cgp 12177 and metoprolol

cgp 12177 has been researched along with metoprolol in 8 studies

Research

Studies (8)

Timeframe	Studies, this research(%)	All Research%
pre-1990	1 (12.50)	18.7374
1990's	4 (50.00)	18.2507
2000's	2 (25.00)	29.6817
2010's	1 (12.50)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Iakovidis, D; Jackman, GP; Louis, SN; Louis, WJ; Nero, TL	1
Baker, JG	1
Charlton, SJ; Dickson, CJ; Duca, JS; Fairhurst, RA; Hornak, V; McKay, DJ; Pearlstein, RA; Reilly, J; Sandham, DA; Shaw, D; Sykes, DA; Velez-Vega, C	1
Nagatomo, T; Tsuchihashi, H; Yokoyama, H	1
Arner, P; Enocksson, S; Lönnqvist, F; Nordenström, J; Shimizu, M	1
Kaila, T; Marttila, R	1
Farias-Silva, E; Grassi-Kassisse, DM; Spadari-Bratfisch, RC; Wolf-Nunes, V	1
Bölck, B; Brixius, K; Bundkirchen, A; Schwinger, RH	1

Trials

1 trial(s) available for cgp 12177 and metoprolol

Article	Year
Receptor occupancy in lumbar CSF as a measure of the antagonist activity of atenolol, metoprolol and propranolol in the CNS. British journal of clinical pharmacology, 1993, Volume: 35, Issue:5 Topics: Adrenergic alpha-Antagonists; Adult; Animals; Atenolol; Central Nervous System; Female; Humans; In Vitro Techniques; Male; Metoprolol; Middle Aged; Propanolamines; Propranolol; Rabbits; Rats; Receptors, Adrenergic, alpha	1993

Article

Year

Receptor occupancy in lumbar CSF as a measure of the antagonist activity of atenolol, metoprolol and propranolol in the CNS.

British journal of clinical pharmacology, 1993, Volume: 35, Issue:5

Topics: Adrenergic alpha-Antagonists; Adult; Animals; Atenolol; Central Nervous System; Female; Humans; In Vitro Techniques; Male; Metoprolol; Middle Aged; Propanolamines; Propranolol; Rabbits; Rats; Receptors, Adrenergic, alpha

1993

Other Studies

7 other study(ies) available for cgp 12177 and metoprolol

Article	Year
LK 204-545, a highly selective beta1-adrenoceptor antagonist at human beta-adrenoceptors. European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3 Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; Cyclopropanes; Female; Humans; Imidazoles; In Vitro Techniques; Ligands; Phenoxypropanolamines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Trachea; Urea	1999
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors. British journal of pharmacology, 2005, Volume: 144, Issue:3 Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3	2005
Uncoupling the Structure-Activity Relationships of β2 Adrenergic Receptor Ligands from Membrane Binding. Journal of medicinal chemistry, 2016, 06-23, Volume: 59, Issue:12 Topics: Binding Sites; Cell Membrane; Dose-Response Relationship, Drug; Humans; Ligands; Models, Molecular; Molecular Structure; Receptors, Adrenergic, beta-2; Structure-Activity Relationship	2016
Binding characteristics of 3H-CGP12177 to beta-adrenoceptors in rat myocardial membranes. Japanese journal of pharmacology, 1989, Volume: 49, Issue:1 Topics: Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; Cell Membrane; Male; Metoprolol; Myocardium; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta	1989
Demonstration of an in vivo functional beta 3-adrenoceptor in man. The Journal of clinical investigation, 1995, Volume: 95, Issue:5 Topics: Adipose Tissue; Adrenergic beta-Antagonists; Adult; Analysis of Variance; Animals; Body Temperature Regulation; Cells, Cultured; Dobutamine; Female; Humans; Isoproterenol; Kinetics; Lipolysis; Male; Mammals; Metoprolol; Microdialysis; Middle Aged; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reference Values; Regional Blood Flow; Terbutaline; Time Factors	1995
Stress-induced alteration in the lipolytic response to beta-adrenoceptor agonists in rat white adipocytes. Journal of lipid research, 1999, Volume: 40, Issue:9 Topics: Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Body Weight; Bucladesine; Eating; Epinephrine; Ethanolamines; Glycerol; Isoproterenol; Lipolysis; Male; Metoprolol; Norepinephrine; Propanolamines; Rats; Rats, Wistar; Stress, Physiological	1999
Bucindolol exerts agonistic activity on the propranolol-insensitive state of beta1-adrenoceptors in human myocardium. The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:3 Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Atrial Function, Right; Benzopyrans; Ethanolamines; Female; Heart; Humans; In Vitro Techniques; Male; Metoprolol; Middle Aged; Myocardial Contraction; Myocardium; Nebivolol; Papillary Muscles; Propanolamines; Propranolol; Receptors, Adrenergic, beta-1; Ventricular Function, Left	2002