cgp 20712a has been researched along with ici 118551 in 133 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 13 (9.77) | 18.7374 |
1990's | 61 (45.86) | 18.2507 |
2000's | 43 (32.33) | 29.6817 |
2010's | 16 (12.03) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Baker, JG | 1 |
Baker, JG; Fischer, PM; Gardiner, SM; Hill, SJ; Kellam, B; Mistry, SN | 1 |
Baker, JG; Gunera, J; Kolb, P; Schmidt, D | 1 |
Bowen, WP; Flint, DJ; Vernon, RG | 2 |
Fraeyman, N; Van de Velde, E; Van Ermen, A; Vanscheeuwijck, P | 1 |
Majewski, H; Mian, MA; Rand, MJ | 1 |
Bals, S; Brodde, OE; Deighton, NM; Motomura, S; Zerkowski, HR | 1 |
Choi, AL; Martínez de la Escalera, G; Weiner, RI | 1 |
Grino, M; Oliver, C | 1 |
Amenta, F; Coppola, L; Ferrante, F; Forlani, A; Gallo, P; Monopoli, A; Napoleone, P | 1 |
Flügge, G; Nazarali, AJ; Pinto, JE; Saavedra, JM; Torda, T; Viglione, PN | 1 |
Leysen, JE; Pauwels, PJ; Van Gompel, P | 1 |
Kim, YS; Molenaar, P; Sainz, RD; Summers, RJ | 1 |
Kaumann, AJ; Lemoine, H | 2 |
Delavier-Klutchko, C; Emorine, LJ; Marullo, S; Strosberg, AD | 1 |
Böhm, M; Erdmann, E; Fruhmann, G; Gengenbach, S; Hauck, RW; Sunder-Plassmann, L | 1 |
Cerbai, E; Masini, I; Mugelli, A | 1 |
Hall, JA; Latimer, M | 1 |
Bühler, FR; Hoyer, D; Jones, CR; Palacios, JM | 1 |
Böhm, M; Erdmann, E; Kemkes, B; Klövekorn, WP; Pieske, B; Schnabel, P; Schwinger, R | 1 |
Brown, MJ; Hall, JA; Kaumann, AJ; Murray, KJ; Wells, FC | 1 |
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
Hollenga, C; Zaagsma, J | 1 |
Dubbin, PN; Dusting, GJ; Macdonald, PS | 1 |
Jones, CR; McMartin, LR; Molenaar, P; Summers, RJ | 1 |
Bos, EA; Knot, HJ; Remie, R; Zaagsma, J | 1 |
Kaumann, AJ | 1 |
Beer, M; Iversen, LL; Poat, J; Richardson, A; Stahl, SM | 1 |
Hadcock, JR; Malbon, CC | 1 |
Molenaar, P; Summers, RJ | 1 |
Canale, E; Molenaar, P; Summers, RJ | 1 |
MacDonald, A; McKean, J | 1 |
Olszewski, MA; Robinson, NE; Zhang, XY | 1 |
Champigneulle, A; Elalouf, JM; Imbert-Teboul, M; Mandon, B; Siga, E | 1 |
Badran, TW; Hoey, AJ; Matthews, ML; Pegg, GG; Sillence, MN | 1 |
Campbell, B; Iakovidis, D; Jackman, G; Louis, S; Louis, WJ; Tung, LH | 1 |
Brown, MJ; Ferro, A; Kaumann, AJ | 1 |
Matthews, ML; Moore, NG; Reich, MM; Sillence, MN | 1 |
Charpentier, F; Rosen, MR | 1 |
Elnatan, J; Molenaar, P; Rosenfeldt, FL; Summers, RJ | 1 |
Collins, S; Daniel, KW; Gettys, TW; Ramkumar, V; Rohlfs, EM; Taylor, IL | 1 |
Carruba, MO; Nisoli, E; Tonello, C | 1 |
Coppes, RP; Dahlöf, C; Tarizzo, VI; Zaagsma, J | 1 |
Kuznetsov, V; Pak, E; Robinson, RB; Steinberg, SF | 1 |
del Monte, F; Harding, SE; Kaumann, AJ; Pepper, J; Poole-Wilson, PA; Wynne, DG | 1 |
Lemoine, H; Rösen, P; Sackmann, B; Zink, S | 1 |
Berry, JL; Chiu, P; Cook, SJ; Downing, SJ; Foster, RW; Small, RC | 1 |
Berry, JL; Carpenter, JR; Chiu, P; Cook, SJ; Downing, SJ; Foster, RW; Miller, AJ; Small, AM; Small, RC | 1 |
Baude, B; Emorine, LJ; Fève, B; Krief, S; Pairault, J; Strosberg, AD; Zilberfarb, V | 1 |
Nash, MS; Osborne, NN | 1 |
Adachi-Akahane, S; Kitagawa, Y; Nagao, T | 1 |
Bültmann, R; Driessen, B; Gonçalves, J; Starke, K | 1 |
Barrionuevo, M; Cenarruzabeitia, E; Martínez, JA; Milagro, FI | 1 |
Pfaffendorf, M; van Zwieten, PA; Winkler Prins, EA; Zwaveling, J | 1 |
Morin, D; Onteniente, B; Sapena, R; Tillement, JP; Zini, R | 1 |
Barker, LA; Spadari-Bratfisch, RC; Zanesco, A | 1 |
Germack, R; Perret, GY; Starzec, AB; Vassy, R | 1 |
Goepel, M; Michel, MC; Rübben, H; Wittmann, A | 1 |
Ahrens, O; Flügge, G; Fuchs, E | 2 |
Altschuld, RA; Billman, GE; Castillo, LC; Hensley, J; Hohl, CM | 1 |
Karim, F; Poucher, SM | 1 |
Bilbe, G; Kellenberger, S; Muller, K; Richener, H | 1 |
Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F | 1 |
Liu, YL; Nwosu, UC; Rice, PJ | 1 |
Doze, P; Elsinga, PH; Ensing, K; Kraan, J; Vaalburg, W; van der Mark, TW; van Waarde, A; Visser, TJ | 1 |
Herzig, S; Schröder, F | 1 |
Ajisawa, Y; Akahane, M; Andersson, KE; Hayakawa, K; Igawa, Y; Nishizawa, O; Takeda, H; Yamazaki, Y; Yoneyama, T | 1 |
Atgié, C; Berlan, M; Carpéné, C; Fontana, E; Galitzky, J; Lafontan, M | 1 |
Cerbai, E; Mugelli, A; Pino, R; Rodriguez, ML | 1 |
Guerrero, SW; Minneman, KP | 1 |
Abuin, L; Cotecchia, S; Lattion, A; Nenniger-Tosato, M | 1 |
Marcondes, FK; Santos, IN; Spadari-Bartfisch, RC; Vanderlei, LC | 1 |
Colucci, WS; Communal, C; Sawyer, DB; Singh, K | 1 |
Ferro, A; Gao, L; Li, J; Xu, B | 1 |
Black, JW; Prendergast, CE; Shankley, NP | 1 |
Giacobino, JP; Jimenez, M; Kaumann, AJ; Moffatt, J; Molenaar, P; Oostendorp, J; Preitner, F | 1 |
Töneke, K | 1 |
Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S | 1 |
Heijenbrok, FJ; Mathy, MJ; Pfaffendorf, M; van Zwieten, PA | 1 |
Danilo, P; Gainullin, RZ; Moise, NS; Rosen, MR; Sosunov, EA; Steinberg, SF | 1 |
Barnes, PJ; Haddad, EB; Mak, JC; Rousell, J | 1 |
Böhm, M; Cremers, B; Dabew, E; Maack, C; Schnabel, P; Südkamp, M; Tyroller, S | 1 |
Huang, Y; Xu, B | 1 |
Graf, EM; Harding, SE; Herzig, S; Heubach, JF; Jäger, A; Molenaar, P; Ravens, U; Schröder, F | 1 |
Beal, AM; Boys, CA | 1 |
Chess-Williams, R; Chong, LK; Peachell, PT | 1 |
Bailey, S; Berhane, Y; Elliott, J; Horn, J; Marr, CM | 1 |
Beal, AM | 1 |
Chapple, CR; Chess-Williams, R; Yamanishi, T; Yasuda, K; Yoshida, K | 3 |
Blaschke, M; Harding, SE; Heubach, JF; Kaumann, AJ; Ravens, U | 1 |
Black, JW; Harper, EA; Hasseldine, AR | 1 |
Chakir, K; Cheng, H; Kobilka, BK; Xiang, Y; Xiao, RP; Yang, D; Zhang, SJ | 1 |
Brahmadevara, N; MacDonald, A; Shaw, AM | 1 |
Callebert, J; Etienne, N; Jaffré, F; Launay, JM; Maroteaux, L; Monassier, L; Nebigil, CG; Sarre, A | 1 |
Ander, AN; Drumm, JD; Duggirala, SK; Roth, DM | 1 |
Battaglia, F; Bonacchi, M; Casini, S; Cerbai, E; Fiorani, B; Giunti, G; Lonardo, G; Mugelli, A; Sani, G; Stefano, PL | 1 |
Caceres, VM; Krieger, MH; Moreira, MF; Santos, IN; Spadari-Bratfisch, RC; Sumitame, M | 1 |
Christ, T; Kaumann, A; Molenaar, P; Ravens, U | 1 |
Badino, P; Barbero, R; Cuniberti, B; Girardi, C; Magistris, G; Odore, R; Pagliasso, S; Re, G | 1 |
Bianchetti, A; Croci, T; Di Marzo, V; Di Palo, S; Ferla, G; Guagnini, F; Matias, I; Mukenge, S; Valenti, M | 1 |
Brodde, OE; Gröner, F; Heinroth-Hoffmann, I; Pönicke, K | 1 |
Allen, BG; Baragli, A; Boivin, B; Ethier, N; Hébert, TE; Lavoie, C; Trieu, P; Vaniotis, G; Villeneuve, LR | 1 |
Jing, Y; Shan, D; Su, Y; Wang, H; Wong, TM | 1 |
Adeoya-Osiguwa, SA; Fraser, LR | 1 |
Horinouchi, T; Koike, K; Michikawa, H; Tanaka, Y; Yamashita, Y | 1 |
Chartier, D; Ehrlich, JR; Hébert, TE; Nattel, S; Qi, X; Yeh, YH | 1 |
Aroca, V; Carceles, MD; Fuentes, T; Hernández, J; Lopez, J | 1 |
Galindo-Tovar, A; Kaumann, AJ | 1 |
Bang, ML; Catalucci, D; Condorelli, G | 1 |
Ali, NN; Brito-Martins, M; Harding, SE | 1 |
Chen, P; Liu, Z; Ma, K; Yang, H; Zhang, Y; Zhou, C | 1 |
Gu, SL; Hao, YL; Sun, H; Wu, Q; Yan, CD; Zhao, Z | 1 |
Fuente, T; Gonzalez-Muñoz, C; Hernández-Cascales, J | 1 |
Cho, KW; Choi, DH; Choi, HR; Cui, HZ; Kang, DG; Lee, HS | 1 |
Candelario-Jalil, E; de Oliveira, AC; Fiebich, BL; Haake, E; Heneka, MT; Hüll, M; Schlachetzki, JC | 1 |
Baker, JG; Fretwell, L; Gardiner, SM; Hill, SJ; Kemp, P; March, J | 1 |
Gao, L; Jiang, X; Li, D; Sun, H; Wang, Y; Xu, C; Yan, C | 1 |
Anderson, ME; He, K; Hell, JW; Koval, OM; Lee, HK; Matt, L; Nguyen, M; Patriarchi, T; Qian, H; Zhang, M | 1 |
Barnes, JL; Ghosh, PM; Ikeno, Y; Kamat, A; Katz, MS; Lu, Z; Shu, ZJ; Yeh, CK; Zhang, BX; Zhu, B | 1 |
Côrrea, FM; Crestani, CC; Fabri, DR; Gomes, FV; Hott, SC; Reis, DG; Resstel, LB | 1 |
Abraham, G; Guenl, B; Jonas, S; Kassahun, WT; Ungemach, FR | 1 |
Cao, K; Chen, Y; Wang, H; Wang, S; Xu, D; Zhang, X; Zhu, H; Zou, J | 1 |
Aflaki, M; Luo, X; Maguy, A; Nattel, S; Ordog, B; Qi, XY; Shi, Y; Tadevosyan, A; Tardif, JC; Xiao, L | 1 |
Belvisi, MG; Birrell, MA; Bonvini, SJ; Buckley, J; Dale, N; Dubuis, ED; Maher, SA; Wortley, MA; Yew-Booth, L | 1 |
Lorenz, K; Newe, M; Propping, S; Ravens, U; Wirth, MP | 1 |
Buonarati, OR; Catterall, WA; Chowdhury, D; Hell, JW; Hofmann, F; Lee, B; Matt, L; Nanou, E; Navedo, MF; Nieves-Cintrón, M; Nystoriak, MA; Patriarchi, T; Poomvanicha, M; Price, JL; Qian, H | 1 |
Kaumann, AJ; Lee, XW; Michel, MC; Mo, W; Molenaar, P | 1 |
Berthiaume, Y; Ferraro, P; Massé, C; Richard, C; Shabbir, W | 1 |
133 other study(ies) available for cgp 20712a and ici 118551
Article | Year |
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The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2005 |
Synthesis and in vitro and in vivo characterization of highly β1-selective β-adrenoceptor partial agonists.
Topics: Adrenergic beta-1 Receptor Agonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Design; Heart Rate; Hemodynamics; Humans; Indicators and Reagents; Ligands; Male; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Structure-Activity Relationship | 2013 |
Similarity- and Substructure-Based Development of β
Topics: | 2017 |
Regional and interspecific differences in the ligand binding properties of beta-adrenergic receptors of individual white adipose tissue depots in the sheep and rat.
Topics: Adipose Tissue; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Imidazoles; Iodocyanopindolol; Lactation; Pindolol; Propanolamines; Proteins; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Sheep | 1992 |
Influence of age on the beta 1- and beta 2-adrenergic receptors in rat liver.
Topics: Adenylyl Cyclases; Aging; Animals; Binding, Competitive; Cell Membrane; Imidazoles; Liver; Liver Glycogen; Male; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1992 |
An inhibitory effect of isoprenaline on stimulation-induced noradrenaline release from rat atria.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Electric Stimulation; Female; Heart Atria; Imidazoles; Indomethacin; Isoproterenol; Male; Norepinephrine; Phentolamine; Propanolamines; Rats; Rats, Inbred Strains | 1992 |
Characterization of the beta adrenoceptor subtype(s) mediating the positive inotropic effects of epinine, dopamine, dobutamine, denopamine and xamoterol in isolated human right atrium.
Topics: Adrenergic beta-Agonists; Adult; Aged; Calcium; Deoxyepinephrine; Dobutamine; Dopamine; Ethanolamines; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Male; Middle Aged; Myocardial Contraction; Propanolamines; Stimulation, Chemical; Xamoterol | 1992 |
Beta 1-adrenergic regulation of the GT1 gonadotropin-releasing hormone (GnRH) neuronal cell lines: stimulation of GnRH release via receptors positively coupled to adenylate cyclase.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Line; Cyclic AMP; Gonadotropin-Releasing Hormone; Imidazoles; Isoproterenol; Kinetics; Mice; Mice, Transgenic; Neurons; Norepinephrine; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, LHRH | 1992 |
Ontogeny of insulin-induced hypoglycemia stimulation of adrenocorticotropin secretion in the rat: role of catecholamines.
Topics: Adrenergic beta-Antagonists; Adrenocorticotropic Hormone; Aging; Animals; Arginine Vasopressin; Catecholamines; Hypoglycemia; Imidazoles; Immunization, Passive; Insulin; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1992 |
Autoradiographic localization of beta-adrenergic receptors in human large coronary arteries.
Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Autoradiography; Binding, Competitive; Coronary Vessels; Female; Humans; Imidazoles; Male; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Silver; Tissue Distribution | 1991 |
Increased beta 2-adrenoceptors in the superior cervical ganglia of genetically hypertensive rats.
Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Enalapril; Ganglia, Sympathetic; Hypertension; Imidazoles; Iodocyanopindolol; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta | 1991 |
Human beta 1- and beta 2-adrenergic receptor binding and mediated accumulation of cAMP in transfected Chinese hamster ovary cells. Profile of nebivolol and known beta-adrenergic blockers.
Topics: Adrenergic beta-Antagonists; Animals; Benzopyrans; Binding Sites; Binding, Competitive; Cell Line; Cricetinae; Cricetulus; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Models, Biological; Nebivolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Stereoisomerism; Transfection | 1991 |
Characterization of beta 1- and beta 2-adrenoceptors in rat skeletal muscles.
Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Imidazoles; Male; Membranes; Muscles; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Regional differences of beta 1- and beta 2-adrenoceptor-mediated functions in feline heart. A beta 2-adrenoceptor-mediated positive inotropic effect possibly unrelated to cyclic AMP.
Topics: Adrenergic beta-Antagonists; Animals; Atrial Function, Left; Cardiotonic Agents; Cats; Cyclic AMP; Epinephrine; Female; Heart; Heart Rate; Imidazoles; Male; Myocardial Contraction; Myocardium; Norepinephrine; Papillary Muscles; Propanolamines; Receptors, Adrenergic, beta; Sinoatrial Node; Ventricular Function, Right | 1991 |
Selective binding of ligands to beta 1, beta 2 or chimeric beta 1/beta 2-adrenergic receptors involves multiple subsites.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Sequence; Animals; Escherichia coli; Ethanolamines; Imidazoles; Kinetics; Molecular Sequence Data; Norepinephrine; Procaterol; Propanolamines; Protein Engineering; Receptors, Adrenergic, beta; Recombinant Fusion Proteins; Structure-Activity Relationship; Thermodynamics | 1990 |
Characterization of the beta-adrenergic receptors of sheep adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Atenolol; Epinephrine; Imidazoles; Isoproterenol; Norepinephrine; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Sheep | 1990 |
Beta 2-adrenoceptors in human lung and peripheral mononuclear leukocytes of untreated and terbutaline-treated patients.
Topics: Adrenergic beta-Antagonists; Bronchial Spasm; Down-Regulation; Female; Humans; Imidazoles; Leukocytes, Mononuclear; Lung; Male; Middle Aged; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Terbutaline | 1990 |
Electrophysiological characterization of cardiac beta 2-adrenoceptors in sheep Purkinje fibers.
Topics: Action Potentials; Adrenergic beta-Antagonists; Animals; Drug Interactions; Imidazoles; Isoproterenol; Propanolamines; Purkinje Fibers; Receptors, Adrenergic, beta; Sheep | 1990 |
Enoximone potentiates the positive inotropic effects of beta-1- and beta-2-adrenoceptor stimulation in human atrial myocardium.
Topics: Adrenergic beta-Antagonists; Diazoxide; Dose-Response Relationship, Drug; Drug Synergism; Enoximone; Humans; Imidazoles; In Vitro Techniques; Myocardial Contraction; Phosphodiesterase Inhibitors; Propanolamines | 1990 |
Receptor modification in the brains of spontaneously hypertensive and Wistar-Kyoto rats: regionally specific and selective increase in cerebellar beta 2-adrenoceptors.
Topics: Animals; Autoradiography; Brain; Cerebellum; Hypertension; Imidazoles; In Vitro Techniques; Iodocyanopindolol; Male; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta | 1990 |
Reduced effects of dopexamine on force of contraction in the failing human heart despite preserved beta 2-adrenoceptor subpopulation.
Topics: Adenylyl Cyclases; Adrenergic Agonists; Adrenergic beta-Antagonists; Binding, Competitive; Dopamine; Female; Heart Failure; Humans; Imidazoles; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Propanolamines; Receptors, Adrenergic, beta | 1989 |
A comparison of the effects of adrenaline and noradrenaline on human heart: the role of beta 1- and beta 2-adrenoceptors in the stimulation of adenylate cyclase and contractile force.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Epinephrine; Heart; Humans; Imidazoles; Myocardial Contraction; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta | 1989 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Direct evidence for the atypical nature of functional beta-adrenoceptors in rat adipocytes.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Epididymis; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1989 |
Beta-adrenoceptors on endothelial cells do not influence release of relaxing factor in dog coronary arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Biological Products; Bradykinin; Coronary Vessels; Dogs; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Isoproterenol; Nitric Oxide; Propanolamines; Prostaglandin Endoperoxides, Synthetic; Receptors, Adrenergic, beta; Vasodilation | 1987 |
Autoradiographic localization and densitometric analysis of beta-1 and beta-2 adrenoceptors in the canine left anterior descending coronary artery.
Topics: Animals; Autoradiography; Coronary Vessels; Dogs; Imidazoles; Iodocyanopindolol; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1988 |
Characterization of presynaptic beta-adrenoceptors facilitating endogenous noradrenaline release in the portal vein of permanently cannulated, freely moving rats.
Topics: Animals; Catheterization; Drug Synergism; Fenoterol; Imidazoles; Male; Norepinephrine; Portal Vein; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Yohimbine | 1988 |
The beta 1-adrenoceptor antagonist CGP 20712 A unmasks beta 2-adrenoceptors activated by (-)-adrenaline in rat sinoatrial node.
Topics: Adrenergic beta-Antagonists; Animals; Catecholamines; Epinephrine; Heart Rate; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sinoatrial Node | 1986 |
Beta 2-adrenoceptor-mediated positive inotropic effect of adrenaline in human ventricular myocardium. Quantitative discrepancies with binding and adenylate cyclase stimulation.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Epinephrine; Humans; Imidazoles; In Vitro Techniques; Myocardial Contraction; Myocardium; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Vasodilator Agents | 1987 |
In vitro selectivity of agonists and antagonists for beta 1- and beta 2-adrenoceptor subtypes in rat brain.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Brain Chemistry; Cerebral Cortex; Clenbuterol; Imidazoles; In Vitro Techniques; Male; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Stereoisomerism | 1988 |
Down-regulation of beta-adrenergic receptors: agonist-induced reduction in receptor mRNA levels.
Topics: Adrenergic beta-Antagonists; Animals; Cell Line; Cricetinae; Cyclic AMP; DNA; Endonucleases; Imidazoles; Isoproterenol; Kinetics; Male; Nucleic Acid Hybridization; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA, Messenger; Single-Strand Specific DNA and RNA Endonucleases; Vas Deferens | 1988 |
Characterization of beta-1 and beta-2 adrenoceptors in guinea pig atrium: functional and receptor binding studies.
Topics: Animals; Electric Stimulation; Ethanolamines; Female; Guinea Pigs; Heart Atria; Heart Rate; Imidazoles; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Pindolol; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Stimulation, Chemical; Uterine Contraction; Uterus | 1987 |
Autoradiographic localization of beta-1 and beta-2 adrenoceptors in guinea pig atrium and regions of the conducting system.
Topics: Animals; Autoradiography; Binding, Competitive; Guinea Pigs; Heart Atria; Heart Conduction System; Imidazoles; Isomerism; Kinetics; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1987 |
Contributions of beta-adrenoceptor subtypes to responses to isoprenaline in rat isolated distal colon.
Topics: Animals; Colon; Imidazoles; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1995 |
Beta 2-adrenoceptor activation augments acetylcholine release from tracheal parasympathetic nerves.
Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Atropine; Electric Stimulation; Horses; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Parasympathetic Nervous System; Propanolamines; Receptors, Adrenergic, beta-2; Trachea | 1995 |
Molecular analysis of beta-adrenergic receptor subtypes in rat collecting duct: effects on cell cAMP and Ca2+ levels.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Calcium; Cyclic AMP; DNA Primers; Epinephrine; Imidazoles; Isoproterenol; Kidney Cortex; Kidney Tubules, Collecting; Male; Molecular Sequence Data; Mutagenesis; Nephrons; Norepinephrine; Pindolol; Polymerase Chain Reaction; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; RNA, Messenger | 1995 |
Cardiovascular effects of clenbuterol are beta 2-adrenoceptor-mediated in steers.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Blood Glucose; Blood Pressure; Cardiovascular Physiological Phenomena; Cardiovascular System; Cattle; Clenbuterol; Dose-Response Relationship, Drug; Heart Atria; Heart Rate; Imidazoles; Infusions, Intravenous; Isoproterenol; Male; Norepinephrine; Potassium; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1995 |
Partial agonist activity of celiprolol.
Topics: Adrenergic beta-Antagonists; Airway Resistance; Animals; Blood Pressure; Celiprolol; Decerebrate State; Guinea Pigs; Heart Rate; Imidazoles; In Vitro Techniques; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1993 |
Beta-adrenoceptor subtypes in human coronary artery: desensitization of beta 2-adrenergic vasorelaxation by chronic beta 1-adrenergic stimulation in vitro.
Topics: Adrenergic beta-Antagonists; Analysis of Variance; Coronary Vessels; Dose-Response Relationship, Drug; Epinephrine; Heart Transplantation; Humans; Imidazoles; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1995 |
Effects of BRL-47672 on growth, beta 2-adrenoceptors, and adenylyl cyclase activation in female rats.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Clenbuterol; Enzyme Activation; Female; Growth; Imidazoles; Organic Chemicals; Propanolamines; Rats; Receptors, Adrenergic, beta; Second Messenger Systems | 1995 |
Beta-adrenergic regulation of action potentials and automaticity in young and adult canine purkinje fibers.
Topics: Action Potentials; Adrenergic beta-Antagonists; Aging; Albuterol; Animals; Cardiac Pacing, Artificial; Dogs; Imidazoles; In Vitro Techniques; Isoproterenol; Propanolamines; Purkinje Fibers; Receptors, Adrenergic, beta | 1994 |
Autoradiographic localization and quantitation of beta 1- and beta 2-adrenoceptors in the human atrioventricular conducting system: a comparison of patients with idiopathic dilated cardiomyopathy and ischemic heart disease.
Topics: Adrenergic beta-Antagonists; Adult; Aged; Atrioventricular Node; Binding, Competitive; Bundle of His; Cardiomyopathy, Dilated; Down-Regulation; Female; Heart Septum; Humans; Imidazoles; Male; Middle Aged; Muscle Proteins; Myocardial Ischemia; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1994 |
Impaired expression and functional activity of the beta 3- and beta 1-adrenergic receptors in adipose tissue of congenitally obese (C57BL/6J ob/ob) mice.
Topics: Adenylyl Cyclases; Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Cells, Cultured; Cyclic AMP; Diabetes Mellitus, Type 2; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Activation; Epinephrine; Gene Expression Regulation; Hyperglycemia; Imidazoles; Lipolysis; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Obesity; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA Splicing; RNA, Messenger | 1994 |
SR 58611A: a novel thermogenic beta-adrenoceptor agonist.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP; Drug Interactions; Glycerol; Imidazoles; Lipid Metabolism; Male; Obesity; Propanolamines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Tetrahydronaphthalenes | 1994 |
Pre- and postganglionic stimulation-induced noradrenaline overflow is markedly facilitated by a prejunctional beta 2-adrenoceptor-mediated control mechanism in the pithed rat.
Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Decerebrate State; Fenoterol; Ganglia; Heart Rate; Imidazoles; Male; Norepinephrine; Portal Vein; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sympathetic Nervous System; Synaptic Transmission | 1994 |
Beta 2-adrenergic receptor actions in neonatal and adult rat ventricular myocytes.
Topics: Age Factors; Animals; Animals, Newborn; Calcium; Cells, Cultured; Cyclic AMP; Ethanolamines; Imidazoles; Isoproterenol; Male; Myocardial Contraction; Myocardium; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1995 |
Coexistence of functioning beta 1- and beta 2-adrenoceptors in single myocytes from human ventricle.
Topics: Adrenergic beta-Antagonists; Animals; Epinephrine; Guinea Pigs; Humans; Imidazoles; In Vitro Techniques; Myocardial Contraction; Myocardium; Propanolamines; Receptors, Adrenergic, beta | 1993 |
Regulation of endothelial permeability by beta-adrenoceptor agonists: contribution of beta 1- and beta 2-adrenoceptors.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cattle; Cell Membrane Permeability; Cells, Cultured; Cyclic AMP; Endothelium, Vascular; Enzyme Activation; Ethanolamines; Formoterol Fumarate; Imidazoles; Propanolamines; Receptors, Adrenergic, beta | 1993 |
Beta-adrenoceptor subtypes and the opening of plasmalemmal K(+)-channels in trachealis muscle: electrophysiological and mechanical studies in guinea-pig tissue.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Benzopyrans; Cell Membrane; Cromakalim; Electrophysiology; Female; Guinea Pigs; Heart; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Myocardium; Norepinephrine; Potassium Channels; Procaterol; Propanolamines; Pyrroles; Receptors, Adrenergic, beta; Rubidium Radioisotopes; Salmeterol Xinafoate; Trachea | 1993 |
Beta-adrenoceptor subtypes and the opening of plasmalemmal K(+)-channels in bovine trachealis muscle: studies of mechanical activity and ion fluxes.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aminophylline; Animals; Cattle; Cell Membrane; Histamine; Imidazoles; In Vitro Techniques; Isometric Contraction; Muscle Relaxation; Muscle, Smooth; Potassium Channels; Propanolamines; Receptors, Adrenergic, beta; Rubidium; Rubidium Radioisotopes; Trachea | 1993 |
Transcriptional modulation by n-butyric acid of beta 1-, beta 2-, and beta 3-adrenergic receptor balance in 3T3-F442A adipocytes.
Topics: 3T3 Cells; Adenylyl Cyclase Inhibitors; Adipocytes; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Animals; Base Sequence; Butyrates; Butyric Acid; DNA Primers; DNA, Complementary; Ethanolamines; Gene Expression Regulation; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Molecular Sequence Data; Oligonucleotides, Antisense; Pindolol; Polymerase Chain Reaction; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Transcription, Genetic | 1994 |
Agonist-induced effects on cyclic AMP metabolism are affected in pigment epithelial cells of the Royal College of Surgeons rat.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprostadil; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dinoprostone; Fibroblast Growth Factor 2; Imidazoles; Isoproterenol; Kinetics; Melatonin; Pigment Epithelium of Eye; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta-2; Receptors, Purinergic P1; Serotonin | 1995 |
Determination of beta-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective beta-antagonists.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cyclic AMP; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Membranes; Myocardium; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Tritium | 1995 |
Opposite modulation of noradrenaline and ATP release in guinea-pig vas deferens through prejunctional beta-adrenoceptors: evidence for the beta 2 subtype.
Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Imidazoles; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Norepinephrine; Prazosin; Propanolamines; Receptors, Adrenergic, beta-2; Suramin; Terbutaline; Vas Deferens | 1996 |
Potential anti-diabetic applications of a new molecule with affinity for beta 3-adrenoceptors.
Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Benzyl Alcohols; Blood Glucose; Diabetes Mellitus, Experimental; Esophagus; Female; Guinea Pigs; Imidazoles; Insulin; Muscle Relaxation; Muscle, Smooth; Oxygen Consumption; Propanolamines; Rats; Rats, Wistar; Triglycerides | 1996 |
The influence of hyperthyroidism on beta-adrenoceptor-mediated relaxation of isolated small mesenteric arteries.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Colforsin; Dose-Response Relationship, Drug; Hyperthyroidism; Imidazoles; Isoproterenol; Male; Mesenteric Arteries; Methoxamine; Muscle Contraction; Muscle Relaxation; Propanolamines; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Wistar; Thromboxane A2; Thyroxine; Vascular Resistance; Vasoconstrictor Agents | 1996 |
Characterization of beta-adrenergic receptors of freshly isolated astrocytes and neurons from rat brain.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Astrocytes; Binding, Competitive; Cells, Cultured; Cerebellum; Imidazoles; Immunohistochemistry; Male; Neurons; Propanolamines; Prosencephalon; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1997 |
Sino-aortic denervation causes right atrial beta adrenoceptor down-regulation.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Down-Regulation; Heart Atria; Heart Rate; Imidazoles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Male; Muscle Denervation; Myocardium; Neurons; Norepinephrine; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Sinoatrial Node | 1997 |
Beta-adrenoceptor subtype expression and function in rat white adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Binding, Competitive; Imidazoles; Lipolysis; Male; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1997 |
Comparison of adrenoceptor subtype expression in porcine and human bladder and prostate.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Humans; Imidazoles; Isoquinolines; Male; Oxymetazoline; Piperazines; Prazosin; Propanolamines; Prostate; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Swine; Urinary Bladder; Yohimbine | 1997 |
Beta-adrenoceptors in the tree shrew brain. I. Distribution and characterization of [125I]iodocyanopindolol binding sites.
Topics: Adrenergic beta-Antagonists; Animals; Brain Chemistry; Imidazoles; Iodocyanopindolol; Nerve Tissue Proteins; Organ Specificity; Pindolol; Propanolamines; Protein Binding; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Serotonin; Serotonin; Substrate Specificity; Tupaiidae | 1997 |
Beta-adrenoceptors in the tree shrew brain. II. Time-dependent effects of chronic psychosocial stress on [125I]iodocyanopindolol bindings sites.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Body Weight; Brain Chemistry; Chronic Disease; Down-Regulation; Hydrocortisone; Imidazoles; Iodocyanopindolol; Male; Norepinephrine; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Social Dominance; Stress, Psychological; Time Factors; Tupaiidae | 1997 |
Beta2-adrenergic receptor antagonists protect against ventricular fibrillation: in vivo and in vitro evidence for enhanced sensitivity to beta2-adrenergic stimulation in animals susceptible to sudden death.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium; Cells, Cultured; Cyclic AMP; Death, Sudden; Dogs; Ethanolamines; Exercise Test; Imidazoles; Isoproterenol; Muscle Fibers, Skeletal; Myocardial Ischemia; Myocardium; Propanolamines; Sensitivity and Specificity; Ventricular Fibrillation | 1997 |
Beta-adrenoceptors in vascular capacitance responses to unloading of carotid baroreceptors in anesthetized dogs.
Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Carotid Arteries; Carotid Sinus; Dogs; Heart Rate; Imidazoles; Pressoreceptors; Propanolamines; Receptors, Adrenergic, beta; Vascular Capacitance | 1997 |
Formoterol and isoproterenol induce c-fos gene expression in osteoblast-like cells by activating beta2-adrenergic receptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DNA, Complementary; Enzyme Activation; Ethanolamines; Formoterol Fumarate; Gene Expression; Genes, fos; Genes, Immediate-Early; Humans; Imidazoles; Isoproterenol; Osteoblasts; Propanolamines; Rats; Receptors, Adrenergic, beta-2; Tumor Cells, Cultured | 1998 |
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1998 |
Relaxation of isolated human myometrial muscle by beta2-adrenergic receptors but not beta1-adrenergic receptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Female; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Myometrium; Potassium Chloride; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1998 |
Characterisation of beta2-adrenoceptors, using the agonist [11C]formoterol and positron emission tomography.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbon Radioisotopes; Ethanolamines; Formoterol Fumarate; Imidazoles; Isoproterenol; Male; Metabolic Clearance Rate; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta-2; Tissue Distribution; Tomography, Emission-Computed | 1998 |
Effects of beta2-adrenergic stimulation on single-channel gating of rat cardiac L-type Ca2+ channels.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium Channels; Calcium Channels, L-Type; Drug Combinations; Electrophysiology; Ethanolamines; Imidazoles; Ion Channel Gating; Isoproterenol; Male; Myocardium; Propanolamines; Rats; Rats, Wistar | 1999 |
Functional and molecular biological evidence for a possible beta3-adrenoceptor in the human detrusor muscle.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colforsin; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 1999 |
Selective activation of beta3-adrenoceptors by octopamine: comparative studies in mammalian fat cells.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adult; Animals; Binding, Competitive; Biogenic Amines; Bupranolol; CHO Cells; Cricetinae; Dioxoles; Dogs; Ethanolamines; Female; Gene Expression; Guinea Pigs; Humans; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lipolysis; Male; Mammals; Mesocricetus; Norepinephrine; Octopamine; Oxygen Consumption; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Species Specificity | 1999 |
Modulation of the pacemaker current If by beta-adrenoceptor subtypes in ventricular myocytes isolated from hypertensive and normotensive rats.
Topics: Action Potentials; Adenosine; Adrenergic alpha-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Cardiomegaly; Catecholamines; GTP-Binding Protein alpha Subunits, Gi-Go; Hypertension; Imidazoles; Isoproterenol; Male; Myocardium; Norepinephrine; Patch-Clamp Techniques; Pertussis Toxin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Virulence Factors, Bordetella | 1999 |
Coupling efficiencies of beta 1- and beta 2-adrenergic receptors expressed alone or together in transfected GH3 pituitary cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Imidazoles; Iodine Radioisotopes; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Pindolol; Pituitary Gland, Anterior; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection | 1999 |
Constitutively active mutants of the beta1-adrenergic receptor.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Betaxolol; Carbazoles; Carvedilol; Cell Line; Cyclic AMP; Epinephrine; Humans; Imidazoles; Isoproterenol; Labetalol; Point Mutation; Practolol; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Timolol | 1999 |
Pharmacological evidence for beta2-adrenoceptor in right atria from stressed female rats.
Topics: Amphetamines; Animals; Dose-Response Relationship, Drug; Estrus; Female; Heart Atria; Heart Rate; Hydroxyquinolines; Imidazoles; Propanolamines; Quinolones; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Stress, Physiological | 1999 |
Opposing effects of beta(1)- and beta(2)-adrenergic receptors on cardiac myocyte apoptosis : role of a pertussis toxin-sensitive G protein.
Topics: Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Apoptosis; Carbachol; Cardiotonic Agents; Cyclic AMP; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Imidazoles; Isoproterenol; Male; Muscarinic Agonists; Myocardium; Pertussis Toxin; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Second Messenger Systems; Virulence Factors, Bordetella | 1999 |
Nitric oxide-dependent vasodilatation of rabbit femoral artery by beta(2)-adrenergic stimulation or cyclic AMP elevation in vivo.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Bucladesine; Colforsin; Cyclic AMP; Enzyme Inhibitors; Femoral Artery; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Tonus; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Propanolamines; Rabbits; Vasodilation | 2000 |
Negative inotropic effects of isoprenaline on isolated left atrial assays from aged transgenic mice with cardiac over-expression of human beta(2)-adrenoceptors.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Aging; Animals; Atrial Function; Cardiotonic Agents; Dose-Response Relationship, Drug; Gene Expression Regulation; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Mice; Mice, Transgenic; Myocardial Contraction; Propanolamines; Receptors, Adrenergic, beta-2 | 2000 |
Contribution of beta-adrenoceptor subtypes to relaxation of colon and oesophagus and pacemaker activity of ureter in wildtype and beta(3)-adrenoceptor knockout mice.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dioxoles; Dose-Response Relationship, Drug; Epinephrine; Esophagus; Female; Imidazoles; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Ureter | 2000 |
Beta-adrenoceptors in equine trachea and heart.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Heart Atria; Heart Ventricles; Horses; Imidazoles; Iodine Radioisotopes; Ligands; Male; Muscle, Smooth; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Regression Analysis; Spectrometry, Gamma; Trachea | 1999 |
Functional assessment of beta adrenoceptor subtypes in human colonic circular and longitudinal (taenia coli) smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Colon; Female; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Terbutaline; Tetrahydronaphthalenes | 2000 |
Beta-adrenergic responses are significantly enhanced in rat carotid artery with intimal hyperplasia.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carotid Artery Injuries; Dose-Response Relationship, Drug; Drug Interactions; Electromyography; Hyperplasia; Imidazoles; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Propanolamines; Rats; Rats, Wistar | 2000 |
beta(1) and beta(2)-adrenergic receptor subtype effects in German shepherd dogs with inherited lethal ventricular arrhythmias.
Topics: Action Potentials; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Death, Sudden, Cardiac; Dog Diseases; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Microelectrodes; Myocardium; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Tachycardia, Ventricular | 2000 |
Transforming growth factor-beta1 inhibits beta2-adrenoceptor gene transcription.
Topics: Adrenergic beta-Antagonists; Binding Sites; Binding, Competitive; Blotting, Northern; Cell Line; Cyclic AMP; Down-Regulation; Embryo, Mammalian; Fibroblasts; Gene Expression; Humans; Imidazoles; Iodine Radioisotopes; Kinetics; Lung; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-2; RNA, Messenger; Transcription, Genetic; Transforming Growth Factor beta; Transforming Growth Factor beta1 | 2000 |
Characterization of beta(1)-selectivity, adrenoceptor-G(s)-protein interaction and inverse agonism of nebivolol in human myocardium.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Benzopyrans; COS Cells; Ethanolamines; GTP-Binding Protein alpha Subunits, Gs; Guanylyl Imidodiphosphate; Heart; Humans; Imidazoles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Myocardial Contraction; Myocardium; Nebivolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Transfection | 2001 |
Different mechanisms mediate beta adrenoceptor stimulated vasorelaxation of coronary and femoral arteries.
Topics: Adrenergic beta-Antagonists; Animals; Arteries; Coronary Vessels; Endothelium, Vascular; Female; Femoral Artery; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; omega-N-Methylarginine; Propanolamines; Swine; Vasodilation | 2000 |
Murine ventricular L-type Ca(2+) current is enhanced by zinterol via beta(1)-adrenoceptors, and is reduced in TG4 mice overexpressing the human beta(2)-adrenoceptor.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Barium; Binding Sites; Calcium; Calcium Channels, L-Type; Electric Conductivity; Ethanolamines; GTP-Binding Protein alpha Subunits, Gi-Go; Heart Ventricles; Humans; Imidazoles; Ion Channel Gating; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Myocardium; Pertussis Toxin; Propanolamines; Protein Binding; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Virulence Factors, Bordetella | 2001 |
Salivary secretion during selective beta-adrenoreceptor stimulation and blockade in the parotid gland of red kangaroos, Macropus rufus.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Electrolytes; Female; Imidazoles; Infusions, Intra-Arterial; Macropodidae; Male; Norepinephrine; Parotid Gland; Phentolamine; Propanolamines; Receptors, Adrenergic, beta; Saliva | 2002 |
Pharmacological characterisation of the beta-adrenoceptor expressed by human lung mast cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Dose-Response Relationship, Drug; Humans; Imidazoles; Isoproterenol; Lung; Mast Cells; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta | 2002 |
Density and binding characteristics of beta-adrenoceptors in the normal and failing equine myocardium.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Heart Diseases; Heart Ventricles; Horse Diseases; Horses; Imidazoles; Iodine Radioisotopes; Male; Myocardium; Propanolamines; Receptors, Adrenergic, beta | 2002 |
Effect of adrenergic antagonists during phenylephrine stimulation of the mandibular gland of red kangaroos, Macropus rufus.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Electrolytes; Extracellular Space; Female; Imidazoles; Macropodidae; Male; Phentolamine; Phenylephrine; Propanolamines; Submandibular Gland | 2002 |
Identification of beta-adrenoceptor subtypes in lower urinary tract of the female pig.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dihydroalprenolol; Ethanolamines; Female; Imidazoles; In Vitro Techniques; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Swine; Urethra; Urinary Bladder | 2002 |
Cardiostimulant and cardiodepressant effects through overexpressed human beta2-adrenoceptors in murine heart: regional differences and functional role of beta1-adrenoceptors.
Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Mice; Mice, Transgenic; Myocardial Contraction; Norepinephrine; Pertussis Toxin; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2003 |
Cardiac-specific overexpression of human beta2 adrenoceptors in mice exposes coupling to both Gs and Gi proteins.
Topics: Adrenergic beta-Antagonists; Animals; Atrial Function, Left; Female; Gene Expression; Genotype; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Humans; Imidazoles; Isoproterenol; Male; Mice; Mice, Transgenic; Models, Theoretical; Pertussis Toxin; Propanolamines; Receptors, Adrenergic, beta-2 | 2003 |
Role of beta-adrenoceptor subtypes in mediating relaxation of the pig bladder trigonal muscle in vitro.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Swine; Urinary Bladder | 2003 |
The third intracellular loop and the carboxyl terminus of beta2-adrenergic receptor confer spontaneous activity of the receptor.
Topics: Adrenergic beta-Antagonists; Animals; Cells, Cultured; Cyclic AMP; Imidazoles; Isoproterenol; Mice; Myocardial Contraction; Myocardium; Propanolamines; Protein Conformation; Protein Structure, Tertiary; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Signal Transduction; Subcellular Fractions | 2003 |
The functional role of beta-adrenoceptor subtypes in mediating relaxation of pig urethral smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Ethanolamines; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Swine; Urethra | 2003 |
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction | 2004 |
Involvement of the serotonin 5-HT2B receptor in cardiac hypertrophy linked to sympathetic stimulation: control of interleukin-6, interleukin-1beta, and tumor necrosis factor-alpha cytokine production by ventricular fibroblasts.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Cardiomegaly; Cells, Cultured; Drug Evaluation, Preclinical; Fibroblasts; Gene Expression Regulation; Heart Ventricles; Imidazoles; Indoles; Interleukin-1; Interleukin-6; Isoproterenol; Mice; Mice, Knockout; Myocytes, Cardiac; Propanolamines; Pyridines; Quinolines; Receptor, Serotonin, 5-HT2B; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Sympathetic Nervous System; Sympathomimetics; Tumor Necrosis Factor-alpha | 2004 |
Natriuretic peptide gene expression after beta-adrenergic stimulation in adult mouse cardiac myocytes.
Topics: Adrenergic beta-Antagonists; Animals; Atrial Natriuretic Factor; Cells, Cultured; Gene Expression; Imidazoles; In Situ Nick-End Labeling; Isoproterenol; Mice; Myocytes, Cardiac; Natriuretic Peptide, Brain; Nerve Tissue Proteins; Propanolamines; RNA, Messenger | 2004 |
Pharmacological modulation of the hyperpolarization-activated current (I f) in human atrial myocytes: focus on G protein-coupled receptors.
Topics: Aged; Arrhythmias, Cardiac; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Ion Transport; Isoproterenol; Male; Membrane Potentials; Middle Aged; Myocytes, Cardiac; Patch-Clamp Techniques; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, G-Protein-Coupled; Receptors, Serotonin, 5-HT4; Serotonin | 2005 |
Evidence for two atypical conformations of beta-adrenoceptors and their interaction with Gi proteins.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Norepinephrine; Pertussis Toxin; Propanolamines; Protein Binding; Protein Conformation; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1 | 2005 |
Carvedilol blocks beta2- more than beta1-adrenoceptors in human heart.
Topics: Adrenergic beta-Antagonists; Calcium Channels, L-Type; Carbazoles; Carvedilol; Dose-Response Relationship, Drug; Epinephrine; Heart Atria; Heart Failure; Heart Ventricles; Humans; Imidazoles; In Vitro Techniques; Metoprolol; Myocardial Contraction; Myocardium; Norepinephrine; Patch-Clamp Techniques; Propanolamines; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 2006 |
Effects of Inflammation upon beta-adrenoceptor concentrations in the common digital artery of the horse: an in vitro study.
Topics: Adrenergic beta-Antagonists; Animals; Arteries; Horse Diseases; Horses; Imidazoles; In Vitro Techniques; Lipopolysaccharides; Muscle, Smooth, Vascular; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Vasculitis | 2005 |
Neural contractions in colonic strips from patients with diverticular disease: role of endocannabinoids and substance P.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Case-Control Studies; Colon; Diverticulum; Endocannabinoids; Female; Glycerides; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Morpholines; Muscle Contraction; Muscle, Smooth; Naphthalenes; Neurokinin-1 Receptor Antagonists; Piperidines; Polyunsaturated Alkamides; Propanolamines; Pyrazoles; Quinuclidines; Rimonabant; Substance P; Tetrodotoxin | 2006 |
Agonist-specific activation of the beta2-adrenoceptor/Gs-protein and beta2-adrenoceptor/Gi-protein pathway in adult rat ventricular cardiomyocytes.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cells, Cultured; Fenoterol; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Heart Ventricles; Imidazoles; In Vitro Techniques; Kinetics; Male; Muscle Proteins; Myocytes, Cardiac; Pertussis Toxin; Phenylalanine; Phenylephrine; Propanolamines; Rats; Rats, Wistar; Signal Transduction; Terbutaline | 2006 |
Functional beta-adrenergic receptor signalling on nuclear membranes in adult rat and mouse ventricular cardiomyocytes.
Topics: Adenylyl Cyclases; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blotting, Western; Dioxoles; Ethanolamines; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Microscopy, Confocal; Myocytes, Cardiac; Nuclear Envelope; Pertussis Toxin; Propanolamines; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Signal Transduction | 2006 |
kappa-opioid receptor stimulation inhibits cardiac hypertrophy induced by beta1-adrenoceptor stimulation in the rat.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Calcium; Cardiomegaly; Cell Size; Cells, Cultured; Imidazoles; Isoproterenol; Leucine; Myocytes, Cardiac; Propanolamines; Proteins; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa | 2007 |
Cathine, an amphetamine-related compound, acts on mammalian spermatozoa via beta1- and alpha2A-adrenergic receptors in a capacitation state-dependent manner.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Benzazepines; Brimonidine Tartrate; Calcium; Cyclic AMP; Imidazoles; Male; Mice; Norepinephrine; Phenylpropanolamine; Phosphorylation; Procaterol; Propanolamines; Quinoxalines; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-1; Sperm Capacitation; Spermatozoa; Tyrosine | 2007 |
Pharmacological characterization of the beta-adrenoceptor that mediates the relaxant response to noradrenaline in guinea-pig tracheal smooth muscle.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Albuterol; Animals; Atenolol; Bupranolol; Butoxamine; Desipramine; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Imidazoles; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Trachea | 2007 |
Adrenergic control of a constitutively active acetylcholine-regulated potassium current in canine atrial cardiomyocytes.
Topics: Acetylcholine; Action Potentials; Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Bee Venoms; Clonidine; Cyclic AMP-Dependent Protein Kinases; Dihydropyridines; Dogs; Dose-Response Relationship, Drug; Estrenes; Heart Atria; Imidazoles; Indoles; Isoproterenol; Isoquinolines; Maleimides; Myocytes, Cardiac; Patch-Clamp Techniques; Phenylephrine; Phorbol 12,13-Dibutyrate; Piperazines; Potassium Channels; Prazosin; Propanolamines; Propranolol; Protein Kinase C; Pyrrolidinones; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Sulfonamides; Type C Phospholipases | 2007 |
Effects of milrinone on contractility and cyclic adenosine monophosphate production induced by beta1- and beta2-adrenergic receptor activation in human myocardium.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Dose-Response Relationship, Drug; Drug Interactions; Epinephrine; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Male; Middle Aged; Milrinone; Myocardial Contraction; Myocardium; Norepinephrine; Phosphodiesterase 3 Inhibitors; Phosphodiesterase Inhibitors; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 2007 |
Phosphodiesterase-4 blunts inotropism and arrhythmias but not sinoatrial tachycardia of (-)-adrenaline mediated through mouse cardiac beta(1)-adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiotonic Agents; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Dose-Response Relationship, Drug; Drug Synergism; Epinephrine; Female; Heart Atria; Heart Rate; Heart Ventricles; Imidazoles; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Myocardial Contraction; Myocytes, Cardiac; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Propanolamines; Quinolones; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Rolipram; Sinoatrial Node; Tachycardia, Sinus; Tachycardia, Ventricular | 2008 |
Deciphering the beta-adrenergic response in human embryonic stem cell-derived-cardiac myocytes: closer to clinical use?
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbachol; Cell Differentiation; Cell Line; Cell Lineage; Dose-Response Relationship, Drug; Embryonic Stem Cells; Heart Failure; Humans; Imidazoles; Isoproterenol; Muscarinic Agonists; Myocardial Contraction; Myocytes, Cardiac; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Stem Cell Transplantation | 2008 |
beta(1)- and beta(2)-adrenoceptor responses in cardiomyocytes derived from human embryonic stem cells: comparison with failing and non-failing adult human heart.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Animals; Carbachol; Cell Differentiation; Cell Line; Cell Lineage; Dose-Response Relationship, Drug; Embryonic Stem Cells; Heart Failure; Humans; Imidazoles; Isoproterenol; Mice; Muscarinic Agonists; Myocardial Contraction; Myocytes, Cardiac; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Stem Cell Transplantation; Time Factors | 2008 |
Mouse embryonic stem cell-derived cardiomyocytes express functional adrenoceptors.
Topics: Animals; Cell Differentiation; Cell Line; Embryonic Stem Cells; Extracellular Signal-Regulated MAP Kinases; Gene Expression; Imidazoles; Isoproterenol; Mice; Myocytes, Cardiac; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptor, Muscarinic M2; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Tyrosine 3-Monooxygenase | 2008 |
Oestrogen changed cardiomyocyte contraction and beta-adrenoceptor expression in rat hearts subjected to ischaemia-reperfusion.
Topics: Adrenergic beta-Antagonists; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Estradiol; Estrogen Antagonists; Estrogens; Female; Fulvestrant; Imidazoles; L-Lactate Dehydrogenase; Myocardial Contraction; Myocardium; Myocytes, Cardiac; Ovariectomy; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Reperfusion Injury | 2008 |
Phosphodiesterases inhibition unmask a positive inotropic effect mediated by beta2-adrenoceptors in rat ventricular myocardium.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Female; GTP-Binding Protein alpha Subunits, Gi-Go; Heart Ventricles; Imidazoles; Male; Myocardial Contraction; Myocardium; Pertussis Toxin; Phosphodiesterase Inhibitors; Propanolamines; Rats; Rats, Sprague-Dawley | 2009 |
Aqueous extract of Zanthoxylum schinifolium elicits contractile and secretory responses via beta1-adrenoceptor activation in beating rabbit atria.
Topics: Animals; Atrial Natriuretic Factor; Blood Pressure; Carbazoles; Cardiotonic Agents; Cardiovascular Agents; Cyclic AMP; Diltiazem; Heart Atria; Hemodynamics; Imidazoles; Plant Extracts; Plant Leaves; Plant Stems; Propanolamines; Propranolol; Pyrroles; Rabbits; Receptors, Adrenergic, beta-1; Stroke Volume; Zanthoxylum | 2009 |
Norepinephrine enhances the LPS-induced expression of COX-2 and secretion of PGE2 in primary rat microglia.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Animals, Newborn; Cells, Cultured; Cerebral Cortex; Cyclooxygenase 2; Dinoprostone; Dose-Response Relationship, Drug; Gene Expression Regulation, Enzymologic; Imidazoles; Immunoenzyme Techniques; Lipopolysaccharides; Microglia; Norepinephrine; Propanolamines; Rats; Rats, Wistar; RNA, Messenger | 2010 |
Predicting in vivo cardiovascular properties of β-blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiovascular Agents; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Heart Rate; Humans; Imidazoles; Isoproterenol; Male; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Rats; Rats, Sprague-Dawley; Vascular Resistance; Xamoterol | 2011 |
β2-adrenoceptor transfection enhances contractile reserve of isolated rat ventricular myocytes exposed to chronic isoprenaline stimulation by improving β1-adrenoceptor responsiveness.
Topics: Adrenergic beta-Antagonists; Animals; Gene Transfer Techniques; Genetic Therapy; Heart Failure; Imidazoles; Isoproterenol; Myocardial Contraction; Myocytes, Cardiac; Primary Cell Culture; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 2012 |
β2-Adrenergic receptor supports prolonged theta tetanus-induced LTP.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Antagonists; Animals; CA1 Region, Hippocampal; Dobutamine; Electric Stimulation; Imidazoles; Long-Term Potentiation; Mice; Mice, Knockout; Phosphorylation; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Synapses; Synaptic Transmission | 2012 |
Role of β-adrenergic receptors in regulation of hepatic fat accumulation during aging.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Cells, Cultured; Enzyme Activation; Fats; Hepatocytes; Imidazoles; Isoproterenol; Lipids; Liver; Male; Mice; Mice, Inbred C57BL; Propanolamines; Propranolol; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction; Time Factors | 2012 |
Both α1- and β1-adrenoceptors in the bed nucleus of the stria terminalis are involved in the expression of conditioned contextual fear.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Conditioning, Psychological; Dioxanes; Electroshock; Fear; Idazoxan; Imidazoles; Male; Phentolamine; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Septal Nuclei | 2012 |
Expression and functional coupling of liver β2 - adrenoceptors in the human hepatocellular carcinoma.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Carcinoma, Hepatocellular; Female; Humans; Imidazoles; Iodocyanopindolol; Liver; Liver Neoplasms; Male; Middle Aged; Propanolamines; Receptors, Adrenergic, beta-2 | 2012 |
Increased response to β₂-adrenoreceptor stimulation augments inhibition of IKr in heart failure ventricular myocytes.
Topics: Action Potentials; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fenoterol; Guinea Pigs; Heart Failure; Heart Ventricles; Imidazoles; Male; Myocardium; Myocytes, Cardiac; Patch-Clamp Techniques; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction; Thionucleotides | 2012 |
Exchange protein directly activated by cAMP mediates slow delayed-rectifier current remodeling by sustained β-adrenergic activation in guinea pig hearts.
Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Calcineurin; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Delayed Rectifier Potassium Channels; Egtazic Acid; Guanine Nucleotide Exchange Factors; Guinea Pigs; Hypertrophy, Left Ventricular; Imidazoles; Ion Channel Gating; Isoproterenol; Myocytes, Cardiac; NFATC Transcription Factors; Patch-Clamp Techniques; Potassium; Propanolamines; Receptors, Adrenergic, beta-1; RNA Interference; RNA, Small Interfering; Second Messenger Systems | 2014 |
The role of adenylyl cyclase isoform 6 in β-adrenoceptor signalling in murine airways.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dinoprostone; Ethanolamines; Fenoterol; Gene Expression Regulation, Enzymologic; Guinea Pigs; Imidazoles; In Vitro Techniques; Isoenzymes; Male; Mice, Knockout; Muscle Contraction; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Receptors, Prostaglandin E, EP2 Subtype; Signal Transduction; Trachea; Vagus Nerve | 2015 |
β-Adrenoceptor-Mediated Relaxation of Carbachol-Pre-Contracted Mouse Detrusor.
Topics: Aminophenols; Animals; Carbachol; Cholinergic Agonists; Colforsin; Homozygote; Imidazoles; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mucous Membrane; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Sulfonamides; Urinary Bladder | 2015 |
Phosphorylation of Ser1928 mediates the enhanced activity of the L-type Ca2+ channel Cav1.2 by the β2-adrenergic receptor in neurons.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium Channels, L-Type; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Female; Imidazoles; Isoproterenol; Long-Term Potentiation; Male; Mice, 129 Strain; Mice, Inbred C57BL; Mice, Transgenic; Myocytes, Cardiac; Neuronal Plasticity; Neurons; Phosphorylation; Propanolamines; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2; Serine; Signal Transduction | 2017 |
The β
Topics: 1-Methyl-3-isobutylxanthine; Acetanilides; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Atrial Function; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Male; Middle Aged; Myocardial Contraction; Propanolamines; Receptors, Adrenergic, beta; Thiazoles | 2017 |
Alveolar liquid clearance in lung injury: Evaluation of the impairment of the β
Topics: Aminophylline; Animals; Blood Pressure; Bronchodilator Agents; Cyclic AMP; Disease Models, Animal; Dogs; Dose-Response Relationship, Drug; Epithelial Sodium Channels; Female; Heart Rate; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Lung Injury; Male; Propanolamines; Protein Binding; Pulmonary Alveoli; Pulmonary Edema; Receptors, Adrenergic, beta-2; Reperfusion Injury; RNA, Messenger | 2019 |