cgp 36742 has been researched along with gamma-aminobutyric acid in 11 studies
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
Studies (cgp 36742) | Trials (cgp 36742) | Recent Studies (post-2010) (cgp 36742) | Studies (gamma-aminobutyric acid) | Trials (gamma-aminobutyric acid) | Recent Studies (post-2010) (gamma-aminobutyric acid) |
---|---|---|---|---|---|
63 | 3 | 2 | 40,215 | 1,423 | 9,631 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 8 (72.73) | 18.2507 |
2000's | 3 (27.27) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chebib, M; Hanrahan, JR; Hibbs, DE; Johnston, GA; Kim, HL; Kumar, RJ; Salam, NK | 1 |
Moshé, SL; Ortíz, J; Ptachewich, Y; Shinnar, S; Velísek, L; Velísková, J | 1 |
Bowery, NG; Malcangio, M | 2 |
Bowery, NG; Da Silva, H; Malcangio, M | 1 |
Bowery, NG; Malcangio, M; Teoh, H | 1 |
Cheng, G; Hu, B; Yu, Z | 1 |
Juhász, G; Kardos, J; Kékesi, KA; Kovács, I; Nyitrai, G; Szárics, E | 1 |
Bonanno, G; Carità, F; Cavazzani, P; Munari, C; Raiteri, M | 1 |
Emri, Z; Juhász, G; Kardos, J; Kékesi, KA; Nyitrai, G; Szárics, E | 1 |
An, G; Höger, H; Lubec, G; Shim, KS; Sunyer, B | 1 |
11 other study(ies) available for cgp 36742 and gamma-aminobutyric acid
Article | Year |
---|---|
Novel gamma-aminobutyric acid rho1 receptor antagonists; synthesis, pharmacological activity and structure-activity relationships.
Topics: Animals; Female; GABA Antagonists; Ligands; Models, Molecular; Molecular Structure; Oocytes; Structure-Activity Relationship; Xenopus laevis | 2008 |
Age-dependent effects of gamma-aminobutyric acid agents on flurothyl seizures.
Topics: Age Factors; Animals; Anticonvulsants; Baclofen; Convulsants; Flurothyl; GABA Agents; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Organophosphorus Compounds; Phenobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Seizures; Vigabatrin | 1995 |
Gamma-aminobutyric acidB, but not gamma-aminobutyric acidA receptor activation, inhibits electrically evoked substance P-like immunoreactivity release from the rat spinal cord in vitro.
Topics: Animals; Baclofen; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Neurotransmitter Uptake Inhibitors; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Substance P | 1993 |
Plasticity of GABAB receptor in rat spinal cord detected by autoradiography.
Topics: Animals; Autoradiography; Baclofen; Binding Sites; gamma-Aminobutyric Acid; Organophosphorus Compounds; Phosphinic Acids; Rats; Receptors, GABA-B; Spinal Cord; Up-Regulation | 1993 |
GABAB receptor-mediated inhibition of forskolin-stimulated cyclic AMP accumulation in rat spinal cord.
Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Capsaicin; Colforsin; Cyclic AMP; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Norepinephrine; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Cord | 1993 |
GABA, glutamate and substance P-like immunoreactivity release: effects of novel GABAB antagonists.
Topics: Animals; Baclofen; Benzoates; Benzylamines; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Nerve Roots; Stereoisomerism; Substance P | 1996 |
Mechanism of colchicine impairment on learning and memory, and protective effect of CGP36742 in mice.
Topics: Animals; Avoidance Learning; Cerebral Cortex; Colchicine; Electroshock; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Infusions, Parenteral; Male; Memory; Mice; Neurons; Neuroprotective Agents; Organophosphorus Compounds; Radioligand Assay; Reaction Time; Receptors, GABA-B; Synaptic Membranes | 1997 |
Effect of CGP 36742 on the extracellular level of neurotransmitter amino acids in the thalamus.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Aspartic Acid; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Kinetics; Male; Microdialysis; Neurotransmitter Agents; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; tau Proteins; Thalamus | 1999 |
Selective block of rat and human neocortex GABA(B) receptors regulating somatostatin release by a GABA(B) antagonist endowed with cognition enhancing activity.
Topics: Adult; Animals; Baclofen; Female; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Humans; Male; Middle Aged; Neocortex; Nootropic Agents; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Somatostatin; Synaptosomes | 1999 |
GABA(B) receptor antagonist CGP-36742 enhances somatostatin release in the rat hippocampus in vivo and in vitro.
Topics: Animals; Electrophysiology; Excitatory Postsynaptic Potentials; Extracellular Space; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Membrane Potentials; Microdialysis; Nerve Endings; Organophosphorus Compounds; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Somatostatin; Somatostatin; Synaptosomes | 2003 |
Hippocampal levels of phosphorylated protein kinase A (phosphor-S96) are linked to spatial memory enhancement by SGS742.
Topics: Amino Acid Sequence; Animals; Cyclic AMP-Dependent Protein Kinases; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Maze Learning; Memory; Memory Disorders; Mice; Neuroprotective Agents; Organophosphorus Compounds; Phosphorylation; Proto-Oncogene Proteins c-fyn; Receptors, GABA-B; Serine; Somatostatin; Space Perception; Up-Regulation | 2009 |