cgp 12177 has been researched along with timolol in 8 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (37.50) | 18.7374 |
1990's | 4 (50.00) | 18.2507 |
2000's | 1 (12.50) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bultsma, T; Donné-Op den Kelder, GM; Rademaker, B; Timmerman, H | 1 |
Baker, JG | 1 |
Kaila, T | 1 |
Wilkinson, DA; Wilkinson, M | 1 |
Baer, M; Chanton, C; Porzig, H | 1 |
Ali-Melkkilä, T; Iisalo, E; Kaila, T; Saari, KM; Vuori, ML | 2 |
Boutilier, RG; Gamperl, AK; Wilkinson, M | 1 |
2 trial(s) available for cgp 12177 and timolol
Article | Year |
---|---|
Absorption of ocular timolol: drug concentrations and beta-receptor binding activity in the aqueous humour of the treated and contralateral eye.
Topics: Absorption; Administration, Topical; Adrenergic beta-Antagonists; Aged; Animals; Aqueous Humor; Cataract Extraction; Heart Rate; Humans; Lenses, Intraocular; Ophthalmic Solutions; Propanolamines; Rabbits; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Timolol | 1993 |
Beta 1- and beta 2-antagonist activity of topically applied betaxolol and timolol in the systemic circulation.
Topics: Administration, Topical; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Aged; Aged, 80 and over; Betaxolol; Humans; Middle Aged; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Timolol | 1993 |
6 other study(ies) available for cgp 12177 and timolol
Article | Year |
---|---|
Mapping of the beta 2-adrenoceptor on Chang liver cells. Differences between high- and low-affinity receptor states.
Topics: Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Hydrogen Bonding; Iodocyanopindolol; Liver; Models, Molecular; Pindolol; Protein Conformation; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship | 1988 |
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2005 |
A sensitive radioligand binding assay for timolol in plasma.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Blood Proteins; Cell Membrane; Female; Gas Chromatography-Mass Spectrometry; Humans; In Vitro Techniques; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Reticulocytes; Timolol | 1991 |
Beta-adrenergic [( 3H]CGP-12177) binding to brain slices and single intact pineal glands.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain; Cerebral Cortex; Cricetinae; In Vitro Techniques; Isoproterenol; Kinetics; Male; Mesocricetus; Phentolamine; Pineal Gland; Propanolamines; Rats; Rats, Inbred Strains; Timolol | 1985 |
Properties of beta-adrenoceptor sites in metabolizing and nonmetabolizing rat reticulocytes and in resealed reticulocyte ghosts.
Topics: Adrenergic beta-Antagonists; Animals; Cell Membrane; Cold Temperature; Cytosol; Dihydroalprenolol; Energy Metabolism; Female; Isoproterenol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reticulocytes; Timolol | 1981 |
Beta-adrenoreceptors in the trout (Oncorhynchus mykiss) heart: characterization, quantification, and effects of repeated catecholamine exposure.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Catecholamines; Down-Regulation; Freezing; Heart; Heart Ventricles; Myocardium; Oncorhynchus mykiss; Propanolamines; Receptors, Adrenergic, beta; Stereoisomerism; Stress, Psychological; Timolol | 1994 |