Compounds > cgp 12177

cgp 12177 and alprenolol

cgp 12177 has been researched along with alprenolol in 19 studies

Research

Studies (19)

Timeframe	Studies, this research(%)	All Research%
pre-1990	10 (52.63)	18.7374
1990's	2 (10.53)	18.2507
2000's	7 (36.84)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Bultsma, T; Donné-Op den Kelder, GM; Rademaker, B; Timmerman, H	1
Baker, JG	1
Coury, A; Guyard, A; Rumigny, JF	1
Creese, I; Riva, MA	1
Korichneva, IL; Krasnikova, TL; Radiukhin, VA	1
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW	1
Affolter, H; Hertel, C; Jaeggi, K; Portenier, M; Staehelin, M	1
Wilkinson, DA; Wilkinson, M	1
Lang, PH; Lemmer, B	1
Arinze, IJ; Graham, SM; Kawai, Y; Yoshioka, H	1
Box, RJ; Staehelin, M	1
Marttila, T; Niina, O; Nikinmaa, M	1
Carlsson, B; Drvota, V; Häggblad, J; Sylvén, C; Wei, H	1
Capuzzo, A; Fabbri, E; Moon, TW; Selva, C	1
Horinouchi, T; Koike, K	1
Brahmadevara, N; MacDonald, A; Shaw, AM	1
Blum, JW; Carron, J; Hammon, HM; Morel, C	1
Desfontis, JC; Gogny, M; Le Coz, O; Mallem, MY; Reculeau, O	1
Hirouchi, M; Katsura, M; Ohkuma, S; Shibasaki, M; Tsujimura, A	1

Other Studies

19 other study(ies) available for cgp 12177 and alprenolol

Article	Year
Mapping of the beta 2-adrenoceptor on Chang liver cells. Differences between high- and low-affinity receptor states. Journal of medicinal chemistry, 1988, Volume: 31, Issue:6 Topics: Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Hydrogen Bonding; Iodocyanopindolol; Liver; Models, Molecular; Pindolol; Protein Conformation; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship	1988
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors. British journal of pharmacology, 2005, Volume: 144, Issue:3 Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3	2005
Characterization of beta-adrenoceptors in synaptoneurosomes from rat brain: [3H]dihydroalprenolol versus [3H]CGP 12177. Biochemical Society transactions, 1990, Volume: 18, Issue:3 Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Synaptosomes; Tritium	1990
Comparison of two putatively selective radioligands for labeling central nervous system beta-adrenergic receptors: inadequacy of [3H]dihydroalprenolol. Molecular pharmacology, 1989, Volume: 36, Issue:1 Topics: Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Kinetics; Male; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin	1989
[Dependence of kinetic constants of intact human lymphocyte beta2-adrenoreceptors on the nature of the radioligands used]. Biokhimiia (Moscow, Russia), 1989, Volume: 54, Issue:2 Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Ethylmaleimide; Humans; Isoproterenol; Kinetics; Lymphocytes; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Temperature	1989
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177. European journal of pharmacology, 1989, Aug-29, Volume: 167, Issue:3 Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta	1989
(-)-S-[3H]CGP-12177 and its use to determine the rate constants of unlabeled beta-adrenergic antagonists. Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:3 Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Cell Line; Computers; Glioma; Kinetics; Pindolol; Propanolamines; Stereoisomerism	1985
Beta-adrenergic [( 3H]CGP-12177) binding to brain slices and single intact pineal glands. Neurochemical research, 1985, Volume: 10, Issue:6 Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain; Cerebral Cortex; Cricetinae; In Vitro Techniques; Isoproterenol; Kinetics; Male; Mesocricetus; Phentolamine; Pineal Gland; Propanolamines; Rats; Rats, Inbred Strains; Timolol	1985
Evidence for two specific affinity states of 3H-antagonist binding to cardiac beta-adrenergic receptors and influence of Gpp(NH)p. Journal of cyclic nucleotide and protein phosphorylation research, 1985, Volume: 10, Issue:4 Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Myocardium; Propanolamines; Rats; Receptors, Adrenergic, beta	1985
Beta-adrenergic receptors in guinea-pig liver plasma membranes and thermal lability of [3H]dihydroalprenolol binding sites. Biochemical pharmacology, 1986, Dec-15, Volume: 35, Issue:24 Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Guinea Pigs; Hot Temperature; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Virulence Factors, Bordetella	1986
Bromoacetylalprenololmenthane binding to beta-receptors modulates the rate of hormone-induced internalization but not desensitization in S49 cells. FEBS letters, 1987, Apr-20, Volume: 214, Issue:2 Topics: Alprenolol; Cell Line; Cell Membrane; Cyclic AMP; Isoproterenol; Kinetics; Lymphoma; Propanolamines; Receptors, Adrenergic, beta	1987
Binding of beta-adrenergic antagonists 3H-DHA and 3H-CGP 12177 to intact rainbow trout (Salmo gairdneri) and carp (Cyprinus carpio) red blood cells. General and comparative endocrinology, 1988, Volume: 70, Issue:3 Topics: Alprenolol; Animals; Carps; Cyprinidae; Dihydroalprenolol; Erythrocytes; Ligands; Membrane Lipids; Propanolamines; Salmonidae; Trout	1988
Beta-adrenergic receptor function in cultured AT-1 cardiomyocytes. Biochemical and biophysical research communications, 1995, Feb-06, Volume: 207, Issue:1 Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Calcium; Cell Line; Cyclic AMP; Cytosol; Heart; Heart Neoplasms; Isoproterenol; Kinetics; Mice; Mice, Transgenic; Myocardial Contraction; Myocardium; Potassium; Propanolamines; Receptors, Adrenergic, beta; Time Factors; Tumor Cells, Cultured	1995
Characterization of [3H]CGP 12177 binding to beta-adrenergic receptors in intact eel hepatocytes. General and comparative endocrinology, 2001, Volume: 121, Issue:3 Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Alprenolol; Anguilla; Animals; Atenolol; Binding Sites; Binding, Competitive; Butoxamine; Cell Count; Colforsin; Cyclic AMP; Epinephrine; Glucose; Guanosine 5'-O-(3-Thiotriphosphate); Hepatocytes; Kinetics; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tritium	2001
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum. European journal of pharmacology, 2001, Mar-23, Volume: 416, Issue:1-2 Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism	2001
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta. British journal of pharmacology, 2004, Volume: 142, Issue:4 Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction	2004
Effects of dexamethasone and colostrum feeding on mRNA levels and binding capacities of beta-adrenergic receptors in the liver of neonatal calves. Domestic animal endocrinology, 2005, Volume: 28, Issue:3 Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Animals, Newborn; Binding, Competitive; Cattle; Colostrum; Dexamethasone; Diet; Glucocorticoids; Liver; Polymerase Chain Reaction; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger	2005
Low-affinity state beta1-adrenoceptor-induced vasodilation in SHR. Peptides, 2005, Volume: 26, Issue:8 Topics: Adrenergic beta-1 Receptor Agonists; Alprenolol; Animals; Aorta; Blood Pressure; Dose-Response Relationship, Drug; Enalapril; Losartan; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta-1; Vasodilation	2005
Expression of beta-adrenergic receptor up-regulation is mediated by two different processes. Brain research, 2006, Sep-27, Volume: 1112, Issue:1 Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Blotting, Western; Cells, Cultured; Cerebral Cortex; Cycloheximide; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Mice; Nadolol; Neurons; Propanolamines; Protein Binding; Protein Synthesis Inhibitors; Receptors, Adrenergic, beta; RNA, Messenger; Signal Transduction; Time Factors; Tritium; Up-Regulation	2006