Page last updated: 2024-09-03

cgp 361a and gr 127935

cgp 361a has been researched along with gr 127935 in 3 studies

Compound Research Comparison

Studies
(cgp 361a)
Trials
(cgp 361a)
Recent Studies (post-2010)
(cgp 361a)
Studies
(gr 127935)
Trials
(gr 127935)
Recent Studies (post-2010) (gr 127935)
2133221028

Protein Interaction Comparison

ProteinTaxonomycgp 361a (IC50)gr 127935 (IC50)
5-hydroxytryptamine receptor 1DHomo sapiens (human)0.052
Sodium-dependent serotonin transporterHomo sapiens (human)1

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davidson, C; Stamford, JA2
Dawson, LA; Nguyen, HQ1

Other Studies

3 other study(ies) available for cgp 361a and gr 127935

ArticleYear
5-HT1B/D antagonists potentiate paroxetine's effect on 5-HT efflux in the lateral geniculate nucleus: in vitro voltammetric data.
    Biochemical Society transactions, 1997, Volume: 25, Issue:1

    Topics: Animals; Electrochemistry; Geniculate Bodies; Male; Methiothepin; Oxadiazoles; Paroxetine; Piperazines; Propanolamines; Pyridines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1997
Synergism of 5-HT 1B/D antagonists with paroxetine on serotonin efflux in rat ventral lateral geniculate nucleus slices.
    Brain research bulletin, 1997, Volume: 43, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Drug Synergism; Geniculate Bodies; Male; Oxadiazoles; Paroxetine; Piperazines; Propanolamines; Rats; Rats, Wistar; Serotonin

1997
The role of 5-HT(1A) and 5-HT(1B/1D) receptors on the modulation of acute fluoxetine-induced changes in extracellular 5-HT: the mechanism of action of (+/-)pindolol.
    Neuropharmacology, 2000, Apr-03, Volume: 39, Issue:6

    Topics: Animals; Autoreceptors; Drug Synergism; Extracellular Space; Fluoxetine; Male; Microdialysis; Oxadiazoles; Pindolol; Piperazines; Propanolamines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists

2000