cgp 12177 and phenylephrine

cgp 12177 has been researched along with phenylephrine in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19903 (25.00)18.7374
1990's5 (41.67)18.2507
2000's4 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cannon, B; Herron, D; Néchad, M; Nedergaard, J; Rehnmark, S1
Hirsch, DJ; Morgunov, NS1
Endoh, M; Hiramoto, T; Kushida, H1
Hiramatsu, Y; Nezu, E; Yoneyama, T; Yoshimura, K1
Clementi, F; Sher, E1
Kajiyama, Y; Ui, M1
Endoh, M; Kohi, M; Norota, I; Takanashi, M1
Berdeaux, A; Bévérelli, F; Gauthier, C; Le Marec, H; Leblais, V; Rautureau, Y; Trochu, JN1
Koivisto, A; Nedergaard, J; Siemen, D1
Horinouchi, T; Koike, K1
Brahmadevara, N; MacDonald, A; Shaw, AM1
Kozłowska, H; Kozłowski, M; Laudański, J; Malinowska, B; Schlicker, E; Siedlecka, U1

Other Studies

12 other study(ies) available for cgp 12177 and phenylephrine

ArticleYear
Alpha- and beta-adrenergic induction of the expression of the uncoupling protein thermogenin in brown adipocytes differentiated in culture.
    The Journal of biological chemistry, 1990, Sep-25, Volume: 265, Issue:27

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Colforsin; Gene Expression; Insulin; Ion Channels; Male; Membrane Proteins; Mice; Mitochondrial Proteins; Norepinephrine; Nucleic Acid Hybridization; Oxymetazoline; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; RNA; RNA, Messenger; Thyroxine; Triiodothyronine; Uncoupling Protein 1

1990
Adenylate cyclase uncoupled beta-adrenergic receptors in salamander proximal tubules.
    Canadian journal of physiology and pharmacology, 1990, Volume: 68, Issue:7

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Ambystoma; Animals; Cyclic AMP; In Vitro Techniques; Isoproterenol; Kidney Tubules, Proximal; Kinetics; Perfusion; Phenylephrine; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta

1990
Preponderance of beta- over alpha-adrenoceptors in mediating the positive inotropic effect of phenylephrine in the ferret ventricular myocardium.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 339, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Bupranolol; Carnivora; Ferrets; Heart; In Vitro Techniques; Myocardial Contraction; Myocardium; Papillary Muscles; Phenylephrine; Prazosin; Propanolamines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1989
Augmentation and inhibition of beta-adrenergic agonists-stimulated tissue cyclic AMP accumulation by alpha-adrenergic agonists in rat parotid gland.
    The Japanese journal of physiology, 1987, Volume: 37, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Calcium; Cyclic AMP; In Vitro Techniques; Isoproterenol; Male; Methoxamine; Parotid Gland; Phenylephrine; Propanolamines; Rats; Rats, Inbred Strains

1987
Agonist-induced internalization of the beta adrenergic receptor in a smooth muscle cell line.
    Biochemical and biophysical research communications, 1984, Nov-14, Volume: 124, Issue:3

    Topics: Animals; Cell Line; Dose-Response Relationship, Drug; Isoproterenol; Kinetics; Muscle, Smooth; Phenylephrine; Propanolamines; Receptors, Adrenergic, beta

1984
Switching from alpha 1- to beta-subtypes in adrenergic response during primary culture of adult-rat hepatocytes as affected by the cell-to-cell interaction through plasma membranes.
    The Biochemical journal, 1994, Oct-01, Volume: 303 ( Pt 1)

    Topics: Adrenergic beta-Antagonists; Angiotensin II; Animals; Cell Communication; Cell Membrane; Cells, Cultured; Cyclic AMP; Inositol 1,4,5-Trisphosphate; Kinetics; Liver; Male; Phenylephrine; Prazosin; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Time Factors; Vasopressins

1994
On the mechanism of action of the beta-1 partial agonist denopamine in regulation of myocardial contractility: effects on myocardial alpha adrenoceptors and intracellular Ca++ transients.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Bupranolol; Calcium; Dogs; Drug Interactions; Ethanolamines; Female; In Vitro Techniques; Male; Myocardial Contraction; Myocardium; Phenylephrine; Prazosin; Propanolamines; Rabbits; Receptors, Adrenergic, alpha

1993
Beta 3-adrenoceptor stimulation induces vasorelaxation mediated essentially by endothelium-derived nitric oxide in rat thoracic aorta.
    British journal of pharmacology, 1999, Volume: 128, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Cyclic GMP; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Nadolol; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Phenylephrine; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes; Vasoconstriction; Vasodilation

1999
Norepinephrine-induced sustained inward current in brown fat cells: alpha(1)-mediated by nonselective cation channels.
    American journal of physiology. Endocrinology and metabolism, 2000, Volume: 279, Issue:5

    Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Calcimycin; Calcium; Cations; Chlorides; Colforsin; Electric Conductivity; Enzyme Activation; Extracellular Space; Imidazoles; Ion Channels; Ionophores; Male; Norepinephrine; Patch-Clamp Techniques; Phenylephrine; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sodium

2000
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
    European journal of pharmacology, 2001, Mar-23, Volume: 416, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism

2001
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction

2004
Ligands at beta2-, beta3-, and the low-affinity state of beta1-adrenoceptors block the alpha1-adrenoceptor-mediated constriction in human pulmonary and rat mesenteric arteries.
    Journal of cardiovascular pharmacology, 2005, Volume: 46, Issue:1

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Ligands; Male; Mesenteric Arteries; Middle Aged; Phenylephrine; Propanolamines; Pulmonary Artery; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Vasoconstriction

2005