Page last updated: 2024-09-03

cgp 28392 and verapamil

cgp 28392 has been researched along with verapamil in 9 studies

Compound Research Comparison

Studies
(cgp 28392)
Trials
(cgp 28392)
Recent Studies (post-2010)
(cgp 28392)
Studies
(verapamil)
Trials
(verapamil)
Recent Studies (post-2010) (verapamil)
761217,6211,5272,067

Protein Interaction Comparison

ProteinTaxonomycgp 28392 (IC50)verapamil (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)6.8
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)0.2
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.297
ATP-dependent translocase ABCB1Mus musculus (house mouse)2
ATP-dependent translocase ABCB1Homo sapiens (human)2.2346
Cytochrome P450 3A4Homo sapiens (human)3.8008
Alpha-2A adrenergic receptorHomo sapiens (human)0.579
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)3.02
ATP-dependent translocase ABCB1Mus musculus (house mouse)10
Catechol O-methyltransferaseHomo sapiens (human)0.2
Potassium voltage-gated channel subfamily A member 3Homo sapiens (human)8
Histamine H2 receptorHomo sapiens (human)2.59
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.442
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.297
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)3.02
Sodium-dependent serotonin transporterHomo sapiens (human)0.24
Multidrug resistance-associated protein 1 Homo sapiens (human)5.598
D(3) dopamine receptorHomo sapiens (human)0.186
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.165
5-hydroxytryptamine receptor 7Cavia porcellus (domestic guinea pig)6.8
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)0.2
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.3945
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)0.2
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)0.175
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)1.1934

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19907 (77.78)18.7374
1990's2 (22.22)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ikemoto, T; Ito, K; Takakura, S1
Barhanin, J; Borsotto, M; Fosset, M; Galizzi, JP; Lazdunski, M; Renaud, JF; Romey, G; Schmid, A1
Matsumura, Y; Morimoto, S; Sasaki, Y; Shinyama, H; Uriu, T1
Jonkman, FA; Korstanje, C; Van Kemenade, JE; Van Zwieten, PA1
Karaki, H; Nagase, H; Ozaki, H; Urakawa, N; Weiss, GB1
Malaisse, WJ; Mathias, PC1
Groth, H; Locher, R; Neyses, L; Stimpel, M; Vetter, W1
Lazdunski, M; Méaux, JP; Renaud, JF; Romey, G; Schmid, A1
Krieger, A1

Other Studies

9 other study(ies) available for cgp 28392 and verapamil

ArticleYear
Involvement of Ca2+ influx-induced Ca2+ release in contractions of intact vascular smooth muscles.
    The American journal of physiology, 1991, Volume: 261, Issue:5 Pt 2

    Topics: Animals; Aorta, Thoracic; Biological Transport, Active; Calcium; Calcium Channel Agonists; Calcium Channels; Guinea Pigs; In Vitro Techniques; Kinetics; Magnesium; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Pyridines; Ryanodine; Verapamil

1991
Dihydropyridine-sensitive Ca2+ channels: molecular properties of interaction with Ca2+ channel blockers, purification, subunit structure, and differentiation.
    Journal of cardiovascular pharmacology, 1986, Volume: 8 Suppl 8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Affinity Labels; Animals; Bepridil; Binding, Competitive; Calcium; Calcium Channel Blockers; Calcium Channels; Chick Embryo; Cholic Acids; Diltiazem; Ion Channels; Isradipine; Kinetics; Macromolecular Substances; Molecular Weight; Muscles; Myocardial Contraction; Oxadiazoles; Pyridines; Pyrrolidines; Receptors, Nicotinic; Verapamil

1986
Inhibitory effects of calcium channel agonists on renin release from rat kidney cortical slices.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dose-Response Relationship, Drug; Imidazoles; Ion Channels; Kidney Cortex; Male; Nifedipine; Pyridines; Rats; Rats, Inbred Strains; Renin; Trifluoperazine; Verapamil

1987
Bay k 8644, a calcium entry promoter, as an antidote in verapamil intoxication in rabbits.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 287, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aminopyridines; Animals; Antidotes; Atrioventricular Node; Blood Pressure; Cardiovascular Agents; Electrocardiography; Female; Heart Rate; Hydrogen-Ion Concentration; In Vitro Techniques; Ion Channels; Male; Pyridines; Rabbits; Verapamil

1987
Effects of the calcium channel facilitator, CGP 28,392, on different modes of contraction in smooth muscle of rabbit and rat aortae and guinea-pig taenia caeci.
    British journal of pharmacology, 1986, Volume: 89, Issue:2

    Topics: Animals; Aorta, Thoracic; Calcium Channel Blockers; Cecum; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Pyridines; Rabbits; Rats; Rats, Inbred Strains; Verapamil

1986
Stimulation of insulin release by an organic calcium agonist.
    Diabetologia, 1985, Volume: 28, Issue:3

    Topics: Animals; Barium; Calcium; Dose-Response Relationship, Drug; Glucose; Insulin; Islets of Langerhans; Pyridines; Rats; Theophylline; Verapamil

1985
Human red blood cells--an ideal model system for the action of calcium agonists and antagonists.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1984, Volume: 2, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Erythrocytes; Humans; Ion Channels; Nicardipine; Nifedipine; Nitrendipine; Pyridines; Stimulation, Chemical; Verapamil

1984
Activation of the voltage-dependent Ca2+ channel in rat heart cells by dihydropyridine derivatives.
    Biochemical and biophysical research communications, 1984, Nov-30, Volume: 125, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bepridil; Calcium; Dose-Response Relationship, Drug; Ion Channels; Myocardium; Nifedipine; Pyridines; Pyrrolidines; Rats; Rats, Inbred Strains; Time Factors; Verapamil

1984
Effect of the Ca2+ channel activator CGP 28392 on reactivation of oxygen evolution of Ca(2+)-depleted photosystem II.
    FEBS letters, 1995, Jun-26, Volume: 367, Issue:2

    Topics: Calcium; Calcium Channel Agonists; Calcium Chloride; Hydrogen-Ion Concentration; Nifedipine; Oxygen; Photosynthetic Reaction Center Complex Proteins; Photosystem II Protein Complex; Pyridines; Verapamil

1995