Page last updated: 2024-09-03

cgp 36742 and colforsin

cgp 36742 has been researched along with colforsin in 2 studies

Compound Research Comparison

Studies
(cgp 36742)
Trials
(cgp 36742)
Recent Studies (post-2010)
(cgp 36742)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
633213,460461,298

Protein Interaction Comparison

ProteinTaxonomycgp 36742 (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bowery, NG; Malcangio, M1
Bowery, NG; Pratt, GD1

Other Studies

2 other study(ies) available for cgp 36742 and colforsin

ArticleYear
GABAB receptor-mediated inhibition of forskolin-stimulated cyclic AMP accumulation in rat spinal cord.
    Neuroscience letters, 1993, Aug-20, Volume: 158, Issue:2

    Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Capsaicin; Colforsin; Cyclic AMP; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Norepinephrine; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Cord

1993
Repeated administration of desipramine and a GABAB receptor antagonist, CGP 36742, discretely up-regulates GABAB receptor binding sites in rat frontal cortex.
    British journal of pharmacology, 1993, Volume: 110, Issue:2

    Topics: Adenylyl Cyclases; Animals; Antidepressive Agents; Autoradiography; Colforsin; Cyclic AMP; Desipramine; GABA-B Receptor Antagonists; Kinetics; Male; Organophosphorus Compounds; Prefrontal Cortex; Rats; Rats, Inbred Strains; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, GABA-B; Transduction, Genetic; Up-Regulation

1993