drug Synergism; Excitatory Amino Acid Antagonists; Glycine; Hallucinogens; Locomotion; Male; Phencyclidine; Phthalazines; Protein Structure, Tertiary; Psychotic Disorders; Pyrrolidinones; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate; Reflex, Startle

1999