Page last updated: 2024-09-03

cgp 36742 and gamma-aminobutyric acid

cgp 36742 has been researched along with gamma-aminobutyric acid in 11 studies

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

Compound Research Comparison

Studies
(cgp 36742)
Trials
(cgp 36742)
Recent Studies (post-2010)
(cgp 36742)
Studies
(gamma-aminobutyric acid)
Trials
(gamma-aminobutyric acid)
Recent Studies (post-2010) (gamma-aminobutyric acid)
633240,2151,4239,631

Protein Interaction Comparison

ProteinTaxonomycgp 36742 (IC50)gamma-aminobutyric acid (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 2Rattus norvegicus (Norway rat)0.0292
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0332
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0323
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)2.152
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0333
Sodium- and chloride-dependent GABA transporter 1Homo sapiens (human)5.2623
Sodium- and chloride-dependent taurine transporterHomo sapiens (human)354
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)2.51
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent GABA transporter 1Mus musculus (house mouse)6.349
Sodium- and chloride-dependent GABA transporter 2Mus musculus (house mouse)7.0795
Sodium- and chloride-dependent GABA transporter 3Mus musculus (house mouse)8.1283
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent betaine transporterHomo sapiens (human)6.4082
Sodium- and chloride-dependent GABA transporter 3Homo sapiens (human)3.9953
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0333
GABA theta subunitRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 1Rattus norvegicus (Norway rat)0.0292

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (72.73)18.2507
2000's3 (27.27)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chebib, M; Hanrahan, JR; Hibbs, DE; Johnston, GA; Kim, HL; Kumar, RJ; Salam, NK1
Moshé, SL; Ortíz, J; Ptachewich, Y; Shinnar, S; Velísek, L; Velísková, J1
Bowery, NG; Malcangio, M2
Bowery, NG; Da Silva, H; Malcangio, M1
Bowery, NG; Malcangio, M; Teoh, H1
Cheng, G; Hu, B; Yu, Z1
Juhász, G; Kardos, J; Kékesi, KA; Kovács, I; Nyitrai, G; Szárics, E1
Bonanno, G; Carità, F; Cavazzani, P; Munari, C; Raiteri, M1
Emri, Z; Juhász, G; Kardos, J; Kékesi, KA; Nyitrai, G; Szárics, E1
An, G; Höger, H; Lubec, G; Shim, KS; Sunyer, B1

Other Studies

11 other study(ies) available for cgp 36742 and gamma-aminobutyric acid

ArticleYear
Novel gamma-aminobutyric acid rho1 receptor antagonists; synthesis, pharmacological activity and structure-activity relationships.
    Journal of medicinal chemistry, 2008, Jul-10, Volume: 51, Issue:13

    Topics: Animals; Female; GABA Antagonists; Ligands; Models, Molecular; Molecular Structure; Oocytes; Structure-Activity Relationship; Xenopus laevis

2008
Age-dependent effects of gamma-aminobutyric acid agents on flurothyl seizures.
    Epilepsia, 1995, Volume: 36, Issue:7

    Topics: Age Factors; Animals; Anticonvulsants; Baclofen; Convulsants; Flurothyl; GABA Agents; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Organophosphorus Compounds; Phenobarbital; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Seizures; Vigabatrin

1995
Gamma-aminobutyric acidB, but not gamma-aminobutyric acidA receptor activation, inhibits electrically evoked substance P-like immunoreactivity release from the rat spinal cord in vitro.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: Animals; Baclofen; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Neurotransmitter Uptake Inhibitors; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Substance P

1993
Plasticity of GABAB receptor in rat spinal cord detected by autoradiography.
    European journal of pharmacology, 1993, Nov-30, Volume: 250, Issue:1

    Topics: Animals; Autoradiography; Baclofen; Binding Sites; gamma-Aminobutyric Acid; Organophosphorus Compounds; Phosphinic Acids; Rats; Receptors, GABA-B; Spinal Cord; Up-Regulation

1993
GABAB receptor-mediated inhibition of forskolin-stimulated cyclic AMP accumulation in rat spinal cord.
    Neuroscience letters, 1993, Aug-20, Volume: 158, Issue:2

    Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Capsaicin; Colforsin; Cyclic AMP; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Norepinephrine; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Cord

1993
GABA, glutamate and substance P-like immunoreactivity release: effects of novel GABAB antagonists.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Animals; Baclofen; Benzoates; Benzylamines; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Isonicotinic Acids; Male; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Nerve Roots; Stereoisomerism; Substance P

1996
Mechanism of colchicine impairment on learning and memory, and protective effect of CGP36742 in mice.
    Brain research, 1997, Mar-07, Volume: 750, Issue:1-2

    Topics: Animals; Avoidance Learning; Cerebral Cortex; Colchicine; Electroshock; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Infusions, Parenteral; Male; Memory; Mice; Neurons; Neuroprotective Agents; Organophosphorus Compounds; Radioligand Assay; Reaction Time; Receptors, GABA-B; Synaptic Membranes

1997
Effect of CGP 36742 on the extracellular level of neurotransmitter amino acids in the thalamus.
    Neurochemistry international, 1999, Volume: 34, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Aspartic Acid; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Kinetics; Male; Microdialysis; Neurotransmitter Agents; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; tau Proteins; Thalamus

1999
Selective block of rat and human neocortex GABA(B) receptors regulating somatostatin release by a GABA(B) antagonist endowed with cognition enhancing activity.
    Neuropharmacology, 1999, Volume: 38, Issue:11

    Topics: Adult; Animals; Baclofen; Female; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Humans; Male; Middle Aged; Neocortex; Nootropic Agents; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Somatostatin; Synaptosomes

1999
GABA(B) receptor antagonist CGP-36742 enhances somatostatin release in the rat hippocampus in vivo and in vitro.
    European journal of pharmacology, 2003, Oct-08, Volume: 478, Issue:2-3

    Topics: Animals; Electrophysiology; Excitatory Postsynaptic Potentials; Extracellular Space; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Membrane Potentials; Microdialysis; Nerve Endings; Organophosphorus Compounds; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Somatostatin; Somatostatin; Synaptosomes

2003
Hippocampal levels of phosphorylated protein kinase A (phosphor-S96) are linked to spatial memory enhancement by SGS742.
    Hippocampus, 2009, Volume: 19, Issue:1

    Topics: Amino Acid Sequence; Animals; Cyclic AMP-Dependent Protein Kinases; GABA Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Maze Learning; Memory; Memory Disorders; Mice; Neuroprotective Agents; Organophosphorus Compounds; Phosphorylation; Proto-Oncogene Proteins c-fyn; Receptors, GABA-B; Serine; Somatostatin; Space Perception; Up-Regulation

2009