Page last updated: 2024-09-03

cgp 28392 and bay-k-8644

cgp 28392 has been researched along with bay-k-8644 in 41 studies

Compound Research Comparison

Studies
(cgp 28392)
Trials
(cgp 28392)
Recent Studies (post-2010)
(cgp 28392)
Studies
(bay-k-8644)
Trials
(bay-k-8644)
Recent Studies (post-2010) (bay-k-8644)
76122,5550144

Research

Studies (41)

TimeframeStudies, this research(%)All Research%
pre-199027 (65.85)18.7374
1990's12 (29.27)18.2507
2000's1 (2.44)29.6817
2010's1 (2.44)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barsys, V; Garaliene, V; Krauze, A; Mačys, A; Vigante, B1
Gainullin, R; Saxon, M1
Kunert-Radek, J; Lyson, K; Pawlikowski, M; Stepien, H1
Bolger, GT; Campbell, N; Crowley, M; McKay, DW; O'Neill, SK; Triggle, CR1
Fraser, S; Kenny, BA; Kilpatrick, AT; Spedding, M1
Frank, GB1
Alonso, MJ; Marín, J; Rico, I; Salaices, M2
Halushka, PV; Mais, DE; Mayeux, PR1
Dannies, PS; Law, GJ; Pachter, JA1
Akimoto, T; Ariyoshi, S; Fujisue, T; Ichida, S; Wada, T1
Marinov, BS; Saxon, ME1
Brooks, HL; Gross, GJ; Preuss, KC; Warltier, DC1
Affolter, H; Coronado, R1
Brill, DM; Fozzard, HA1
Criscione, L; Meier, M; Rogg, H; Truog, A1
Schramm, M; Towart, R1
Jakobsen, P; Mikkelsen, EO; Nyborg, NC1
Carpenter, CL; Greenberg, DA; Messing, RO1
Bevan, JA; Hwa, JJ1
Aunis, D; Gandía, L; García, AG; Ladona, MG1
Barhanin, J; Borsotto, M; Fosset, M; Galizzi, JP; Lazdunski, M; Renaud, JF; Romey, G; Schmid, A1
Matsumura, Y; Morimoto, S; Sasaki, Y; Shinyama, H; Uriu, T1
Malaisse, WJ; Malaisse-Lagae, F; Sener, A1
Asem, EK; Tsang, BK1
Jonkman, FA; Korstanje, C; Van Kemenade, JE; Van Zwieten, PA1
Costa, G; Mikkelsen, EO; Nyborg, NC1
Heisler, S; MacDonald, JF; Miljkovic, Z1
Alonso, MJ; Fernández-Alfonso, MS; Marín, J; Rico, I; Salaices, M; Sánchez-Ferrer, CF1
Filippov, A; Kobrinsky, E; Porotikov, V; Saxon, M1
Panzer-Knodle, S; Papaioannou, S; Yang, PC1
Fichtner, H; Herzig, JW; Kohlhardt, M1
Groth, H; Locher, R; Neyses, L; Stimpel, M; Vetter, W1
Kokubun, S; Reuter, H1
Freedman, SB; Miller, RJ1
Lazdunski, M; Méaux, JP; Renaud, JF; Romey, G; Schmid, A1
Hof, A; Hof, RP; Loutzenhiser, R; Rüegg, UT1
Nakamura, KT; Pichoff, BE; Uyehara, CF1
Caviedes, P; Caviedes, R; Jaimovich, E; Olivares, E; Salas, K1
Kanno, M; Nakaya, H; Takeda, Y; Tohse, N1
Brochu, M; Cadorette, C; Poterek, M; Simaan, M; St-Louis, J1

Reviews

2 review(s) available for cgp 28392 and bay-k-8644

ArticleYear
Slow channel calcium activators, a new group of pharmacological agents.
    Life sciences, 1985, Oct-07, Volume: 37, Issue:14

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Blood Pressure; Calcium; Calcium Channel Blockers; Cells, Cultured; Heart; Heart Rate; Ion Channels; Muscle Contraction; Muscle, Smooth, Vascular; Myocardium; Nifedipine; Pyridines; Stimulation, Chemical; Vascular Resistance

1985
Modulation of calcium channel function by drugs.
    Life sciences, 1985, Nov-18, Volume: 37, Issue:20

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Dihydropyridines; Electric Conductivity; Heart Rate; Homeostasis; Humans; Ion Channels; Membrane Potentials; Nifedipine; Pyridines; Receptors, Cell Surface; Structure-Activity Relationship

1985

Other Studies

39 other study(ies) available for cgp 28392 and bay-k-8644

ArticleYear
Effect of 4-aryl-2-methyl-5-nitro-1,4-dihydropyridine-3-carboxylates on the guinea pig papillary muscle and isolated human vena saphena magna that is used for coronary artery bypass grafting.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:9

    Topics: Animals; Coronary Artery Bypass; Dihydropyridines; Guinea Pigs; Humans; In Vitro Techniques; Muscle, Smooth, Vascular; Saphenous Vein

2011
Two subtypes of dihydropyridine-sensitive calcium channels in rat ventricular muscle.
    European journal of pharmacology, 1990, Mar-13, Volume: 178, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Animals; Calcium Channel Agonists; Calcium Channels; Dihydropyridines; Female; Heart; In Vitro Techniques; Magnesium; Male; Myocardial Contraction; Myocardium; Nifedipine; Potassium Chloride; Pyridines; Rats; Rats, Inbred Strains; Sarcoplasmic Reticulum

1990
Effects of calcium channel modulators on the proliferation of mouse spleen lymphocytes in vitro.
    Agents and actions, 1990, Volume: 29, Issue:3-4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Chloride; Cell Division; DNA; Lymphocytes; Male; Mice; Mice, Inbred BALB C; Nimodipine; Pyridines; Spleen

1990
Comparative behavioral, neurochemical and pharmacological activities of dihydropyridine calcium channel activating drugs.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Brain; Calcium Channel Agonists; Catecholamines; Chromatography, High Pressure Liquid; Dihydropyridines; Guinea Pigs; Injections, Intraperitoneal; Male; Mice; Motor Activity; Muscle Contraction; Muscle, Smooth; Nicotinic Acids; Nifedipine; Oxadiazoles; Pyridines; Stereoisomerism; Structure-Activity Relationship

1990
Selective antagonism of calcium channel activators by fluspirilene.
    British journal of pharmacology, 1990, Volume: 100, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding Sites; Binding, Competitive; Calcium Channel Agonists; Calcium Channel Blockers; Cecum; Cerebral Cortex; Female; Fluspirilene; Guinea Pigs; In Vitro Techniques; Isradipine; Kinetics; Muscle, Smooth; Oxadiazoles; Potassium; Pyridines; Radioligand Assay; Spiro Compounds

1990
Dihydropyridine calcium channel antagonists block and agonists potentiate high potassium contractures but not twitches in frog skeletal muscle.
    The Japanese journal of physiology, 1990, Volume: 40, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; In Vitro Techniques; Muscle Contraction; Nifedipine; Nitrendipine; Potassium; Pyridines; Rana pipiens

1990
Pharmacological dissection of Ca2+ channels in the rat aorta by Ca2+ entry modulators.
    Pharmacology, 1990, Volume: 40, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Female; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Potassium; Pyridines; Rats; Rats, Inbred Strains; Time Factors

1990
Interactions of dihydropyridine Ca2+ channel agonists with the human platelet thromboxane A2/prostaglandin H2 receptor.
    European journal of pharmacology, 1991, Jan-25, Volume: 206, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Affinity Labels; Blood Platelets; Calcium Channel Agonists; Calcium Channel Blockers; Dihydropyridines; Fura-2; Humans; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Manganese; Prostaglandin Endoperoxides, Synthetic; Prostaglandin H2; Prostaglandins H; Pyridines; Radioligand Assay; Receptors, Prostaglandin; Receptors, Thromboxane; Stereoisomerism

1991
Ca2+ channel agonists enhance thyrotropin-releasing hormone-induced inositol phosphates and prolactin secretion.
    European journal of pharmacology, 1991, Apr-03, Volume: 195, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Radioisotopes; Dihydropyridines; Female; In Vitro Techniques; Inositol Phosphates; Nimodipine; Perfusion; Prolactin; Pyridines; Rats; Rats, Inbred Strains; Receptors, Purinergic; Thyrotropin-Releasing Hormone

1991
Effects of calcium channel agonists (BAY K 8644, CGP28392 and YC-170) on 45Ca uptake by rat uterine segments.
    Japanese journal of pharmacology, 1991, Volume: 56, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Female; Nifedipine; Nitrendipine; Potassium Chloride; Pyridines; Rats; Rats, Inbred Strains; Uterus

1991
Dihydropyridine Ca2+ agonists and channel blockers interact in the opposite manner with photogenerated unpaired electrons.
    FEBS letters, 1985, Jul-08, Volume: 186, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Electron Transport; Eosine Yellowish-(YS); Heme; Ion Channels; Kinetics; Myoglobin; Nifedipine; Pyridines; Structure-Activity Relationship; Whales

1985
Agonists Bay-K8644 and CGP-28392 open calcium channels reconstituted from skeletal muscle transverse tubules.
    Biophysical journal, 1985, Volume: 48, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Electric Conductivity; Ion Channels; Kinetics; Muscles; Nifedipine; Pyridines

1985
Calcium channel blocking drugs. Part I: The calcium channel.
    Comprehensive therapy, 1985, Volume: 11, Issue:10

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Action Potentials; Biological Transport, Active; Calcium; Calcium Channel Blockers; Cell Membrane Permeability; Electric Conductivity; Humans; Ion Channels; Muscle, Smooth; Muscle, Smooth, Vascular; Muscles; Nifedipine; Pyridines

1985
In vitro comparative studies of the calcium-entry activators YC-170, CGP 28392, and BAY K 8644.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Biological Transport; Calcium; Guinea Pigs; Heart Rate; In Vitro Techniques; Ion Channels; Male; Mesentery; Myocardial Contraction; Nifedipine; Nitrendipine; Pyridines; Rats; Vasoconstriction

1985
A comparison of effects of BAY K 8644 and CGP 28392, dihydropyridines with Ca agonistic properties, on spontaneous mechanical activity in rat portal vein: modification of effect by ultraviolet radiation.
    Acta pharmacologica et toxicologica, 1985, Volume: 57, Issue:5

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Chromatography, High Pressure Liquid; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Portal Vein; Pyridines; Rats; Rats, Inbred WKY; Ultraviolet Rays

1985
Depolarization-dependent binding of the calcium channel antagonist, (+)-[3H]PN200-110, to intact cultured PC12 cells.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Cells, Cultured; Isradipine; Kinetics; Membrane Potentials; Nifedipine; Nitrendipine; Onium Compounds; Organophosphorus Compounds; Oxadiazoles; Potassium; Pyridines; Tritium

1986
Dihydropyridine calcium agonists selectively enhance resistance artery myogenic tone.
    European journal of pharmacology, 1986, Jul-31, Volume: 126, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Arteries; Calcium; In Vitro Techniques; Ion Channels; Male; Nimodipine; Potassium; Pyridines; Rabbits; Vasoconstriction

1986
Dihydropyridine modulation of the chromaffin cell secretory response.
    Journal of neurochemistry, 1987, Volume: 48, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cats; Cell Membrane Permeability; Chromaffin Granules; Chromaffin System; Female; Male; Muscarine; Nicotine; Nitrendipine; Norepinephrine; Perfusion; Potassium; Pyridines

1987
Dihydropyridine-sensitive Ca2+ channels: molecular properties of interaction with Ca2+ channel blockers, purification, subunit structure, and differentiation.
    Journal of cardiovascular pharmacology, 1986, Volume: 8 Suppl 8

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Affinity Labels; Animals; Bepridil; Binding, Competitive; Calcium; Calcium Channel Blockers; Calcium Channels; Chick Embryo; Cholic Acids; Diltiazem; Ion Channels; Isradipine; Kinetics; Macromolecular Substances; Molecular Weight; Muscles; Myocardial Contraction; Oxadiazoles; Pyridines; Pyrrolidines; Receptors, Nicotinic; Verapamil

1986
Inhibitory effects of calcium channel agonists on renin release from rat kidney cortical slices.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Dose-Response Relationship, Drug; Imidazoles; Ion Channels; Kidney Cortex; Male; Nifedipine; Pyridines; Rats; Rats, Inbred Strains; Renin; Trifluoperazine; Verapamil

1987
Stimulation of insulin release by organic calcium-agonists.
    Advances in experimental medicine and biology, 1986, Volume: 211

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Ion Channels; Islets of Langerhans; Kinetics; Nifedipine; Pyridines

1986
Effects of calcium channel activators BAY-K8644 and CGP-28392 on steroidogenesis in granulosa cells of the domestic hen.
    Biochemical and biophysical research communications, 1987, Jul-15, Volume: 146, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bucladesine; Calcium; Chickens; Colforsin; Female; Granulosa Cells; Luteinizing Hormone; Progesterone; Pyridines; Steroids

1987
Bay k 8644, a calcium entry promoter, as an antidote in verapamil intoxication in rabbits.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 287, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 4-Aminopyridine; Aminopyridines; Animals; Antidotes; Atrioventricular Node; Blood Pressure; Cardiovascular Agents; Electrocardiography; Female; Heart Rate; Hydrogen-Ion Concentration; In Vitro Techniques; Ion Channels; Male; Pyridines; Rabbits; Verapamil

1987
Influence of endothelium on the response to calcium agonists, calcium, potassium and noradrenaline in rat aorta.
    Pharmacology & toxicology, 1988, Volume: 62, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Calcium; Calcium Channel Agonists; Endothelium, Vascular; Ion Channels; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Pyridines; Rats; Rats, Inbred Strains

1988
Opposing actions of the enantiomers of BAY-K-8644 on calcium currents and ACTH secretion in clonal pituitary corticotrophs.
    Canadian journal of physiology and pharmacology, 1987, Volume: 65, Issue:12

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenocorticotropic Hormone; Animals; Calcium Channel Agonists; Cells, Cultured; Electrophysiology; Ion Channels; Mice; Pituitary Gland; Pyridines; Stereoisomerism

1987
Effects of the Ca2+ agonists, Bay K 8644 and CGP 28392, on isolated cat cerebral and peripheral arteries.
    Brain research, 1988, Nov-22, Volume: 474, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic Fibers; Animals; Arteries; Cats; Cerebral Arteries; Female; Male; Pyridines

1988
Paradoxical reversion of the inhibitory effects of dihydropyridine enantiomers on the calcium current in frog heart by CGP 28861.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Drug Interactions; Female; Heart Atria; In Vitro Techniques; Male; Membrane Potentials; Pyridines; Rana ridibunda; Receptors, Nicotinic

1989
Calcium uptake studies of 1,4-dihydropyridine agonists into rabbit aortic smooth muscle cells in culture.
    Life sciences, 1989, Volume: 44, Issue:23

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta; Calcium; Calcium Channels; Cells, Cultured; Dihydropyridines; Dose-Response Relationship, Drug; Muscle, Smooth, Vascular; Potassium; Pyridines; Rabbits

1989
The response of single cardiac sodium channels in neonatal rats to the dihydropyridines CGP 28392 and (-)-Bay K 8644.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Calcium Channel Agonists; Cell Membrane; Cytoplasm; Dihydropyridines; Ethanol; Heart; In Vitro Techniques; Male; Myocardium; Pyridines; Rats; Sodium Channels

1989
Effects of the Ca agonists Bay K 8644 and CGP 28392 on vascular smooth muscle tone.
    General pharmacology, 1989, Volume: 20, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Calcium; Calcium Channel Agonists; Calcium Channels; Calcium Radioisotopes; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Nifedipine; Pyridines; Rats; Rats, Inbred Strains

1989
Human red blood cells--an ideal model system for the action of calcium agonists and antagonists.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1984, Volume: 2, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Erythrocytes; Humans; Ion Channels; Nicardipine; Nifedipine; Nitrendipine; Pyridines; Stimulation, Chemical; Verapamil

1984
Dihydropyridine derivatives prolong the open state of Ca channels in cultured cardiac cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:15

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Blockers; Cells, Cultured; Heart; Ion Channels; Kinetics; Nifedipine; Pyridines; Rats

1984
Calcium channel activation: a different type of drug action.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:17

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cadmium; Calcium; Calcium Channel Blockers; Cell Line; Diltiazem; Gallopamil; Glioma; Hybrid Cells; Ion Channels; Kinetics; Mice; Neuroblastoma; Nifedipine; Nitrendipine; Pyridines; Rats

1984
Activation of the voltage-dependent Ca2+ channel in rat heart cells by dihydropyridine derivatives.
    Biochemical and biophysical research communications, 1984, Nov-30, Volume: 125, Issue:1

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Bepridil; Calcium; Dose-Response Relationship, Drug; Ion Channels; Myocardium; Nifedipine; Pyridines; Pyrrolidines; Rats; Rats, Inbred Strains; Time Factors; Verapamil

1984
Studies on the mechanism of action of the vasoconstrictive dihydropyridine, CGP 28392.
    European journal of pharmacology, 1984, Oct-15, Volume: 105, Issue:3-4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Nifedipine; Potassium Chloride; Pyridines; Rabbits; Vasoconstriction; Vasoconstrictor Agents

1984
Effect of calcium agonists, BAY K 8644 and CGP 28392, on guinea pig airway smooth muscle function during development.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aspirin; Calcium Channel Agonists; Drug Antagonism; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle Development; Muscle, Smooth; Pyridines; Trachea

1993
Calcium fluxes, ion currents and dihydropyridine receptors in a new immortal cell line from rat heart muscle.
    Journal of molecular and cellular cardiology, 1993, Volume: 25, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Calcium Channels, L-Type; Cell Differentiation; Cell Division; Cell Line; Heart; Immunohistochemistry; Male; Membrane Potentials; Muscle Proteins; Myocardium; Nitrendipine; Pyridines; Rats; Rats, Inbred F344; Time Factors; Tritium

1993
Voltage-dependence of Ca2+ agonist effect of YC-170 on cardiac L-type Ca2+ channels.
    British journal of pharmacology, 1995, Volume: 116, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channel Agonists; Calcium Channels; Heart; Myocardium; Nifedipine; Patch-Clamp Techniques; Pyridines; Rabbits

1995
Calcium channels contribute to the decrease in blood pressure of pregnant rats.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Blood Pressure; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Female; Hypotension; Male; Nifedipine; Pregnancy; Pregnancy Complications, Cardiovascular; Pyridines; Rats; Rats, Sprague-Dawley

2002