cgp 12177 and betaxolol

cgp 12177 has been researched along with betaxolol in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19901 (20.00)18.7374
1990's3 (60.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Iakovidis, D; Jackman, GP; Louis, SN; Louis, WJ; Nero, TL1
Belz, GG; Palm, D; Wellstein, A1
Iisalo, E; Kaila, T; Saari, KM; Vuori, ML1
Ali-Melkkilä, T; Iisalo, E; Kaila, T; Saari, KM; Vuori, ML1
McLean, AJ; Milligan, G1

Trials

2 trial(s) available for cgp 12177 and betaxolol

ArticleYear
Concentrations and antagonist activity of topically applied betaxolol in aqueous humour.
    Acta ophthalmologica, 1993, Volume: 71, Issue:5

    Topics: Absorption; Administration, Topical; Adrenergic beta-Antagonists; Aged; Aged, 80 and over; Aqueous Humor; Betaxolol; Cataract Extraction; Humans; Lenses, Intraocular; Ophthalmic Solutions; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta

1993
Beta 1- and beta 2-antagonist activity of topically applied betaxolol and timolol in the systemic circulation.
    Acta ophthalmologica, 1993, Volume: 71, Issue:5

    Topics: Administration, Topical; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Aged; Aged, 80 and over; Betaxolol; Humans; Middle Aged; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Timolol

1993

Other Studies

3 other study(ies) available for cgp 12177 and betaxolol

ArticleYear
LK 204-545, a highly selective beta1-adrenoceptor antagonist at human beta-adrenoceptors.
    European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; Cyclopropanes; Female; Humans; Imidazoles; In Vitro Techniques; Ligands; Phenoxypropanolamines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Trachea; Urea

1999
Affinity and selectivity of beta-adrenoceptor antagonists in vitro.
    Journal of cardiovascular pharmacology, 1986, Volume: 8 Suppl 11

    Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Betaxolol; Binding, Competitive; Bisoprolol; Propanolamines; Propranolol; Rats; Salivary Glands; Tritium

1986
Ligand regulation of green fluorescent protein-tagged forms of the human beta(1)- and beta(2)-adrenoceptors; comparisons with the unmodified receptors.
    British journal of pharmacology, 2000, Volume: 130, Issue:8

    Topics: Betaxolol; Binding, Competitive; Cell Line; Dihydroalprenolol; Endocytosis; Green Fluorescent Proteins; Humans; Isoproterenol; Kinetics; Ligands; Luminescent Proteins; Microscopy, Confocal; Oligopeptides; Peptides; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Recombinant Fusion Proteins; Tritium

2000