cgp 12177 has been researched along with cgp 20712a in 30 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 1 (3.33) | 18.7374 |
| 1990's | 19 (63.33) | 18.2507 |
| 2000's | 8 (26.67) | 29.6817 |
| 2010's | 2 (6.67) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Guillaume, JL; Méjean, A; Strosberg, AD | 1 |
| Iakovidis, D; Jackman, GP; Louis, SN; Louis, WJ; Nero, TL | 1 |
| Baker, JG | 1 |
| Baker, JG; Fischer, PM; Gardiner, SM; Hill, SJ; Kellam, B; Mistry, SN | 1 |
| Blanksma, PK; Bouwer, J; Elsinga, PH; Lie, KI; Meeder, JG; Paans, AM; Vaalburg, W; van Waarde, A; Visser, GM | 1 |
| Blanksma, PK; Brodde, OE; Elsinga, PH; Lie, KI; Meeder, JG; Paans, AM; Vaalburg, W; Van Waarde, A; Visser, GM | 1 |
| Leysen, JE; Pauwels, PJ; Van Gompel, P | 1 |
| Baude, B; Blin, N; Emorine, LJ; Fève, B; Lasnier, F; Nahmias, C; Pairault, J; Strosberg, AD | 1 |
| Johnson, AM; Nelson, DR; Palmer, KJ | 1 |
| Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
| Langer, L; Lemmer, B; Olbrich, HG; Witte, K | 1 |
| Döring, V; Kalmár, P; Lavicky, J; Schmitz, W; Scholz, H; Steinfath, M | 1 |
| Bohl, J; Langer, L; Lemmer, B; Ohm, T | 1 |
| Adachi-Akahane, S; Kitagawa, Y; Nagao, T | 1 |
| Gardner, ML; Körner, C; Pittelkow, MR; Schallreuter, KU; Swanson, NN | 1 |
| Morin, C; Morin, D; Sapena, R; Tillement, JP; Zini, R | 1 |
| Morin, D; Onteniente, B; Sapena, R; Tillement, JP; Zini, R | 1 |
| Germack, R; Perret, GY; Starzec, AB; Vassy, R | 1 |
| Malinowska, B; Schlicker, E | 1 |
| Nürnberger, F; Pleschka, K | 1 |
| Atlan, G; Collet, F; Féve, B; Frisdal, E; Pavoine, C; Pecker, F | 1 |
| Ajisawa, Y; Akahane, M; Andersson, KE; Hayakawa, K; Igawa, Y; Nishizawa, O; Takeda, H; Yamazaki, Y; Yoneyama, T | 1 |
| Giacobino, JP; Jimenez, M; Kaumann, AJ; Moffatt, J; Molenaar, P; Oostendorp, J; Preitner, F | 1 |
| Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S | 1 |
| Santos, IN; Spadari-Bratfisch, RC | 1 |
| Brørs, O; Jørgen, J; Sharikabad, MN | 1 |
| Brahmadevara, N; MacDonald, A; Shaw, AM | 1 |
| Caceres, VM; Krieger, MH; Moreira, MF; Santos, IN; Spadari-Bratfisch, RC; Sumitame, M | 1 |
| Badino, P; Barbero, R; Cuniberti, B; Girardi, C; Magistris, G; Odore, R; Pagliasso, S; Re, G | 1 |
| Abraham, G; Guenl, B; Jonas, S; Kassahun, WT; Ungemach, FR | 1 |
30 other study(ies) available for cgp 12177 and cgp 20712a
| Article | Year |
|---|---|
Carazolol: a potent, selective beta 3-adrenoceptor agonist.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cells, Cultured; CHO Cells; Cricetinae; Dithiothreitol; Lipolysis; Propanolamines; Receptors, Adrenergic, beta | 1995 |
LK 204-545, a highly selective beta1-adrenoceptor antagonist at human beta-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; Cyclopropanes; Female; Humans; Imidazoles; In Vitro Techniques; Ligands; Phenoxypropanolamines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Trachea; Urea | 1999 |
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2005 |
Synthesis and in vitro and in vivo characterization of highly β1-selective β-adrenoceptor partial agonists.
Topics: Adrenergic beta-1 Receptor Agonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Design; Heart Rate; Hemodynamics; Humans; Indicators and Reagents; Ligands; Male; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Structure-Activity Relationship | 2013 |
Suitability of CGP-12177 and CGP-26505 for quantitative imaging of beta-adrenoceptors.
Topics: Adrenergic beta-Antagonists; Animals; Imidazoles; Male; Metabolic Clearance Rate; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Time Factors; Tissue Distribution; Tritium | 1992 |
Uptake of radioligands by rat heart and lung in vivo: CGP 12177 does and CGP 26505 does not reflect binding to beta-adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Imidazoles; In Vitro Techniques; Lung; Male; Myocardium; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Tissue Distribution | 1992 |
Human beta 1- and beta 2-adrenergic receptor binding and mediated accumulation of cAMP in transfected Chinese hamster ovary cells. Profile of nebivolol and known beta-adrenergic blockers.
Topics: Adrenergic beta-Antagonists; Animals; Benzopyrans; Binding Sites; Binding, Competitive; Cell Line; Cricetinae; Cricetulus; Cyclic AMP; Ethanolamines; Humans; Imidazoles; Isoproterenol; Models, Biological; Nebivolol; Propanolamines; Propranolol; Radioligand Assay; Receptors, Adrenergic, beta; Stereoisomerism; Transfection | 1991 |
Atypical beta-adrenergic receptor in 3T3-F442A adipocytes. Pharmacological and molecular relationship with the human beta 3-adrenergic receptor.
Topics: 3T3 Cells; Adipose Tissue; Adrenergic beta-Antagonists; Animals; Base Sequence; Binding, Competitive; Blotting, Northern; DNA; Ethanolamines; Humans; Imidazoles; Mice; Molecular Sequence Data; Oxprenolol; Pindolol; Polymerase Chain Reaction; Propanolamines; Receptors, Adrenergic, beta; RNA, Messenger | 1991 |
Effect of prolonged 5-hydroxytryptamine uptake inhibition by paroxetine on cortical beta 1 and beta 2-adrenoceptors in rat brain.
Topics: Adrenergic beta-Antagonists; Amitriptyline; Animals; Antidepressive Agents; Cerebral Cortex; Dose-Response Relationship, Drug; Imidazoles; Kinetics; Male; Neurotransmitter Uptake Inhibitors; Paroxetine; Piperidines; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin | 1990 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
Uncoupling of beta 1-adrenoceptors from cardiac adenylyl cyclase in cardiomyopathic and control hamsters.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cardiomyopathies; Cricetinae; Heart Ventricles; Imidazoles; Isoproterenol; Male; Membranes; Mesocricetus; Myocardium; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1 | 1993 |
Changes in cardiac beta-adrenoceptors in human heart diseases: relationship to the degree of heart failure and further evidence for etiology-related regulation of beta 1 and beta 2 subtypes.
Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Aortic Valve; Cardiomyopathy, Hypertrophic; Down-Regulation; Female; Heart Failure; Heart Valve Diseases; Heart Ventricles; Humans; Imidazoles; Iodocyanopindolol; Male; Middle Aged; Mitral Valve; Muscular Dystrophies; Myocardium; Pindolol; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Tetralogy of Fallot | 1993 |
Beta-adrenoceptor density and subtype distribution in cerebellum and hippocampus from patients with Alzheimer's disease.
Topics: Adrenergic beta-Antagonists; Aged; Aged, 80 and over; Alzheimer Disease; Binding, Competitive; Cerebellum; Dementia; Female; Hippocampus; Humans; Imidazoles; Kinetics; Male; Middle Aged; Propanolamines; Receptors, Adrenergic, beta; Tritium | 1993 |
Determination of beta-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective beta-antagonists.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Binding, Competitive; Cyclic AMP; Heart Ventricles; Imidazoles; Iodocyanopindolol; Isoproterenol; Kinetics; Male; Membranes; Myocardium; Pindolol; Propanolamines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Stimulation, Chemical; Tritium | 1995 |
The induction of the alpha-1-adrenoceptor signal transduction system on human melanocytes.
Topics: Adrenergic beta-Antagonists; Adult; Cells, Cultured; Gene Expression Regulation; Humans; Imidazoles; Infant, Newborn; Keratinocytes; Melanocytes; Norepinephrine; Prazosin; Propanolamines; Receptors, Adrenergic, alpha-1; Signal Transduction | 1996 |
Desipramine treatment differently down-regulates beta-adrenoceptors of freshly isolated neurons and astrocytes.
Topics: Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Animals; Astrocytes; Binding Sites; Brain; Desipramine; Down-Regulation; Imidazoles; Male; Neurons; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1996 |
Characterization of beta-adrenergic receptors of freshly isolated astrocytes and neurons from rat brain.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Astrocytes; Binding, Competitive; Cells, Cultured; Cerebellum; Imidazoles; Immunohistochemistry; Male; Neurons; Propanolamines; Prosencephalon; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1997 |
Beta-adrenoceptor subtype expression and function in rat white adipocytes.
Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Binding, Competitive; Imidazoles; Lipolysis; Male; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 1997 |
Further evidence for differences between cardiac atypical beta-adrenoceptors and brown adipose tissue beta3-adrenoceptors in the pithed rat.
Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dioxoles; Dose-Response Relationship, Drug; Heart Rate; Imidazoles; Male; Pindolol; Propanolamines; Rats; Rats, Wistar; Temperature | 1997 |
Beta-adrenergic signal transduction in the hypothalamus of the European hamster: relation with the seasonal hibernation cycle and the diurnal activity cycle.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Arousal; Chlorides; Circadian Rhythm; Colforsin; Cricetinae; Cyclic AMP; Enzyme Activation; Guanylyl Imidodiphosphate; Hibernation; Hypothalamus; Imidazoles; Light; Male; Manganese Compounds; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Seasons; Signal Transduction | 1997 |
Pharmacological and molecular characterisation of beta-adrenoceptors in adult rat diaphragm muscle.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aging; Animals; Dose-Response Relationship, Drug; Fenoterol; Imidazoles; Isoproterenol; Male; Muscle, Smooth; Pindolol; Prenalterol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 1998 |
Functional and molecular biological evidence for a possible beta3-adrenoceptor in the human detrusor muscle.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Aged, 80 and over; Colforsin; Dioxoles; Dobutamine; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Female; Gene Expression; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 1999 |
Contribution of beta-adrenoceptor subtypes to relaxation of colon and oesophagus and pacemaker activity of ureter in wildtype and beta(3)-adrenoceptor knockout mice.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Colon; Dioxoles; Dose-Response Relationship, Drug; Epinephrine; Esophagus; Female; Imidazoles; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Ureter | 2000 |
Functional assessment of beta adrenoceptor subtypes in human colonic circular and longitudinal (taenia coli) smooth muscle.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Colon; Female; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Terbutaline; Tetrahydronaphthalenes | 2000 |
Chronotropic response to (+/-)-CGP12177 in right atria of stressed rats.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Heart Atria; Heart Rate; Imidazoles; In Vitro Techniques; Male; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Stress, Physiological; Time Factors | 2001 |
Sarcolemmal beta-adrenoceptors determined in rat ventricular heart biopsies with (-)-[3H]CGP-12177.
Topics: Adrenergic beta-Antagonists; Animals; Binding, Competitive; Heart Ventricles; Imidazoles; In Vitro Techniques; Propanolamines; Rats; Rats, Wistar; Rats, Zucker; Receptors, Adrenergic, beta | 2002 |
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction | 2004 |
Evidence for two atypical conformations of beta-adrenoceptors and their interaction with Gi proteins.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Heart Atria; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; Norepinephrine; Pertussis Toxin; Propanolamines; Protein Binding; Protein Conformation; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1 | 2005 |
Effects of Inflammation upon beta-adrenoceptor concentrations in the common digital artery of the horse: an in vitro study.
Topics: Adrenergic beta-Antagonists; Animals; Arteries; Horse Diseases; Horses; Imidazoles; In Vitro Techniques; Lipopolysaccharides; Muscle, Smooth, Vascular; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Vasculitis | 2005 |
Expression and functional coupling of liver β2 - adrenoceptors in the human hepatocellular carcinoma.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adult; Aged; Carcinoma, Hepatocellular; Female; Humans; Imidazoles; Iodocyanopindolol; Liver; Liver Neoplasms; Male; Middle Aged; Propanolamines; Receptors, Adrenergic, beta-2 | 2012 |