cgp 12177 has been researched along with colforsin in 31 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (9.68) | 18.7374 |
1990's | 20 (64.52) | 18.2507 |
2000's | 8 (25.81) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bronnikov, G; Houstĕk, J; Nedergaard, J | 1 |
Bouanani, N; Corsin, A; Crozatier, B; Gilson, N | 1 |
Cannon, B; Herron, D; Néchad, M; Nedergaard, J; Rehnmark, S | 1 |
Gierschik, P; Jakobs, KH; Müller, U; Reithmann, C; Werdan, K | 1 |
Reithmann, C; Werdan, K | 1 |
Anakwe, OO; Moger, WH; Murphy, PR | 1 |
Henneberry, RC; Jahangeer, S; Lysko, PG | 1 |
Bouloumie, A; Galitzky, J; Lafontan, M; Langin, D; Remaury, A; Tavernier, G; Valet, P | 1 |
Bronnikov, G; Mohell, N; Nedergaard, J; Unelius, L | 1 |
Brunello, N; Perez, J; Racagni, G; Rovescalli, AC; Steardo, L; Vitali, S | 1 |
Baumgold, J; Curran, P; Fishman, PH; Zhou, XM | 1 |
Matheny, M; Scarpace, PJ | 1 |
el Hadri, K; Fève, B; Pairault, J | 1 |
Arner, P; Hellström, L; Langin, D; Reynisdottir, S; Rössner, S | 1 |
Baamonde, C; Dierssen, M; Flórez, J; García-Calatayud, S; Lumbreras, MA; Vallina, IF | 1 |
Berg, L; Hershman, JM; Ohta, K; Pang, XP | 1 |
Nürnberger, F; Pleschka, K | 1 |
Lisá, V; Myslivecek, J; Trojan, S; Tucek, S | 1 |
Gerhardt, CC; Gros, J; Issad, T; Strosberg, AD | 1 |
Bergström, D; Fowler, CJ; Jacobsson, SO | 1 |
Ajisawa, Y; Akahane, M; Andersson, KE; Hayakawa, K; Igawa, Y; Nishizawa, O; Takeda, H; Yamazaki, Y; Yoneyama, T | 1 |
Agarwal, D; Glasel, JA | 1 |
Germack, R; Perret, GY; Starzec, A | 1 |
Coussin, F; Macrez, N; Mironneau, J; Morel, JL; Viard, P | 1 |
Ito, M; Nakagawa, M; Saikawa, T; Takahashi, N; Teshima, Y; Yasunaga, S; Yonemochi, H | 1 |
Baamonde, C; Dierssen, M; Flórez, J; García-Calatayud, S; Lumbreras, MA; Martínez-Cué, C; Vallina, IF | 1 |
Koivisto, A; Nedergaard, J; Siemen, D | 1 |
Bourin, MC; Crozatier, B; Germack, R; León-Velarde, F; Mohammadi, K; Richalet, JP | 1 |
Capuzzo, A; Fabbri, E; Moon, TW; Selva, C | 1 |
Frontera, M; Gianotti, M; Justo, R; Oliver, J; Pujol, E; Roca, P; Rodriguez-Cuenca, S | 1 |
Carter, AA; Hill, SJ | 1 |
31 other study(ies) available for cgp 12177 and colforsin
Article | Year |
---|---|
Beta-adrenergic, cAMP-mediated stimulation of proliferation of brown fat cells in primary culture. Mediation via beta 1 but not via beta 3 adrenoceptors.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bucladesine; Cell Division; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; DNA Replication; Imidazoles; Mice; Mice, Inbred Strains; Norepinephrine; Oxymetazoline; Propanolamines; Receptors, Adrenergic, beta; Thymidine | 1992 |
Beta-adrenoceptors and adenylate cyclase activity in hypertrophied and failing rabbit left ventricle.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cardiomegaly; Colforsin; Cyclic AMP; Female; GTP-Binding Proteins; Heart Arrest; Isoproterenol; Male; Nucleotidases; Propanolamines; Rabbits; Receptors, Adrenergic, beta; Sodium Fluoride | 1991 |
Alpha- and beta-adrenergic induction of the expression of the uncoupling protein thermogenin in brown adipocytes differentiated in culture.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Colforsin; Gene Expression; Insulin; Ion Channels; Male; Membrane Proteins; Mice; Mitochondrial Proteins; Norepinephrine; Nucleic Acid Hybridization; Oxymetazoline; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; RNA; RNA, Messenger; Thyroxine; Triiodothyronine; Uncoupling Protein 1 | 1990 |
Pseudomonas exotoxin A prevents beta-adrenoceptor-induced upregulation of Gi protein alpha-subunits and adenylyl cyclase desensitization in rat heart muscle cells.
Topics: Adenosine Diphosphate Ribose; Adenylyl Cyclases; ADP Ribose Transferases; Adrenergic beta-Antagonists; Animals; Bacterial Toxins; Cells, Cultured; Colforsin; Exotoxins; GTP-Binding Proteins; Heart; Isoproterenol; Kinetics; Macromolecular Substances; Muscle, Smooth; Myocardium; NAD; Norepinephrine; Propanolamines; Pseudomonas aeruginosa Exotoxin A; Rats; Receptors, Adrenergic, beta; Virulence Factors | 1990 |
Homologous vs. heterologous desensitization of the adenylate cyclase system in heart cells.
Topics: Adenylyl Cyclases; Alprostadil; Animals; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Isoproterenol; Myocardium; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta | 1988 |
Characterization of beta-adrenergic binding sites on rodent Leydig cells.
Topics: Adrenergic beta-Antagonists; Androgens; Animals; Binding, Competitive; Cell Separation; Cells, Cultured; Colforsin; Isoproterenol; Kinetics; Leydig Cells; Luteinizing Hormone; Male; Mice; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1985 |
Transport of beta-adrenergic antagonists in the absence of beta-adrenergic receptors in rat pituitary tumor cells.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Biological Transport; Cell Line; Colforsin; Cyclic AMP; Dihydroalprenolol; Epinephrine; Hydrogen-Ion Concentration; Imipramine; Kinetics; Monensin; Norepinephrine; Nucleotides; Oligomycins; Ouabain; Pituitary Neoplasms; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta; Reserpine; Serotonin; Temperature | 1986 |
Molecular mechanisms underlying regional variations of catecholamine-induced lipolysis in rat adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Base Sequence; Brimonidine Tartrate; Bucladesine; Catecholamines; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Dioxanes; DNA Primers; Epididymis; Gene Expression; Idazoxan; Isoproterenol; Lipase; Lipolysis; Male; Molecular Sequence Data; Organ Specificity; Polymerase Chain Reaction; Propanolamines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; RNA, Messenger; Skin | 1995 |
Physiological desensitization of beta 3-adrenergic responses in brown fat cells: involvement of a postreceptor process.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Acclimatization; Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cells, Cultured; Cold Temperature; Colforsin; Cricetinae; Cyclic AMP; Ethanolamines; Isoproterenol; Kinetics; Male; Mesocricetus; Norepinephrine; Oxygen Consumption; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3 | 1993 |
Heterologous sensitization of adenylate cyclase activity by serotonin in the rat cerebral cortex.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Cerebral Cortex; Colforsin; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoproterenol; Male; Phorbol 12,13-Dibutyrate; Propanolamines; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Somatostatin; Tetradecanoylphorbol Acetate; Vasoactive Intestinal Peptide | 1993 |
Modulation of adenylylcyclase by protein kinase C in human neurotumor SK-N-MC cells: evidence that the alpha isozyme mediates both potentiation and desensitization.
Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Alkaloids; Aluminum Compounds; Animals; Brain; Cell Line; Cell Membrane; Cholera Toxin; Colforsin; Cyclic AMP; Dopamine; Drug Synergism; Fluorides; GTP-Binding Proteins; Humans; Isoenzymes; Isoproterenol; Kinetics; Manganese; Neuroblastoma; Neuropeptide Y; Propanolamines; Protein Kinase C; Rats; Sphingosine; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1994 |
Thermogenesis in brown adipose tissue with age: post-receptor activation by forskolin.
Topics: Adipose Tissue, Brown; Adrenergic beta-Antagonists; Aging; Animals; Binding Sites; Body Temperature Regulation; Carrier Proteins; Colforsin; Guanosine Diphosphate; Ion Channels; Male; Membrane Proteins; Mitochondria; Mitochondrial Proteins; Oxygen Consumption; Propanolamines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; RNA, Messenger; Uncoupling Agents; Uncoupling Protein 1 | 1996 |
Triiodothyronine regulates beta 3-adrenoceptor expression in 3T3-F442A differentiating adipocytes.
Topics: 3T3 Cells; Adenylyl Cyclases; Adipocytes; Adrenergic beta-Antagonists; Animals; Base Sequence; Cell Differentiation; Cell Nucleus; Colforsin; Dactinomycin; DNA Primers; Gene Expression; Glycerolphosphate Dehydrogenase; Guanosine 5'-O-(3-Thiotriphosphate); Isoproterenol; Kinetics; Mice; Molecular Sequence Data; Propanolamines; Protein Biosynthesis; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Recombinant Proteins; RNA, Messenger; Transcription, Genetic; Transfection; Triiodothyronine | 1996 |
Regulation of lipolysis in fat cells of obese women during long-term hypocaloric diet.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipocytes; Adrenergic beta-Agonists; Adult; Brimonidine Tartrate; Bucladesine; Catecholamines; Colforsin; Dobutamine; Energy Intake; Female; Food Deprivation; Glucose; Humans; Insulin; Insulin Resistance; Isoproterenol; Lipolysis; Middle Aged; Obesity; Propanolamines; Quinoxalines; Terbutaline; Time Factors | 1996 |
Alterations of central noradrenergic transmission in Ts65Dn mouse, a model for Down syndrome.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Agonists; Animals; Brain; Cell Membrane; Cerebellum; Cerebral Cortex; Chromosome Mapping; Chromosomes, Human, Pair 21; Colforsin; Cyclic AMP; Down Syndrome; Hippocampus; Humans; In Vitro Techniques; Isoproterenol; Kinetics; Mice; Mice, Neurologic Mutants; Norepinephrine; Organ Specificity; Propanolamines; Receptors, Adrenergic, beta; Reference Values; Signal Transduction | 1997 |
Growth inhibition of new human thyroid carcinoma cell lines by activation of adenylate cyclase through the beta-adrenergic receptor.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adult; Animals; Cell Division; Colforsin; Cyclic AMP; DNA-Binding Proteins; DNA, Neoplasm; Enzyme Activation; Female; Humans; Nuclear Proteins; Paired Box Transcription Factors; PAX8 Transcription Factor; Propanolamines; Rats; Receptors, Adrenergic, beta; RNA, Messenger; Thyroid Neoplasms; Thyroid Nuclear Factor 1; Trans-Activators; Transcription Factors; Tumor Cells, Cultured | 1997 |
Beta-adrenergic signal transduction in the hypothalamus of the European hamster: relation with the seasonal hibernation cycle and the diurnal activity cycle.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Arousal; Chlorides; Circadian Rhythm; Colforsin; Cricetinae; Cyclic AMP; Enzyme Activation; Guanylyl Imidodiphosphate; Hibernation; Hypothalamus; Imidazoles; Light; Male; Manganese Compounds; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Seasons; Signal Transduction | 1997 |
Heterologous regulation of muscarinic and beta-adrenergic receptors in rat cardiomyocytes in culture.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding Sites; Binding, Competitive; Bucladesine; Carbachol; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Inhibitors; Female; Indoles; Isoproterenol; Isoquinolines; Kinetics; Male; Maleimides; Muscarinic Agonists; Myocardium; N-Methylscopolamine; Propanolamines; Protein Kinase C; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Sulfonamides; Thionucleotides; Tritium | 1998 |
Stimulation of the extracellular signal-regulated kinase 1/2 pathway by human beta-3 adrenergic receptor: new pharmacological profile and mechanism of activation.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Colforsin; Cricetinae; Dioxoles; Enzyme Activation; Epinephrine; Ethanolamines; Humans; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Norepinephrine; Phentolamine; Prazosin; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction; Yohimbine | 1999 |
The effect of hydrogen peroxide upon beta-adrenoceptor density and function in C6 rat glioma cells.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Cell Death; Colforsin; Culture Media, Serum-Free; Cyclic AMP; Glioma; GTP-Binding Protein alpha Subunits, Gs; Hydrogen Peroxide; Isoproterenol; L-Lactate Dehydrogenase; Propanolamines; Rats; Receptors, Adrenergic, beta; Tumor Cells, Cultured | 1999 |
Functional and molecular biological evidence for a possible beta3-adrenoceptor in the human detrusor muscle.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colforsin; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 1999 |
Differential effects of opioid and adrenergic agonists on proliferation in a cultured cell line.
Topics: 3T3 Cells; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Analgesics, Opioid; Animals; Cell Culture Techniques; Cell Division; Cloning, Molecular; Colforsin; Cyclic AMP; Gene Expression Regulation, Enzymologic; Hypoglycemic Agents; Insulin; JNK Mitogen-Activated Protein Kinases; MAP Kinase Kinase 4; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Morphine; Procaterol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-2; Receptors, Opioid, delta; RNA, Messenger; Second Messenger Systems; Transfection; Tritium | 1999 |
Regulation of beta 1- and beta 3-adrenergic agonist-stimulated lipolytic response in hyperthyroid and hypothyroid rat white adipocytes.
Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Agonists; Animals; Blotting, Northern; Cell Membrane; Colforsin; Hyperthyroidism; Hypothyroidism; Kinetics; Lipolysis; Male; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; RNA, Messenger; Thyroidectomy | 2000 |
Beta-3 adrenergic stimulation of L-type Ca(2+) channels in rat portal vein myocytes.
Topics: 1-Propanol; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Barium; Calcium Channels, L-Type; Cells, Cultured; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; Isoproterenol; Isoquinolines; Membrane Potentials; Muscle, Smooth, Vascular; Phorbol 12,13-Dibutyrate; Portal Vein; Propanolamines; Rats; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Sulfonamides | 2000 |
Rapid electrical stimulation of contraction reduces the density of beta-adrenergic receptors and responsiveness of cultured neonatal rat cardiomyocytes. Possible involvement of microtubule disassembly secondary to mechanical stress.
Topics: Acetylcholine; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Antineoplastic Agents, Phytogenic; Cells, Cultured; Colforsin; Diacetyl; Dihydroalprenolol; Down-Regulation; Electric Stimulation; Enzyme Inhibitors; Heart Failure; Isoproterenol; Microtubules; Muscle Fibers, Skeletal; Myocardial Contraction; Myocardium; Pacemaker, Artificial; Paclitaxel; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stress, Mechanical; Tritium; Vasodilator Agents | 2000 |
Short-term effects of postnatal manipulation on central beta-adrenoceptor transmission.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenocorticotropic Hormone; Animals; Animals, Suckling; Cerebellum; Cerebral Cortex; Colforsin; Corticosterone; Cyclic AMP; Emotions; Female; Handling, Psychological; Hippocampus; Isoproterenol; Male; Norepinephrine; Pregnancy; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Restraint, Physical; Signal Transduction; Stress, Physiological; Tritium | 1999 |
Norepinephrine-induced sustained inward current in brown fat cells: alpha(1)-mediated by nonselective cation channels.
Topics: Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Calcimycin; Calcium; Cations; Chlorides; Colforsin; Electric Conductivity; Enzyme Activation; Extracellular Space; Imidazoles; Ion Channels; Ionophores; Male; Norepinephrine; Patch-Clamp Techniques; Phenylephrine; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sodium | 2000 |
Differential alterations in cardiac adrenergic signaling in chronic hypoxia or norepinephrine infusion.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Cholera Toxin; Chronic Disease; Colforsin; GTP-Binding Proteins; Guanosine Triphosphate; Heart Rate; Heart Ventricles; Hypertrophy, Left Ventricular; Hypertrophy, Right Ventricular; Hypoxia; Isoproterenol; Male; Myocardium; Norepinephrine; Pertussis Toxin; Propanolamines; Protein Kinase C; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Signal Transduction; Sodium Fluoride; Sympathomimetics; Tritium; Virulence Factors, Bordetella; Weight Gain | 2001 |
Characterization of [3H]CGP 12177 binding to beta-adrenergic receptors in intact eel hepatocytes.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Alprenolol; Anguilla; Animals; Atenolol; Binding Sites; Binding, Competitive; Butoxamine; Cell Count; Colforsin; Cyclic AMP; Epinephrine; Glucose; Guanosine 5'-O-(3-Thiotriphosphate); Hepatocytes; Kinetics; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tritium | 2001 |
Sex-dependent thermogenesis, differences in mitochondrial morphology and function, and adrenergic response in brown adipose tissue.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Weight; Bucladesine; Calorimetry, Indirect; Colforsin; DNA; Female; Isoproterenol; Light; Lipolysis; Male; Mitochondria; Norepinephrine; Organ Size; Oxygen Consumption; Propanolamines; Rats; Rats, Wistar; Respiratory Mechanics; Sex Characteristics; Thermogenesis; Triglycerides | 2002 |
Characterization of isoprenaline- and salmeterol-stimulated interactions between beta2-adrenoceptors and beta-arrestin 2 using beta-galactosidase complementation in C2C12 cells.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Arrestins; beta-Arrestin 2; beta-Arrestins; beta-Galactosidase; Cell Line; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Genetic Complementation Test; Humans; Isoproterenol; Mutation; Propanolamines; Propranolol; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Salmeterol Xinafoate; Transfection | 2005 |