Page last updated: 2024-09-03

cgp 28392 and nicardipine

cgp 28392 has been researched along with nicardipine in 2 studies

Compound Research Comparison

Studies
(cgp 28392)
Trials
(cgp 28392)
Recent Studies (post-2010)
(cgp 28392)
Studies
(nicardipine)
Trials
(nicardipine)
Recent Studies (post-2010) (nicardipine)
76122,646444312

Protein Interaction Comparison

ProteinTaxonomycgp 28392 (IC50)nicardipine (IC50)
Bile salt export pumpHomo sapiens (human)8.314
ATP-dependent translocase ABCB1Mus musculus (house mouse)8
ATP-dependent translocase ABCB1Homo sapiens (human)4.2992
Cytochrome P450 3A4Homo sapiens (human)0.42
Cytochrome P450 2C9 Homo sapiens (human)1.69
ATP-dependent translocase ABCB1Mus musculus (house mouse)2.5
Cytochrome P450 2J2Homo sapiens (human)1.69
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)4.925
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)4.8

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19901 (50.00)18.7374
1990's1 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ikeda, M; Karaki, H; Koike, H; Ozaki, H; Sada, T; Sato, K1
Groth, H; Locher, R; Neyses, L; Stimpel, M; Vetter, W1

Other Studies

2 other study(ies) available for cgp 28392 and nicardipine

ArticleYear
Cytosolic free calcium of aorta in hypertensive rats. Chronic inhibition of angiotensin converting enzyme.
    Hypertension (Dallas, Tex. : 1979), 1990, Volume: 16, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Aorta; Calcium; Cytosol; Hypertension; Male; Muscle Contraction; Nicardipine; Pyridines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Thiazepines

1990
Human red blood cells--an ideal model system for the action of calcium agonists and antagonists.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1984, Volume: 2, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Erythrocytes; Humans; Ion Channels; Nicardipine; Nifedipine; Nitrendipine; Pyridines; Stimulation, Chemical; Verapamil

1984