cgp 12177 has been researched along with alprenolol in 19 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 10 (52.63) | 18.7374 |
1990's | 2 (10.53) | 18.2507 |
2000's | 7 (36.84) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bultsma, T; Donné-Op den Kelder, GM; Rademaker, B; Timmerman, H | 1 |
Baker, JG | 1 |
Coury, A; Guyard, A; Rumigny, JF | 1 |
Creese, I; Riva, MA | 1 |
Korichneva, IL; Krasnikova, TL; Radiukhin, VA | 1 |
Cheetham, SC; Crompton, MR; De Paermentier, F; Horton, RW | 1 |
Affolter, H; Hertel, C; Jaeggi, K; Portenier, M; Staehelin, M | 1 |
Wilkinson, DA; Wilkinson, M | 1 |
Lang, PH; Lemmer, B | 1 |
Arinze, IJ; Graham, SM; Kawai, Y; Yoshioka, H | 1 |
Box, RJ; Staehelin, M | 1 |
Marttila, T; Niina, O; Nikinmaa, M | 1 |
Carlsson, B; Drvota, V; Häggblad, J; Sylvén, C; Wei, H | 1 |
Capuzzo, A; Fabbri, E; Moon, TW; Selva, C | 1 |
Horinouchi, T; Koike, K | 1 |
Brahmadevara, N; MacDonald, A; Shaw, AM | 1 |
Blum, JW; Carron, J; Hammon, HM; Morel, C | 1 |
Desfontis, JC; Gogny, M; Le Coz, O; Mallem, MY; Reculeau, O | 1 |
Hirouchi, M; Katsura, M; Ohkuma, S; Shibasaki, M; Tsujimura, A | 1 |
19 other study(ies) available for cgp 12177 and alprenolol
Article | Year |
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Mapping of the beta 2-adrenoceptor on Chang liver cells. Differences between high- and low-affinity receptor states.
Topics: Cell Membrane; Cells, Cultured; Guanylyl Imidodiphosphate; Hydrogen Bonding; Iodocyanopindolol; Liver; Models, Molecular; Pindolol; Protein Conformation; Receptors, Adrenergic, beta; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Structure-Activity Relationship | 1988 |
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors.
Topics: Adrenergic beta-1 Receptor Agonists; Adrenergic beta-2 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Algorithms; Animals; Cell Line; CHO Cells; Cricetinae; Dioxoles; Humans; Propanolamines; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3 | 2005 |
Characterization of beta-adrenoceptors in synaptoneurosomes from rat brain: [3H]dihydroalprenolol versus [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Propanolamines; Radioligand Assay; Rats; Receptors, Adrenergic, beta; Synaptosomes; Tritium | 1990 |
Comparison of two putatively selective radioligands for labeling central nervous system beta-adrenergic receptors: inadequacy of [3H]dihydroalprenolol.
Topics: Alprenolol; Animals; Brain Chemistry; Dihydroalprenolol; Guanosine Triphosphate; Isoproterenol; Kinetics; Male; Propanolamines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, Serotonin | 1989 |
[Dependence of kinetic constants of intact human lymphocyte beta2-adrenoreceptors on the nature of the radioligands used].
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Ethylmaleimide; Humans; Isoproterenol; Kinetics; Lymphocytes; Pindolol; Propanolamines; Radioligand Assay; Receptors, Adrenergic, beta; Temperature | 1989 |
Beta-adrenoceptors in human brain labelled with [3H]dihydroalprenolol and [3H]CGP 12177.
Topics: Adrenergic beta-Antagonists; Alprenolol; Binding, Competitive; Brain Chemistry; Dihydroalprenolol; Humans; Imidazoles; In Vitro Techniques; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Practolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta | 1989 |
(-)-S-[3H]CGP-12177 and its use to determine the rate constants of unlabeled beta-adrenergic antagonists.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Cell Line; Computers; Glioma; Kinetics; Pindolol; Propanolamines; Stereoisomerism | 1985 |
Beta-adrenergic [( 3H]CGP-12177) binding to brain slices and single intact pineal glands.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Brain; Cerebral Cortex; Cricetinae; In Vitro Techniques; Isoproterenol; Kinetics; Male; Mesocricetus; Phentolamine; Pineal Gland; Propanolamines; Rats; Rats, Inbred Strains; Timolol | 1985 |
Evidence for two specific affinity states of 3H-antagonist binding to cardiac beta-adrenergic receptors and influence of Gpp(NH)p.
Topics: Alprenolol; Animals; Binding, Competitive; Dihydroalprenolol; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Isoproterenol; Kinetics; Male; Myocardium; Propanolamines; Rats; Receptors, Adrenergic, beta | 1985 |
Beta-adrenergic receptors in guinea-pig liver plasma membranes and thermal lability of [3H]dihydroalprenolol binding sites.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Alprenolol; Animals; Binding, Competitive; Cell Membrane; Cholera Toxin; Dihydroalprenolol; Guanylyl Imidodiphosphate; Guinea Pigs; Hot Temperature; Iodocyanopindolol; Isoproterenol; Liver; Male; Pindolol; Propanolamines; Receptors, Adrenergic, beta; Virulence Factors, Bordetella | 1986 |
Bromoacetylalprenololmenthane binding to beta-receptors modulates the rate of hormone-induced internalization but not desensitization in S49 cells.
Topics: Alprenolol; Cell Line; Cell Membrane; Cyclic AMP; Isoproterenol; Kinetics; Lymphoma; Propanolamines; Receptors, Adrenergic, beta | 1987 |
Binding of beta-adrenergic antagonists 3H-DHA and 3H-CGP 12177 to intact rainbow trout (Salmo gairdneri) and carp (Cyprinus carpio) red blood cells.
Topics: Alprenolol; Animals; Carps; Cyprinidae; Dihydroalprenolol; Erythrocytes; Ligands; Membrane Lipids; Propanolamines; Salmonidae; Trout | 1988 |
Beta-adrenergic receptor function in cultured AT-1 cardiomyocytes.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Calcium; Cell Line; Cyclic AMP; Cytosol; Heart; Heart Neoplasms; Isoproterenol; Kinetics; Mice; Mice, Transgenic; Myocardial Contraction; Myocardium; Potassium; Propanolamines; Receptors, Adrenergic, beta; Time Factors; Tumor Cells, Cultured | 1995 |
Characterization of [3H]CGP 12177 binding to beta-adrenergic receptors in intact eel hepatocytes.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Alprenolol; Anguilla; Animals; Atenolol; Binding Sites; Binding, Competitive; Butoxamine; Cell Count; Colforsin; Cyclic AMP; Epinephrine; Glucose; Guanosine 5'-O-(3-Thiotriphosphate); Hepatocytes; Kinetics; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Tritium | 2001 |
Functional properties of atypical beta-adrenoceptors on the guinea pig duodenum.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Albuterol; Alprenolol; Animals; Bupranolol; Carteolol; Clenbuterol; Dobutamine; Dopamine; Dose-Response Relationship, Drug; Duodenum; Epinephrine; Ethanolamines; Fenoterol; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Nadolol; Norepinephrine; Phenylephrine; Pindolol; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Stereoisomerism | 2001 |
ALpha1-adrenoceptor antagonist properties of CGP 12177A and other beta-adrenoceptor ligands: evidence against beta(3)- or atypical beta-adrenoceptors in rat aorta.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic beta-Antagonists; Alprenolol; Animals; Aorta, Thoracic; Binding Sites; Bupranolol; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle, Smooth, Vascular; Phenylephrine; Pindolol; Prazosin; Propanolamines; Propranolol; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-3; Tritium; United Kingdom; Vasoconstriction | 2004 |
Effects of dexamethasone and colostrum feeding on mRNA levels and binding capacities of beta-adrenergic receptors in the liver of neonatal calves.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Animals, Newborn; Binding, Competitive; Cattle; Colostrum; Dexamethasone; Diet; Glucocorticoids; Liver; Polymerase Chain Reaction; Propanolamines; Propranolol; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger | 2005 |
Low-affinity state beta1-adrenoceptor-induced vasodilation in SHR.
Topics: Adrenergic beta-1 Receptor Agonists; Alprenolol; Animals; Aorta; Blood Pressure; Dose-Response Relationship, Drug; Enalapril; Losartan; Male; Muscle Relaxation; Pindolol; Propanolamines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, beta-1; Vasodilation | 2005 |
Expression of beta-adrenergic receptor up-regulation is mediated by two different processes.
Topics: Adrenergic beta-Antagonists; Alprenolol; Animals; Blotting, Western; Cells, Cultured; Cerebral Cortex; Cycloheximide; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Mice; Nadolol; Neurons; Propanolamines; Protein Binding; Protein Synthesis Inhibitors; Receptors, Adrenergic, beta; RNA, Messenger; Signal Transduction; Time Factors; Tritium; Up-Regulation | 2006 |