cgp 12177 and pyrroles

cgp 12177 has been researched along with pyrroles in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chang, FR; Chen, IJ; Kuo, RY; Wu, CC; Wu, YC; Yeh, JL1
Kinsella, BT; O'Meara, SJ1
Briddon, SJ; Gherbi, K; Hill, SJ1
Baker, JG; Briddon, SJ; Gherbi, K; Hill, SJ; May, LT1

Other Studies

4 other study(ies) available for cgp 12177 and pyrroles

ArticleYear
Antiplatelet activity of synthetic pyrrolo-benzylisoquinolines.
    Bioorganic & medicinal chemistry letters, 2003, Mar-10, Volume: 13, Issue:5

    Topics: Adrenergic Antagonists; Animals; Arachidonic Acid; Aspirin; Benzyl Compounds; Collagen; Guinea Pigs; Humans; Inhibitory Concentration 50; Isoquinolines; Platelet Aggregation; Platelet Aggregation Inhibitors; Propanolamines; Pyrroles; Structure-Activity Relationship; Tumor Cells, Cultured

2003
Effect of the statin atorvastatin on intracellular signalling by the prostacyclin receptor in vitro and in vivo.
    British journal of pharmacology, 2004, Volume: 143, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenylyl Cyclases; Animals; Atorvastatin; Blood Platelets; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cell Line; Cell Line, Tumor; Cholesterol; Clinical Trials as Topic; Cyclic AMP; Drug Evaluation, Preclinical; Fatty Acids, Unsaturated; Female; Heptanoic Acids; Humans; Hydantoins; Hydrazines; Iloprost; Ireland; Lipids; Male; Mice; Middle Aged; Propanolamines; Protein Prenylation; Pyrroles; Radioligand Assay; Receptor Cross-Talk; Receptors, Epoprostenol; Receptors, Immunologic; Receptors, Prostaglandin; Signal Transduction; Tritium

2004
Detection of the secondary, low-affinity β1 -adrenoceptor site in living cells using the fluorescent CGP 12177 derivative BODIPY-TMR-CGP.
    British journal of pharmacology, 2014, Volume: 171, Issue:23

    Topics: Adrenergic beta-1 Receptor Agonists; Animals; Boron Compounds; CHO Cells; Cricetulus; Cyclic AMP; Cyclopentanes; Fluorescent Dyes; Genes, Reporter; Humans; Membrane Proteins; Propanolamines; Pyrroles; Receptors, Adrenergic, beta-1; Response Elements

2014
Negative cooperativity across β1-adrenoceptor homodimers provides insights into the nature of the secondary low-affinity CGP 12177 β1-adrenoceptor binding conformation.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2015, Volume: 29, Issue:7

    Topics: Adrenergic beta-Antagonists; Animals; Binding Sites; Boron Compounds; CHO Cells; Cricetinae; Cricetulus; Cyclopentanes; Humans; Kinetics; Ligands; Mutagenesis, Site-Directed; Propanolamines; Protein Conformation; Protein Multimerization; Protein Structure, Quaternary; Pyrroles; Receptors, Adrenergic, beta-1; Recombinant Proteins

2015