cgp 12177 has been researched along with prazosin in 27 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 6 (22.22) | 18.7374 |
| 1990's | 12 (44.44) | 18.2507 |
| 2000's | 8 (29.63) | 29.6817 |
| 2010's | 1 (3.70) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Endoh, M; Norota, I; Takanashi, M | 1 |
| Kinami, J; Maruyama, K; Nagatomo, T; Sugita, Y; Sugiyama, E; Takada, Y; Tsuchihashi, H | 1 |
| Cannon, B; Herron, D; Néchad, M; Nedergaard, J; Rehnmark, S | 1 |
| Endoh, M; Hiramoto, T; Kushida, H | 1 |
| Böhm, M; Erdmann, E; Feiler, G; Geist, BJ; Lauk, S | 1 |
| Mohell, N; Nedergaard, J | 1 |
| Limas, C; Limas, CJ | 1 |
| Ganas, L; Studer, RK | 1 |
| Raasmaja, A; York, DA | 2 |
| Kajiyama, Y; Ui, M | 1 |
| Chalecka-Franaszek, E; Dikshit, M; Nalepa, I | 1 |
| Endoh, M; Kohi, M; Norota, I; Takanashi, M | 1 |
| Gardner, ML; Körner, C; Pittelkow, MR; Schallreuter, KU; Swanson, NN | 1 |
| Barbin, L; Capuzzo, A; Fabbri, E | 1 |
| Gerhardt, CC; Gros, J; Issad, T; Strosberg, AD | 1 |
| Arioli, F; Badino, P; Belloli, C; Caloni, F; Carcano, R; Odore, R; Re, G | 1 |
| Badino, P; Bergamasco, L; Borgarelli, M; Girardi, C; Odore, R; Re, G; Tarducci, A; Zanatta, R | 1 |
| Hébert, C; Lalonde, R; Reader, TA; Strazielle, C | 1 |
| Hagmüller, K; Hofer, D; Korsatko, W; Porta, S; Raíces, M; Schauenstein, K; Zaninovich, A | 1 |
| Guibert, C; Ivorra, MD; Leblais, V; Marthan, R; Muller, B; Pourageaud, F | 1 |
| Brahmadevara, N; MacDonald, A; Shaw, AM | 1 |
| Bönisch, H; Caron, MG; Drozdowska, E; Dziedzicka-Wasylewska, M; Faron-Górecka, A; Kuśmider, M; Rogóz, Z; Siwanowicz, J | 1 |
| Bronnikov, GE; Cannon, B; Ignat'ev, DA; Kramarova, LI; Nedergaard, J | 1 |
| Borea, PA; Dorigo, P; Floreani, M; Quintieri, L; Varani, K | 1 |
| Huang, Y; O'Donnell, JM; Whisler, LR; Xiang, Y; Zhang, HT | 1 |
| Daly, CJ; Henstridge, CM; Irving, AJ; McGrath, JC; Ross, RA; Whyte, J | 1 |
27 other study(ies) available for cgp 12177 and prazosin
| Article | Year |
|---|---|
Effect of (+)-niguldipine on myocardial alpha 1-adrenoceptors in the rabbit.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Calcium Channel Blockers; Dihydropyridines; Dose-Response Relationship, Drug; Heart; Male; Myocardial Contraction; Prazosin; Propanolamines; Rabbits; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Stimulation, Chemical | 1992 |
MCI-9042: high affinity for serotonergic receptors as assessed by radioligand binding assay.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Brain Chemistry; Clonidine; Hippocampus; In Vitro Techniques; Ketanserin; Kinetics; Platelet Aggregation Inhibitors; Prazosin; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Muscarinic; Receptors, Serotonin; Succinates | 1991 |
Alpha- and beta-adrenergic induction of the expression of the uncoupling protein thermogenin in brown adipocytes differentiated in culture.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Colforsin; Gene Expression; Insulin; Ion Channels; Male; Membrane Proteins; Mice; Mitochondrial Proteins; Norepinephrine; Nucleic Acid Hybridization; Oxymetazoline; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; RNA; RNA, Messenger; Thyroxine; Triiodothyronine; Uncoupling Protein 1 | 1990 |
Preponderance of beta- over alpha-adrenoceptors in mediating the positive inotropic effect of phenylephrine in the ferret ventricular myocardium.
Topics: Adrenergic beta-Antagonists; Animals; Bupranolol; Carnivora; Ferrets; Heart; In Vitro Techniques; Myocardial Contraction; Myocardium; Papillary Muscles; Phenylephrine; Prazosin; Propanolamines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta | 1989 |
Increased number of cardiac adrenergic receptors following local heart irradiation.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Heart; Male; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tritium | 1989 |
Comparison of the pharmacological profiles of adrenergic drugs (including BRL-agonists) at [3H]prazosin and [3H]CGP-12177 binding sites in brown adipose tissue.
Topics: Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Cricetinae; In Vitro Techniques; Membranes; Mesocricetus; Prazosin; Propanolamines; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sympathomimetics | 1989 |
Altered intracellular adrenoceptor distribution in myocardium of spontaneously hypertensive rats.
Topics: Adrenergic beta-Agonists; Animals; Cardiomegaly; Cell Membrane; Cytosol; Dihydroalprenolol; Hypertension; Myocardial Contraction; Myocardium; Prazosin; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tissue Distribution | 1987 |
Adrenergic receptor properties of hepatocytes from male and female rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Female; Liver; Male; Prazosin; Propanolamines; Rats; Receptors, Adrenergic; Sex Characteristics | 1988 |
Alpha 1- and beta-adrenergic receptors in brown adipose tissue of lean (Fa/?) and obese (fa/fa) Zucker rats. Effects of cold-acclimation, sucrose feeding and adrenalectomy.
Topics: Adipose Tissue, Brown; Adrenalectomy; Adrenergic beta-Antagonists; Animals; Binding Sites; Cell Membrane; Cold Temperature; Female; Male; Obesity; Prazosin; Propanolamines; Rats; Rats, Zucker; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sucrose | 1988 |
Switching from alpha 1- to beta-subtypes in adrenergic response during primary culture of adult-rat hepatocytes as affected by the cell-to-cell interaction through plasma membranes.
Topics: Adrenergic beta-Antagonists; Angiotensin II; Animals; Cell Communication; Cell Membrane; Cells, Cultured; Cyclic AMP; Inositol 1,4,5-Trisphosphate; Kinetics; Liver; Male; Phenylephrine; Prazosin; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Time Factors; Vasopressins | 1994 |
Centpropazine affinity to cortical noradrenergic receptors and effect on their responsiveness in the rat.
Topics: Adrenergic beta-Antagonists; Animals; Antidepressive Agents; Binding, Competitive; Cerebral Cortex; In Vitro Techniques; Inositol Phosphates; Male; Membranes; Norepinephrine; Piperazines; Prazosin; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic; Second Messenger Systems | 1993 |
On the mechanism of action of the beta-1 partial agonist denopamine in regulation of myocardial contractility: effects on myocardial alpha adrenoceptors and intracellular Ca++ transients.
Topics: Adrenergic beta-Agonists; Animals; Bupranolol; Calcium; Dogs; Drug Interactions; Ethanolamines; Female; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Phenylephrine; Prazosin; Propanolamines; Rabbits; Receptors, Adrenergic, alpha | 1993 |
The induction of the alpha-1-adrenoceptor signal transduction system on human melanocytes.
Topics: Adrenergic beta-Antagonists; Adult; Cells, Cultured; Gene Expression Regulation; Humans; Imidazoles; Infant, Newborn; Keratinocytes; Melanocytes; Norepinephrine; Prazosin; Propanolamines; Receptors, Adrenergic, alpha-1; Signal Transduction | 1996 |
Coexistence of alpha1 and beta adrenergic receptors in the liver of the frog Rana esculenta, the toad Bufo bufo, the lizard Podarcis sicula campestris, and the turtle Pseudemys picta elegans.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Bufo bufo; In Vitro Techniques; Kinetics; Liver; Lizards; Membranes; Prazosin; Propanolamines; Rana esculenta; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Species Specificity; Turtles | 1997 |
Stimulation of the extracellular signal-regulated kinase 1/2 pathway by human beta-3 adrenergic receptor: new pharmacological profile and mechanism of activation.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Colforsin; Cricetinae; Dioxoles; Enzyme Activation; Epinephrine; Ethanolamines; Humans; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Norepinephrine; Phentolamine; Prazosin; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction; Yohimbine | 1999 |
Investigations on the stereoselective action of isoxsuprine on alpha- and beta-adrenoceptors in equine common digital artery.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Arteries; Binding, Competitive; Female; Forelimb; Horses; In Vitro Techniques; Isoxsuprine; Male; Membranes; Norepinephrine; Prazosin; Propanolamines; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Stereoisomerism; Toes; Tritium; Vasoconstriction | 1999 |
Canine dilated cardiomyopathy: lymphocyte and cardiac alpha(1)- and beta-adrenoceptor concentrations in normal and affected great danes.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathy, Dilated; Catecholamines; Dog Diseases; Dogs; Electrocardiography; Female; Heart Failure; Lymphocyte Count; Lymphocytes; Male; Myocardium; Prazosin; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1999 |
Regional brain distribution of noradrenaline uptake sites, and of alpha1-alpha2- and beta-adrenergic receptors in PCD mutant mice: a quantitative autoradiographic study.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Autoradiography; Basal Ganglia; Brain Stem; Cerebral Cortex; Disease Models, Animal; Female; Fluoxetine; Hypothalamus; Idazoxan; Limbic System; Mice; Mice, Neurologic Mutants; Norepinephrine; Prazosin; Propanolamines; Purkinje Cells; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Spinocerebellar Degenerations; Thalamus; Tritium | 1999 |
The in vivo effects of beta-3-receptor agonist CGP-12177 on thyroxine deiodination in cold-exposed, sympathectomized rat brown fat.
Topics: Adipose Tissue, Brown; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cold Temperature; Drug Implants; Enzyme Activation; Iodide Peroxidase; Iodine; Iodine Radioisotopes; Male; Norepinephrine; Prazosin; Propanolamines; Propranolol; Rats; Rats, Wistar; Sympathectomy; Thyroxine | 2000 |
Role of alpha-adrenergic receptors in the effect of the beta-adrenergic receptor ligands, CGP 12177, bupranolol, and SR 59230A, on the contraction of rat intrapulmonary artery.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Bupranolol; Calcium; Dinoprost; Female; Male; Prazosin; Propanolamines; Pulmonary Artery; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tritium; Vasoconstriction | 2004 |
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction | 2004 |
Effect of antidepressant drugs in mice lacking the norepinephrine transporter.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antidepressive Agents; Autoradiography; Behavior, Animal; Cerebral Cortex; Hindlimb Suspension; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Norepinephrine Plasma Membrane Transport Proteins; Prazosin; Propanolamines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Swimming; Time Factors; Tritium | 2006 |
Pharmacological characterization of alpha1- and beta-adrenergic synergism of 5'DII activity in rat brown adipocytes.
Topics: Adipose Tissue, Brown; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Cell Membrane; Drug Synergism; Ethanolamines; Female; Imidazoles; Iodide Peroxidase; Male; Oxathiins; Piperazines; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Rats, Zucker; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Triiodothyronine | 2006 |
Adrenergic receptor density in brown adipose tissue of active and hibernating hamsters and ground squirrels.
Topics: Acclimatization; Adipose Tissue, Brown; Animals; Arousal; Cold Temperature; Cricetinae; Female; Hibernation; Male; Mesocricetus; Prazosin; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sciuridae | 2007 |
Comparison of the binding affinity of CGP-12177A at recombinant rat alpha(1D)-adrenoceptors expressed in BHK-21 cell membranes and alpha(1)-adrenoceptors present in rat cerebral cortex membranes.
Topics: Animals; Aorta, Thoracic; Cells, Cultured; Cerebral Cortex; Cricetinae; Dose-Response Relationship, Drug; Male; Prazosin; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Vasoconstriction | 2008 |
Postsynaptic alpha-2 adrenergic receptors are critical for the antidepressant-like effects of desipramine on behavior.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Antidepressive Agents, Tricyclic; Depression; Desipramine; Idazoxan; Male; Mice; Mice, Knockout; Motor Activity; Prazosin; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Synapses | 2009 |
Fluorescent ligand binding reveals heterogeneous distribution of adrenoceptors and 'cannabinoid-like' receptors in small arteries.
Topics: Angiotensin II; Animals; Boron Compounds; Connective Tissue; Endothelium, Vascular; Fluorescent Dyes; Ligands; Male; Mesenteric Arteries; Mice; Mice, Inbred C57BL; Mice, Knockout; Microscopy, Confocal; Molecular Imaging; Molecular Probe Techniques; Muscle, Smooth, Vascular; Prazosin; Propanolamines; Pyrazoles; Rats; Rats, Wistar; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Receptors, Cannabinoid; Tail | 2010 |