cgp 12177 has been researched along with propranolol in 75 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 17 (22.67) | 18.7374 |
1990's | 27 (36.00) | 18.2507 |
2000's | 28 (37.33) | 29.6817 |
2010's | 3 (4.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Batink, HD; Boer, GJ; Doornbos, T; Dubois, EA; Janssen, AG; Pfaffendorf, M; Somsen, GA; van den Bos, JC; van Doremalen, PA; van Royen, EA; van Zwieten, PA; Vekemans, JA | 1 |
Iakovidis, D; Jackman, GP; Louis, SN; Louis, WJ; Nero, TL | 1 |
Baker, JG | 2 |
Charlton, SJ; Dickson, CJ; Duca, JS; Fairhurst, RA; Hornak, V; McKay, DJ; Pearlstein, RA; Reilly, J; Sandham, DA; Shaw, D; Sykes, DA; Velez-Vega, C | 1 |
Van Liefde, I; Van Witzenburg, A; Vauquelin, G | 1 |
Blanksma, PK; Bouwer, J; Elsinga, PH; Lie, KI; Meeder, JG; Paans, AM; Vaalburg, W; van Waarde, A; Visser, GM | 1 |
Leysen, JE; Pauwels, PJ; Van Gompel, P | 1 |
Lenz, T; Strobel, G; Weicker, H; Werle, E | 1 |
Mauz, AB; Pelzer, H | 1 |
Cannon, B; Herron, D; Néchad, M; Nedergaard, J; Rehnmark, S | 1 |
Dunn, AJ; Yang, XM | 1 |
Bouscarel, B; Cortinovis, C; Mayer, D; Murat, JC; Paris, H | 1 |
Belz, GG; Palm, D; Wellstein, A | 1 |
Marsh, JD; Sweeney, KA | 1 |
Nose, M; Scholz, H; Steinkraus, V; Thormählen, K | 1 |
Francendese, A; Hjeresen, DL; O'Donnell, JM | 1 |
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
Graafsma, SJ; Rodrigues de Miranda, JF; Snijders, PJ; Thien, T | 1 |
O'Donnell, JM | 1 |
Anakwe, OO; Moger, WH; Murphy, PR | 1 |
Henneberry, RC; Jahangeer, S; Lysko, PG | 1 |
Molinoff, PB; Reynolds, EE | 1 |
Akamatsu, N; Oikawa, S; Okeyama, N; Shima, S | 1 |
Belz, GG; Palm, D; Pitschner, HF; Wellstein, A | 1 |
Cunningham, EM; DeBlasi, A; Insel, PA; Motulsky, HJ | 1 |
De Blasi, A; Fratelli, M; Lipartiti, M; Wielosz, M | 1 |
Delavier-Klutchko, C; Hoebeke, J; Strosberg, AD | 1 |
Mutschler, E; Palm, D; Schäfer-Korting, M; Wellstein, A; Wiemer, G | 1 |
Brodde, OE; Elsinga, PH; Vaalburg, W; Van Waarde, A; Visser, GM | 1 |
Arner, P; Enocksson, S; Lönnqvist, F; Nordenström, J; Shimizu, M | 1 |
Hirsch, DJ; Morgunov, NS; You, YD | 1 |
Change, HT; Chen, CF; Liao, JF | 1 |
Berlan, M; Carpéné, C; Galitzky, J; Lafontan, M; Portillo, M; Reverte, M | 1 |
Kaila, T; Marttila, R | 1 |
Law, MP | 1 |
Fujii, N; Homma, S; Ikegami, H; Miyazaki, H | 1 |
Kashiwada, K; Ogata, H; Ohira, M; Someya, K; Takahashi, H | 1 |
el Borai, N; Ito, K; Nakano, S; Nakazawa, H; Tanaka, E; Yamakawa, A; Yamamura, M | 1 |
Kaumann, AJ | 1 |
Hattori, K; Hosohata, Y; Maruyama, K; Nagatomo, T; Ohnuki, T; Sasaki, K; Suzuki, J; Watanabe, K | 1 |
Garnier, V; Tillement, JP; Zini, R | 1 |
Crema, F; de Ponti, F; Frigo, G; Gibelli, G; Modini, C | 1 |
Faundez, V; Kelly, RB; Marullo, S | 1 |
Gao, BB; Han, QD | 1 |
Brown, D; Freestone, NS; Heubach, JF; Kaumann, AJ; Ravens, U; Wettwer, E | 1 |
Kanda, Y; Kuroki, Y; Mizuno, K; Tomiyama, K; Watanabe, Y | 1 |
Koike, K; Yamamoto, Y | 1 |
Brawley, L; MacDonald, A; Shaw, AM | 1 |
Hagmüller, K; Hofer, D; Korsatko, W; Porta, S; Raíces, M; Schauenstein, K; Zaninovich, A | 1 |
Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S | 1 |
Horinouchi, T; Koike, K | 4 |
Gibbs, ME; Summers, RJ | 1 |
Capuzzo, A; Fabbri, E; Moon, TW; Selva, C | 1 |
Bach, TJ; Brady, E; Candelore, MR; Cascieri, MA; Fisher, MH; Fletcher, DJ; Forrest, MJ; Hom, GJ; Iliff, SA; MacIntyre, DE; Mathvink, R; Metzger, J; Pecore, V; Saperstein, R; Shih, T; Weber, AE; Wyvratt, M; Zafian, P | 1 |
Santos, IN; Spadari-Bratfisch, RC | 1 |
Malo, A; Puerta, M | 1 |
Busch, M; Funsch, B; Gradl, G; Lohse, MJ; Pschorr, J; Scheel, AA | 1 |
Bölck, B; Brixius, K; Bundkirchen, A; Schwinger, RH | 1 |
Fong, KM; Kaumann, AJ; Li, L; Lynham, JA; Molenaar, P; Rabnott, G; Russell, FD; Sarsero, D; Yang, I | 1 |
Marcondes, FK; Santos, IN; Spadari-Bratfisch, RC | 1 |
Huang, Y; O'Donnell, JM; Zhang, HT | 1 |
Kolár, F; Myslivecek, J; Rícný, J; Tucek, S | 1 |
Colledge, WH; Grace, AA; Joseph, SS; Kaumann, AJ; Lynham, JA; Molenaar, P | 1 |
Brahmadevara, N; MacDonald, A; Shaw, AM | 1 |
Beigi, F; Chakir, K; Wainer, IW; Xiao, RP | 1 |
Blum, JW; Carron, J; Hammon, HM; Morel, C | 1 |
Carter, AA; Hill, SJ | 1 |
Koike, K; Matsushita, M; Tanaka, Y | 1 |
Huang, Y; O'Donnell, JM; Whisler, LR; Xiang, Y; Zhang, HT | 1 |
Granzow, M; Heller, J; Hennenberg, M; Klein, S; Laleman, W; Nevens, F; Sauerbruch, T; Schulze Pröbsting, A; Trebicka, J; Zaagsma, J | 1 |
Abdelkrim, MA; Chatagnon, G; Desfontis, JC; Gogny, M; Mallem, MY; Noireaud, J | 1 |
2 trial(s) available for cgp 12177 and propranolol
Article | Year |
---|---|
Receptor binding of propranolol is the missing link between plasma concentration kinetics and the effect-time course in man.
Topics: Adult; Animals; Blood Pressure; Double-Blind Method; Half-Life; Heart Rate; Humans; In Vitro Techniques; Kinetics; Male; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta | 1985 |
Receptor occupancy in lumbar CSF as a measure of the antagonist activity of atenolol, metoprolol and propranolol in the CNS.
Topics: Adrenergic alpha-Antagonists; Adult; Animals; Atenolol; Central Nervous System; Female; Humans; In Vitro Techniques; Male; Metoprolol; Middle Aged; Propanolamines; Propranolol; Rabbits; Rats; Receptors, Adrenergic, alpha | 1993 |
73 other study(ies) available for cgp 12177 and propranolol
Article | Year |
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Synthesis and in vitro and in vivo characteristics of an iodinated analogue of the beta-adrenoceptor antagonist carazolol.
Topics: Adrenergic beta-Antagonists; Animals; Brain; Carbazoles; Cell Membrane; Heart Ventricles; Indicators and Reagents; Iodine Radioisotopes; Lung; Magnetic Resonance Spectroscopy; Male; Myocardium; Propanolamines; Rabbits; Radioligand Assay; Receptors, Adrenergic, beta; Tissue Distribution | 1996 |
LK 204-545, a highly selective beta1-adrenoceptor antagonist at human beta-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; Cyclopropanes; Female; Humans; Imidazoles; In Vitro Techniques; Ligands; Phenoxypropanolamines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Trachea; Urea | 1999 |
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2005 |
Uncoupling the Structure-Activity Relationships of β2 Adrenergic Receptor Ligands from Membrane Binding.
Topics: Binding Sites; Cell Membrane; Dose-Response Relationship, Drug; Humans; Ligands; Models, Molecular; Molecular Structure; Receptors, Adrenergic, beta-2; Structure-Activity Relationship | 2016 |
Multiple beta adrenergic receptor subclasses mediate the l-isoproterenol-induced lipolytic response in rat adipocytes.
Topics: Adipose Tissue; Animals; Dose-Response Relationship, Drug; Ethanolamines; In Vitro Techniques; Isoproterenol; Lipolysis; Male; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1992 |
Suitability of CGP-12177 and CGP-26505 for quantitative imaging of beta-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Imidazoles; Male; Metabolic Clearance Rate; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Time Factors; Tissue Distribution; Tritium | 1992 |
Human beta 1- and beta 2-adrenergic receptor binding and mediated accumulation of cAMP in transfected Chinese hamster ovary cells. Profile of nebivolol and known beta-adrenergic blockers.
Topics: Adrenergic beta-Antagonists; Animals; Benzopyrans; Binding Sites; Binding, Competitive; Cell Line; Cricetinae; Cricetulus; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Models, Biological; Nebivolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Stereoisomerism; Transfection | 1991 |
O-Methylated and sulfoconjugated catecholamines: differential activities at human platelet alpha 2-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Adult; Binding, Competitive; Blood Platelets; Catecholamines; Dopamine; Humans; In Vitro Techniques; Lipids; Mandelic Acids; Methylation; Platelet Aggregation; Platelet Aggregation Inhibitors; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, alpha; Sulfur; Yohimbine | 1991 |
Beta-adrenoceptor-binding studies of the cardioselective beta blockers bisoprolol, H-I 42 BS, and HX-CH 44 BS to heart membranes and intact ventricular myocytes of adult rats: two beta 1-binding sites for bisoprolol.
Topics: Adrenergic beta-Antagonists; Animals; Bisoprolol; Cell Membrane; In Vitro Techniques; Isoquinolines; Male; Myocardium; Propanolamines; Propranolol; Quinazolinones; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1990 |
Alpha- and beta-adrenergic induction of the expression of the uncoupling protein thermogenin in brown adipocytes differentiated in culture.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Colforsin; Gene Expression; Insulin; Ion Channels; Male; Membrane Proteins; Mice; Mitochondrial Proteins; Norepinephrine; Nucleic Acid Hybridization; Oxymetazoline; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; RNA; RNA, Messenger; Thyroxine; Triiodothyronine; Uncoupling Protein 1 | 1990 |
Central beta 1-adrenergic receptors are involved in CRF-induced defensive withdrawal.
Topics: Animals; Atenolol; Behavior, Animal; Corticotropin-Releasing Hormone; Injections, Intraperitoneal; Injections, Intraventricular; Male; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1990 |
Study of beta-adrenoceptors and beta-adrenergic responsiveness in cultured "preneoplastic-like" and neoplastic rat hepatocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Antagonists; Albuterol; Animals; Atenolol; Binding, Competitive; Cells, Cultured; Cyclic AMP; Epinephrine; Isoproterenol; Kinetics; Liver Neoplasms, Experimental; Norepinephrine; Precancerous Conditions; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta | 1985 |
Affinity and selectivity of beta-adrenoceptor antagonists in vitro.
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Betaxolol; Binding, Competitive; Bisoprolol; Propanolamines; Propranolol; Rats; Salivary Glands; Tritium | 1986 |
Beta-adrenergic receptor regulation during hypoxia in intact cultured heart cells.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Cells, Cultured; Chick Embryo; Cyclic AMP; Heart; Hypoxia; Myocardium; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Time course and extent of alpha 1-adrenoceptor density changes in rat heart after beta-adrenoceptor blockade.
Topics: Adrenergic beta-Antagonists; Animals; Cycloheximide; Heart; Heart Rate; Male; Myocardial Contraction; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1989 |
Microwave attenuation of ethanol-induced interactions with noradrenergic neurotransmitter systems.
Topics: Adrenergic beta-Antagonists; Animals; Ethanol; Female; Hypothermia, Induced; Male; Microwaves; Neurotransmitter Agents; Propanolamines; Propranolol; Rats | 1989 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Complications of (-)125I-iodocyanopindolol binding to human mononuclear cells.
Topics: Binding, Competitive; Humans; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Leukocytes, Mononuclear; Models, Biological; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Sonication; Stereoisomerism | 1987 |
Behavioral consequences of activation of beta adrenergic receptors by clenbuterol: evidence for mediation by the central nervous system.
Topics: Animals; Behavior, Animal; Binding, Competitive; Central Nervous System; Clenbuterol; Ethanolamines; Male; Pindolol; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1988 |
Characterization of beta-adrenergic binding sites on rodent Leydig cells.
Topics: Adrenergic beta-Antagonists; Androgens; Animals; Binding, Competitive; Cell Separation; Cells, Cultured; Colforsin; Isoproterenol; Kinetics; Leydig Cells; Luteinizing Hormone; Male; Mice; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1985 |
Transport of beta-adrenergic antagonists in the absence of beta-adrenergic receptors in rat pituitary tumor cells.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Biological Transport; Cell Line; Colforsin; Cyclic AMP; Dihydroalprenolol; Epinephrine; Hydrogen-Ion Concentration; Imipramine; Kinetics; Monensin; Norepinephrine; Nucleotides; Oligomycins; Ouabain; Pituitary Neoplasms; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta; Reserpine; Serotonin; Temperature | 1986 |
Down regulation of beta adrenergic receptors in S49 lymphoma cells induced by atypical agonists.
Topics: Adrenergic beta-Agonists; Animals; Binding Sites; Celiprolol; Cell Division; Cell Line; Isoproterenol; Kinetics; Lymphoma; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Time Factors | 1986 |
Effects of chronic propranolol treatment on hepatic adenylate cyclase system in the rat.
Topics: Adenosine Diphosphate; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Blood Glucose; Cell Membrane; Electrophoresis, Polyacrylamide Gel; Glucagon; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Liver; Liver Glycogen; Male; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Sodium Fluoride | 1987 |
Desensitization and redistribution of beta-adrenergic receptors on human mononuclear leukocytes.
Topics: Adolescent; Adult; Binding, Competitive; Cyclic AMP; Drug Tolerance; Female; Humans; Iodocyanopindolol; Isoproterenol; Leukocytes; Male; Monocytes; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1986 |
Regulation of beta adrenergic receptors on rat mononuclear leukocytes by stress: receptor redistribution and down-regulation are altered with aging.
Topics: Aging; Animals; Cyclic AMP; Dihydroalprenolol; Isoproterenol; Male; Monocytes; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Restraint, Physical; Stress, Physiological; Time Factors | 1987 |
The human carcinoma cell line A431 possesses large numbers of functional beta-adrenergic receptors.
Topics: Adrenergic beta-Antagonists; Binding, Competitive; Carcinoma, Squamous Cell; Cell Line; Dihydroalprenolol; Humans; Isoproterenol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 1984 |
Simple and reliable radioreceptor assay for beta-adrenoceptor antagonists and active metabolites in native human plasma.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Carteolol; Dihydroalprenolol; Erythrocyte Membrane; Female; Humans; Male; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Time Factors | 1984 |
Myocardial and pulmonary uptake of S-1'-[18F]fluorocarazolol in intact rats reflects radioligand binding to beta-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Carbazoles; Chlorpromazine; Fluorine Radioisotopes; Isoproterenol; Lung; Male; Myocardium; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Tomography, Emission-Computed | 1995 |
Demonstration of an in vivo functional beta 3-adrenoceptor in man.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adult; Analysis of Variance; Animals; Body Temperature Regulation; Cells, Cultured; Dobutamine; Female; Humans; Isoproterenol; Kinetics; Lipolysis; Male; Mammals; Metoprolol; Microdialysis; Middle Aged; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reference Values; Regional Blood Flow; Terbutaline; Time Factors | 1995 |
Response of mouse proximal straight tubule and medullary thick ascending limb to beta-agonist.
Topics: Adrenergic beta-Antagonists; Animals; Electrophysiology; Furosemide; In Vitro Techniques; Isoproterenol; Kidney Medulla; Kidney Tubules; Kidney Tubules, Proximal; Kinetics; Membrane Potentials; Mice; Perfusion; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta | 1993 |
Characterization of agonist-induced internalization and down-regulation of beta-adrenergic receptors in isolated rat lung and heart preparations.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Cycloheximide; Down-Regulation; Endocytosis; Heart; Hypertonic Solutions; Iodocyanopindolol; Isoproterenol; Lung; Male; Myocardium; Organ Specificity; Pindolol; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Sucrose; Terbutaline | 1993 |
Coexistence of beta 1-, beta 2-, and beta 3-adrenoceptors in dog fat cells and their differential activation by catecholamines.
Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamines; Cell Membrane; Dogs; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Isoproterenol; Norepinephrine; Procaterol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tetrahydronaphthalenes | 1993 |
Demonstration of the suitability of CGP 12177 for in vivo studies of beta-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Heart Ventricles; Liver; Lung; Male; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Stereoisomerism; Tissue Distribution; Tomography, Emission-Computed | 1993 |
Dynamic exercise induces translocation of beta-adrenergic receptors in human lymphocytes.
Topics: Adrenergic beta-Antagonists; Adult; Cell Membrane; Cyclic AMP; Exercise; Exercise Test; Humans; Isoproterenol; Lymphocytes; Propanolamines; Propranolol; Radioimmunoassay; Receptors, Adrenergic, beta | 1993 |
Dosing rate-dependent relationship between propranolol plasma concentration and beta-blockade.
Topics: Adult; Animals; Delayed-Action Preparations; Dose-Response Relationship, Drug; Female; Guinea Pigs; Heart Atria; Heart Rate; Humans; In Vitro Techniques; Male; Propanolamines; Propranolol; Rabbits | 1993 |
Regulation of heat production of brown adipocytes via typical and atypical beta-adrenoceptors in the rat.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Calorimetry; Ethanolamines; In Vitro Techniques; Isoproterenol; Male; Phenoxyacetates; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1995 |
(-)-CGP 12177-induced increase of human atrial contraction through a putative third beta-adrenoceptor.
Topics: Adrenergic beta-Antagonists; Adult; Aged; Bupranolol; Female; Heart Atria; Humans; In Vitro Techniques; Male; Middle Aged; Myocardial Contraction; Propanolamines; Propranolol; Receptors, Adrenergic; Stimulation, Chemical | 1996 |
Effects of chronic administration of bopindolol on the binding characteristics of cardiac alpha 1H-, alpha 1L-, beta 1- and beta 2-adrenoceptor subtypes in cardiac muscles of spontaneously hypertensive rats (SHR).
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Hypertension; In Vitro Techniques; Membranes; Myocardium; Pindolol; Propanolamines; Propranolol; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1996 |
A GppNHp-insensitivity factor modulates the activation of beta-adrenoceptor-coupled Gs protein in rat cortex and cerebellum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Astrocytes; Cerebellum; Cerebral Cortex; Cholic Acids; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Kinetics; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Synaptosomes | 1999 |
Atypical beta-adrenoceptors mediating relaxation in the human colon: functional evidence for beta3-rather than beta4-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colon; Ethanolamines; Female; Humans; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes | 1999 |
Beta 2-adrenergic receptor endocytic pathway is controlled by a saturable mechanism distinct from that of transferrin receptor.
Topics: 3,3'-Diaminobenzidine; Adrenergic beta-Agonists; Arrestin; Cell Line; Centrifugation, Density Gradient; Endocytosis; Humans; Iodocyanopindolol; Isoproterenol; Microscopy, Fluorescence; Phosphorylation; Propanolamines; Propranolol; Protein Processing, Post-Translational; Receptors, Adrenergic, beta-2; Receptors, Transferrin; Recombinant Fusion Proteins; Temperature; Transfection | 1999 |
No functional beta 3-adrenergic receptors expressed in rat skeletal muscle cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Cells, Cultured; Cyclic AMP; Isoproterenol; Muscle, Skeletal; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1998 |
Beta4-adrenoceptors are more effective than beta1-adrenoceptors in mediating arrhythmic Ca2+ transients in mouse ventricular myocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Arrhythmias, Cardiac; Calcium; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Mice; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Time Factors | 1999 |
Phosphorylation of extracellular signal-regulated kinases 1 and 2 in 3T3-L1 adipocytes by stimulation of beta(3)-adrenoceptor.
Topics: 3T3 Cells; Adipocytes; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethanolamines; Flavonoids; Glycerol; Isoquinolines; Mice; Mitogen-Activated Protein Kinases; Phosphorylation; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Sulfonamides; Tetrahydronaphthalenes | 1999 |
The effects of beta-adrenoceptor agonists on KCl-induced rhythmic contraction in the ureter of guinea pig.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Calcium Channels, L-Type; Dose-Response Relationship, Drug; Guinea Pigs; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Periodicity; Potassium Chloride; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Ureter | 2000 |
Role of endothelium/nitric oxide in atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Norepinephrine; Oxadiazoles; Phenoxyacetates; Phenoxypropanolamines; Phenylacetates; Pindolol; Propanolamines; Propranolol; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Vasodilation | 2000 |
The in vivo effects of beta-3-receptor agonist CGP-12177 on thyroxine deiodination in cold-exposed, sympathectomized rat brown fat.
Topics: Adipose Tissue, Brown; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cold Temperature; Drug Implants; Enzyme Activation; Iodide Peroxidase; Iodine; Iodine Radioisotopes; Male; Norepinephrine; Prazosin; Propanolamines; Propranolol; Rats; Rats, Wistar; Sympathectomy; Thyroxine | 2000 |
Functional assessment of beta adrenoceptor subtypes in human colonic circular and longitudinal (taenia coli) smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Colon; Female; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Terbutaline; Tetrahydronaphthalenes | 2000 |
Partial agonist activity of carteolol on atypical beta-adrenoceptors in the guinea pig duodenum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Carteolol; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Vasodilator Agents | 2000 |
Enhancement of memory consolidation in chicks by beta(3)-adrenoceptor agonists.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Avoidance Learning; Chickens; Discrimination Learning; Dose-Response Relationship, Drug; Ethanolamines; Female; Memory; Propanolamines; Propranolol; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes | 2001 |
(+/-)-Pindolol acts as a partial agonist at atypical beta-adrenoceptors in the guinea pig duodenum.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamines; Duodenum; Ethanolamines; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 2001 |
Characterization of [3H]CGP 12177 binding to beta-adrenergic receptors in intact eel hepatocytes.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Alprenolol; Anguilla; Animals; Atenolol; Binding Sites; Binding, Competitive; Butoxamine; Cell Count; Colforsin; Cyclic AMP; Epinephrine; Glucose; Guanosine 5'-O-(3-Thiotriphosphate); Hepatocytes; Kinetics; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tritium | 2001 |
Beta(3)-adrenoceptor agonist-induced increases in lipolysis, metabolic rate, facial flushing, and reflex tachycardia in anesthetized rhesus monkeys.
Topics: Adenylyl Cyclases; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Anesthesia; Animals; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Flushing; Heart Rate; Indomethacin; Lipolysis; Macaca mulatta; Male; Propanolamines; Propranolol; Reflex | 2001 |
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 2001 |
Chronotropic response to (+/-)-CGP12177 in right atria of stressed rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Heart Atria; Heart Rate; Imidazoles; In Vitro Techniques; Male; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stress, Physiological; Time Factors | 2001 |
Oestradiol and progesterone change beta3-adrenergic receptor affinity and density in brown adipocytes.
Topics: Adipocytes; Adipose Tissue, Brown; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Cold Temperature; Estradiol; Female; Norepinephrine; Progesterone; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta-3; Statistics, Nonparametric | 2001 |
Receptor-ligand interactions studied with homogeneous fluorescence-based assays suitable for miniaturized screening.
Topics: Betacellulin; Cell Line; Drug Evaluation, Preclinical; Epidermal Growth Factor; ErbB Receptors; Fluorescence; Fluorescent Dyes; Growth Substances; Humans; Intercellular Signaling Peptides and Proteins; Ligands; Miniaturization; Optics and Photonics; Propanolamines; Propranolol; Receptors, Adrenergic, beta-2; Receptors, Cell Surface; Recombinant Proteins; Sensitivity and Specificity | 2001 |
Bucindolol exerts agonistic activity on the propranolol-insensitive state of beta1-adrenoceptors in human myocardium.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Atrial Function, Right; Benzopyrans; Ethanolamines; Female; Heart; Humans; In Vitro Techniques; Male; Metoprolol; Middle Aged; Myocardial Contraction; Myocardium; Nebivolol; Papillary Muscles; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Ventricular Function, Left | 2002 |
Cyclic AMP-independent relaxation mediated by beta3-adrenoceptors on guinea pig gastrointestine.
Topics: Adenine; Adenylyl Cyclase Inhibitors; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Butoxamine; Catecholamines; Cyclic AMP; Digestive System; Digestive System Physiological Phenomena; Dose-Response Relationship, Drug; Duodenum; Enzyme Inhibitors; Ethanolamines; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Propanolamines; Propranolol; Receptors, Adrenergic, beta-3 | 2002 |
(-)-CGP 12177 increases contractile force and hastens relaxation of human myocardial preparations through a propranolol-resistant state of the beta 1-adrenoceptor.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adult; Aged; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Relaxation; Myocardial Contraction; Myocardium; Propanolamines; Propranolol; Protein Binding; Receptors, Adrenergic, beta-1; Stimulation, Chemical | 2003 |
The beta1-adrenoceptor site activated by CGP12177 varies in behavior according to the estrous cycle phase and stress.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Animals; Atrial Function, Right; Corticosterone; Dose-Response Relationship, Drug; Electroshock; Estradiol; Estrous Cycle; Female; Heart Rate; In Vitro Techniques; Male; Progesterone; Propanolamines; Propranolol; Rats; Rats, Wistar; Stress, Physiological | 2003 |
Antagonism of the antidepressant-like effects of clenbuterol by central administration of beta-adrenergic antagonists in rats.
Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Antidepressive Agents; Clenbuterol; Dose-Response Relationship, Drug; Drug Interactions; Hippocampus; Male; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2; Reinforcement, Psychology | 2003 |
The effects of hydrocortisone on rat heart muscarinic and adrenergic alpha 1, beta 1 and beta 2 receptors, propranolol-resistant binding sites and on some subsequent steps in intracellular signalling.
Topics: Adrenergic beta-Antagonists; Animals; Binding Sites; Glucocorticoids; Heart Ventricles; Hydrocortisone; Injections, Subcutaneous; Male; Myocardium; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Muscarinic; Signal Transduction | 2003 |
Intrinsic sympathomimetic activity of (-)-pindolol mediated through a (-)-propranolol-resistant site of the beta1-adrenoceptor in human atrium and recombinant receptors.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Animals; Binding Sites; CHO Cells; Cricetinae; Cyclic AMP; Drug Interactions; Drug Resistance; Female; Heart; Heart Atria; Humans; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Norepinephrine; omega-N-Methylarginine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Recombinant Proteins; Stereoisomerism; Sympathomimetics | 2003 |
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction | 2004 |
G-protein-coupled receptor chromatographic stationary phases. 2. Ligand-induced conformational mobility in an immobilized beta2-adrenergic receptor.
Topics: Adrenergic beta-Antagonists; Animals; Binding Sites; Butoxamine; Cell Line; Chromatography, Affinity; Ligands; Membrane Proteins; Mice; Nadolol; Propanolamines; Propranolol; Protein Conformation; Receptors, Adrenergic; Receptors, G-Protein-Coupled; Time Factors | 2004 |
Effects of dexamethasone and colostrum feeding on mRNA levels and binding capacities of beta-adrenergic receptors in the liver of neonatal calves.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Animals, Newborn; Binding, Competitive; Cattle; Colostrum; Dexamethasone; Diet; Glucocorticoids; Liver; Polymerase Chain Reaction; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger | 2005 |
Characterization of isoprenaline- and salmeterol-stimulated interactions between beta2-adrenoceptors and beta-arrestin 2 using beta-galactosidase complementation in C2C12 cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Arrestins; beta-Arrestin 2; beta-Arrestins; beta-Galactosidase; Cell Line; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Genetic Complementation Test; Humans; Isoproterenol; Mutation; Propanolamines; Propranolol; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Salmeterol Xinafoate; Transfection | 2005 |
Studies on the mechanisms underlying beta-adrenoceptor-mediated relaxation of rat abdominal aorta.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Abdominal; Cyclic AMP; In Vitro Techniques; Isoproterenol; Large-Conductance Calcium-Activated Potassium Channels; Male; Muscle Relaxation; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 2006 |
Postsynaptic alpha-2 adrenergic receptors are critical for the antidepressant-like effects of desipramine on behavior.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Antidepressive Agents, Tricyclic; Depression; Desipramine; Idazoxan; Male; Mice; Mice, Knockout; Motor Activity; Prazosin; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Synapses | 2009 |
Role of beta3-adrenoceptors for intrahepatic resistance and portal hypertension in liver cirrhosis.
Topics: Animals; Cyclic AMP; Cyclic GMP-Dependent Protein Kinases; Hepatic Stellate Cells; Humans; Hypertension, Portal; Liver Cirrhosis; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Vascular Resistance | 2009 |
A full pharmacological analysis of the three turkey β-adrenoceptors and comparison with the human β-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Sequence; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Molecular Sequence Data; Mutation; Propanolamines; Propranolol; Protein Isoforms; Radioligand Assay; Receptors, Adrenergic, beta; Sequence Homology, Amino Acid; Tritium; Turkey | 2010 |
Autoantibodies against cardiac β(1)-adrenoceptor do not affect the low-affinity state β(1)-adrenoceptor-mediated inotropy in rat cardiomyocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Animals; Autoantibodies; Bisoprolol; Isoproterenol; Male; Myocardial Contraction; Myocytes, Cardiac; Phosphodiesterase Inhibitors; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1 | 2012 |