cgp 12177 and amibegron

cgp 12177 has been researched along with amibegron in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (50.00)18.2507
2000's5 (41.67)29.6817
2010's1 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blin, N; Camoin, L; Maigret, B; Strosberg, AD1
Benarese, M; Carruba, MO; Nisoli, E; Tonello, C1
Berlan, M; Carpéné, C; Galitzky, J; Lafontan, M; Portillo, M; Reverte, M1
Berlan, M; Galitzky, J; Lafontan, M; Langin, D; Montastruc, JL; Verwaerde, P1
Berdeaux, A; Bévérelli, F; Gauthier, C; Le Marec, H; Leblais, V; Rautureau, Y; Trochu, JN1
Kanda, Y; Kuroki, Y; Mizuno, K; Tomiyama, K; Watanabe, Y1
Aureggi, G; Croci, T; Ferla, G; Guagnini, F; Le Fur, G; Maffrand, JP; Manara, L; Mukenge, S1
Gibbs, ME; Summers, RJ1
Danner, I; Escande, D; Gauthier, C1
Balligand, JL; Donckier, JE; Gauthier, C; Heyndrickx, GR; Massart, PE; Van Mechelen, H1
Desfontis, JC; Gogny, M; Holopherne, D; Le Coz, O; Mallem, Y; Reculeau, O1
Christ, T; Kaumann, AJ; Klenowski, PM; Molenaar, P; Ravens, U1

Other Studies

12 other study(ies) available for cgp 12177 and amibegron

ArticleYear
Structural and conformational features determining selective signal transduction in the beta 3-adrenergic receptor.
    Molecular pharmacology, 1993, Volume: 44, Issue:6

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; CHO Cells; Cricetinae; GTP-Binding Proteins; Humans; Models, Molecular; Protein Conformation; Receptors, Adrenergic, beta; Signal Transduction; Structure-Activity Relationship

1993
Rat frontal cortex beta 1-adrenoceptors are activated by the beta 3-adrenoceptor agonists SR 58611A and SR 58878A but not by BRL 37344 or ICI 215,001.
    Journal of neurochemistry, 1995, Volume: 65, Issue:4

    Topics: Adipose Tissue, Brown; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Base Sequence; Cyclic AMP; Frontal Lobe; Imipramine; Male; Molecular Sequence Data; Oligonucleotide Probes; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; RNA, Messenger; Tetrahydronaphthalenes

1995
Coexistence of beta 1-, beta 2-, and beta 3-adrenoceptors in dog fat cells and their differential activation by catecholamines.
    The American journal of physiology, 1993, Volume: 264, Issue:3 Pt 1

    Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Catecholamines; Cell Membrane; Dogs; Dose-Response Relationship, Drug; Epinephrine; Ethanolamines; Isoproterenol; Norepinephrine; Procaterol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tetrahydronaphthalenes

1993
Lipolytic effects of conventional beta 3-adrenoceptor agonists and of CGP 12,177 in rat and human fat cells: preliminary pharmacological evidence for a putative beta 4-adrenoceptor.
    British journal of pharmacology, 1997, Volume: 122, Issue:6

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Dioxoles; Humans; Lipolysis; Male; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes

1997
Beta 3-adrenoceptor stimulation induces vasorelaxation mediated essentially by endothelium-derived nitric oxide in rat thoracic aorta.
    British journal of pharmacology, 1999, Volume: 128, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Cyclic GMP; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Nadolol; Nitric Oxide; Nitric Oxide Synthase; omega-N-Methylarginine; Phenylephrine; Propanolamines; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes; Vasoconstriction; Vasodilation

1999
Phosphorylation of extracellular signal-regulated kinases 1 and 2 in 3T3-L1 adipocytes by stimulation of beta(3)-adrenoceptor.
    European journal of pharmacology, 1999, Nov-26, Volume: 385, Issue:1

    Topics: 3T3 Cells; Adipocytes; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethanolamines; Flavonoids; Glycerol; Isoquinolines; Mice; Mitogen-Activated Protein Kinases; Phosphorylation; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Sulfonamides; Tetrahydronaphthalenes

1999
Functional assessment of beta adrenoceptor subtypes in human colonic circular and longitudinal (taenia coli) smooth muscle.
    Gut, 2000, Volume: 47, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Colon; Female; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Terbutaline; Tetrahydronaphthalenes

2000
Enhancement of memory consolidation in chicks by beta(3)-adrenoceptor agonists.
    European journal of pharmacology, 2001, Feb-16, Volume: 413, Issue:2-3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Avoidance Learning; Chickens; Discrimination Learning; Dose-Response Relationship, Drug; Ethanolamines; Female; Memory; Propanolamines; Propranolol; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes

2001
Beta(3)-adrenoceptors control Cl(-) conductance in rabbit nasal epithelium.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Agonists; Amiloride; Animals; Chlorides; Isoproterenol; Membrane Potentials; Nasal Mucosa; Propanolamines; Rabbits; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes

2001
Cardiovascular effects of beta 3-adrenoceptor stimulation in perinephritic hypertension.
    European journal of clinical investigation, 2001, Volume: 31, Issue:8

    Topics: Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Aorta; Atropine Derivatives; Blood Pressure; Bupranolol; Dogs; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Hexamethonium; Hypertension, Renal; Lipolysis; Myocardial Contraction; Nadolol; Propanolamines; Receptors, Adrenergic, beta-3; Tetrahydronaphthalenes; Time Factors

2001
Beta-adrenoceptor-mediated vascular relaxation in spontaneously hypertensive rats.
    Autonomic neuroscience : basic & clinical, 2005, Mar-31, Volume: 118, Issue:1-2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta; Tetrahydronaphthalenes

2005
Human atrial β(1L)-adrenoceptor but not β₃-adrenoceptor activation increases force and Ca(2+) current at physiological temperature.
    British journal of pharmacology, 2011, Volume: 162, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Atrial Appendage; Calcium Channels, L-Type; Calcium Signaling; Ethanolamines; Female; Humans; In Vitro Techniques; Kinetics; Male; Middle Aged; Myocardial Contraction; Myocytes, Cardiac; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Temperature; Tetrahydronaphthalenes

2011