Page last updated: 2024-09-03

cgp 28392 and nitrendipine

cgp 28392 has been researched along with nitrendipine in 14 studies

Compound Research Comparison

Studies
(cgp 28392)
Trials
(cgp 28392)
Recent Studies (post-2010)
(cgp 28392)
Studies
(nitrendipine)
Trials
(nitrendipine)
Recent Studies (post-2010) (nitrendipine)
76122,17037883

Protein Interaction Comparison

ProteinTaxonomycgp 28392 (IC50)nitrendipine (IC50)
G-protein coupled receptor 55Homo sapiens (human)1.4652
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)0.0152
Cytochrome P450 2C9 Homo sapiens (human)0.3
Voltage-dependent L-type calcium channel subunit alpha-1CRattus norvegicus (Norway rat)0.0013
Voltage-dependent L-type calcium channel subunit alpha-1DRattus norvegicus (Norway rat)0.0013
Cytochrome P450 2C19Homo sapiens (human)3
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)0.0152
Voltage-dependent L-type calcium channel subunit alpha-1SRattus norvegicus (Norway rat)0.0013
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)10
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)0.0152
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)0.0152
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1CHomo sapiens (human)1.85

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-199010 (71.43)18.7374
1990's4 (28.57)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Frank, GB1
Akimoto, T; Ariyoshi, S; Fujisue, T; Ichida, S; Wada, T1
Criscione, L; Meier, M; Rogg, H; Truog, A1
Carpenter, CL; Greenberg, DA; Messing, RO1
Aunis, D; Gandía, L; García, AG; Ladona, MG1
Plant, TD2
Montague, W; Morgan, NG; Rumford, GM; Short, CD1
Bühler, FR; Erne, P; Resink, TJ1
Groth, H; Locher, R; Neyses, L; Stimpel, M; Vetter, W1
Freedman, SB; Miller, RJ1
Bühler, FR; Bürgisser, E; Dubach, B; Erne, P; Kühnis, H; Meier, M; Rogg, H1
Caviedes, P; Caviedes, R; Jaimovich, E; Olivares, E; Salas, K1
Chaylakhyan, LM; Grishchenko, VM; Zherelova, OM1

Other Studies

14 other study(ies) available for cgp 28392 and nitrendipine

ArticleYear
Dihydropyridine calcium channel antagonists block and agonists potentiate high potassium contractures but not twitches in frog skeletal muscle.
    The Japanese journal of physiology, 1990, Volume: 40, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; In Vitro Techniques; Muscle Contraction; Nifedipine; Nitrendipine; Potassium; Pyridines; Rana pipiens

1990
Effects of calcium channel agonists (BAY K 8644, CGP28392 and YC-170) on 45Ca uptake by rat uterine segments.
    Japanese journal of pharmacology, 1991, Volume: 56, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Female; Nifedipine; Nitrendipine; Potassium Chloride; Pyridines; Rats; Rats, Inbred Strains; Uterus

1991
In vitro comparative studies of the calcium-entry activators YC-170, CGP 28392, and BAY K 8644.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Biological Transport; Calcium; Guinea Pigs; Heart Rate; In Vitro Techniques; Ion Channels; Male; Mesentery; Myocardial Contraction; Nifedipine; Nitrendipine; Pyridines; Rats; Vasoconstriction

1985
Depolarization-dependent binding of the calcium channel antagonist, (+)-[3H]PN200-110, to intact cultured PC12 cells.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Cells, Cultured; Isradipine; Kinetics; Membrane Potentials; Nifedipine; Nitrendipine; Onium Compounds; Organophosphorus Compounds; Oxadiazoles; Potassium; Pyridines; Tritium

1986
Dihydropyridine modulation of the chromaffin cell secretory response.
    Journal of neurochemistry, 1987, Volume: 48, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cats; Cell Membrane Permeability; Chromaffin Granules; Chromaffin System; Female; Male; Muscarine; Nicotine; Nitrendipine; Norepinephrine; Perfusion; Potassium; Pyridines

1987
Ion channels in pancreatic B cells.
    Journal of protein chemistry, 1989, Volume: 8, Issue:3

    Topics: Action Potentials; Adenosine Triphosphate; Animals; Calcium Channels; Cell Membrane; Cell Membrane Permeability; Ion Channels; Islets of Langerhans; Membrane Potentials; Mice; Nitrendipine; Potassium Channels; Pyridines; Sodium Channels

1989
Properties and calcium-dependent inactivation of calcium currents in cultured mouse pancreatic B-cells.
    The Journal of physiology, 1988, Volume: 404

    Topics: Action Potentials; Animals; Barium; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Egtazic Acid; Islets of Langerhans; Membrane Potentials; Mice; Nitrendipine; Pyridines; Sodium; Time Factors

1988
Effects of the calcium-channel agonist CGP 28392 on insulin secretion from isolated rat islets of Langerhans.
    The Biochemical journal, 1985, Nov-01, Volume: 231, Issue:3

    Topics: Animals; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nifedipine; Nitrendipine; Norepinephrine; Pyridines; Rats; Rats, Inbred Strains; Stimulation, Chemical

1985
The influence of CGP 28392, a 1,4-dihydropyridine, on human platelet calcium and cyclic AMP metabolism.
    European journal of pharmacology, 1985, Jul-31, Volume: 113, Issue:3

    Topics: Alprostadil; Blood Platelets; Calcium; Calcium Channel Blockers; Cyclic AMP; Humans; In Vitro Techniques; Kinetics; Nifedipine; Nitrendipine; Phosphorylation; Protein Kinases; Pyridines

1985
Human red blood cells--an ideal model system for the action of calcium agonists and antagonists.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1984, Volume: 2, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Erythrocytes; Humans; Ion Channels; Nicardipine; Nifedipine; Nitrendipine; Pyridines; Stimulation, Chemical; Verapamil

1984
Calcium channel activation: a different type of drug action.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:17

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cadmium; Calcium; Calcium Channel Blockers; Cell Line; Diltiazem; Gallopamil; Glioma; Hybrid Cells; Ion Channels; Kinetics; Mice; Neuroblastoma; Nifedipine; Nitrendipine; Pyridines; Rats

1984
Enhancement of calcium influx in human platelets by CGP 28392, a novel dihydropyridine.
    Biochemical and biophysical research communications, 1984, Feb-14, Volume: 118, Issue:3

    Topics: Animals; Blood Platelets; Calcium; Calcium Channel Blockers; Cell Membrane; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Ion Channels; Myocardium; Nifedipine; Nitrendipine; Pyridines

1984
Calcium fluxes, ion currents and dihydropyridine receptors in a new immortal cell line from rat heart muscle.
    Journal of molecular and cellular cardiology, 1993, Volume: 25, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Calcium Channels, L-Type; Cell Differentiation; Cell Division; Cell Line; Heart; Immunohistochemistry; Male; Membrane Potentials; Muscle Proteins; Myocardium; Nitrendipine; Pyridines; Rats; Rats, Inbred F344; Time Factors; Tritium

1993
Blockers of Ca2+ channels in the plasmalemma of perfused Characeae cells.
    Comparative biochemistry and physiology. Pharmacology, toxicology and endocrinology, 1994, Volume: 107, Issue:3

    Topics: Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Chlorophyta; Dihydropyridines; Membrane Potentials; Nifedipine; Nitrendipine; Perfusion; Pyridines

1994