Page last updated: 2024-08-24

ceronapril and proline

ceronapril has been researched along with proline in 42 studies

Research

Studies (42)

TimeframeStudies, this research(%)All Research%
pre-19905 (11.90)18.7374
1990's34 (80.95)18.2507
2000's3 (7.14)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, BZ; Mendelsohn, FA1
Feldon, J; Rawlins, JN; Smith, AD; Weiner, I1
Kaneko, K; Osugi, S; Shimamura, K; Sunano, S; Yamamoto, K1
Barnes, JM; Barnes, NM; Costall, B; Coughlan, J; Kelly, ME; Naylor, RJ; Tomkins, DM; Williams, TJ1
Brennan, J; Mantha, S; Stouffer, B; Tsay, HM; Tu, JI; Turabi, N1
Katsumura, H; Ogawa, N; Ohara, N; Ono, H; Takizawa, M; Yokota, S1
Grupp, LA1
Chikugo, T; Morita, N; Ohta, Y; Okamoto, K; Shiokawa, H1
Barnes, NM; Costall, B; Egli, P; Horovitz, ZP; Ironside, JW; Naylor, RJ; Williams, TJ2
Barnes, NM; Cheng, CH; Costall, B; Naylor, RJ; Williams, TJ; Wischik, CM1
DeForrest, JM; Hammerstone, S; Harvey, C; Karanewsky, D; Powell, JR; Scalese, R; Waldron, TL1
Chikugo, T; Hamada, Y; Morita, N; Ohta, Y; Okamoto, K; Shiokawa, H1
Konishi, C; Ohara, N; Ono, H; Shukunobe, K; Yokota, S1
Costall, B; Domeney, AM; Gerrard, PA; Horovitz, ZP; Kelly, ME; Naylor, RJ; Tomkins, DM1
Hiwada, K; Inoue, Y; Kokubu, T1
Badia, MC; Cushman, DW; DeForrest, JM; Dejneka, T; Karanewsky, DS; Lee, VG; Loots, MJ; Petrillo, EW1
Cushman, DW; DeForrest, JM; Fung, WC; Grover, GJ; Harvey, CM; Mitch, SL; Scalese, RJ; Wang, FL1
Amidon, GL; Friedman, DI1
Costall, B; Coughlan, J; Horovitz, ZP; Kelly, ME; Naylor, RJ; Tomkins, DM1
Brittain, HG; Cohen, AI; Ivashkiv, E; Kadin, H1
Badia, MC; Cushman, DW; DeForrest, JM; Dejneka, T; Karanewsky, DS; Loots, MJ; Perri, MG; Petrillo, EW; Powell, JR1
Higashimori, K; Katahira, K; Kohara, K; Mikami, H; Moriguchi, A; Morishita, R; Nagano, M; Ogihara, T; Okuda, N; Otsuka, A1
Higaki, J; Katsuya, T; Mikami, H; Morishita, R; Nakamura, F; Ogihara, T; Rakugi, H; Tomita, N; Yu, H1
Minck, KO; Raddatz, P; Rippmann, F; Schmitges, CJ1
Fujishima, M; Ibayashi, S; Nagao, T; Sadoshima, S1
Ikeda, M; Kishi, K1
Cutler, NR; Markowitz, J; Mickelson, W; Repetti, S; Sramek, JJ; Sudilovsky, A; Veroff, AE; Wardle, T1
Fujii, K; Fujishima, M; Ibayashi, S; Ooboshi, H; Sadoshima, S1
Paulson, OB; Torup, M; Waldemar, G1
Doi, Y; Kagimoto, M; Kato, K; Kawasaki, K; Koga, S; Sakai, K; Sakaue, A; Sasaki, J; Takada, K; Takii, M1
Bathala, MS; Chong, S; Dando, SA; Kripalani, KJ; Marino, AM; Morrison, RA1
Brass, EP; Brennan, JJ; Cutler, NR; Kurtz, NM; Luna, A; Mena, I; Sramek, JJ1
Chong, S; Irwin, WJ; Marino, AM; Moore, VA; Morrison, RA; Timmins, P; Wasserman, MA1
Chalas, A; Conway, EL1
Chikugo, TA; Hamada, Y; Niisato, E; Ohta, Y; Okamoto, K; Otori, T; Suzuki, T1
Chichibu, S; Chikugo, T; Ohta, Y; Suzuki, T1
Akhtar, S; Brown, T; Dunnion, DJ; Irwin, WJ; Moore, VA1
Costall, B; Naylor, RJ1
Chong, S; Dando, SA; Irwin, WJ; Moore, VA; Morrison, RA; Timmins, P1
Chong, S; Dando, SA; Irwin, WJ; Lambert, PA; Moore, VA; Morrison, RA; Timmins, P1
Kinsella, BT; O'Meara, SJ1

Trials

3 trial(s) available for ceronapril and proline

ArticleYear
A pilot clinical trial of the angiotensin-converting enzyme inhibitor ceranapril in Alzheimer disease.
    Alzheimer disease and associated disorders, 1993,Summer, Volume: 7, Issue:2

    Topics: Aged; Alzheimer Disease; Angiotensin-Converting Enzyme Inhibitors; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Male; Middle Aged; Neuropsychological Tests; Organophosphorus Compounds; Pilot Projects; Proline

1993
Hypotensive effects and influence on serum lipids of SQ29,852, a new angiotensin converting enzyme inhibitor, in patients with essential hypertension: a comparison with atenolol.
    International journal of clinical pharmacology, therapy, and toxicology, 1993, Volume: 31, Issue:2

    Topics: Adult; Aged; Analysis of Variance; Angiotensin-Converting Enzyme Inhibitors; Apolipoproteins; Arteriosclerosis; Atenolol; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Lipids; Lipoproteins; Male; Middle Aged; Organophosphorus Compounds; Phosphatidylcholine-Sterol O-Acyltransferase; Proline

1993
Effect of the ACE inhibitor ceronapril on cerebral blood flow in hypertensive patients.
    The Annals of pharmacotherapy, 1996, Volume: 30, Issue:6

    Topics: Aged; Angiotensin-Converting Enzyme Inhibitors; Blood Pressure; Cerebrovascular Circulation; Chlorthalidone; Diuretics; Drug Therapy, Combination; Female; Homeostasis; Humans; Hypertension; Male; Middle Aged; Organophosphorus Compounds; Proline; Xenon Radioisotopes

1996

Other Studies

39 other study(ies) available for ceronapril and proline

ArticleYear
Effect of acute and chronic administration of ceronapril on angiotensin converting enzyme in plasma, kidney, lung, brain regions and cerebrospinal fluid of rats.
    Neuropharmacology, 1992, Volume: 31, Issue:9

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Autoradiography; Brain; Iodine Radioisotopes; Kidney; Lung; Male; Organophosphorus Compounds; Peptidyl-Dipeptidase A; Proline; Rats; Rats, Sprague-Dawley

1992
A neuroleptic-like effect of ceronapril on latent inhibition.
    Neuroscience, 1992, Volume: 49, Issue:2

    Topics: Acoustic Stimulation; Animals; Antipsychotic Agents; Conditioning, Operant; Dextroamphetamine; Emotions; Handling, Psychological; Male; Organophosphorus Compounds; Proline; Rats; Rats, Wistar

1992
Effects of chronic treatment with SQ29852 on spontaneous smooth muscle tone and endothelium-dependent relaxation in aorta of stroke-prone spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:4

    Topics: Acetylcholine; Angiotensin-Converting Enzyme Inhibitors; Animals; Aorta; Blood Pressure; Captopril; Endothelium, Vascular; Hypertension; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Organophosphorus Compounds; Proline; Rats; Rats, Inbred SHR

1992
Angiotensin-converting enzyme inhibition, angiotensin, and cognition.
    Journal of cardiovascular pharmacology, 1992, Volume: 19 Suppl 6

    Topics: Acetylcholine; Angiotensin II; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Behavior, Animal; Brain; Catecholamines; Cognition; Female; Habituation, Psychophysiologic; Humans; Mice; Organophosphorus Compounds; Potassium; Proline; Rats; Scopolamine

1992
Radioimmunoassay for ceronapril, a new angiotensin-converting enzyme inhibitor, and its application to a pharmacokinetic study in healthy male volunteers.
    Therapeutic drug monitoring, 1992, Volume: 14, Issue:3

    Topics: Adult; Angiotensin-Converting Enzyme Inhibitors; Blood Proteins; Drug Tolerance; Glutaral; Humans; Iodine Radioisotopes; Male; Organophosphorus Compounds; Proline; Protein Binding; Radioimmunoassay; Reference Standards; Thyroglobulin

1992
Hypotensive effect of a phosphorus-containing novel angiotensin converting enzyme inhibitor, (S)-1-[6-amino-2[[hydroxy(4-phenylbutyl)phosphinyl] oxy]-1-oxohexyl]-L-proline (SQ 29,852) in conscious hypertensive dogs.
    Journal of pharmacobio-dynamics, 1992, Volume: 15, Issue:6

    Topics: Administration, Oral; Angiotensin-Converting Enzyme Inhibitors; Angiotensins; Animals; Dogs; Enalapril; Female; Hypertension; Organophosphorus Compounds; Proline; Renin

1992
Effects of angiotensin II and an angiotensin converting enzyme inhibitor on alcohol intake in P and NP rats.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:1

    Topics: Alcohol Drinking; Angiotensin II; Angiotensin-Converting Enzyme Inhibitors; Animals; Dose-Response Relationship, Drug; Male; Organophosphorus Compounds; Proline; Rats; Renin-Angiotensin System; Species Specificity

1992
Chronic treatment with captopril, SQ29,852, hydralazine and a 33% fish meal diet in malignant stroke-prone spontaneously hypertensive rats.
    Journal of hypertension, 1991, Volume: 9, Issue:12

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Body Weight; Captopril; Cerebrovascular Disorders; Fish Products; Hydralazine; Hypertension, Malignant; Life Expectancy; Male; Organophosphorus Compounds; Proline; Rats; Rats, Inbred SHR; Rats, Inbred WKY

1991
Characterisation of [3H]ceranapril recognition sites in rat and human brain tissue.
    Neuropharmacology, 1991, Volume: 30, Issue:8

    Topics: Adult; Aged; Angiotensin-Converting Enzyme Inhibitors; Animals; Binding Sites; Brain; Captopril; Enalapril; Female; Fosinopril; Humans; Kinetics; Lisinopril; Male; Middle Aged; Organophosphorus Compounds; Proline; Rats; Thiorphan

1991
Angiotensin converting enzyme density is increased in temporal cortex from patients with Alzheimer's disease.
    European journal of pharmacology, 1991, Aug-06, Volume: 200, Issue:2-3

    Topics: Aged; Alzheimer Disease; Angiotensin-Converting Enzyme Inhibitors; Captopril; Cerebellum; Female; Frontal Lobe; Humans; Male; Organophosphorus Compounds; Peptidyl-Dipeptidase A; Proline; Temporal Lobe; Tritium

1991
Ceranapril (SQ 29,852), an orally active inhibitor of angiotensin converting enzyme (ACE).
    Journal of cardiovascular pharmacology, 1990, Volume: 16, Issue:1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Captopril; Dogs; Female; Hypertension; Hypertension, Renovascular; Lung; Macaca fascicularis; Male; Nephrectomy; Organophosphorus Compounds; Proline; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Renal Circulation; Species Specificity

1990
Therapy and prevention of hypertension of M-SHRSP.
    Clinical and experimental hypertension. Part A, Theory and practice, 1991, Volume: 13, Issue:5

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Captopril; Cerebrovascular Disorders; Diet; Disease Models, Animal; Disease Susceptibility; Fish Flour; Hydralazine; Hypertension, Malignant; Male; Organophosphorus Compounds; Proline; Rats; Rats, Inbred SHR

1991
Pharmacology of a phosphorus-containing novel angiotensin converting enzyme inhibitor, SQ 29 852 in anesthetized dogs.
    Journal of pharmacobio-dynamics, 1991, Volume: 14, Issue:12

    Topics: Anesthesia; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Flow Velocity; Captopril; Dogs; Female; Hemodynamics; Infusions, Intravenous; Male; Organophosphorus Compounds; Proline; Vascular Resistance; Vasodilation

1991
Effects of captopril and SQ29,852 on anxiety-related behaviours in rodent and marmoset.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Anxiety; Behavior, Animal; Callitrichinae; Captopril; Diazepam; Drug Interactions; Female; Male; Mice; Organophosphorus Compounds; Proline; Rats; Species Specificity; Substance Withdrawal Syndrome

1990
Effect of SQ29,852, a new angiotensin converting enzyme (ACE) inhibitor with a phosphonic acid group, on the activity of angiotensin converting enzyme from human kidney.
    General pharmacology, 1990, Volume: 21, Issue:4

    Topics: Angiotensin-Converting Enzyme Inhibitors; Captopril; Enalapril; Enalaprilat; Humans; Kidney; Kinetics; Organophosphorus Compounds; Peptidyl-Dipeptidase A; Proline; Protease Inhibitors

1990
The ACE inhibitor [3H]SQ29,852 identifies a high affinity recognition site located in the human temporal cortex.
    Brain research bulletin, 1990, Volume: 25, Issue:1

    Topics: Adult; Aged; Angiotensin-Converting Enzyme Inhibitors; Binding Sites; Cerebral Cortex; Humans; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Male; Middle Aged; Organophosphorus Compounds; Proline; Temporal Lobe

1990
(Phosphinyloxy)acyl amino acid inhibitors of angiotensin converting enzyme. 2. Terminal amino acid analogues of (S)-1-[6-amino-2 [[hydroxy(4-phenylbutyl)phosphinyl]oxy]-1-oxohexyl]-L-proline.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:5

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Chemical Phenomena; Chemistry; Indoles; Male; Organophosphorus Compounds; Proline; Rabbits; Rats; Rats, Inbred Strains; Stereoisomerism; Structure-Activity Relationship

1990
Comparisons in vitro, ex vivo, and in vivo of the actions of seven structurally diverse inhibitors of angiotensin converting enzyme (ACE).
    British journal of clinical pharmacology, 1989, Volume: 28 Suppl 2

    Topics: Administration, Oral; Angiotensin-Converting Enzyme Inhibitors; Animals; Bridged Bicyclo Compounds; Captopril; Chemotherapy, Cancer, Regional Perfusion; Dose-Response Relationship, Drug; Enalapril; Fosinopril; Heart; Hypertension; Lisinopril; Male; Organophosphorus Compounds; Proline; Ramipril; Rats; Time Factors; Tissue Distribution

1989
Intestinal absorption mechanism of dipeptide angiotensin converting enzyme inhibitors of the lysyl-proline type: lisinopril and SQ 29,852.
    Journal of pharmaceutical sciences, 1989, Volume: 78, Issue:12

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Cephradine; Chromatography, High Pressure Liquid; Enalapril; In Vitro Techniques; Intestinal Absorption; Kinetics; Lisinopril; Organophosphorus Compounds; Proline; Rats; Spectrophotometry, Ultraviolet

1989
The effects of ACE inhibitors captopril and SQ29,852 in rodent tests of cognition.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:3

    Topics: Age Factors; Angiotensin-Converting Enzyme Inhibitors; Animals; Behavior, Animal; Captopril; Cognition; Drug Interactions; Habituation, Psychophysiologic; Male; Mice; Organophosphorus Compounds; Proline; Rats; Scopolamine; Time Factors

1989
Body fluid analysis of a phosphonic acid angiotensin-converting enzyme inhibitor using high-performance liquid chromatography and post-column derivatization with o-phthalaldehyde.
    Journal of chromatography, 1989, Jan-27, Volume: 487, Issue:1

    Topics: Chemical Phenomena; Chemistry; Chromatography, High Pressure Liquid; Humans; Indicators and Reagents; o-Phthalaldehyde; Organophosphorus Compounds; Proline; Spectrometry, Fluorescence

1989
(Phosphinyloxy)acyl amino acid inhibitors of angiotensin converting enzyme (ACE). 1. Discovery of (S)-1-[6-amino-2-[[hydroxy(4-phenylbutyl)phosphinyl]oxy]-1-oxohexyl]-L -proline a novel orally active inhibitor of ACE.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:1

    Topics: Administration, Oral; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Indicators and Reagents; Lung; Magnetic Resonance Spectroscopy; Male; Optical Rotation; Organophosphorus Compounds; Proline; Rabbits; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1988
Differential control of vascular tone and heart rate by different amino acid neurotransmitters in the rostral ventrolateral medulla of the rat.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:7

    Topics: Anesthesia; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Heart Rate; Injections; Male; Medulla Oblongata; Microdialysis; Muscle Tonus; Muscle, Smooth, Vascular; Neurotransmitter Agents; Nitroglycerin; Organophosphorus Compounds; Proline; Rats; Rats, Wistar

1994
Differential regulation of brain angiotensin II in genetically hypertensive and normotensive rats after nephrectomy.
    Blood pressure, 1994, Volume: 3, Issue:4

    Topics: Angiotensin II; Animals; Blood Pressure; Brain Chemistry; Hypertension; Male; Nephrectomy; Organophosphorus Compounds; Proline; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Renin; Renin-Angiotensin System

1994
Non-peptide renin inhibitors containing 2-(((3-phenylpropyl)phosphoryl)oxy)alkanoic acid moieties as P2-P3 replacements.
    Journal of medicinal chemistry, 1994, Feb-18, Volume: 37, Issue:4

    Topics: Amino Acid Sequence; Angiotensin-Converting Enzyme Inhibitors; Animals; Binding Sites; Blood Pressure; Cathepsin D; Female; Humans; Macaca fascicularis; Models, Molecular; Molecular Sequence Data; Organophosphorus Compounds; Pepsin A; Proline; Renin; Stereoisomerism; Structure-Activity Relationship

1994
Inhibition of angiotensin-converting enzyme modulates the autoregulation of regional cerebral blood flow in hypertensive rats.
    Hypertension (Dallas, Tex. : 1979), 1994, Volume: 23, Issue:6 Pt 1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Captopril; Cerebrovascular Circulation; Homeostasis; Hypertension; Male; Organophosphorus Compounds; Proline; Rats; Rats, Inbred SHR

1994
Chronic effects of SQ29,852, a new angiotensin converting enzyme (ACE) inhibitor with a phosphonic acid group, in experimental hypertensive rats.
    General pharmacology, 1993, Volume: 24, Issue:4

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Blood Pressure; Captopril; Enalapril; Hypertension, Renovascular; Male; Organophosphorus Compounds; Proline; Rats; Rats, Inbred SHR

1993
Angiotensin converting enzyme inhibitors attenuate ischemic brain metabolism in hypertensive rats.
    Stroke, 1993, Volume: 24, Issue:10

    Topics: Adenosine Triphosphate; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Brain; Captopril; Cerebrovascular Circulation; Female; Ischemic Attack, Transient; Lactates; Organophosphorus Compounds; Parietal Lobe; Proline; Pyruvates; Rats; Rats, Inbred SHR; Regional Blood Flow

1993
Ceranapril and cerebral blood flow autoregulation.
    Journal of hypertension, 1993, Volume: 11, Issue:4

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Cerebrovascular Circulation; Homeostasis; Hypertension; Male; Organophosphorus Compounds; Proline; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Time Factors

1993
Distribution of the dipeptide transporter system along the gastrointestinal tract of rats based on absorption of a stable and specific probe, SQ-29852.
    Journal of pharmaceutical sciences, 1996, Volume: 85, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Digestive System; Dipeptides; Dose-Response Relationship, Drug; Male; Organophosphorus Compounds; Proline; Rats; Rats, Sprague-Dawley

1996
Suitability of enalapril as a probe of the dipeptide transporter system: in vitro and in vivo studies.
    Pharmaceutical research, 1996, Volume: 13, Issue:7

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Biological Transport; Caco-2 Cells; Cefaclor; Dipeptides; Dogs; Dose-Response Relationship, Drug; Enalapril; Humans; In Vitro Techniques; Intestinal Absorption; Jejunum; Male; Models, Biological; Organophosphorus Compounds; Permeability; Proline; Rats

1996
No evidence for involvement of angiotensin II in spatial learning in water maze in rats.
    Behavioural brain research, 1996, Volume: 81, Issue:1-2

    Topics: Angiotensin II; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Biphenyl Compounds; Cholinergic Antagonists; Diazepam; GABA Modulators; Imidazoles; Injections, Intraventricular; Losartan; Maze Learning; Memory; Organophosphorus Compounds; Proline; Psychomotor Performance; Rats; Renin; Scopolamine; Tetrazoles

1996
Ocular fundus changes in malignant or precocious stroke-prone spontaneously hypertensive rats after administration of antihypertensive drugs.
    Clinical and experimental pharmacology & physiology. Supplement, 1995, Volume: 22, Issue:1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Arterioles; Blood Pressure; Calcium Channel Blockers; Cerebrovascular Disorders; Dihydropyridines; Fundus Oculi; Histocytochemistry; Hypertension; Male; Nitrobenzenes; Organophosphorus Compounds; Piperazines; Proline; Rats; Rats, Inbred SHR; Rats, Inbred WKY

1995
Electroencephalographic evaluation of the therapeutic efficiency of antihypertensive agents on M-SHRSP.
    Clinical and experimental pharmacology & physiology. Supplement, 1995, Volume: 22, Issue:1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Antihypertensive Agents; Blood Pressure; Body Weight; Calcium Channel Blockers; Dihydropyridines; Electroencephalography; Hypertension, Malignant; Longevity; Male; Nitrobenzenes; Organophosphorus Compounds; Piperazines; Proline; Rats; Rats, Inbred SHR

1995
Interaction of oligonucleotide-conjugates with the dipeptide transporter system in Caco-2 cells.
    Biochemical pharmacology, 1997, May-09, Volume: 53, Issue:9

    Topics: Angiotensin-Converting Enzyme Inhibitors; Biological Transport; Caco-2 Cells; Dipeptides; Dose-Response Relationship, Drug; Glyceryl Ethers; Humans; Oligodeoxyribonucleotides; Organophosphorus Compounds; Proline; Thionucleotides; Vitamin E

1997
The influence of 5-HT2 and 5-HT4 receptor antagonists to modify drug induced disinhibitory effects in the mouse light/dark test.
    British journal of pharmacology, 1997, Volume: 122, Issue:6

    Topics: Animals; Avoidance Learning; Behavior, Animal; Benzodiazepinones; Darkness; Devazepide; Diazepam; Drug Antagonism; Fenclonine; Indoles; Light; Losartan; Male; Meglumine; Mice; Organophosphorus Compounds; Proline; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Ritanserin; Serotonin Antagonists; Sulfonamides

1997
A rapid screening system to determine drug affinities for the intestinal dipeptide transporter 1: system characterisation.
    International journal of pharmaceutics, 2000, Dec-04, Volume: 210, Issue:1-2

    Topics: Algorithms; Angiotensin-Converting Enzyme Inhibitors; Anti-Bacterial Agents; Caco-2 Cells; Cadherins; Carrier Proteins; Dipeptides; Drug Evaluation, Preclinical; Humans; Kinetics; Lactams; Membrane Transport Proteins; Organophosphorus Compounds; Proline; Substrate Specificity

2000
A rapid screening system to determine drug affinities for the intestinal dipeptide transporter 2: affinities of ACE inhibitors.
    International journal of pharmaceutics, 2000, Dec-04, Volume: 210, Issue:1-2

    Topics: Algorithms; Angiotensin-Converting Enzyme Inhibitors; ATP Binding Cassette Transporter, Subfamily B, Member 2; ATP-Binding Cassette Transporters; Caco-2 Cells; Culture Media; Dipeptides; Drug Evaluation, Preclinical; Humans; Models, Biological; Organophosphorus Compounds; Proline; Structure-Activity Relationship

2000
The effect of the farnesyl protein transferase inhibitor SCH66336 on isoprenylation and signalling by the prostacyclin receptor.
    The Biochemical journal, 2005, Feb-15, Volume: 386, Issue:Pt 1

    Topics: Adrenergic beta-Agonists; Alkyl and Aryl Transferases; Amino Acid Motifs; Animals; Calcium Signaling; Carrier Proteins; Cell Line; Cell Line, Tumor; Cyclic AMP; Dose-Response Relationship, Drug; Endocytosis; Epoprostenol; Farnesyltranstransferase; Heat-Shock Proteins; HSP40 Heat-Shock Proteins; Humans; Iloprost; Isoproterenol; Kidney; Leukemia, Erythroblastic, Acute; Mice; Mutagenesis, Site-Directed; Organophosphorus Compounds; Piperidines; Proline; Propanolamines; Protein Prenylation; Protein Processing, Post-Translational; Proto-Oncogene Proteins p21(ras); Pyridines; Receptors, Adrenergic, beta-2; Receptors, Epoprostenol; Receptors, Thromboxane A2, Prostaglandin H2; Recombinant Fusion Proteins; Signal Transduction; Transfection

2005