cgp 12177 and cl 316243

cgp 12177 has been researched along with cl 316243 in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (57.14)18.2507
2000's6 (42.86)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Begin-Heick, N; Ghorbani, M; Himms-Hagen, J; Kates, AL; Triandafillou, J1
Berlan, M; Bousquet-Melou, A; Galitzky, J; Lafontan, M; Montastruc, JL1
Arner, P; Blaak, E; Hoffstedt, J; Lönnqvist, F; Shimizu, M1
Berlan, M; Galitzky, J; Lafontan, M; Langin, D; Montastruc, JL; Verwaerde, P1
Malinowska, B; Schlicker, E1
Gerhardt, CC; Gros, J; Issad, T; Strosberg, AD1
Ajisawa, Y; Akahane, M; Andersson, KE; Hayakawa, K; Igawa, Y; Nishizawa, O; Takeda, H; Yamazaki, Y; Yoneyama, T1
Bloomquist, W; Calligaro, D; Cohen, ML; Kriauciunas, A; Shuker, A1
Asano, A; Fushiki, T; Kawada, T; Kayahashi, S; Kimura, K; Mizukami, J; Morimatsu, M; Saito, M; Sasaki, N; Yoshida, T1
Giacobino, JP; Jimenez, M; Kaumann, AJ; Moffatt, J; Molenaar, P; Oostendorp, J; Preitner, F1
Ajisawa, Y; Akahane, M; Igawa, Y; Komatsu, Y; Nishizawa, O; Takeda, H; Yamazaki, Y1
Akahane, M; Kojima, M; Murakami, M; Tomiyama, Y; Yamazaki, Y1
Baker, JG1
Badawi, JK; Bross, S; Haferkamp, A; Hatzinger, M; Michel, MS; Uecelehan, H1

Other Studies

14 other study(ies) available for cgp 12177 and cl 316243

ArticleYear
Apparent lack of beta 3-adrenoceptors and of insulin regulation of glucose transport in brown adipose tissue of guinea pigs.
    The American journal of physiology, 1995, Volume: 268, Issue:1 Pt 2

    Topics: Acclimatization; Adenylyl Cyclases; Adipose Tissue, Brown; Adrenergic alpha-Agonists; Animals; Body Temperature Regulation; Cell Membrane; Dioxoles; Epinephrine; Ethanolamines; Female; Glucose Transporter Type 4; Guinea Pigs; Insulin; Isoproterenol; Monosaccharide Transport Proteins; Muscle Proteins; Norepinephrine; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Temperature; Time Factors

1995
Beta-3 adrenoceptor-mediated increase in cutaneous blood flow in the dog.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Bupranolol; Dioxoles; Dogs; Ethanolamines; Heart Rate; Isoproterenol; Male; Nitroprusside; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Regional Blood Flow; Skin

1994
Effects of several putative beta 3-adrenoceptor agonists on lipolysis in human omental adipocytes.
    International journal of obesity and related metabolic disorders : journal of the International Association for the Study of Obesity, 1996, Volume: 20, Issue:5

    Topics: Adipocytes; Adrenergic beta-Agonists; Catechols; Dioxoles; Ethanolamines; Glycerol; Humans; Isoproterenol; Lipolysis; Omentum; Propanolamines; Serine

1996
Lipolytic effects of conventional beta 3-adrenoceptor agonists and of CGP 12,177 in rat and human fat cells: preliminary pharmacological evidence for a putative beta 4-adrenoceptor.
    British journal of pharmacology, 1997, Volume: 122, Issue:6

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Dioxoles; Humans; Lipolysis; Male; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes

1997
Further evidence for differences between cardiac atypical beta-adrenoceptors and brown adipose tissue beta3-adrenoceptors in the pithed rat.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Male; Pindolol; Propanolamines; Rats; Rats, Wistar; Temperature

1997
Stimulation of the extracellular signal-regulated kinase 1/2 pathway by human beta-3 adrenergic receptor: new pharmacological profile and mechanism of activation.
    Molecular pharmacology, 1999, Volume: 55, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Colforsin; Cricetinae; Dioxoles; Enzyme Activation; Epinephrine; Ethanolamines; Humans; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Norepinephrine; Phentolamine; Prazosin; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction; Yohimbine

1999
Functional and molecular biological evidence for a possible beta3-adrenoceptor in the human detrusor muscle.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colforsin; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

1999
Aryl propanolamines: comparison of activity at human beta3 receptors, rat beta3 receptors and rat atrial receptors mediating tachycardia.
    British journal of pharmacology, 1999, Volume: 126, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Dioxoles; Humans; Male; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Tachycardia

1999
Mutated human beta3-adrenergic receptor (Trp64Arg) lowers the response to beta3-adrenergic agonists in transfected 3T3-L1 preadipocytes.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 2000, Volume: 32, Issue:3

    Topics: 3T3 Cells; Adenylyl Cyclases; Adipocytes; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amino Acid Substitution; Animals; Cyclic AMP; Dioxoles; Epinephrine; Humans; Isoproterenol; Kinetics; Mice; Mutagenesis, Site-Directed; Norepinephrine; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Recombinant Proteins; Sulfonamides; Transfection

2000
Contribution of beta-adrenoceptor subtypes to relaxation of colon and oesophagus and pacemaker activity of ureter in wildtype and beta(3)-adrenoceptor knockout mice.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dioxoles; Dose-Response Relationship, Drug; Epinephrine; Esophagus; Female; Imidazoles; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Ureter

2000
Characterization of beta-adrenoceptor subtypes in the ferret urinary bladder in vitro and in vivo.
    European journal of pharmacology, 2000, Sep-01, Volume: 403, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Anesthesia; Animals; Blood Pressure; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Ethanolamines; Ferrets; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pressure; Procaterol; Propanolamines; Receptors, Adrenergic, beta; Time Factors; Urinary Bladder

2000
Comparison between CL-316243- and CGP-12177A-induced relaxations in isolated canine ureter.
    Pharmacology, 2003, Volume: 68, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Dogs; Female; In Vitro Techniques; Male; Muscle Relaxation; Propanolamines; Receptors, Adrenergic, beta; Substrate Specificity; Ureter; Vasodilator Agents

2003
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
    British journal of pharmacology, 2005, Volume: 144, Issue:3

    Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3

2005
Relaxant effects of beta-adrenergic agonists on porcine and human detrusor muscle.
    Acta physiologica Scandinavica, 2005, Volume: 185, Issue:2

    Topics: Adrenergic beta-Agonists; Aged; Albuterol; Animals; Dioxoles; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Humans; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Procaterol; Propanolamines; Swine

2005