Page last updated: 2024-08-26

cgp 35348 and phaclofen

cgp 35348 has been researched along with phaclofen in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's23 (92.00)18.2507
2000's2 (8.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Douglas, WW; Kongsamut, S; Shibuya, I1
Bonanno, G; Raiteri, M2
Bonanno, G; Gemignani, A; Lanza, M; Pende, M; Raiteri, M; Vellebuona, F1
Bartolini, A; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P1
Howson, W; Lacey, MG; Seabrook, GR1
Karlsson, G; Olpe, HR1
Bittiger, H; Brugger, F; Fagg, G; Froestl, W; Hall, RG; Karlsson, G; Olpe, HR; Pozza, MF; Steinmann, M; Van Riezen, H1
Humeniuk, RE; Kerr, DI; Ong, J; White, JM1
Banerjee, PK; Snead, OC1
Slaughter, MM; Tian, N1
Bonanno, G; Cavazzani, P; Fassio, A; Raiteri, M1
Humeniuk, RE; Ong, J; White, JM1
Bonanno, G; Gemignani, A; Paudice, P; Raiteri, M1
Finch, DM; Gigg, J; Tan, AM1
Bonanno, G; Lanza, M; Pende, M; Raiteri, M1
Lewis, DV; Mott, DD; Swartzwelder, HS; Wilson, WA; Xie, CW1
Hammond, DL; McGowan, MK1
DiScenna, PG; Nowicky, AV; Teyler, TJ1
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G1
Brailowsky, S; Di Scala, G; Meneses, S; Montiel, T1
Snead, OC1
Chowdhury, SA; Kawashima, T; Konishi, T; Matsunami, K1
Chowdhury, SA; Matsunami, KI1
Balcar, VJ; Griffin, JL; Nasrallah, FA; Rae, C1

Other Studies

25 other study(ies) available for cgp 35348 and phaclofen

ArticleYear
Effectiveness of GABAB antagonists in inhibiting baclofen-induced reductions in cytosolic free Ca concentration in isolated melanotrophs of rat.
    British journal of pharmacology, 1992, Volume: 105, Issue:4

    Topics: Animals; Baclofen; Calcium; Cytosol; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Organophosphorus Compounds; Pituitary Gland, Anterior; Rats; Rats, Inbred Strains

1992
Functional evidence for multiple gamma-aminobutyric acidB receptor subtypes in the rat cerebral cortex.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:1

    Topics: Animals; Baclofen; Cerebral Cortex; Chromatography, High Pressure Liquid; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Male; Organophosphorus Compounds; Peptides; Rats; Rats, Inbred Strains; Receptors, GABA-A

1992
Pharmacologically distinct GABAB receptor subtypes modulate neurotransmitter release in the rat brain cortex.
    Advances in biochemical psychopharmacology, 1992, Volume: 47

    Topics: Animals; Baclofen; Bicuculline; Cerebral Cortex; GABA-A Receptor Antagonists; Glutamates; Glutamic Acid; Muscimol; Neurotransmitter Agents; Organophosphorus Compounds; Rats; Receptors, GABA-A; Somatostatin; Synaptosomes

1992
CGP 35348, a new GABAB antagonist, prevents antinociception and muscle-relaxant effect induced by baclofen.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Analgesics; Animals; Baclofen; GABA Antagonists; GABA-A Receptor Antagonists; Injections, Intraventricular; Male; Mice; Morphine; Muscle Relaxation; Muscles; Organophosphorus Compounds; Oxotremorine; Postural Balance; Rats; Rats, Inbred Strains; Reaction Time

1991
Electrophysiological characterization of potent agonists and antagonists at pre- and postsynaptic GABAB receptors on neurones in rat brain slices.
    British journal of pharmacology, 1990, Volume: 101, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Brain; Corpus Striatum; Electrophysiology; GABA-A Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Neurons; Organophosphorus Compounds; Rats; Receptors, GABA-A; Substantia Nigra; Synapses

1990
The effects of baclofen and two GABAB-receptor antagonists on long-term potentiation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:2

    Topics: Animals; Baclofen; Electric Stimulation; GABA-A Receptor Antagonists; Hippocampus; In Vitro Techniques; Male; Neurons; Organophosphorus Compounds; Rats; Rats, Inbred Strains; Synapses

1990
CGP 35348: a centrally active blocker of GABAB receptors.
    European journal of pharmacology, 1990, Oct-02, Volume: 187, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Animals, Newborn; Anticonvulsants; Baclofen; Behavior, Animal; Brain Chemistry; Cyclic AMP; Electrophysiology; Hippocampus; In Vitro Techniques; Iontophoresis; Organophosphorus Compounds; Postural Balance; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spinal Cord

1990
Characterization of GABAB ligands in vivo.
    General pharmacology, 1995, Volume: 26, Issue:2

    Topics: Animals; Baclofen; beta-Alanine; Drug Interactions; Female; GABA Antagonists; GABA-B Receptor Antagonists; Ligands; Mice; Mice, Inbred BALB C; Muscle Relaxation; Organophosphorus Compounds

1995
Presynaptic gamma-hydroxybutyric acid (GHB) and gamma-aminobutyric acidB (GABAB) receptor-mediated release of GABA and glutamate (GLU) in rat thalamic ventrobasal nucleus (VB): a possible mechanism for the generation of absence-like seizures induced by GH
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 273, Issue:3

    Topics: Action Potentials; Animals; Baclofen; Epilepsy, Absence; Extracellular Space; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Male; Organophosphorus Compounds; Potassium; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, GABA-B; Sodium Oxybate; Thalamic Nuclei

1995
Pharmacology of the GABAB receptor in amphibian retina.
    Brain research, 1994, Oct-17, Volume: 660, Issue:2

    Topics: Ambystoma; Animals; Baclofen; Butylamines; Evoked Potentials; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Membrane Potentials; Necturus; Organophosphorus Compounds; Propylamines; Receptors, GABA-B; Retina; Retinal Ganglion Cells; Stereoisomerism; Structure-Activity Relationship

1994
Characterization of the GABA autoreceptor in human neocortex as a pharmacological subtype of the GABAB receptor.
    European journal of pharmacology, 1994, Oct-03, Volume: 263, Issue:3

    Topics: Adolescent; Adult; Aged; Animals; Baclofen; Benzylamines; Binding, Competitive; Brain Neoplasms; Cerebral Cortex; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Humans; Male; Middle Aged; Organophosphorus Compounds; Phosphinic Acids; Rats; Receptors, GABA-B

1994
The effects of GABAB ligands on alcohol withdrawal in mice.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:3

    Topics: Animals; Baclofen; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Ethanol; Female; GABA Antagonists; GABA-B Receptor Antagonists; Mice; Mice, Inbred C57BL; Organophosphorus Compounds; Phenylalanine; Receptors, GABA-B; Seizures; Substance Withdrawal Syndrome; Tremor

1994
Pharmacological discrimination between gamma-aminobutyric acid type B receptors regulating cholecystokinin and somatostatin release from rat neocortex synaptosomes.
    Molecular pharmacology, 1994, Volume: 46, Issue:3

    Topics: Animals; Baclofen; Benzylamines; Cerebral Cortex; Cholecystokinin; GABA Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Ligands; Male; Organophosphorus Compounds; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Somatostatin; Synaptosomes

1994
Glutamatergic hippocampal formation projections to prefrontal cortex in the rat are regulated by GABAergic inhibition and show convergence with glutamatergic projections from the limbic thalamus.
    Hippocampus, 1994, Volume: 4, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Brain Mapping; Electric Stimulation; Electrophysiology; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Limbic System; Male; Neurons; Organophosphorus Compounds; Piperazines; Prefrontal Cortex; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Thalamus

1994
Release of endogenous glutamic and aspartic acids from cerebrocortex synaptosomes and its modulation through activation of a gamma-aminobutyric acidB (GABAB) receptor subtype.
    Brain research, 1993, Feb-26, Volume: 604, Issue:1-2

    Topics: Animals; Aspartic Acid; Baclofen; Bicuculline; Cerebral Cortex; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Kinetics; Male; Organophosphorus Compounds; Picrotoxin; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptosomes

1993
GABAB autoreceptors mediate activity-dependent disinhibition and enhance signal transmission in the dentate gyrus.
    Journal of neurophysiology, 1993, Volume: 69, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Culture Techniques; GABA-A Receptor Antagonists; Hippocampus; Male; Membrane Potentials; Nerve Fibers; Neural Inhibition; Organophosphorus Compounds; Picrotoxin; Quinoxalines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Synaptic Transmission; Theta Rhythm

1993
Intrathecal GABAB antagonists attenuate the antinociception produced by microinjection of L-glutamate into the ventromedial medulla of the rat.
    Brain research, 1993, Apr-02, Volume: 607, Issue:1-2

    Topics: Analgesics; Animals; Baclofen; Basal Ganglia; Behavior, Animal; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA-A Receptor Antagonists; Glutamates; Glutamic Acid; Injections, Spinal; Medulla Oblongata; Methysergide; Microinjections; Organophosphorus Compounds; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-A; Skin Temperature

1993
The development of GABAB-mediated activity in the rat dentate gyrus.
    Brain research. Developmental brain research, 1994, Feb-18, Volume: 77, Issue:2

    Topics: Animals; Baclofen; Electric Stimulation; Evoked Potentials; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Hippocampus; In Vitro Techniques; Organophosphorus Compounds; Rats; Receptors, GABA-A; Receptors, GABA-B

1994
gamma-Aminobutyric acid (GABA) autoreceptors in rat cerebral cortex and spinal cord represent pharmacologically distinct subtypes of the GABAB receptor.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: Animals; Baclofen; Cerebral Cortex; gamma-Aminobutyric Acid; Male; Organophosphorus Compounds; Potassium; Rats; Rats, Wistar; Receptors, GABA-A; Spinal Cord; Synaptosomes

1993
Role of peripheral GABAB receptors in the regulation of pepsinogen secretion in anaesthetized rats.
    European journal of pharmacology, 1995, Dec-27, Volume: 294, Issue:1

    Topics: Anesthesia; Animals; Baclofen; Capsaicin; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Gastric Mucosa; Male; Organophosphorus Compounds; p-Methoxy-N-methylphenethylamine; Pepsinogens; Perfusion; Rats; Rats, Wistar; Receptors, GABA-B; Vagotomy

1995
Effects of GABAB receptor antagonists on two models of focal epileptogenesis.
    Brain research, 1995, Dec-08, Volume: 702, Issue:1-2

    Topics: Animals; Baclofen; Disease Models, Animal; Epilepsies, Partial; GABA Antagonists; GABA-B Receptor Antagonists; Male; Organophosphorus Compounds; Rats; Rats, Wistar; Time Factors

1995
Relation of the [3H] gamma-hydroxybutyric acid (GHB) binding site to the gamma-aminobutyric acidB (GABAB) receptor in rat brain.
    Biochemical pharmacology, 1996, Oct-25, Volume: 52, Issue:8

    Topics: Animals; Autoradiography; Baclofen; Benzocycloheptenes; Binding Sites; Brain; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Guanosine Triphosphate; In Vitro Techniques; Male; Organophosphorus Compounds; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Seizures; Sodium Oxybate; Stereoisomerism

1996
GABAergic characteristics of transcallosal activity of cat motor cortical neurons.
    Neuroscience research, 1996, Volume: 26, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Cats; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Motor Cortex; Organophosphorus Compounds

1996
GABA-B-related activity in processing of transcallosal response in cat motor cortex.
    Journal of neuroscience research, 2002, May-15, Volume: 68, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Cats; Corpus Callosum; Female; GABA Agonists; GABA Antagonists; Male; Motor Cortex; Organophosphorus Compounds; Receptors, GABA-A; Receptors, GABA-B; Receptors, Presynaptic; Synaptic Transmission

2002
Understanding your inhibitions: modulation of brain cortical metabolism by GABA(B) receptors.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2007, Volume: 27, Issue:8

    Topics: Animals; Baclofen; Benzylamines; Carbon Isotopes; Cerebral Cortex; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; Guinea Pigs; Molecular Structure; Morpholines; Nuclear Magnetic Resonance, Biomolecular; Organophosphorus Compounds; Phosphinic Acids; Principal Component Analysis; Receptors, GABA-B

2007