cgp 20712a and ici 118551

cgp 20712a has been researched along with ici 118551 in 133 studies

Research

Studies (133)

TimeframeStudies, this research(%)All Research%
pre-199013 (9.77)18.7374
1990's61 (45.86)18.2507
2000's43 (32.33)29.6817
2010's16 (12.03)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baker, JG1
Baker, JG; Fischer, PM; Gardiner, SM; Hill, SJ; Kellam, B; Mistry, SN1
Baker, JG; Gunera, J; Kolb, P; Schmidt, D1
Bowen, WP; Flint, DJ; Vernon, RG2
Fraeyman, N; Van de Velde, E; Van Ermen, A; Vanscheeuwijck, P1
Majewski, H; Mian, MA; Rand, MJ1
Bals, S; Brodde, OE; Deighton, NM; Motomura, S; Zerkowski, HR1
Choi, AL; Martínez de la Escalera, G; Weiner, RI1
Grino, M; Oliver, C1
Amenta, F; Coppola, L; Ferrante, F; Forlani, A; Gallo, P; Monopoli, A; Napoleone, P1
Flügge, G; Nazarali, AJ; Pinto, JE; Saavedra, JM; Torda, T; Viglione, PN1
Leysen, JE; Pauwels, PJ; Van Gompel, P1
Kim, YS; Molenaar, P; Sainz, RD; Summers, RJ1
Kaumann, AJ; Lemoine, H2
Delavier-Klutchko, C; Emorine, LJ; Marullo, S; Strosberg, AD1
Böhm, M; Erdmann, E; Fruhmann, G; Gengenbach, S; Hauck, RW; Sunder-Plassmann, L1
Cerbai, E; Masini, I; Mugelli, A1
Hall, JA; Latimer, M1
Bühler, FR; Hoyer, D; Jones, CR; Palacios, JM1
Böhm, M; Erdmann, E; Kemkes, B; Klövekorn, WP; Pieske, B; Schnabel, P; Schwinger, R1
Brown, MJ; Hall, JA; Kaumann, AJ; Murray, KJ; Wells, FC1
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW1
Hollenga, C; Zaagsma, J1
Dubbin, PN; Dusting, GJ; Macdonald, PS1
Jones, CR; McMartin, LR; Molenaar, P; Summers, RJ1
Bos, EA; Knot, HJ; Remie, R; Zaagsma, J1
Kaumann, AJ1
Beer, M; Iversen, LL; Poat, J; Richardson, A; Stahl, SM1
Hadcock, JR; Malbon, CC1
Molenaar, P; Summers, RJ1
Canale, E; Molenaar, P; Summers, RJ1
MacDonald, A; McKean, J1
Olszewski, MA; Robinson, NE; Zhang, XY1
Champigneulle, A; Elalouf, JM; Imbert-Teboul, M; Mandon, B; Siga, E1
Badran, TW; Hoey, AJ; Matthews, ML; Pegg, GG; Sillence, MN1
Campbell, B; Iakovidis, D; Jackman, G; Louis, S; Louis, WJ; Tung, LH1
Brown, MJ; Ferro, A; Kaumann, AJ1
Matthews, ML; Moore, NG; Reich, MM; Sillence, MN1
Charpentier, F; Rosen, MR1
Elnatan, J; Molenaar, P; Rosenfeldt, FL; Summers, RJ1
Collins, S; Daniel, KW; Gettys, TW; Ramkumar, V; Rohlfs, EM; Taylor, IL1
Carruba, MO; Nisoli, E; Tonello, C1
Coppes, RP; Dahlöf, C; Tarizzo, VI; Zaagsma, J1
Kuznetsov, V; Pak, E; Robinson, RB; Steinberg, SF1
del Monte, F; Harding, SE; Kaumann, AJ; Pepper, J; Poole-Wilson, PA; Wynne, DG1
Lemoine, H; Rösen, P; Sackmann, B; Zink, S1
Berry, JL; Chiu, P; Cook, SJ; Downing, SJ; Foster, RW; Small, RC1
Berry, JL; Carpenter, JR; Chiu, P; Cook, SJ; Downing, SJ; Foster, RW; Miller, AJ; Small, AM; Small, RC1
Baude, B; Emorine, LJ; Fève, B; Krief, S; Pairault, J; Strosberg, AD; Zilberfarb, V1
Nash, MS; Osborne, NN1
Adachi-Akahane, S; Kitagawa, Y; Nagao, T1
Bültmann, R; Driessen, B; Gonçalves, J; Starke, K1
Barrionuevo, M; Cenarruzabeitia, E; Martínez, JA; Milagro, FI1
Pfaffendorf, M; van Zwieten, PA; Winkler Prins, EA; Zwaveling, J1
Morin, D; Onteniente, B; Sapena, R; Tillement, JP; Zini, R1
Barker, LA; Spadari-Bratfisch, RC; Zanesco, A1
Germack, R; Perret, GY; Starzec, AB; Vassy, R1
Goepel, M; Michel, MC; Rübben, H; Wittmann, A1
Ahrens, O; Flügge, G; Fuchs, E2
Altschuld, RA; Billman, GE; Castillo, LC; Hensley, J; Hohl, CM1
Karim, F; Poucher, SM1
Bilbe, G; Kellenberger, S; Muller, K; Richener, H1
Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F1
Liu, YL; Nwosu, UC; Rice, PJ1
Doze, P; Elsinga, PH; Ensing, K; Kraan, J; Vaalburg, W; van der Mark, TW; van Waarde, A; Visser, TJ1
Herzig, S; Schröder, F1
Ajisawa, Y; Akahane, M; Andersson, KE; Hayakawa, K; Igawa, Y; Nishizawa, O; Takeda, H; Yamazaki, Y; Yoneyama, T1
Atgié, C; Berlan, M; Carpéné, C; Fontana, E; Galitzky, J; Lafontan, M1
Cerbai, E; Mugelli, A; Pino, R; Rodriguez, ML1
Guerrero, SW; Minneman, KP1
Abuin, L; Cotecchia, S; Lattion, A; Nenniger-Tosato, M1
Marcondes, FK; Santos, IN; Spadari-Bartfisch, RC; Vanderlei, LC1
Colucci, WS; Communal, C; Sawyer, DB; Singh, K1
Ferro, A; Gao, L; Li, J; Xu, B1
Black, JW; Prendergast, CE; Shankley, NP1
Giacobino, JP; Jimenez, M; Kaumann, AJ; Moffatt, J; Molenaar, P; Oostendorp, J; Preitner, F1
Töneke, K1
Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S1
Heijenbrok, FJ; Mathy, MJ; Pfaffendorf, M; van Zwieten, PA1
Danilo, P; Gainullin, RZ; Moise, NS; Rosen, MR; Sosunov, EA; Steinberg, SF1
Barnes, PJ; Haddad, EB; Mak, JC; Rousell, J1
Böhm, M; Cremers, B; Dabew, E; Maack, C; Schnabel, P; Südkamp, M; Tyroller, S1
Huang, Y; Xu, B1
Graf, EM; Harding, SE; Herzig, S; Heubach, JF; Jäger, A; Molenaar, P; Ravens, U; Schröder, F1
Beal, AM; Boys, CA1
Chess-Williams, R; Chong, LK; Peachell, PT1
Bailey, S; Berhane, Y; Elliott, J; Horn, J; Marr, CM1
Beal, AM1
Chapple, CR; Chess-Williams, R; Yamanishi, T; Yasuda, K; Yoshida, K3
Blaschke, M; Harding, SE; Heubach, JF; Kaumann, AJ; Ravens, U1
Black, JW; Harper, EA; Hasseldine, AR1
Chakir, K; Cheng, H; Kobilka, BK; Xiang, Y; Xiao, RP; Yang, D; Zhang, SJ1
Brahmadevara, N; MacDonald, A; Shaw, AM1
Callebert, J; Etienne, N; Jaffré, F; Launay, JM; Maroteaux, L; Monassier, L; Nebigil, CG; Sarre, A1
Ander, AN; Drumm, JD; Duggirala, SK; Roth, DM1
Battaglia, F; Bonacchi, M; Casini, S; Cerbai, E; Fiorani, B; Giunti, G; Lonardo, G; Mugelli, A; Sani, G; Stefano, PL1
Caceres, VM; Krieger, MH; Moreira, MF; Santos, IN; Spadari-Bratfisch, RC; Sumitame, M1
Christ, T; Kaumann, A; Molenaar, P; Ravens, U1
Badino, P; Barbero, R; Cuniberti, B; Girardi, C; Magistris, G; Odore, R; Pagliasso, S; Re, G1
Bianchetti, A; Croci, T; Di Marzo, V; Di Palo, S; Ferla, G; Guagnini, F; Matias, I; Mukenge, S; Valenti, M1
Brodde, OE; Gröner, F; Heinroth-Hoffmann, I; Pönicke, K1
Allen, BG; Baragli, A; Boivin, B; Ethier, N; Hébert, TE; Lavoie, C; Trieu, P; Vaniotis, G; Villeneuve, LR1
Jing, Y; Shan, D; Su, Y; Wang, H; Wong, TM1
Adeoya-Osiguwa, SA; Fraser, LR1
Horinouchi, T; Koike, K; Michikawa, H; Tanaka, Y; Yamashita, Y1
Chartier, D; Ehrlich, JR; Hébert, TE; Nattel, S; Qi, X; Yeh, YH1
Aroca, V; Carceles, MD; Fuentes, T; Hernández, J; Lopez, J1
Galindo-Tovar, A; Kaumann, AJ1
Bang, ML; Catalucci, D; Condorelli, G1
Ali, NN; Brito-Martins, M; Harding, SE1
Chen, P; Liu, Z; Ma, K; Yang, H; Zhang, Y; Zhou, C1
Gu, SL; Hao, YL; Sun, H; Wu, Q; Yan, CD; Zhao, Z1
Fuente, T; Gonzalez-Muñoz, C; Hernández-Cascales, J1
Cho, KW; Choi, DH; Choi, HR; Cui, HZ; Kang, DG; Lee, HS1
Candelario-Jalil, E; de Oliveira, AC; Fiebich, BL; Haake, E; Heneka, MT; Hüll, M; Schlachetzki, JC1
Baker, JG; Fretwell, L; Gardiner, SM; Hill, SJ; Kemp, P; March, J1
Gao, L; Jiang, X; Li, D; Sun, H; Wang, Y; Xu, C; Yan, C1
Anderson, ME; He, K; Hell, JW; Koval, OM; Lee, HK; Matt, L; Nguyen, M; Patriarchi, T; Qian, H; Zhang, M1
Barnes, JL; Ghosh, PM; Ikeno, Y; Kamat, A; Katz, MS; Lu, Z; Shu, ZJ; Yeh, CK; Zhang, BX; Zhu, B1
Côrrea, FM; Crestani, CC; Fabri, DR; Gomes, FV; Hott, SC; Reis, DG; Resstel, LB1
Abraham, G; Guenl, B; Jonas, S; Kassahun, WT; Ungemach, FR1
Cao, K; Chen, Y; Wang, H; Wang, S; Xu, D; Zhang, X; Zhu, H; Zou, J1
Aflaki, M; Luo, X; Maguy, A; Nattel, S; Ordog, B; Qi, XY; Shi, Y; Tadevosyan, A; Tardif, JC; Xiao, L1
Belvisi, MG; Birrell, MA; Bonvini, SJ; Buckley, J; Dale, N; Dubuis, ED; Maher, SA; Wortley, MA; Yew-Booth, L1
Lorenz, K; Newe, M; Propping, S; Ravens, U; Wirth, MP1
Buonarati, OR; Catterall, WA; Chowdhury, D; Hell, JW; Hofmann, F; Lee, B; Matt, L; Nanou, E; Navedo, MF; Nieves-Cintrón, M; Nystoriak, MA; Patriarchi, T; Poomvanicha, M; Price, JL; Qian, H1
Kaumann, AJ; Lee, XW; Michel, MC; Mo, W; Molenaar, P1
Berthiaume, Y; Ferraro, P; Massé, C; Richard, C; Shabbir, W1

Other Studies

133 other study(ies) available for cgp 20712a and ici 118551

ArticleYear
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
    British journal of pharmacology, 2005, Volume: 144, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

2005
Synthesis and in vitro and in vivo characterization of highly β1-selective β-adrenoceptor partial agonists.
    Journal of medicinal chemistry, 2013, May-23, Volume: 56, Issue:10

    Topics: Adrenergic beta-1 Receptor Agonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Design; Heart Rate; Hemodynamics; Humans; Indicators and Reagents; Ligands; Male; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Structure-Activity Relationship

2013
Similarity- and Substructure-Based Development of β
    ACS medicinal chemistry letters, 2017, May-11, Volume: 8, Issue:5

    Topics:

2017
Regional and interspecific differences in the ligand binding properties of beta-adrenergic receptors of individual white adipose tissue depots in the sheep and rat.
    Biochemical pharmacology, 1992, Aug-18, Volume: 44, Issue:4

    Topics: Adipose Tissue; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Imidazoles; Iodocyanopindolol; Lactation; Pindolol; Propanolamines; Proteins; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Sheep

1992
Influence of age on the beta 1- and beta 2-adrenergic receptors in rat liver.
    Molecular pharmacology, 1992, Volume: 42, Issue:4

    Topics: Adenylyl Cyclases; Aging; Animals; Binding, Competitive; Cell Membrane; Imidazoles; Liver; Liver Glycogen; Male; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1992
An inhibitory effect of isoprenaline on stimulation-induced noradrenaline release from rat atria.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Electric Stimulation; Female; Heart Atria; Imidazoles; Indomethacin; Isoproterenol; Male; Norepinephrine; Phentolamine; Propanolamines; Rats; Rats, Inbred Strains

1992
Characterization of the beta adrenoceptor subtype(s) mediating the positive inotropic effects of epinine, dopamine, dobutamine, denopamine and xamoterol in isolated human right atrium.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: Adrenergic beta-Agonists; Adult; Aged; Calcium; Deoxyepinephrine; Dobutamine; Dopamine; Ethanolamines; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Male; Middle Aged; Myocardial Contraction; Propanolamines; Stimulation, Chemical; Xamoterol

1992
Beta 1-adrenergic regulation of the GT1 gonadotropin-releasing hormone (GnRH) neuronal cell lines: stimulation of GnRH release via receptors positively coupled to adenylate cyclase.
    Endocrinology, 1992, Volume: 131, Issue:3

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Line; Cyclic AMP; Gonadotropin-Releasing Hormone; Imidazoles; Isoproterenol; Kinetics; Mice; Mice, Transgenic; Neurons; Norepinephrine; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, LHRH

1992
Ontogeny of insulin-induced hypoglycemia stimulation of adrenocorticotropin secretion in the rat: role of catecholamines.
    Endocrinology, 1992, Volume: 131, Issue:6

    Topics: Adrenergic beta-Antagonists; Adrenocorticotropic Hormone; Aging; Animals; Arginine Vasopressin; Catecholamines; Hypoglycemia; Imidazoles; Immunization, Passive; Insulin; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta

1992
Autoradiographic localization of beta-adrenergic receptors in human large coronary arteries.
    Circulation research, 1991, Volume: 68, Issue:6

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Autoradiography; Binding, Competitive; Coronary Vessels; Female; Humans; Imidazoles; Male; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Silver; Tissue Distribution

1991
Increased beta 2-adrenoceptors in the superior cervical ganglia of genetically hypertensive rats.
    Brain research, 1991, Feb-22, Volume: 542, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Enalapril; Ganglia, Sympathetic; Hypertension; Imidazoles; Iodocyanopindolol; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta

1991
Human beta 1- and beta 2-adrenergic receptor binding and mediated accumulation of cAMP in transfected Chinese hamster ovary cells. Profile of nebivolol and known beta-adrenergic blockers.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Benzopyrans; Binding Sites; Binding, Competitive; Cell Line; Cricetinae; Cricetulus; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Models, Biological; Nebivolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Stereoisomerism; Transfection

1991
Characterization of beta 1- and beta 2-adrenoceptors in rat skeletal muscles.
    Biochemical pharmacology, 1991, Oct-09, Volume: 42, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Imidazoles; Male; Membranes; Muscles; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Regional differences of beta 1- and beta 2-adrenoceptor-mediated functions in feline heart. A beta 2-adrenoceptor-mediated positive inotropic effect possibly unrelated to cyclic AMP.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Atrial Function, Left; Cardiotonic Agents; Cats; Cyclic AMP; Epinephrine; Female; Heart; Heart Rate; Imidazoles; Male; Myocardial Contraction; Myocardium; Norepinephrine; Papillary Muscles; Propanolamines; Receptors, Adrenergic, beta; Sinoatrial Node; Ventricular Function, Right

1991
Selective binding of ligands to beta 1, beta 2 or chimeric beta 1/beta 2-adrenergic receptors involves multiple subsites.
    The EMBO journal, 1990, Volume: 9, Issue:5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Sequence; Animals; Escherichia coli; Ethanolamines; Imidazoles; Kinetics; Molecular Sequence Data; Norepinephrine; Procaterol; Propanolamines; Protein Engineering; Receptors, Adrenergic, beta; Recombinant Fusion Proteins; Structure-Activity Relationship; Thermodynamics

1990
Characterization of the beta-adrenergic receptors of sheep adipocytes.
    Biochemical Society transactions, 1990, Volume: 18, Issue:3

    Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Atenolol; Epinephrine; Imidazoles; Isoproterenol; Norepinephrine; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Sheep

1990
Beta 2-adrenoceptors in human lung and peripheral mononuclear leukocytes of untreated and terbutaline-treated patients.
    Chest, 1990, Volume: 98, Issue:2

    Topics: Adrenergic beta-Antagonists; Bronchial Spasm; Down-Regulation; Female; Humans; Imidazoles; Leukocytes, Mononuclear; Lung; Male; Middle Aged; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Terbutaline

1990
Electrophysiological characterization of cardiac beta 2-adrenoceptors in sheep Purkinje fibers.
    Journal of molecular and cellular cardiology, 1990, Volume: 22, Issue:8

    Topics: Action Potentials; Adrenergic beta-Antagonists; Animals; Drug Interactions; Imidazoles; Isoproterenol; Propanolamines; Purkinje Fibers; Receptors, Adrenergic, beta; Sheep

1990
Enoximone potentiates the positive inotropic effects of beta-1- and beta-2-adrenoceptor stimulation in human atrial myocardium.
    Cardiology, 1990, Volume: 77 Suppl 3

    Topics: Adrenergic beta-Antagonists; Diazoxide; Dose-Response Relationship, Drug; Drug Synergism; Enoximone; Humans; Imidazoles; In Vitro Techniques; Myocardial Contraction; Phosphodiesterase Inhibitors; Propanolamines

1990
Receptor modification in the brains of spontaneously hypertensive and Wistar-Kyoto rats: regionally specific and selective increase in cerebellar beta 2-adrenoceptors.
    British journal of clinical pharmacology, 1990, Volume: 30 Suppl 1

    Topics: Animals; Autoradiography; Brain; Cerebellum; Hypertension; Imidazoles; In Vitro Techniques; Iodocyanopindolol; Male; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta

1990
Reduced effects of dopexamine on force of contraction in the failing human heart despite preserved beta 2-adrenoceptor subpopulation.
    Journal of cardiovascular pharmacology, 1989, Volume: 14, Issue:4

    Topics: Adenylyl Cyclases; Adrenergic Agonists; Adrenergic beta-Antagonists; Binding, Competitive; Dopamine; Female; Heart Failure; Humans; Imidazoles; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Propanolamines; Receptors, Adrenergic, beta

1989
A comparison of the effects of adrenaline and noradrenaline on human heart: the role of beta 1- and beta 2-adrenoceptors in the stimulation of adenylate cyclase and contractile force.
    European heart journal, 1989, Volume: 10 Suppl B

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Epinephrine; Heart; Humans; Imidazoles; Myocardial Contraction; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta

1989
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
    European journal of pharmacology, 1989, Aug-29, Volume: 167, Issue:3

    Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta

1989
Direct evidence for the atypical nature of functional beta-adrenoceptors in rat adipocytes.
    British journal of pharmacology, 1989, Volume: 98, Issue:4

    Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Epididymis; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1989
Beta-adrenoceptors on endothelial cells do not influence release of relaxing factor in dog coronary arteries.
    Clinical and experimental pharmacology & physiology, 1987, Volume: 14, Issue:6

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Biological Products; Bradykinin; Coronary Vessels; Dogs; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Isoproterenol; Nitric Oxide; Propanolamines; Prostaglandin Endoperoxides, Synthetic; Receptors, Adrenergic, beta; Vasodilation

1987
Autoradiographic localization and densitometric analysis of beta-1 and beta-2 adrenoceptors in the canine left anterior descending coronary artery.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1

    Topics: Animals; Autoradiography; Coronary Vessels; Dogs; Imidazoles; Iodocyanopindolol; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1988
Characterization of presynaptic beta-adrenoceptors facilitating endogenous noradrenaline release in the portal vein of permanently cannulated, freely moving rats.
    European journal of pharmacology, 1988, Nov-15, Volume: 157, Issue:1

    Topics: Animals; Catheterization; Drug Synergism; Fenoterol; Imidazoles; Male; Norepinephrine; Portal Vein; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Yohimbine

1988
The beta 1-adrenoceptor antagonist CGP 20712 A unmasks beta 2-adrenoceptors activated by (-)-adrenaline in rat sinoatrial node.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Catecholamines; Epinephrine; Heart Rate; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Sinoatrial Node

1986
Beta 2-adrenoceptor-mediated positive inotropic effect of adrenaline in human ventricular myocardium. Quantitative discrepancies with binding and adenylate cyclase stimulation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:4

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Epinephrine; Humans; Imidazoles; In Vitro Techniques; Myocardial Contraction; Myocardium; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Vasodilator Agents

1987
In vitro selectivity of agonists and antagonists for beta 1- and beta 2-adrenoceptor subtypes in rat brain.
    Biochemical pharmacology, 1988, Mar-15, Volume: 37, Issue:6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Brain Chemistry; Cerebral Cortex; Clenbuterol; Imidazoles; In Vitro Techniques; Male; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Stereoisomerism

1988
Down-regulation of beta-adrenergic receptors: agonist-induced reduction in receptor mRNA levels.
    Proceedings of the National Academy of Sciences of the United States of America, 1988, Volume: 85, Issue:14

    Topics: Adrenergic beta-Antagonists; Animals; Cell Line; Cricetinae; Cyclic AMP; DNA; Endonucleases; Imidazoles; Isoproterenol; Kinetics; Male; Nucleic Acid Hybridization; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA, Messenger; Single-Strand Specific DNA and RNA Endonucleases; Vas Deferens

1988
Characterization of beta-1 and beta-2 adrenoceptors in guinea pig atrium: functional and receptor binding studies.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Animals; Electric Stimulation; Ethanolamines; Female; Guinea Pigs; Heart Atria; Heart Rate; Imidazoles; Isoproterenol; Kinetics; Myocardial Contraction; Myocardium; Pindolol; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Stimulation, Chemical; Uterine Contraction; Uterus

1987
Autoradiographic localization of beta-1 and beta-2 adrenoceptors in guinea pig atrium and regions of the conducting system.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:3

    Topics: Animals; Autoradiography; Binding, Competitive; Guinea Pigs; Heart Atria; Heart Conduction System; Imidazoles; Isomerism; Kinetics; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1987
Contributions of beta-adrenoceptor subtypes to responses to isoprenaline in rat isolated distal colon.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:5

    Topics: Animals; Colon; Imidazoles; In Vitro Techniques; Isometric Contraction; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

1995
Beta 2-adrenoceptor activation augments acetylcholine release from tracheal parasympathetic nerves.
    The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 1

    Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Atropine; Electric Stimulation; Horses; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Contraction; Muscle, Smooth; Parasympathetic Nervous System; Propanolamines; Receptors, Adrenergic, beta-2; Trachea

1995
Molecular analysis of beta-adrenergic receptor subtypes in rat collecting duct: effects on cell cAMP and Ca2+ levels.
    The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 2

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Calcium; Cyclic AMP; DNA Primers; Epinephrine; Imidazoles; Isoproterenol; Kidney Cortex; Kidney Tubules, Collecting; Male; Molecular Sequence Data; Mutagenesis; Nephrons; Norepinephrine; Pindolol; Polymerase Chain Reaction; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; RNA, Messenger

1995
Cardiovascular effects of clenbuterol are beta 2-adrenoceptor-mediated in steers.
    Journal of animal science, 1995, Volume: 73, Issue:6

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Blood Glucose; Blood Pressure; Cardiovascular Physiological Phenomena; Cardiovascular System; Cattle; Clenbuterol; Dose-Response Relationship, Drug; Heart Atria; Heart Rate; Imidazoles; Infusions, Intravenous; Isoproterenol; Male; Norepinephrine; Potassium; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

1995
Partial agonist activity of celiprolol.
    Journal of cardiovascular pharmacology, 1993, Volume: 21, Issue:3

    Topics: Adrenergic beta-Antagonists; Airway Resistance; Animals; Blood Pressure; Celiprolol; Decerebrate State; Guinea Pigs; Heart Rate; Imidazoles; In Vitro Techniques; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta

1993
Beta-adrenoceptor subtypes in human coronary artery: desensitization of beta 2-adrenergic vasorelaxation by chronic beta 1-adrenergic stimulation in vitro.
    Journal of cardiovascular pharmacology, 1995, Volume: 25, Issue:1

    Topics: Adrenergic beta-Antagonists; Analysis of Variance; Coronary Vessels; Dose-Response Relationship, Drug; Epinephrine; Heart Transplantation; Humans; Imidazoles; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

1995
Effects of BRL-47672 on growth, beta 2-adrenoceptors, and adenylyl cyclase activation in female rats.
    The American journal of physiology, 1995, Volume: 268, Issue:1 Pt 1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Clenbuterol; Enzyme Activation; Female; Growth; Imidazoles; Organic Chemicals; Propanolamines; Rats; Receptors, Adrenergic, beta; Second Messenger Systems

1995
Beta-adrenergic regulation of action potentials and automaticity in young and adult canine purkinje fibers.
    The American journal of physiology, 1994, Volume: 266, Issue:6 Pt 2

    Topics: Action Potentials; Adrenergic beta-Antagonists; Aging; Albuterol; Animals; Cardiac Pacing, Artificial; Dogs; Imidazoles; In Vitro Techniques; Isoproterenol; Propanolamines; Purkinje Fibers; Receptors, Adrenergic, beta

1994
Autoradiographic localization and quantitation of beta 1- and beta 2-adrenoceptors in the human atrioventricular conducting system: a comparison of patients with idiopathic dilated cardiomyopathy and ischemic heart disease.
    Journal of molecular and cellular cardiology, 1994, Volume: 26, Issue:3

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Atrioventricular Node; Binding, Competitive; Bundle of His; Cardiomyopathy, Dilated; Down-Regulation; Female; Heart Septum; Humans; Imidazoles; Male; Middle Aged; Muscle Proteins; Myocardial Ischemia; Pindolol; Propanolamines; Receptors, Adrenergic, beta

1994
Impaired expression and functional activity of the beta 3- and beta 1-adrenergic receptors in adipose tissue of congenitally obese (C57BL/6J ob/ob) mice.
    Molecular endocrinology (Baltimore, Md.), 1994, Volume: 8, Issue:4

    Topics: Adenylyl Cyclases; Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Cells, Cultured; Cyclic AMP; Diabetes Mellitus, Type 2; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Activation; Epinephrine; Gene Expression Regulation; Hyperglycemia; Imidazoles; Lipolysis; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Obesity; Propanolamines; Propranolol; Receptors, Adrenergic, beta; RNA Splicing; RNA, Messenger

1994
SR 58611A: a novel thermogenic beta-adrenoceptor agonist.
    European journal of pharmacology, 1994, Jul-01, Volume: 259, Issue:2

    Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP; Drug Interactions; Glycerol; Imidazoles; Lipid Metabolism; Male; Obesity; Propanolamines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Tetrahydronaphthalenes

1994
Pre- and postganglionic stimulation-induced noradrenaline overflow is markedly facilitated by a prejunctional beta 2-adrenoceptor-mediated control mechanism in the pithed rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1994, Volume: 349, Issue:6

    Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Decerebrate State; Fenoterol; Ganglia; Heart Rate; Imidazoles; Male; Norepinephrine; Portal Vein; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sympathetic Nervous System; Synaptic Transmission

1994
Beta 2-adrenergic receptor actions in neonatal and adult rat ventricular myocytes.
    Circulation research, 1995, Volume: 76, Issue:1

    Topics: Age Factors; Animals; Animals, Newborn; Calcium; Cells, Cultured; Cyclic AMP; Ethanolamines; Imidazoles; Isoproterenol; Male; Myocardial Contraction; Myocardium; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

1995
Coexistence of functioning beta 1- and beta 2-adrenoceptors in single myocytes from human ventricle.
    Circulation, 1993, Volume: 88, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Epinephrine; Guinea Pigs; Humans; Imidazoles; In Vitro Techniques; Myocardial Contraction; Myocardium; Propanolamines; Receptors, Adrenergic, beta

1993
Regulation of endothelial permeability by beta-adrenoceptor agonists: contribution of beta 1- and beta 2-adrenoceptors.
    Biochimica et biophysica acta, 1993, Sep-13, Volume: 1178, Issue:3

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cattle; Cell Membrane Permeability; Cells, Cultured; Cyclic AMP; Endothelium, Vascular; Enzyme Activation; Ethanolamines; Formoterol Fumarate; Imidazoles; Propanolamines; Receptors, Adrenergic, beta

1993
Beta-adrenoceptor subtypes and the opening of plasmalemmal K(+)-channels in trachealis muscle: electrophysiological and mechanical studies in guinea-pig tissue.
    British journal of pharmacology, 1993, Volume: 109, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Benzopyrans; Cell Membrane; Cromakalim; Electrophysiology; Female; Guinea Pigs; Heart; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Myocardium; Norepinephrine; Potassium Channels; Procaterol; Propanolamines; Pyrroles; Receptors, Adrenergic, beta; Rubidium Radioisotopes; Salmeterol Xinafoate; Trachea

1993
Beta-adrenoceptor subtypes and the opening of plasmalemmal K(+)-channels in bovine trachealis muscle: studies of mechanical activity and ion fluxes.
    British journal of pharmacology, 1993, Volume: 109, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aminophylline; Animals; Cattle; Cell Membrane; Histamine; Imidazoles; In Vitro Techniques; Isometric Contraction; Muscle Relaxation; Muscle, Smooth; Potassium Channels; Propanolamines; Receptors, Adrenergic, beta; Rubidium; Rubidium Radioisotopes; Trachea

1993
Transcriptional modulation by n-butyric acid of beta 1-, beta 2-, and beta 3-adrenergic receptor balance in 3T3-F442A adipocytes.
    The Journal of biological chemistry, 1994, Mar-04, Volume: 269, Issue:9

    Topics: 3T3 Cells; Adenylyl Cyclase Inhibitors; Adipocytes; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Animals; Base Sequence; Butyrates; Butyric Acid; DNA Primers; DNA, Complementary; Ethanolamines; Gene Expression Regulation; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Molecular Sequence Data; Oligonucleotides, Antisense; Pindolol; Polymerase Chain Reaction; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Transcription, Genetic

1994
Agonist-induced effects on cyclic AMP metabolism are affected in pigment epithelial cells of the Royal College of Surgeons rat.
    Neurochemistry international, 1995, Volume: 27, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprostadil; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dinoprostone; Fibroblast Growth Factor 2; Imidazoles; Isoproterenol; Kinetics; Melatonin; Pigment Epithelium of Eye; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta-2; Receptors, Purinergic P1; Serotonin

1995
Determination of beta-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective beta-antagonists.
    British journal of pharmacology, 1995, Volume: 116, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cyclic AMP; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Membranes; Myocardium; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Tritium

1995
Opposite modulation of noradrenaline and ATP release in guinea-pig vas deferens through prejunctional beta-adrenoceptors: evidence for the beta 2 subtype.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Imidazoles; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Norepinephrine; Prazosin; Propanolamines; Receptors, Adrenergic, beta-2; Suramin; Terbutaline; Vas Deferens

1996
Potential anti-diabetic applications of a new molecule with affinity for beta 3-adrenoceptors.
    Life sciences, 1996, Volume: 59, Issue:11

    Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Benzyl Alcohols; Blood Glucose; Diabetes Mellitus, Experimental; Esophagus; Female; Guinea Pigs; Imidazoles; Insulin; Muscle Relaxation; Muscle, Smooth; Oxygen Consumption; Propanolamines; Rats; Rats, Wistar; Triglycerides

1996
The influence of hyperthyroidism on beta-adrenoceptor-mediated relaxation of isolated small mesenteric arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Colforsin; Dose-Response Relationship, Drug; Hyperthyroidism; Imidazoles; Isoproterenol; Male; Mesenteric Arteries; Methoxamine; Muscle Contraction; Muscle Relaxation; Propanolamines; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Wistar; Thromboxane A2; Thyroxine; Vascular Resistance; Vasoconstrictor Agents

1996
Characterization of beta-adrenergic receptors of freshly isolated astrocytes and neurons from rat brain.
    Life sciences, 1997, Volume: 60, Issue:4-5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Astrocytes; Binding, Competitive; Cells, Cultured; Cerebellum; Imidazoles; Immunohistochemistry; Male; Neurons; Propanolamines; Prosencephalon; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1997
Sino-aortic denervation causes right atrial beta adrenoceptor down-regulation.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 280, Issue:2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Down-Regulation; Heart Atria; Heart Rate; Imidazoles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Male; Muscle Denervation; Myocardium; Neurons; Norepinephrine; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Sinoatrial Node

1997
Beta-adrenoceptor subtype expression and function in rat white adipocytes.
    British journal of pharmacology, 1997, Volume: 120, Issue:2

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Binding, Competitive; Imidazoles; Lipolysis; Male; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta

1997
Comparison of adrenoceptor subtype expression in porcine and human bladder and prostate.
    Urological research, 1997, Volume: 25, Issue:3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Humans; Imidazoles; Isoquinolines; Male; Oxymetazoline; Piperazines; Prazosin; Propanolamines; Prostate; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Swine; Urinary Bladder; Yohimbine

1997
Beta-adrenoceptors in the tree shrew brain. I. Distribution and characterization of [125I]iodocyanopindolol binding sites.
    Cellular and molecular neurobiology, 1997, Volume: 17, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Brain Chemistry; Imidazoles; Iodocyanopindolol; Nerve Tissue Proteins; Organ Specificity; Pindolol; Propanolamines; Protein Binding; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Serotonin; Serotonin; Substrate Specificity; Tupaiidae

1997
Beta-adrenoceptors in the tree shrew brain. II. Time-dependent effects of chronic psychosocial stress on [125I]iodocyanopindolol bindings sites.
    Cellular and molecular neurobiology, 1997, Volume: 17, Issue:4

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Body Weight; Brain Chemistry; Chronic Disease; Down-Regulation; Hydrocortisone; Imidazoles; Iodocyanopindolol; Male; Norepinephrine; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Social Dominance; Stress, Psychological; Time Factors; Tupaiidae

1997
Beta2-adrenergic receptor antagonists protect against ventricular fibrillation: in vivo and in vitro evidence for enhanced sensitivity to beta2-adrenergic stimulation in animals susceptible to sudden death.
    Circulation, 1997, Sep-16, Volume: 96, Issue:6

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium; Cells, Cultured; Cyclic AMP; Death, Sudden; Dogs; Ethanolamines; Exercise Test; Imidazoles; Isoproterenol; Muscle Fibers, Skeletal; Myocardial Ischemia; Myocardium; Propanolamines; Sensitivity and Specificity; Ventricular Fibrillation

1997
Beta-adrenoceptors in vascular capacitance responses to unloading of carotid baroreceptors in anesthetized dogs.
    The American journal of physiology, 1997, Volume: 273, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Carotid Arteries; Carotid Sinus; Dogs; Heart Rate; Imidazoles; Pressoreceptors; Propanolamines; Receptors, Adrenergic, beta; Vascular Capacitance

1997
Formoterol and isoproterenol induce c-fos gene expression in osteoblast-like cells by activating beta2-adrenergic receptors.
    Bone, 1998, Volume: 22, Issue:5

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DNA, Complementary; Enzyme Activation; Ethanolamines; Formoterol Fumarate; Gene Expression; Genes, fos; Genes, Immediate-Early; Humans; Imidazoles; Isoproterenol; Osteoblasts; Propanolamines; Rats; Receptors, Adrenergic, beta-2; Tumor Cells, Cultured

1998
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
    Respiration physiology, 1998, Volume: 112, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

1998
Relaxation of isolated human myometrial muscle by beta2-adrenergic receptors but not beta1-adrenergic receptors.
    American journal of obstetrics and gynecology, 1998, Volume: 179, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Female; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Myometrium; Potassium Chloride; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

1998
Characterisation of beta2-adrenoceptors, using the agonist [11C]formoterol and positron emission tomography.
    European journal of pharmacology, 1998, Nov-13, Volume: 361, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbon Radioisotopes; Ethanolamines; Formoterol Fumarate; Imidazoles; Isoproterenol; Male; Metabolic Clearance Rate; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta-2; Tissue Distribution; Tomography, Emission-Computed

1998
Effects of beta2-adrenergic stimulation on single-channel gating of rat cardiac L-type Ca2+ channels.
    The American journal of physiology, 1999, Volume: 276, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium Channels; Calcium Channels, L-Type; Drug Combinations; Electrophysiology; Ethanolamines; Imidazoles; Ion Channel Gating; Isoproterenol; Male; Myocardium; Propanolamines; Rats; Rats, Wistar

1999
Functional and molecular biological evidence for a possible beta3-adrenoceptor in the human detrusor muscle.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colforsin; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

1999
Selective activation of beta3-adrenoceptors by octopamine: comparative studies in mammalian fat cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adult; Animals; Binding, Competitive; Biogenic Amines; Bupranolol; CHO Cells; Cricetinae; Dioxoles; Dogs; Ethanolamines; Female; Gene Expression; Guinea Pigs; Humans; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Lipolysis; Male; Mammals; Mesocricetus; Norepinephrine; Octopamine; Oxygen Consumption; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Species Specificity

1999
Modulation of the pacemaker current If by beta-adrenoceptor subtypes in ventricular myocytes isolated from hypertensive and normotensive rats.
    Cardiovascular research, 1999, Volume: 42, Issue:1

    Topics: Action Potentials; Adenosine; Adrenergic alpha-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Cardiomegaly; Catecholamines; GTP-Binding Protein alpha Subunits, Gi-Go; Hypertension; Imidazoles; Isoproterenol; Male; Myocardium; Norepinephrine; Patch-Clamp Techniques; Pertussis Toxin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Virulence Factors, Bordetella

1999
Coupling efficiencies of beta 1- and beta 2-adrenergic receptors expressed alone or together in transfected GH3 pituitary cells.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Imidazoles; Iodine Radioisotopes; Isopropyl Thiogalactoside; Isoproterenol; Kinetics; Pindolol; Pituitary Gland, Anterior; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Transfection

1999
Constitutively active mutants of the beta1-adrenergic receptor.
    FEBS letters, 1999, Sep-03, Volume: 457, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Betaxolol; Carbazoles; Carvedilol; Cell Line; Cyclic AMP; Epinephrine; Humans; Imidazoles; Isoproterenol; Labetalol; Point Mutation; Practolol; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Proteins; Timolol

1999
Pharmacological evidence for beta2-adrenoceptor in right atria from stressed female rats.
    Canadian journal of physiology and pharmacology, 1999, Volume: 77, Issue:6

    Topics: Amphetamines; Animals; Dose-Response Relationship, Drug; Estrus; Female; Heart Atria; Heart Rate; Hydroxyquinolines; Imidazoles; Propanolamines; Quinolones; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Stress, Physiological

1999
Opposing effects of beta(1)- and beta(2)-adrenergic receptors on cardiac myocyte apoptosis : role of a pertussis toxin-sensitive G protein.
    Circulation, 1999, Nov-30, Volume: 100, Issue:22

    Topics: Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Apoptosis; Carbachol; Cardiotonic Agents; Cyclic AMP; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Imidazoles; Isoproterenol; Male; Muscarinic Agonists; Myocardium; Pertussis Toxin; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Second Messenger Systems; Virulence Factors, Bordetella

1999
Nitric oxide-dependent vasodilatation of rabbit femoral artery by beta(2)-adrenergic stimulation or cyclic AMP elevation in vivo.
    British journal of pharmacology, 2000, Volume: 129, Issue:5

    Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Bucladesine; Colforsin; Cyclic AMP; Enzyme Inhibitors; Femoral Artery; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Tonus; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Propanolamines; Rabbits; Vasodilation

2000
Negative inotropic effects of isoprenaline on isolated left atrial assays from aged transgenic mice with cardiac over-expression of human beta(2)-adrenoceptors.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Aging; Animals; Atrial Function; Cardiotonic Agents; Dose-Response Relationship, Drug; Gene Expression Regulation; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Mice; Mice, Transgenic; Myocardial Contraction; Propanolamines; Receptors, Adrenergic, beta-2

2000
Contribution of beta-adrenoceptor subtypes to relaxation of colon and oesophagus and pacemaker activity of ureter in wildtype and beta(3)-adrenoceptor knockout mice.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dioxoles; Dose-Response Relationship, Drug; Epinephrine; Esophagus; Female; Imidazoles; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Ureter

2000
Beta-adrenoceptors in equine trachea and heart.
    Veterinary research communications, 1999, Volume: 23, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Heart Atria; Heart Ventricles; Horses; Imidazoles; Iodine Radioisotopes; Ligands; Male; Muscle, Smooth; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Regression Analysis; Spectrometry, Gamma; Trachea

1999
Functional assessment of beta adrenoceptor subtypes in human colonic circular and longitudinal (taenia coli) smooth muscle.
    Gut, 2000, Volume: 47, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Colon; Female; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Terbutaline; Tetrahydronaphthalenes

2000
Beta-adrenergic responses are significantly enhanced in rat carotid artery with intimal hyperplasia.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 362, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carotid Artery Injuries; Dose-Response Relationship, Drug; Drug Interactions; Electromyography; Hyperplasia; Imidazoles; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Propanolamines; Rats; Rats, Wistar

2000
beta(1) and beta(2)-adrenergic receptor subtype effects in German shepherd dogs with inherited lethal ventricular arrhythmias.
    Cardiovascular research, 2000, Volume: 48, Issue:2

    Topics: Action Potentials; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Death, Sudden, Cardiac; Dog Diseases; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Ethanolamines; Imidazoles; In Vitro Techniques; Isoproterenol; Microelectrodes; Myocardium; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Tachycardia, Ventricular

2000
Transforming growth factor-beta1 inhibits beta2-adrenoceptor gene transcription.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 362, Issue:6

    Topics: Adrenergic beta-Antagonists; Binding Sites; Binding, Competitive; Blotting, Northern; Cell Line; Cyclic AMP; Down-Regulation; Embryo, Mammalian; Fibroblasts; Gene Expression; Humans; Imidazoles; Iodine Radioisotopes; Kinetics; Lung; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-2; RNA, Messenger; Transcription, Genetic; Transforming Growth Factor beta; Transforming Growth Factor beta1

2000
Characterization of beta(1)-selectivity, adrenoceptor-G(s)-protein interaction and inverse agonism of nebivolol in human myocardium.
    British journal of pharmacology, 2001, Volume: 132, Issue:8

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Benzopyrans; COS Cells; Ethanolamines; GTP-Binding Protein alpha Subunits, Gs; Guanylyl Imidodiphosphate; Heart; Humans; Imidazoles; In Vitro Techniques; Iodocyanopindolol; Isoproterenol; Myocardial Contraction; Myocardium; Nebivolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Transfection

2001
Different mechanisms mediate beta adrenoceptor stimulated vasorelaxation of coronary and femoral arteries.
    Acta pharmacologica Sinica, 2000, Volume: 21, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Arteries; Coronary Vessels; Endothelium, Vascular; Female; Femoral Artery; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; omega-N-Methylarginine; Propanolamines; Swine; Vasodilation

2000
Murine ventricular L-type Ca(2+) current is enhanced by zinterol via beta(1)-adrenoceptors, and is reduced in TG4 mice overexpressing the human beta(2)-adrenoceptor.
    British journal of pharmacology, 2001, Volume: 133, Issue:1

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Barium; Binding Sites; Calcium; Calcium Channels, L-Type; Electric Conductivity; Ethanolamines; GTP-Binding Protein alpha Subunits, Gi-Go; Heart Ventricles; Humans; Imidazoles; Ion Channel Gating; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Myocardium; Pertussis Toxin; Propanolamines; Protein Binding; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Virulence Factors, Bordetella

2001
Salivary secretion during selective beta-adrenoreceptor stimulation and blockade in the parotid gland of red kangaroos, Macropus rufus.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 2002, Volume: 172, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Electrolytes; Female; Imidazoles; Infusions, Intra-Arterial; Macropodidae; Male; Norepinephrine; Parotid Gland; Phentolamine; Propanolamines; Receptors, Adrenergic, beta; Saliva

2002
Pharmacological characterisation of the beta-adrenoceptor expressed by human lung mast cells.
    European journal of pharmacology, 2002, Feb-15, Volume: 437, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Dose-Response Relationship, Drug; Humans; Imidazoles; Isoproterenol; Lung; Mast Cells; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta

2002
Density and binding characteristics of beta-adrenoceptors in the normal and failing equine myocardium.
    Equine veterinary journal, 2002, Volume: 34, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Heart Diseases; Heart Ventricles; Horse Diseases; Horses; Imidazoles; Iodine Radioisotopes; Male; Myocardium; Propanolamines; Receptors, Adrenergic, beta

2002
Effect of adrenergic antagonists during phenylephrine stimulation of the mandibular gland of red kangaroos, Macropus rufus.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 2002, Volume: 172, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Electrolytes; Extracellular Space; Female; Imidazoles; Macropodidae; Male; Phentolamine; Phenylephrine; Propanolamines; Submandibular Gland

2002
Identification of beta-adrenoceptor subtypes in lower urinary tract of the female pig.
    The Journal of urology, 2002, Volume: 168, Issue:6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dihydroalprenolol; Ethanolamines; Female; Imidazoles; In Vitro Techniques; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Swine; Urethra; Urinary Bladder

2002
Cardiostimulant and cardiodepressant effects through overexpressed human beta2-adrenoceptors in murine heart: regional differences and functional role of beta1-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 367, Issue:4

    Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Mice; Mice, Transgenic; Myocardial Contraction; Norepinephrine; Pertussis Toxin; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

2003
Cardiac-specific overexpression of human beta2 adrenoceptors in mice exposes coupling to both Gs and Gi proteins.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Adrenergic beta-Antagonists; Animals; Atrial Function, Left; Female; Gene Expression; Genotype; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Humans; Imidazoles; Isoproterenol; Male; Mice; Mice, Transgenic; Models, Theoretical; Pertussis Toxin; Propanolamines; Receptors, Adrenergic, beta-2

2003
Role of beta-adrenoceptor subtypes in mediating relaxation of the pig bladder trigonal muscle in vitro.
    Neurourology and urodynamics, 2003, Volume: 22, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Dose-Response Relationship, Drug; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Swine; Urinary Bladder

2003
The third intracellular loop and the carboxyl terminus of beta2-adrenergic receptor confer spontaneous activity of the receptor.
    Molecular pharmacology, 2003, Volume: 64, Issue:5

    Topics: Adrenergic beta-Antagonists; Animals; Cells, Cultured; Cyclic AMP; Imidazoles; Isoproterenol; Mice; Myocardial Contraction; Myocardium; Propanolamines; Protein Conformation; Protein Structure, Tertiary; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Signal Transduction; Subcellular Fractions

2003
The functional role of beta-adrenoceptor subtypes in mediating relaxation of pig urethral smooth muscle.
    The Journal of urology, 2003, Volume: 170, Issue:6 Pt 1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Ethanolamines; Female; Imidazoles; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Swine; Urethra

2003
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction

2004
Involvement of the serotonin 5-HT2B receptor in cardiac hypertrophy linked to sympathetic stimulation: control of interleukin-6, interleukin-1beta, and tumor necrosis factor-alpha cytokine production by ventricular fibroblasts.
    Circulation, 2004, Aug-24, Volume: 110, Issue:8

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Animals; Cardiomegaly; Cells, Cultured; Drug Evaluation, Preclinical; Fibroblasts; Gene Expression Regulation; Heart Ventricles; Imidazoles; Indoles; Interleukin-1; Interleukin-6; Isoproterenol; Mice; Mice, Knockout; Myocytes, Cardiac; Propanolamines; Pyridines; Quinolines; Receptor, Serotonin, 5-HT2B; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Sympathetic Nervous System; Sympathomimetics; Tumor Necrosis Factor-alpha

2004
Natriuretic peptide gene expression after beta-adrenergic stimulation in adult mouse cardiac myocytes.
    DNA and cell biology, 2004, Volume: 23, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Atrial Natriuretic Factor; Cells, Cultured; Gene Expression; Imidazoles; In Situ Nick-End Labeling; Isoproterenol; Mice; Myocytes, Cardiac; Natriuretic Peptide, Brain; Nerve Tissue Proteins; Propanolamines; RNA, Messenger

2004
Pharmacological modulation of the hyperpolarization-activated current (I f) in human atrial myocytes: focus on G protein-coupled receptors.
    Journal of molecular and cellular cardiology, 2005, Volume: 38, Issue:3

    Topics: Aged; Arrhythmias, Cardiac; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Ion Transport; Isoproterenol; Male; Membrane Potentials; Middle Aged; Myocytes, Cardiac; Patch-Clamp Techniques; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, G-Protein-Coupled; Receptors, Serotonin, 5-HT4; Serotonin

2005
Evidence for two atypical conformations of beta-adrenoceptors and their interaction with Gi proteins.
    European journal of pharmacology, 2005, Apr-18, Volume: 513, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Norepinephrine; Pertussis Toxin; Propanolamines; Protein Binding; Protein Conformation; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1

2005
Carvedilol blocks beta2- more than beta1-adrenoceptors in human heart.
    Cardiovascular research, 2006, Volume: 69, Issue:1

    Topics: Adrenergic beta-Antagonists; Calcium Channels, L-Type; Carbazoles; Carvedilol; Dose-Response Relationship, Drug; Epinephrine; Heart Atria; Heart Failure; Heart Ventricles; Humans; Imidazoles; In Vitro Techniques; Metoprolol; Myocardial Contraction; Myocardium; Norepinephrine; Patch-Clamp Techniques; Propanolamines; Propranolol; Receptors, Adrenergic; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

2006
Effects of Inflammation upon beta-adrenoceptor concentrations in the common digital artery of the horse: an in vitro study.
    Veterinary research communications, 2005, Volume: 29 Suppl 2

    Topics: Adrenergic beta-Antagonists; Animals; Arteries; Horse Diseases; Horses; Imidazoles; In Vitro Techniques; Lipopolysaccharides; Muscle, Smooth, Vascular; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Vasculitis

2005
Neural contractions in colonic strips from patients with diverticular disease: role of endocannabinoids and substance P.
    Gut, 2006, Volume: 55, Issue:7

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Case-Control Studies; Colon; Diverticulum; Endocannabinoids; Female; Glycerides; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Morpholines; Muscle Contraction; Muscle, Smooth; Naphthalenes; Neurokinin-1 Receptor Antagonists; Piperidines; Polyunsaturated Alkamides; Propanolamines; Pyrazoles; Quinuclidines; Rimonabant; Substance P; Tetrodotoxin

2006
Agonist-specific activation of the beta2-adrenoceptor/Gs-protein and beta2-adrenoceptor/Gi-protein pathway in adult rat ventricular cardiomyocytes.
    British journal of pharmacology, 2006, Volume: 147, Issue:7

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cells, Cultured; Fenoterol; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Heart Ventricles; Imidazoles; In Vitro Techniques; Kinetics; Male; Muscle Proteins; Myocytes, Cardiac; Pertussis Toxin; Phenylalanine; Phenylephrine; Propanolamines; Rats; Rats, Wistar; Signal Transduction; Terbutaline

2006
Functional beta-adrenergic receptor signalling on nuclear membranes in adult rat and mouse ventricular cardiomyocytes.
    Cardiovascular research, 2006, Jul-01, Volume: 71, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blotting, Western; Dioxoles; Ethanolamines; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Mice; Microscopy, Confocal; Myocytes, Cardiac; Nuclear Envelope; Pertussis Toxin; Propanolamines; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Signal Transduction

2006
kappa-opioid receptor stimulation inhibits cardiac hypertrophy induced by beta1-adrenoceptor stimulation in the rat.
    European journal of pharmacology, 2007, Jan-26, Volume: 555, Issue:2-3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Calcium; Cardiomegaly; Cell Size; Cells, Cultured; Imidazoles; Isoproterenol; Leucine; Myocytes, Cardiac; Propanolamines; Proteins; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

2007
Cathine, an amphetamine-related compound, acts on mammalian spermatozoa via beta1- and alpha2A-adrenergic receptors in a capacitation state-dependent manner.
    Human reproduction (Oxford, England), 2007, Volume: 22, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Benzazepines; Brimonidine Tartrate; Calcium; Cyclic AMP; Imidazoles; Male; Mice; Norepinephrine; Phenylpropanolamine; Phosphorylation; Procaterol; Propanolamines; Quinoxalines; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-1; Sperm Capacitation; Spermatozoa; Tyrosine

2007
Pharmacological characterization of the beta-adrenoceptor that mediates the relaxant response to noradrenaline in guinea-pig tracheal smooth muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Albuterol; Animals; Atenolol; Bupranolol; Butoxamine; Desipramine; Desoxycorticosterone; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Imidazoles; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Trachea

2007
Adrenergic control of a constitutively active acetylcholine-regulated potassium current in canine atrial cardiomyocytes.
    Cardiovascular research, 2007, Jun-01, Volume: 74, Issue:3

    Topics: Acetylcholine; Action Potentials; Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Bee Venoms; Clonidine; Cyclic AMP-Dependent Protein Kinases; Dihydropyridines; Dogs; Dose-Response Relationship, Drug; Estrenes; Heart Atria; Imidazoles; Indoles; Isoproterenol; Isoquinolines; Maleimides; Myocytes, Cardiac; Patch-Clamp Techniques; Phenylephrine; Phorbol 12,13-Dibutyrate; Piperazines; Potassium Channels; Prazosin; Propanolamines; Propranolol; Protein Kinase C; Pyrrolidinones; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Sulfonamides; Type C Phospholipases

2007
Effects of milrinone on contractility and cyclic adenosine monophosphate production induced by beta1- and beta2-adrenergic receptor activation in human myocardium.
    Clinical therapeutics, 2007, Volume: 29, Issue:8

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Dose-Response Relationship, Drug; Drug Interactions; Epinephrine; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Male; Middle Aged; Milrinone; Myocardial Contraction; Myocardium; Norepinephrine; Phosphodiesterase 3 Inhibitors; Phosphodiesterase Inhibitors; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

2007
Phosphodiesterase-4 blunts inotropism and arrhythmias but not sinoatrial tachycardia of (-)-adrenaline mediated through mouse cardiac beta(1)-adrenoceptors.
    British journal of pharmacology, 2008, Volume: 153, Issue:4

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiotonic Agents; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Dose-Response Relationship, Drug; Drug Synergism; Epinephrine; Female; Heart Atria; Heart Rate; Heart Ventricles; Imidazoles; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Myocardial Contraction; Myocytes, Cardiac; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 4 Inhibitors; Phosphodiesterase Inhibitors; Propanolamines; Quinolones; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Rolipram; Sinoatrial Node; Tachycardia, Sinus; Tachycardia, Ventricular

2008
Deciphering the beta-adrenergic response in human embryonic stem cell-derived-cardiac myocytes: closer to clinical use?
    British journal of pharmacology, 2008, Volume: 153, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Carbachol; Cell Differentiation; Cell Line; Cell Lineage; Dose-Response Relationship, Drug; Embryonic Stem Cells; Heart Failure; Humans; Imidazoles; Isoproterenol; Muscarinic Agonists; Myocardial Contraction; Myocytes, Cardiac; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Stem Cell Transplantation

2008
beta(1)- and beta(2)-adrenoceptor responses in cardiomyocytes derived from human embryonic stem cells: comparison with failing and non-failing adult human heart.
    British journal of pharmacology, 2008, Volume: 153, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Animals; Carbachol; Cell Differentiation; Cell Line; Cell Lineage; Dose-Response Relationship, Drug; Embryonic Stem Cells; Heart Failure; Humans; Imidazoles; Isoproterenol; Mice; Muscarinic Agonists; Myocardial Contraction; Myocytes, Cardiac; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Stem Cell Transplantation; Time Factors

2008
Mouse embryonic stem cell-derived cardiomyocytes express functional adrenoceptors.
    Biochemical and biophysical research communications, 2008, Apr-18, Volume: 368, Issue:4

    Topics: Animals; Cell Differentiation; Cell Line; Embryonic Stem Cells; Extracellular Signal-Regulated MAP Kinases; Gene Expression; Imidazoles; Isoproterenol; Mice; Myocytes, Cardiac; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptor, Muscarinic M2; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Tyrosine 3-Monooxygenase

2008
Oestrogen changed cardiomyocyte contraction and beta-adrenoceptor expression in rat hearts subjected to ischaemia-reperfusion.
    Experimental physiology, 2008, Volume: 93, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Estradiol; Estrogen Antagonists; Estrogens; Female; Fulvestrant; Imidazoles; L-Lactate Dehydrogenase; Myocardial Contraction; Myocardium; Myocytes, Cardiac; Ovariectomy; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Reperfusion Injury

2008
Phosphodiesterases inhibition unmask a positive inotropic effect mediated by beta2-adrenoceptors in rat ventricular myocardium.
    European journal of pharmacology, 2009, Apr-01, Volume: 607, Issue:1-3

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Female; GTP-Binding Protein alpha Subunits, Gi-Go; Heart Ventricles; Imidazoles; Male; Myocardial Contraction; Myocardium; Pertussis Toxin; Phosphodiesterase Inhibitors; Propanolamines; Rats; Rats, Sprague-Dawley

2009
Aqueous extract of Zanthoxylum schinifolium elicits contractile and secretory responses via beta1-adrenoceptor activation in beating rabbit atria.
    Journal of ethnopharmacology, 2009, Nov-12, Volume: 126, Issue:2

    Topics: Animals; Atrial Natriuretic Factor; Blood Pressure; Carbazoles; Cardiotonic Agents; Cardiovascular Agents; Cyclic AMP; Diltiazem; Heart Atria; Hemodynamics; Imidazoles; Plant Extracts; Plant Leaves; Plant Stems; Propanolamines; Propranolol; Pyrroles; Rabbits; Receptors, Adrenergic, beta-1; Stroke Volume; Zanthoxylum

2009
Norepinephrine enhances the LPS-induced expression of COX-2 and secretion of PGE2 in primary rat microglia.
    Journal of neuroinflammation, 2010, Jan-11, Volume: 7

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Animals, Newborn; Cells, Cultured; Cerebral Cortex; Cyclooxygenase 2; Dinoprostone; Dose-Response Relationship, Drug; Gene Expression Regulation, Enzymologic; Imidazoles; Immunoenzyme Techniques; Lipopolysaccharides; Microglia; Norepinephrine; Propanolamines; Rats; Rats, Wistar; RNA, Messenger

2010
Predicting in vivo cardiovascular properties of β-blockers from cellular assays: a quantitative comparison of cellular and cardiovascular pharmacological responses.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2011, Volume: 25, Issue:12

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiovascular Agents; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Heart Rate; Humans; Imidazoles; Isoproterenol; Male; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Rats; Rats, Sprague-Dawley; Vascular Resistance; Xamoterol

2011
β2-adrenoceptor transfection enhances contractile reserve of isolated rat ventricular myocytes exposed to chronic isoprenaline stimulation by improving β1-adrenoceptor responsiveness.
    Journal of receptor and signal transduction research, 2012, Volume: 32, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Gene Transfer Techniques; Genetic Therapy; Heart Failure; Imidazoles; Isoproterenol; Myocardial Contraction; Myocytes, Cardiac; Primary Cell Culture; Propanolamines; Rats; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2

2012
β2-Adrenergic receptor supports prolonged theta tetanus-induced LTP.
    Journal of neurophysiology, 2012, Volume: 107, Issue:10

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Antagonists; Animals; CA1 Region, Hippocampal; Dobutamine; Electric Stimulation; Imidazoles; Long-Term Potentiation; Mice; Mice, Knockout; Phosphorylation; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Synapses; Synaptic Transmission

2012
Role of β-adrenergic receptors in regulation of hepatic fat accumulation during aging.
    The Journal of endocrinology, 2012, Volume: 213, Issue:3

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Cells, Cultured; Enzyme Activation; Fats; Hepatocytes; Imidazoles; Isoproterenol; Lipids; Liver; Male; Mice; Mice, Inbred C57BL; Propanolamines; Propranolol; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction; Time Factors

2012
Both α1- and β1-adrenoceptors in the bed nucleus of the stria terminalis are involved in the expression of conditioned contextual fear.
    British journal of pharmacology, 2012, Volume: 167, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Conditioning, Psychological; Dioxanes; Electroshock; Fear; Idazoxan; Imidazoles; Male; Phentolamine; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Septal Nuclei

2012
Expression and functional coupling of liver β2 - adrenoceptors in the human hepatocellular carcinoma.
    Pharmacology, 2012, Volume: 89, Issue:5-6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Carcinoma, Hepatocellular; Female; Humans; Imidazoles; Iodocyanopindolol; Liver; Liver Neoplasms; Male; Middle Aged; Propanolamines; Receptors, Adrenergic, beta-2

2012
Increased response to β₂-adrenoreceptor stimulation augments inhibition of IKr in heart failure ventricular myocytes.
    PloS one, 2012, Volume: 7, Issue:9

    Topics: Action Potentials; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fenoterol; Guinea Pigs; Heart Failure; Heart Ventricles; Imidazoles; Male; Myocardium; Myocytes, Cardiac; Patch-Clamp Techniques; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction; Thionucleotides

2012
Exchange protein directly activated by cAMP mediates slow delayed-rectifier current remodeling by sustained β-adrenergic activation in guinea pig hearts.
    Circulation research, 2014, Mar-14, Volume: 114, Issue:6

    Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Calcineurin; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Delayed Rectifier Potassium Channels; Egtazic Acid; Guanine Nucleotide Exchange Factors; Guinea Pigs; Hypertrophy, Left Ventricular; Imidazoles; Ion Channel Gating; Isoproterenol; Myocytes, Cardiac; NFATC Transcription Factors; Patch-Clamp Techniques; Potassium; Propanolamines; Receptors, Adrenergic, beta-1; RNA Interference; RNA, Small Interfering; Second Messenger Systems

2014
The role of adenylyl cyclase isoform 6 in β-adrenoceptor signalling in murine airways.
    British journal of pharmacology, 2015, Volume: 172, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dinoprostone; Ethanolamines; Fenoterol; Gene Expression Regulation, Enzymologic; Guinea Pigs; Imidazoles; In Vitro Techniques; Isoenzymes; Male; Mice, Knockout; Muscle Contraction; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Receptors, Prostaglandin E, EP2 Subtype; Signal Transduction; Trachea; Vagus Nerve

2015
β-Adrenoceptor-Mediated Relaxation of Carbachol-Pre-Contracted Mouse Detrusor.
    Urologia internationalis, 2015, Volume: 95, Issue:1

    Topics: Aminophenols; Animals; Carbachol; Cholinergic Agonists; Colforsin; Homozygote; Imidazoles; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Mucous Membrane; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Sulfonamides; Urinary Bladder

2015
Phosphorylation of Ser1928 mediates the enhanced activity of the L-type Ca2+ channel Cav1.2 by the β2-adrenergic receptor in neurons.
    Science signaling, 2017, 01-24, Volume: 10, Issue:463

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium Channels, L-Type; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Female; Imidazoles; Isoproterenol; Long-Term Potentiation; Male; Mice, 129 Strain; Mice, Inbred C57BL; Mice, Transgenic; Myocytes, Cardiac; Neuronal Plasticity; Neurons; Phosphorylation; Propanolamines; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2; Serine; Signal Transduction

2017
The β
    British journal of pharmacology, 2017, Volume: 174, Issue:16

    Topics: 1-Methyl-3-isobutylxanthine; Acetanilides; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Atrial Function; Female; Heart Atria; Humans; Imidazoles; In Vitro Techniques; Male; Middle Aged; Myocardial Contraction; Propanolamines; Receptors, Adrenergic, beta; Thiazoles

2017
Alveolar liquid clearance in lung injury: Evaluation of the impairment of the β
    Respiratory physiology & neurobiology, 2019, Volume: 259

    Topics: Aminophylline; Animals; Blood Pressure; Bronchodilator Agents; Cyclic AMP; Disease Models, Animal; Dogs; Dose-Response Relationship, Drug; Epithelial Sodium Channels; Female; Heart Rate; Imidazoles; Iodine Radioisotopes; Iodocyanopindolol; Lung Injury; Male; Propanolamines; Protein Binding; Pulmonary Alveoli; Pulmonary Edema; Receptors, Adrenergic, beta-2; Reperfusion Injury; RNA, Messenger

2019