cgp 12177 has been researched along with pindolol in 59 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 22 (37.29) | 18.7374 |
1990's | 26 (44.07) | 18.2507 |
2000's | 10 (16.95) | 29.6817 |
2010's | 1 (1.69) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bultsma, T; Donné-Op den Kelder, GM; Rademaker, B; Timmerman, H | 1 |
Bersohn, MM; Doshi, RN | 1 |
McNeel, RL; Mersmann, HJ | 1 |
Morin, D; Sapena, R; Tillement, JP; Urien, S; Zini, R | 1 |
Duman, RS; Fishman, PH; Nussbaum, E | 1 |
Lafontan, M; Langin, D; Portillo, MP; Saulnier-Blache, JS | 1 |
Bowery, NG; Johnson, AM; Nelson, DR; Palmer, KJ; Pratt, GD | 1 |
Baude, B; Blin, N; Emorine, LJ; Fève, B; Lasnier, F; Nahmias, C; Pairault, J; Strosberg, AD | 1 |
Akashi, H; Hosohata, Y; Kinami, J; Nagatomo, T; Sakuma, N; Tsuchihashi, H | 1 |
Olson, MF; Pon, DJ; Schimmer, BP; Tsao, J | 1 |
Korichneva, IL; Krasnikova, TL; Radiukhin, VA | 1 |
Cardone, F; Cignarelli, M; Corso, M; De Pergola, G; Di Paolo, S; Garruti, G; Giorgino, R; Nardelli, G | 1 |
Kashiwagi, A; Kida, Y; Kodama, M; Nishio, Y; Saeki, Y; Shigeta, Y | 1 |
Imai, S; Nagotomo, T; Tsuchihashi, H | 1 |
Graafsma, SJ; Rodrigues de Miranda, JF; Snijders, PJ; Thien, T | 1 |
O'Donnell, JM | 1 |
Affolter, H; Hertel, C; Jaeggi, K; Portenier, M; Staehelin, M | 1 |
Contreras, ML; Molinoff, PB; Wolfe, BB | 1 |
Feldman, RD; Motulsky, HJ; Thede-Reynolds, KR | 1 |
Molinoff, PB; Reynolds, EE | 1 |
Brunswick, DJ; Conway, PG; Tejani-Butt, S | 1 |
Jacobsen, FW; Jacobsen, S; Sandnes, D | 1 |
Freissmuth, M; Nanoff, C; Schütz, W | 1 |
Jacobsen, S; Refsnes, M; Sager, G; Sand, TE; Sandnes, D | 1 |
Coulter, SJ; Hertel, C; Perkins, JP | 1 |
Cunningham, EM; DeBlasi, A; Insel, PA; Motulsky, HJ | 1 |
Arinze, IJ; Graham, SM; Kawai, Y; Yoshioka, H | 1 |
Insel, PA; Maisel, AS; Motulsky, HJ | 1 |
Gjerde, I; Jacobsen, S; Refsnes, M; Sandnes, D | 1 |
Harden, TK; Perkins, JP; Toews, ML; Waldo, GL | 1 |
Hertel, C; Perkins, JP; Staehelin, M | 1 |
Hosohata, Y; Karakisawa, Y; Maruyama, K; Nagatomo, T; Suzuki, M | 1 |
Nunnally, MH; Parker, EM; Perkins, JP; Ross, EM; Swigart, P | 1 |
Hirsch, DJ; Morgunov, NS; You, YD | 1 |
Döring, V; Kalmár, P; Lavicky, J; Schmitz, W; Scholz, H; Steinfath, M | 1 |
Ambid, L; Carpéné, C; Lafontan, M | 1 |
Change, HT; Chen, CF; Liao, JF | 1 |
Laurent, S; Nicolas, P; Perret, GY; Vassy, R; Yin, Y | 1 |
Hattori, K; Hosohata, Y; Nagatomo, T; Sasaki, K; Shen, Y; Suzuki, J | 1 |
Adachi-Akahane, S; Kitagawa, Y; Nagao, T | 1 |
Barak, LS; Bertrand, L; Caron, MG; Colapietro, AM; Ferguson, SS; Lefkowitz, RJ; Ménard, L; Premont, RT | 1 |
el Borai, N; Ito, K; Nakano, S; Nakazawa, H; Tanaka, E; Yamakawa, A; Yamamura, M | 1 |
Mersmann, HJ | 1 |
Hattori, K; Hosohata, Y; Maruyama, K; Nagatomo, T; Ohnuki, T; Sasaki, K; Suzuki, J; Watanabe, K | 1 |
Malinowska, B; Schlicker, E | 2 |
Kaumann, AJ; Molenaar, P | 1 |
Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F | 1 |
Brawley, L; MacDonald, A; Shaw, AM | 1 |
Engelhardt, S; Hein, L; Kaumann, AJ; Lohse, M; Molenaar, P | 1 |
Horinouchi, T; Koike, K | 2 |
Colledge, WH; Grace, AA; Joseph, SS; Kaumann, AJ; Lynham, JA; Molenaar, P | 1 |
Brahmadevara, N; MacDonald, A; Shaw, AM | 1 |
Desfontis, JC; Gauthier, C; Gautier, F; Gogny, M; Mallem, MY; Serpillon, S; Toumaniantz, G | 1 |
Desfontis, JC; Gogny, M; Holopherne, D; Le Coz, O; Mallem, Y; Reculeau, O | 1 |
Desfontis, JC; Gogny, M; Le Coz, O; Mallem, MY; Reculeau, O | 1 |
Kozłowska, H; Kwolek, G; Malinowska, B; Schlicker, E; Zakrzeska, A | 1 |
Abdelkrim, MA; Chatagnon, G; Desfontis, JC; Gogny, M; Mallem, MY; Noireaud, J | 1 |
1 review(s) available for cgp 12177 and pindolol
Article | Year |
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Life cycles of cardiac alpha 1- and beta-adrenergic receptors.
Topics: Animals; Cyclic AMP; Heart; Iodocyanopindolol; Myocardial Contraction; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Time Factors | 1987 |
58 other study(ies) available for cgp 12177 and pindolol
Article | Year |
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Mapping of the beta 2-adrenoceptor on Chang liver cells. Differences between high- and low-affinity receptor states.
Topics: Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Hydrogen Bonding; Iodocyanopindolol; Liver; Models, Molecular; Pindolol; Protein Conformation; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship | 1988 |
Measurement of sarcolemmal vesicle orientation by beta-adrenergic receptor binding.
Topics: Animals; Binding Sites; Heart; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Methods; Ouabain; Pindolol; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Sarcolemma; Sodium-Potassium-Exchanging ATPase; Tritium | 1992 |
Ligand binding to the porcine adipose tissue beta-adrenergic receptor.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Kinetics; Ligands; Molecular Conformation; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Swine; Temperature; Time Factors | 1992 |
Labelling of rat brain beta-adrenoceptors: (3H)CGP-12177 or (125I)iodocyanopindolol?
Topics: Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Hippocampus; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Male; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Serotonin; Tritium | 1992 |
Characterization and regulation of beta 1-adrenergic receptors in a human neuroepithelioma cell line.
Topics: Adrenergic beta-Antagonists; Binding, Competitive; Cell Membrane; Cyclic AMP; DNA Probes; Down-Regulation; Epinephrine; Humans; Iodine Radioisotopes; Iodocyanopindolol; Isoproterenol; Neuroectodermal Tumors, Primitive, Peripheral; Norepinephrine; Nucleic Acid Hybridization; Pindolol; Propanolamines; Receptors, Adrenergic, beta; RNA, Messenger; Tumor Cells, Cultured | 1991 |
Coexistence of three beta-adrenoceptor subtypes in white fat cells of various mammalian species.
Topics: Adipose Tissue; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cell Membrane; Cricetinae; Dogs; Ethanolamines; Humans; Iodine Radioisotopes; Isoproterenol; Kinetics; Lipolysis; Male; Mesocricetus; Muscle, Smooth; Pindolol; Propanolamines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Effect of paroxetine, a selective 5-hydroxytryptamine uptake inhibitor, on beta-adrenoceptors in rat brain: autoradiographic and functional studies.
Topics: Adrenergic beta-Antagonists; Amitriptyline; Animals; Autoradiography; Brain Chemistry; Cyclic AMP; Desipramine; Iodine Radioisotopes; Iodocyanopindolol; Kinetics; Male; Membranes; Paroxetine; Pindolol; Piperidines; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Serotonin Antagonists | 1991 |
Atypical beta-adrenergic receptor in 3T3-F442A adipocytes. Pharmacological and molecular relationship with the human beta 3-adrenergic receptor.
Topics: 3T3 Cells; Adipose Tissue; Adrenergic beta-Antagonists; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; DNA; Ethanolamines; Humans; Imidazoles; Mice; Molecular Sequence Data; Oxprenolol; Pindolol; Polymerase Chain Reaction; Propanolamines; Receptors, Adrenergic, beta; RNA, Messenger | 1991 |
Beta-blocking potency and selectivity of bopindolol and its two metabolites for beta 1- and beta 2-adrenergic receptors as assessed by radioligand binding assay.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Brain; Guinea Pigs; Heart Rate; In Vitro Techniques; Iodocyanopindolol; Kinetics; Muscle Contraction; Myocardium; Pindolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Trachea | 1991 |
Regulation of adenylyl cyclase activity by beta-adrenergic agonists in a desensitization-resistant mutant cell line.
Topics: Adenylyl Cyclases; Adrenal Cortex Neoplasms; Adrenocorticotropic Hormone; Animals; Gene Expression; Iodocyanopindolol; Isoproterenol; Mice; Mutation; Pindolol; Plasmids; Propanolamines; Receptors, Adrenergic, beta; Sodium Fluoride; Transfection; Tumor Cells, Cultured | 1991 |
[Dependence of kinetic constants of intact human lymphocyte beta2-adrenoreceptors on the nature of the radioligands used].
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Ethylmaleimide; Humans; Isoproterenol; Kinetics; Lymphocytes; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Temperature | 1989 |
Influence of lactate on isoproterenol-induced lipolysis and beta-adrenoceptors distribution in human fat cells.
Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adult; Cell Membrane; Cells, Cultured; Humans; Isoproterenol; Lactates; Lipolysis; Middle Aged; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Serotonin Antagonists | 1989 |
Plasma membrane-specific deficiency in cardiac beta-adrenergic receptor in streptozocin-diabetic rats.
Topics: Adrenergic beta-Antagonists; Animals; Cell Membrane; Cells, Cultured; Diabetes Mellitus, Experimental; Insulin; Iodocyanopindolol; Kinetics; Male; Myocardium; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Reference Values | 1989 |
Selectivity of bunitrolol for beta 1- and beta 2-adrenergic receptors and 5HT1B-receptors: assessment by biphasic Scatchard plots and biphasic displacement curve analysis with 125I-iodocyanopindolol and 3H-CGP12177.
Topics: Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Heart; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Kinetics; Lung; Male; Myocardium; Pindolol; Propanolamines; Rats; Receptors, Adrenergic, beta; Receptors, Serotonin | 1989 |
Complications of (-)125I-iodocyanopindolol binding to human mononuclear cells.
Topics: Binding, Competitive; Humans; In Vitro Techniques; Iodine Radioisotopes; Iodocyanopindolol; Leukocytes, Mononuclear; Models, Biological; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Sonication; Stereoisomerism | 1987 |
Behavioral consequences of activation of beta adrenergic receptors by clenbuterol: evidence for mediation by the central nervous system.
Topics: Animals; Behavior, Animal; Binding, Competitive; Central Nervous System; Clenbuterol; Ethanolamines; Male; Pindolol; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1988 |
(-)-S-[3H]CGP-12177 and its use to determine the rate constants of unlabeled beta-adrenergic antagonists.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Cell Line; Computers; Glioma; Kinetics; Pindolol; Propanolamines; Stereoisomerism | 1985 |
Kinetic analysis of the interactions of agonists and antagonists with beta adrenergic receptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Bupranolol; Cell Line; Computers; Dihydroalprenolol; Kinetics; Mathematics; Pindolol; Propanolamines; Time Factors | 1986 |
Temperature-dependent binding of hydrophilic beta-adrenergic receptor ligands to intact human lymphocytes.
Topics: Adolescent; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Binding, Competitive; Cell Membrane; Humans; In Vitro Techniques; Isoproterenol; Ligands; Lymphocytes; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Temperature | 1986 |
Down regulation of beta adrenergic receptors in S49 lymphoma cells induced by atypical agonists.
Topics: Adrenergic beta-Agonists; Animals; Binding Sites; Celiprolol; Cell Division; Cell Line; Isoproterenol; Kinetics; Lymphoma; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Time Factors | 1986 |
Interaction of beta adrenergic agonists and antagonists with brain beta adrenergic receptors in vivo.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Brain; Butoxamine; Drug Interactions; Male; Pindolol; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1987 |
Modes of determining beta-adrenoceptor number in human mononuclear leucocytes.
Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Female; Humans; Iodine Radioisotopes; Iodocyanopindolol; Male; Middle Aged; Neutrophils; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Subcellular Fractions; Temperature | 1987 |
The role of a low beta 1-adrenoceptor selectivity of [3H]CGP-12177 for resolving subtype-selectivity of competitive ligands.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Iodocyanopindolol; Microsomes; Pindolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta | 1987 |
Elevated level of beta-adrenoceptors in intact hepatocytes from partially hepatectomized rats.
Topics: Adrenergic beta-Antagonists; Animals; Hepatectomy; Iodocyanopindolol; Liver; Male; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1988 |
A comparison of catecholamine-induced internalization of beta-adrenergic receptors and receptor-mediated endocytosis of epidermal growth factor in human astrocytoma cells. Inhibition by phenylarsine oxide.
Topics: Adenosine Triphosphate; Arsenicals; Astrocytoma; Catecholamines; Cell Line; Dithiothreitol; Endocytosis; Epidermal Growth Factor; Humans; Iodocyanopindolol; Isoproterenol; Pindolol; Propanolamines; Receptors, Adrenergic, beta | 1985 |
Desensitization and redistribution of beta-adrenergic receptors on human mononuclear leukocytes.
Topics: Adolescent; Adult; Binding, Competitive; Cyclic AMP; Drug Tolerance; Female; Humans; Iodocyanopindolol; Isoproterenol; Leukocytes; Male; Monocytes; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1986 |
Beta-adrenergic receptors in guinea-pig liver plasma membranes and thermal lability of [3H]dihydroalprenolol binding sites.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Guinea Pigs; Hot Temperature; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Virulence Factors, Bordetella | 1986 |
Down-regulation of surface beta-adrenoceptors on intact human mononuclear leukocytes. Time-course and isoproterenol concentration dependence.
Topics: Adenylyl Cyclases; Adolescent; Adult; Dose-Response Relationship, Drug; Female; Humans; Iodocyanopindolol; Isoproterenol; Leukocytes; Male; Middle Aged; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Time Factors | 1987 |
Relationship between an altered membrane form and a low affinity form of the beta-adrenergic receptor occurring during catecholamine-induced desensitization. Evidence for receptor internalization.
Topics: Astrocytoma; Cell Line; Centrifugation, Density Gradient; Concanavalin A; Humans; Isoproterenol; Methylmannosides; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Time Factors | 1984 |
Evidence for intravesicular beta-adrenergic receptors in membrane fractions from desensitized cells: binding of the hydrophilic ligand CGP-12177 only in the presence of alamethicin.
Topics: Alamethicin; Animals; Anti-Bacterial Agents; Cells, Cultured; Centrifugation, Density Gradient; Glioma; Isoproterenol; Pindolol; Propanolamines; Rats; Receptors, Adrenergic, beta | 1983 |
The affinity of bopindolol and its two metabolites for a beta 2-adrenoceptor in the bovine mesenteric artery.
Topics: Adrenergic beta-Antagonists; Animals; Cattle; In Vitro Techniques; Mesenteric Arteries; Muscle, Smooth, Vascular; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-2 | 1994 |
Carboxyl-terminal domains in the avian beta 1-adrenergic receptor that regulate agonist-promoted endocytosis.
Topics: Animals; Endocytosis; Iodocyanopindolol; Isoproterenol; Mice; Peptide Fragments; Pindolol; Propanolamines; Receptors, Adrenergic, beta-1; Turkeys | 1995 |
Response of mouse proximal straight tubule and medullary thick ascending limb to beta-agonist.
Topics: Adrenergic beta-Antagonists; Animals; Electrophysiology; Furosemide; In Vitro Techniques; Isoproterenol; Kidney Medulla; Kidney Tubules; Kidney Tubules, Proximal; Kinetics; Membrane Potentials; Mice; Perfusion; Pindolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta | 1993 |
Changes in cardiac beta-adrenoceptors in human heart diseases: relationship to the degree of heart failure and further evidence for etiology-related regulation of beta 1 and beta 2 subtypes.
Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Aortic Valve; Cardiomyopathy, Hypertrophic; Down-Regulation; Female; Heart Failure; Heart Valve Diseases; Heart Ventricles; Humans; Imidazoles; Iodocyanopindolol; Male; Middle Aged; Mitral Valve; Muscular Dystrophies; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Tetralogy of Fallot | 1993 |
Predominance of beta 3-adrenergic component in catecholamine activation of lipolysis in garden dormouse adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Catecholamines; Female; Iodocyanopindolol; Lipolysis; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Rodentia | 1994 |
Characterization of agonist-induced internalization and down-regulation of beta-adrenergic receptors in isolated rat lung and heart preparations.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Cycloheximide; Down-Regulation; Endocytosis; Heart; Hypertonic Solutions; Iodocyanopindolol; Isoproterenol; Lung; Male; Myocardium; Organ Specificity; Pindolol; Propanolamines; Propranolol; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Sucrose; Terbutaline | 1993 |
Antagonism between T3 and amiodarone on the contractility and the density of beta-adrenoceptors of chicken cardiac myocytes.
Topics: Adrenergic beta-Antagonists; Amiodarone; Animals; Calcium; Chick Embryo; Heart; Iodocyanopindolol; Isoproterenol; Myocardial Contraction; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Triiodothyronine | 1994 |
Bopindolol is a slowly dissociating beta 1-adrenoceptor antagonist when compared to other beta-blockers.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Brain; Guinea Pigs; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Pindolol; Propanolamines; Radioligand Assay; Rats; Tritium | 1995 |
Determination of beta-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective beta-antagonists.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cyclic AMP; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Membranes; Myocardium; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Tritium | 1995 |
Members of the G protein-coupled receptor kinase family that phosphorylate the beta2-adrenergic receptor facilitate sequestration.
Topics: Adrenergic beta-Antagonists; Cell Line; Cloning, Molecular; GTP-Binding Proteins; Humans; Immunoblotting; Iodine Radioisotopes; Kidney; Phosphates; Phosphorus Radioisotopes; Phosphorylation; Pindolol; Point Mutation; Propanolamines; Receptor Protein-Tyrosine Kinases; Receptors, Adrenergic, beta-2; Recombinant Proteins; Sequence Tagged Sites; Substrate Specificity; Transfection | 1996 |
Regulation of heat production of brown adipocytes via typical and atypical beta-adrenoceptors in the rat.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Calorimetry; Ethanolamines; In Vitro Techniques; Isoproterenol; Male; Phenoxyacetates; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1995 |
Evidence of classic beta 3-adrenergic receptors in porcine adipocytes.
Topics: Adipocytes; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Dihydroalprenolol; Iodocyanopindolol; Magnesium Chloride; Male; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; RNA; Swine; Tritium | 1996 |
Effects of chronic administration of bopindolol on the binding characteristics of cardiac alpha 1H-, alpha 1L-, beta 1- and beta 2-adrenoceptor subtypes in cardiac muscles of spontaneously hypertensive rats (SHR).
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Hypertension; In Vitro Techniques; Membranes; Myocardium; Pindolol; Propanolamines; Propranolol; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2 | 1996 |
Mediation of the positive chronotropic effect of CGP 12177 and cyanopindolol in the pithed rat by atypical beta-adrenoceptors, different from beta 3-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Male; Pindolol; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stimulation, Chemical | 1996 |
Differences between the third cardiac beta-adrenoceptor and the colonic beta 3-adrenoceptor in the rat.
Topics: Adrenergic beta-Antagonists; Animals; Colon; Dose-Response Relationship, Drug; Female; Heart; Male; Norepinephrine; Pindolol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta | 1996 |
Further evidence for differences between cardiac atypical beta-adrenoceptors and brown adipose tissue beta3-adrenoceptors in the pithed rat.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Male; Pindolol; Propanolamines; Rats; Rats, Wistar; Temperature | 1997 |
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1998 |
Role of endothelium/nitric oxide in atypical beta-adrenoceptor-mediated relaxation in rat isolated aorta.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitroprusside; Norepinephrine; Oxadiazoles; Phenoxyacetates; Phenoxypropanolamines; Phenylacetates; Pindolol; Propanolamines; Propranolol; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Vasodilation | 2000 |
Abolition of (-)-CGP 12177-evoked cardiostimulation in double beta1/beta2-adrenoceptor knockout mice. Obligatory role of beta1-adrenoceptors for putative beta4-adrenoceptor pharmacology.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Binding, Competitive; Bucladesine; Dose-Response Relationship, Drug; Female; Genotype; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Membranes; Mice; Mice, Knockout; Myocardial Contraction; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Sinoatrial Node; Tritium | 2001 |
(+/-)-Pindolol acts as a partial agonist at atypical beta-adrenoceptors in the guinea pig duodenum.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamines; Duodenum; Ethanolamines; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 2001 |
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 2001 |
Intrinsic sympathomimetic activity of (-)-pindolol mediated through a (-)-propranolol-resistant site of the beta1-adrenoceptor in human atrium and recombinant receptors.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Animals; Binding Sites; CHO Cells; Cricetinae; Cyclic AMP; Drug Interactions; Drug Resistance; Female; Heart; Heart Atria; Humans; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Myocardial Contraction; Norepinephrine; omega-N-Methylarginine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Recombinant Proteins; Stereoisomerism; Sympathomimetics | 2003 |
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction | 2004 |
Impairment of the low-affinity state beta1-adrenoceptor-induced relaxation in spontaneously hypertensive rats.
Topics: Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hypertension; Immunohistochemistry; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; omega-N-Methylarginine; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta-1 | 2004 |
Beta-adrenoceptor-mediated vascular relaxation in spontaneously hypertensive rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Tetrahydronaphthalenes | 2005 |
Low-affinity state beta1-adrenoceptor-induced vasodilation in SHR.
Topics: Adrenergic beta-1 Receptor Agonists; Alprenolol; Animals; Aorta; Blood Pressure; Dose-Response Relationship, Drug; Enalapril; Losartan; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta-1; Vasodilation | 2005 |
Positive inotropic and lusitropic effects mediated via the low-affinity state of beta1-adrenoceptors in pithed rats.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Animals; Decerebrate State; Humans; Male; Myocardial Contraction; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1 | 2005 |
Autoantibodies against cardiac β(1)-adrenoceptor do not affect the low-affinity state β(1)-adrenoceptor-mediated inotropy in rat cardiomyocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Animals; Autoantibodies; Bisoprolol; Isoproterenol; Male; Myocardial Contraction; Myocytes, Cardiac; Phosphodiesterase Inhibitors; Pindolol; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1 | 2012 |