Page last updated: 2024-09-03

cercosporamide and cgp 57380

cercosporamide has been researched along with cgp 57380 in 2 studies

Compound Research Comparison

Studies
(cercosporamide)
Trials
(cercosporamide)
Recent Studies (post-2010)
(cercosporamide)
Studies
(cgp 57380)
Trials
(cgp 57380)
Recent Studies (post-2010) (cgp 57380)
2602064044

Protein Interaction Comparison

ProteinTaxonomycercosporamide (IC50)cgp 57380 (IC50)
Serine/threonine-protein kinase Sgk1Homo sapiens (human)2.7
Dual specificity tyrosine-phosphorylation-regulated kinase 3Homo sapiens (human)3.2
Cytochrome P450 1A2Homo sapiens (human)1.6
Proto-oncogene tyrosine-protein kinase LCK Mus musculus (house mouse)2.5
Eukaryotic translation initiation factor 4EHomo sapiens (human)3
Cytochrome P450 2D6Homo sapiens (human)1.6
Interferon-induced, double-stranded RNA-activated protein kinaseHomo sapiens (human)5
Casein kinase I isoform deltaHomo sapiens (human)0.51
Serine/threonine-protein kinase BRSK2Homo sapiens (human)1.1
Aurora kinase BHomo sapiens (human)2.5
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)1.2182
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)2.06

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's2 (100.00)2.80

Authors

AuthorsStudies
Kannan, S; Nacro, K; Verma, CS; Xu, W1
Alarcon, H; Borrell, JI; Bou-Petit, E; Cano-Galietero, M; Estrada-Tejedor, R; Fuentes, P; Guijarro, PJ; Hümmer, S; Muñoz, MJ; Ramón Y Cajal, S; Santamaria, A; Slobodnyuk, K; Suarez-Cabrera, L1

Reviews

1 review(s) available for cercosporamide and cgp 57380

ArticleYear
Update on the Development of MNK Inhibitors as Therapeutic Agents.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Animals; Humans; Inflammation; Intracellular Signaling Peptides and Proteins; Neoplasms; Nervous System Diseases; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2022

Other Studies

1 other study(ies) available for cercosporamide and cgp 57380

ArticleYear
Overcoming Paradoxical Kinase Priming by a Novel MNK1 Inhibitor.
    Journal of medicinal chemistry, 2022, 04-28, Volume: 65, Issue:8

    Topics: Adenosine Triphosphate; Intracellular Signaling Peptides and Proteins; Models, Molecular; Protein Serine-Threonine Kinases; Signal Transduction

2022