cgp 20712a and sr 59230a

cgp 20712a has been researched along with sr 59230a in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (15.38)18.2507
2000's10 (76.92)29.6817
2010's1 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Amend, A; Candelore, MR; Cascieri, MA; Deng, L; Guan, XM; Liu, Y; Newbold, R; Tota, L; Weber, AE1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Atgié, C; Berlan, M; Carpéné, C; Fontana, E; Galitzky, J; Lafontan, M1
Brawley, L; MacDonald, A; Shaw, AM1
Giacobino, JP; Jimenez, M; Kaumann, AJ; Moffatt, J; Molenaar, P; Oostendorp, J; Preitner, F1
Beiler, RJ; Commins, SP; Gettys, TW; Levin, N; Watson, PM1
Brown, KJ; Summers, RJ1
Chapple, CR; Chess-Williams, R; Yamanishi, T; Yasuda, K; Yoshida, K3
Brahmadevara, N; MacDonald, A; Shaw, AM1
Chan, O; Dziura, J; Horblitt, A; Sherwin, RS; Szepietowska, B; Zhu, W1

Other Studies

13 other study(ies) available for cgp 20712a and sr 59230a

ArticleYear
Potent and selective human beta(3)-adrenergic receptor antagonists.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:2

    Topics: Adipocytes; Adrenergic beta-Antagonists; Aminophenols; Animals; Binding, Competitive; CHO Cells; Cloning, Molecular; Cricetinae; Cyclic AMP; Humans; Ligands; Lipolysis; Macaca mulatta; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Structure-Activity Relationship; Sulfonamides

1999
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Selective activation of beta3-adrenoceptors by octopamine: comparative studies in mammalian fat cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adult; Animals; Binding, Competitive; Biogenic Amines; Bupranolol; CHO Cells; Cricetinae; Dioxoles; Dogs; Ethanolamines; Female; Gene Expression; Guinea Pigs; Humans; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lipolysis; Male; Mammals; Mesocricetus; Norepinephrine; Octopamine; Oxygen Consumption; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Species Specificity

1999
Beta 1-, beta 2- and atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
    British journal of pharmacology, 2000, Volume: 129, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Bupranolol; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Substrate Specificity; Vasodilator Agents

2000
Contribution of beta-adrenoceptor subtypes to relaxation of colon and oesophagus and pacemaker activity of ureter in wildtype and beta(3)-adrenoceptor knockout mice.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dioxoles; Dose-Response Relationship, Drug; Epinephrine; Esophagus; Female; Imidazoles; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Ureter

2000
Central leptin regulates the UCP1 and ob genes in brown and white adipose tissue via different beta-adrenoceptor subtypes.
    The Journal of biological chemistry, 2000, Oct-20, Volume: 275, Issue:42

    Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Carrier Proteins; Cell Membrane; Cerebral Ventricles; Gene Expression Regulation; Imidazoles; Injections, Intraventricular; Ion Channels; Leptin; Male; Membrane Proteins; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Mitochondrial Proteins; Propanolamines; Propranolol; Receptors, Adrenergic, beta-3; Receptors, Leptin; RNA, Messenger; Transcription, Genetic; Uncoupling Protein 1

2000
beta(1)- and beta(3)-adrenoceptor mediated smooth muscle relaxation in hypothyroid rat ileum.
    European journal of pharmacology, 2001, Volume: 415, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Hypothyroidism; Ileum; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3; RNA, Messenger

2001
Identification of beta-adrenoceptor subtypes in lower urinary tract of the female pig.
    The Journal of urology, 2002, Volume: 168, Issue:6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dihydroalprenolol; Ethanolamines; Female; Imidazoles; In Vitro Techniques; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Swine; Urethra; Urinary Bladder

2002
Role of beta-adrenoceptor subtypes in mediating relaxation of the pig bladder trigonal muscle in vitro.
    Neurourology and urodynamics, 2003, Volume: 22, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Swine; Urinary Bladder

2003
The functional role of beta-adrenoceptor subtypes in mediating relaxation of pig urethral smooth muscle.
    The Journal of urology, 2003, Volume: 170, Issue:6 Pt 1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Ethanolamines; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Swine; Urethra

2003
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction

2004
Modulation of β-adrenergic receptors in the ventromedial hypothalamus influences counterregulatory responses to hypoglycemia.
    Diabetes, 2011, Volume: 60, Issue:12

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Blood Glucose; Epinephrine; Ethanolamines; Formoterol Fumarate; Glucagon; Glucose Clamp Technique; Hypoglycemia; Imidazoles; Insulin; Male; Norepinephrine; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Ventromedial Hypothalamic Nucleus

2011