Page last updated: 2024-09-03

cgp 36742 and glutamic acid

cgp 36742 has been researched along with glutamic acid in 5 studies

Compound Research Comparison

Studies
(cgp 36742)
Trials
(cgp 36742)
Recent Studies (post-2010)
(cgp 36742)
Studies
(glutamic acid)
Trials
(glutamic acid)
Recent Studies (post-2010) (glutamic acid)
633241,75745212,876

Protein Interaction Comparison

ProteinTaxonomycgp 36742 (IC50)glutamic acid (IC50)
Chain A, GLUTAMATE RECEPTOR SUBUNIT 2Rattus norvegicus (Norway rat)0.821
Chain A, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.821
Chain B, Glutamate Receptor Subunit 2Rattus norvegicus (Norway rat)0.821
Metabotropic glutamate receptor 8Homo sapiens (human)0.0057
Glutamate receptor ionotropic, NMDA 2DHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 3BHomo sapiens (human)0.07
Glutamate receptor 1Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 2Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 3Rattus norvegicus (Norway rat)0.5885
Glutamate receptor 4Rattus norvegicus (Norway rat)0.5885
Glutamate receptor ionotropic, kainate 1Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 2Rattus norvegicus (Norway rat)0.38
Glutamate receptor 1Homo sapiens (human)0.613
Glutamate receptor 2Homo sapiens (human)0.613
Glutamate receptor 3Homo sapiens (human)0.613
Glutamate receptor ionotropic, kainate 3Rattus norvegicus (Norway rat)0.38
Excitatory amino acid transporter 1Homo sapiens (human)207
Glutamate receptor 4Homo sapiens (human)0.613
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 4Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2CHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, kainate 5Rattus norvegicus (Norway rat)0.38
Glutamate receptor ionotropic, NMDA 3AHomo sapiens (human)0.07
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.1533
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.1533

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bowery, NG; Malcangio, M; Teoh, H1
Cheng, G; Hu, B; Yu, Z1
Juhász, G; Kardos, J; Kékesi, KA; Kovács, I; Nyitrai, G; Szárics, E1
Bonanno, G; Carità, F; Cavazzani, P; Munari, C; Raiteri, M1
Emri, Z; Juhász, G; Kardos, J; Kékesi, KA; Nyitrai, G; Szárics, E1

Other Studies

5 other study(ies) available for cgp 36742 and glutamic acid

ArticleYear
GABA, glutamate and substance P-like immunoreactivity release: effects of novel GABAB antagonists.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Animals; Baclofen; Benzoates; Benzylamines; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Nerve Roots; Stereoisomerism; Substance P

1996
Mechanism of colchicine impairment on learning and memory, and protective effect of CGP36742 in mice.
    Brain research, 1997, Mar-07, Volume: 750, Issue:1-2

    Topics: Animals; Avoidance Learning; Cerebral Cortex; Colchicine; Electroshock; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Infusions, Parenteral; Male; Memory; Mice; Neurons; Neuroprotective Agents; Organophosphorus Compounds; Radioligand Assay; Reaction Time; Receptors, GABA-B; Synaptic Membranes

1997
Effect of CGP 36742 on the extracellular level of neurotransmitter amino acids in the thalamus.
    Neurochemistry international, 1999, Volume: 34, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Aspartic Acid; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Kinetics; Male; Microdialysis; Neurotransmitter Agents; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; tau Proteins; Thalamus

1999
Selective block of rat and human neocortex GABA(B) receptors regulating somatostatin release by a GABA(B) antagonist endowed with cognition enhancing activity.
    Neuropharmacology, 1999, Volume: 38, Issue:11

    Topics: Adult; Animals; Baclofen; Female; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Humans; Male; Middle Aged; Neocortex; Nootropic Agents; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Somatostatin; Synaptosomes

1999
GABA(B) receptor antagonist CGP-36742 enhances somatostatin release in the rat hippocampus in vivo and in vitro.
    European journal of pharmacology, 2003, Oct-08, Volume: 478, Issue:2-3

    Topics: Animals; Electrophysiology; Excitatory Postsynaptic Potentials; Extracellular Space; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Membrane Potentials; Microdialysis; Nerve Endings; Organophosphorus Compounds; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Somatostatin; Somatostatin; Synaptosomes

2003