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cgp 35348 and sk&f 97541

cgp 35348 has been researched along with sk&f 97541 in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (33.33)18.2507
2000's6 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baumann, PA; Bernasconi, R; Diel, PJ; Froestl, W; Hall, RG; Maier, L; Melillo, V; Mickel, SJ; Strub, D; von Sprecher, G1
Howson, W; Lacey, MG; Seabrook, GR1
Bon, C; Galvan, M1
Carter, LP; Chen, W; Coop, A; France, CP; Koek, W; Lamb, RJ; Wu, H1
Carter, LP; Coop, A; France, CP; Koek, W; Wu, H1
Carter, LP; Chen, W; Coop, A; France, CP; Koek, W1
Coop, A; Koek, W; Mercer, SL1
Balcar, VJ; Griffin, JL; Nasrallah, FA; Rae, C1
Coop, A; France, CP; Koek, W; Mercer, SL1

Other Studies

9 other study(ies) available for cgp 35348 and sk&f 97541

ArticleYear
Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.
    Journal of medicinal chemistry, 1995, Aug-18, Volume: 38, Issue:17

    Topics: Administration, Oral; Amnesia; Animals; Cerebral Cortex; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Learning; Long-Term Potentiation; Magnetic Resonance Spectroscopy; Phosphinic Acids; Protein Binding; Radioligand Assay; Rats; Receptors, GABA-B; Structure-Activity Relationship

1995
Electrophysiological characterization of potent agonists and antagonists at pre- and postsynaptic GABAB receptors on neurones in rat brain slices.
    British journal of pharmacology, 1990, Volume: 101, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Brain; Corpus Striatum; Electrophysiology; GABA-A Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Neurons; Organophosphorus Compounds; Rats; Receptors, GABA-A; Substantia Nigra; Synapses

1990
Electrophysiological actions of GABAB agonists and antagonists in rat dorso-lateral septal neurones in vitro.
    British journal of pharmacology, 1996, Volume: 118, Issue:4

    Topics: Analysis of Variance; Animals; Baclofen; Benzylamines; Dose-Response Relationship, Drug; Electrophysiology; GABA Agonists; GABA Antagonists; GABA-B Receptor Antagonists; In Vitro Techniques; Male; Membrane Potentials; Organophosphorus Compounds; Phosphinic Acids; Propanolamines; Rats; Receptors, GABA-B; Septal Nuclei

1996
Discriminative stimulus effects of gamma-hydroxybutyrate (GHB) in rats discriminating GHB from baclofen and diazepam.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:1

    Topics: 4-Butyrolactone; Anesthetics, Intravenous; Animals; Baclofen; Benzocycloheptenes; Benzylamines; Butylene Glycols; Diazepam; Discrimination, Psychological; Dithiothreitol; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Sodium Oxybate

2005
Discriminative stimulus effects of flumazenil: perceptual masking by baclofen, and lack of substitution with gamma-hydroxybutyrate and its precursors 1,4-butanediol and gamma-butyrolactone.
    Behavioural pharmacology, 2006, Volume: 17, Issue:3

    Topics: 4-Butyrolactone; Animals; Baclofen; Benzocycloheptenes; Butylene Glycols; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Flumazenil; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Organophosphorus Compounds; Sodium Oxybate

2006
Discriminative stimulus effects of GHB and GABA(B) agonists are differentially attenuated by CGP35348.
    European journal of pharmacology, 2006, May-24, Volume: 538, Issue:1-3

    Topics: Analysis of Variance; Animals; Baclofen; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Male; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Sodium Oxybate

2006
Cataleptic effects of gamma-hydroxybutyrate (GHB), its precursor gamma-butyrolactone (GBL), and GABAB receptor agonists in mice: differential antagonism by the GABAB receptor antagonist CGP35348.
    Psychopharmacology, 2007, Volume: 192, Issue:3

    Topics: 4-Butyrolactone; Animals; Baclofen; Catalepsy; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Male; Mice; Mice, Inbred C57BL; Narcolepsy; Organophosphorus Compounds; Receptors, GABA-B; Sodium Oxybate; Substance-Related Disorders

2007
Understanding your inhibitions: modulation of brain cortical metabolism by GABA(B) receptors.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2007, Volume: 27, Issue:8

    Topics: Animals; Baclofen; Benzylamines; Carbon Isotopes; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Guinea Pigs; Molecular Structure; Morpholines; Nuclear Magnetic Resonance, Biomolecular; Organophosphorus Compounds; Phosphinic Acids; Principal Component Analysis; Receptors, GABA-B

2007
Behavioral effects of gamma-hydroxybutyrate, its precursor gamma-butyrolactone, and GABA(B) receptor agonists: time course and differential antagonism by the GABA(B) receptor antagonist 3-aminopropyl(diethoxymethyl)phosphinic acid (CGP35348).
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 330, Issue:3

    Topics: 4-Butyrolactone; Anesthetics, Intravenous; Animals; Baclofen; Columbidae; Conditioning, Operant; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Injections, Intramuscular; Kinetics; Organophosphorus Compounds; Sodium Oxybate

2009