cgp 12177 and atenolol

cgp 12177 has been researched along with atenolol in 15 studies

Research

Studies (15)

Timeframe	Studies, this research(%)	All Research%
pre-1990	2 (13.33)	18.7374
1990's	9 (60.00)	18.2507
2000's	3 (20.00)	29.6817
2010's	1 (6.67)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Iakovidis, D; Jackman, GP; Louis, SN; Louis, WJ; Nero, TL	1
Colledge, WH; Joseph, SS; Kaumann, AJ; Lynham, JA	1
Baker, JG	1
Charlton, SJ; Dickson, CJ; Duca, JS; Fairhurst, RA; Hornak, V; McKay, DJ; Pearlstein, RA; Reilly, J; Sandham, DA; Shaw, D; Sykes, DA; Velez-Vega, C	1
Heibel, B; Lücker, PW; Palm, D; Sitzler, G	1
Dunn, AJ; Yang, XM	1
Bouscarel, B; Cortinovis, C; Mayer, D; Murat, JC; Paris, H	1
Belz, GG; Palm, D; Wellstein, A	1
Horinouchi, T; Koike, K; Muramatsu, M; Ohki, S; Takayanagi, I	1
Anctil, M; Awad, EW	1
Kaila, T; Marttila, R	1
Hattori, K; Hosohata, Y; Maruyama, K; Nagatomo, T; Ohnuki, T; Sasaki, K; Suzuki, J; Watanabe, K	1
Chen, CM; Ko, FN; Lin, CH; Teng, CM; Yang, CM	1
Horinouchi, T; Koike, K	1
Capuzzo, A; Fabbri, E; Moon, TW; Selva, C	1

Trials

2 trial(s) available for cgp 12177 and atenolol

Article	Year
Bioequivalence of two atenolol formulations in healthy volunteers. Evaluation and prediction of effect kinetics at beta-adrenoceptors in vivo by means of a radioreceptor assay. Methods and findings in experimental and clinical pharmacology, 1991, Volume: 13, Issue:2 Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Atenolol; Chromatography, Gas; Double-Blind Method; Heart Rate; Humans; Male; Propanolamines; Radioligand Assay; Random Allocation; Receptors, Adrenergic, beta; Therapeutic Equivalency	1991
Receptor occupancy in lumbar CSF as a measure of the antagonist activity of atenolol, metoprolol and propranolol in the CNS. British journal of clinical pharmacology, 1993, Volume: 35, Issue:5 Topics: Adrenergic alpha-Antagonists; Adult; Animals; Atenolol; Central Nervous System; Female; Humans; In Vitro Techniques; Male; Metoprolol; Middle Aged; Propanolamines; Propranolol; Rabbits; Rats; Receptors, Adrenergic, alpha	1993

Article

Year

Bioequivalence of two atenolol formulations in healthy volunteers. Evaluation and prediction of effect kinetics at beta-adrenoceptors in vivo by means of a radioreceptor assay.

Methods and findings in experimental and clinical pharmacology, 1991, Volume: 13, Issue:2

Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Atenolol; Chromatography, Gas; Double-Blind Method; Heart Rate; Humans; Male; Propanolamines; Radioligand Assay; Random Allocation; Receptors, Adrenergic, beta; Therapeutic Equivalency

1991

Receptor occupancy in lumbar CSF as a measure of the antagonist activity of atenolol, metoprolol and propranolol in the CNS.

British journal of clinical pharmacology, 1993, Volume: 35, Issue:5

Topics: Adrenergic alpha-Antagonists; Adult; Animals; Atenolol; Central Nervous System; Female; Humans; In Vitro Techniques; Male; Metoprolol; Middle Aged; Propanolamines; Propranolol; Rabbits; Rats; Receptors, Adrenergic, alpha

1993

Other Studies

13 other study(ies) available for cgp 12177 and atenolol

Article	Year
LK 204-545, a highly selective beta1-adrenoceptor antagonist at human beta-adrenoceptors. European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3 Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; Cyclopropanes; Female; Humans; Imidazoles; In Vitro Techniques; Ligands; Phenoxypropanolamines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Trachea; Urea	1999
Binding of (-)-[3H]-CGP12177 at two sites in recombinant human beta 1-adrenoceptors and interaction with beta-blockers. Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 369, Issue:5 Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Binding Sites; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Interactions; Humans; Propanolamines; Receptors, Adrenergic, beta-1	2004
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors. British journal of pharmacology, 2005, Volume: 144, Issue:3 Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3	2005
Uncoupling the Structure-Activity Relationships of β2 Adrenergic Receptor Ligands from Membrane Binding. Journal of medicinal chemistry, 2016, 06-23, Volume: 59, Issue:12 Topics: Binding Sites; Cell Membrane; Dose-Response Relationship, Drug; Humans; Ligands; Models, Molecular; Molecular Structure; Receptors, Adrenergic, beta-2; Structure-Activity Relationship	2016
Central beta 1-adrenergic receptors are involved in CRF-induced defensive withdrawal. Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4 Topics: Animals; Atenolol; Behavior, Animal; Corticotropin-Releasing Hormone; Injections, Intraperitoneal; Injections, Intraventricular; Male; Propanolamines; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta	1990
Study of beta-adrenoceptors and beta-adrenergic responsiveness in cultured "preneoplastic-like" and neoplastic rat hepatocytes. General pharmacology, 1985, Volume: 16, Issue:3 Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Antagonists; Albuterol; Animals; Atenolol; Binding, Competitive; Cells, Cultured; Cyclic AMP; Epinephrine; Isoproterenol; Kinetics; Liver Neoplasms, Experimental; Norepinephrine; Precancerous Conditions; Propanolamines; Propranolol; Rats; Receptors, Adrenergic, beta	1985
Affinity and selectivity of beta-adrenoceptor antagonists in vitro. Journal of cardiovascular pharmacology, 1986, Volume: 8 Suppl 11 Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Betaxolol; Binding, Competitive; Bisoprolol; Propanolamines; Propranolol; Rats; Salivary Glands; Tritium	1986
Involvement of beta 3-adrenoceptor in the relaxation response in guinea pig taenia caecum. Japanese journal of pharmacology, 1994, Volume: 66, Issue:2 Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Binding, Competitive; Butoxamine; Cecum; Dose-Response Relationship, Drug; Epinephrine; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Microsomes; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phentolamine; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta	1994
Distribution of beta 2-like adrenergic receptors in the cnidarian Renilla koellikeri as revealed by autoradiography and in situ hybridization. Cell and tissue research, 1994, Volume: 278, Issue:2 Topics: Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Atenolol; Autoradiography; Cnidaria; Endoderm; In Situ Hybridization; Luminescent Measurements; Propanolamines; Receptors, Adrenergic, beta-2; Tritium	1994
Effects of chronic administration of bopindolol on the binding characteristics of cardiac alpha 1H-, alpha 1L-, beta 1- and beta 2-adrenoceptor subtypes in cardiac muscles of spontaneously hypertensive rats (SHR). Biological & pharmaceutical bulletin, 1996, Volume: 19, Issue:7 Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Hypertension; In Vitro Techniques; Membranes; Myocardium; Pindolol; Propanolamines; Propranolol; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2	1996
Pharmacological characteristics of BDTI, a new isoquinoline-derived beta 2-adrenoceptor agonist, in canine trachea and rat heart. Pharmacology, 1996, Volume: 53, Issue:1 Topics: Adrenergic beta-2 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Animals; Atenolol; Carbachol; Cells, Cultured; Dogs; Dose-Response Relationship, Drug; Female; Heart; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Myocardium; Propanolamines; Radioligand Assay; Rats; Rats, Wistar; Trachea; Tretoquinol	1996
Pharmacological analysis of atypical beta-adrenoceptors in the guinea pig gastric fundus using the beta(3)-adrenoceptor antagonist bupranolol. Pharmacology, 1999, Volume: 59, Issue:6 Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atenolol; Bupranolol; Butoxamine; Catecholamines; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Gastric Fundus; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle Relaxation; Norepinephrine; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-3	1999
Characterization of [3H]CGP 12177 binding to beta-adrenergic receptors in intact eel hepatocytes. General and comparative endocrinology, 2001, Volume: 121, Issue:3 Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Alprenolol; Anguilla; Animals; Atenolol; Binding Sites; Binding, Competitive; Butoxamine; Cell Count; Colforsin; Cyclic AMP; Epinephrine; Glucose; Guanosine 5'-O-(3-Thiotriphosphate); Hepatocytes; Kinetics; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tritium	2001