cephalosporin c has been researched along with ly 163892 in 103 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 13 (12.62) | 18.7374 |
1990's | 81 (78.64) | 18.2507 |
2000's | 6 (5.83) | 29.6817 |
2010's | 3 (2.91) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Jacobs, NF; Moellering, RC | 1 |
Burman, LG; Kallings, I; Olsson-Liljequist, B | 1 |
Fah, YS; Powell, M; Seymour, A; Williams, JD; Yuan, M | 1 |
Boeckh, M; Deppermann, KM; Koeppe, P; Lode, H; Roller, S; Stelzer, I | 1 |
Barry, AL; Doern, GV; Ferraro, MJ; Jorgensen, JH; Murray, PR | 1 |
Dolence, EK; McKee, JA; Miller, MJ; Minnick, AA | 1 |
Gwaltney, J; Huck, W; Nielsen, RW; Scheld, WM; Sydnor, TA; Therasse, DG | 1 |
Foshee, WS; Qvarnberg, Y | 1 |
Disney, FA; Hanfling, MJ; Hausinger, SA | 1 |
Hanfling, MJ; Hausinger, SA; Squires, J | 1 |
Indelicato, JM; Pasini, CE | 1 |
Foshee, WS | 1 |
Syrop, J | 1 |
DeSante, KA; Zeckel, ML | 1 |
Copper, RD | 1 |
Therasse, DG | 1 |
Dere, WH | 1 |
Zeckel, ML | 1 |
Hyslop, DL | 1 |
Doern, G | 1 |
Nielsen, RW | 1 |
McCarty, J | 1 |
Jacobson, KD; McCarty, J; Ruoff, GE | 1 |
Bischoff, W; Hyslop, DL | 1 |
Bischoff, W; Iravani, A | 1 |
Van der Auwera, P | 1 |
Brumfitt, W; Hamilton-Miller, JM | 1 |
Eckernäs, SA; Grahnen, A; Nord, CE | 1 |
Gan, VN; Kusmiesz, H; Nelson, JD; Shelton, S | 1 |
Akaniro, JC; Arguedas, AG; Arrieta, AC; Marks, MI; Stutman, HR | 1 |
Brier, G; Kovach, PM; Lantz, RJ | 1 |
Doern, GV; Parker, D; Torres, B; Tubert, T; Vautour, R | 1 |
Iravani, A | 1 |
Adinolfi, LE; Marrone, A; Ruggiero, G; Tripodi, MF; Utili, R | 1 |
Brown, O; Kusmiesz, H; Manning, S; Nelson, JD; Shelton, S | 1 |
Hirata, T; Matsukuma, I; Mochida, K; Okachi, R; Sato, K | 1 |
Dunkin, KT; Howard, AJ | 1 |
Nelson, JD; Shelton, S | 1 |
Gratton, CA; Kibsey, PC; Knight, VE; Wenman, WM | 1 |
Fontana, R; Pelosi, E | 1 |
Barry, AL; Jones, RN | 3 |
Jorgensen, JH; Maher, LA; Redding, JS | 1 |
Kusmiesz, H; Nelson, JD; Shelton, S | 1 |
Cao, C; Chin, NX; Neu, HC | 1 |
Knapp, CC; Washington, JA | 1 |
Baertschi, SW; Collins, MW; Dorman, DE; Lorenz, LJ; Spangle, LA | 1 |
Brogden, RN; McTavish, D | 1 |
Anderson, RL; McKnight, JT; Rodman, DP | 1 |
Chen, J; Dantzig, AH; Hu, M; Kuhfeld, MT; Stratford, RE; Zhu, Y | 1 |
Doern, GV; Gerlach, EH; Hindler, J; Jones, RN; St Amand, R | 1 |
Aoki, FY; Hoban, DJ; Sitar, DS | 1 |
Beumer, H; Floor, M; Kolsters, A; Rozenberg-Arska, M; van Akkeren, F; Verhoef, J; Visser, M | 1 |
Rodriguez, WJ; Wiedermann, BL | 1 |
Andrews, JM; Lees, AS; Wise, R | 1 |
Biedenbach, DJ; Jones, RN | 1 |
Dantzig, AH; Duckworth, DC; Tabas, LB | 1 |
Bilton, D; Hill, SL; Johnson, MM; Mitchell, JL; Pye, A; Stockley, RA | 1 |
Bass, JW; Chan, DS; Demers, DM | 1 |
Baertschi, SW; Collins, MW; Dorman, DE; Lorenz, LJ; Occolowitz, JL; Paschal, JW; Skibic, MJ; Spangle, LA; Taylor, KW | 1 |
Belcher, J; Cole, PJ; Kanthakumar, K; Lund, V; Read, RC; Roberts, DE; Rutman, A; Tsang, KW; Wilson, R | 1 |
Greenfield, RA | 1 |
Cerimele, BJ; Davidson, RL; DeSante, KA; Farlow, DS; Hatcher, BL; Quadracci, LJ; Therasse, DG | 1 |
Berman, S; Roark, R | 1 |
Hussar, DA | 1 |
Bendele, A; Buening, M; Clemens, J; Colbert, W; Deldar, A; Helton, D; McGrath, J; Shannon, H; Shetler, T; Turk, J | 1 |
Force, RW; Nahata, MC | 1 |
Kamme, C; Petersson, AC | 1 |
Borner, K; Fassbender, M; Koeppe, P; Lode, H; Schaberg, T | 1 |
Aspinall, S; Connell, C; Corkill, J | 1 |
Caldwell, SA; Lum, GM; Thieme, RE | 1 |
Fravert, D; Hsu, CY; Tune, BM | 1 |
Daniel, H; Thwaites, DT; Wenzel, U | 1 |
Cappelletty, DM; Rybak, MJ | 1 |
Chen, J; Dantzig, AH; Hu, M; Stratford, RE; Zheng, L | 1 |
Chen, J; Dantzig, AH; Hu, M; Li, Y; Liu, L; Stratford, RE; Zheng, L | 1 |
Itokazu, GS; Karavokiros, KT; Schatz, BS; Taeubel, MA | 1 |
Gonzales, J; Overturf, GD; Shandler, L | 1 |
Björnsson, E; Olsson, R | 1 |
Benn, RA; Fernandes, CJ; Nimmo, GR | 1 |
Larsson, P; Roos, K | 1 |
Berry, DM; Dantzig, AH; Duckworth, DC; Snyder, NJ; Spry, DO; Tabas, LB | 1 |
Preston, DA; Turik, M | 1 |
Gould, IM; Mackenzie, FM; Milne, KE | 1 |
Abdel-Rahman, SM; Blowey, DL; Kauffmann, RE; Kearns, GL | 1 |
Blondeau, JM; Borsos, S; Suter, M | 1 |
Adelglass, J; Gooch, WM; Johns, D; Kelsey, DK; Masica, D; Weinberg, BC | 1 |
Allen, BS; Bandak, SI; Bolzon, LD; Preston, DA; Turnak, MR | 1 |
Griffin, TJ; Keyserling, CH; McAdoo, MA; Nemeth, MA; Paster, RZ; Tack, KJ | 1 |
Kalich, S; Nilsson-Ehle, I; Nord, CE; Ochs, HR; Odenholt, I; Vogel, F; Wettich, K | 1 |
Arghittu, M; Colombo, R; Conio, F; Gagliardi, L; Garlaschi, ML; Rusconi, F; Sala, A; Sideri, S; Varotto, F | 1 |
Aljitawi, OS; Aster, RH; Bougie, DW; Curtis, BR; Krishnan, K | 1 |
Kamme, C; Orrling, A; Stjernquist-Desatnik, A | 1 |
Heidron, F; Knothe, H; Sammann, A; Schäfer, V | 1 |
Balatsouras, DG; Eliopoulos, P; Ferekidis, E; Korres, S; Rallis, E | 1 |
Correra, TC; Hu, CQ; Li, J; Maître, P; Qian, JQ; Song, DQ | 1 |
Amicosante, G; Bottoni, C; Celenza, G; Colapietro, M; Galleni, M; Kerff, F; Marcoccia, F; Matagne, A; Mercuri, PS; Perilli, M; Sabatini, A | 1 |
Cattrall, JWS; Kirby, A; Robinson, AV | 1 |
18 review(s) available for cephalosporin c and ly 163892
Article | Year |
---|---|
Comparative United States and European trials of loracarbef in the treatment of acute otitis media.
Topics: Acute Disease; Amoxicillin; Cephalosporins; Clinical Trials as Topic; Europe; Humans; Otitis Media; United States | 1992 |
Pharmacokinetic profile of loracarbef.
Topics: Adult; Age Factors; Biological Availability; Cephalosporins; Child; Clinical Trials as Topic; Food; Humans; Kidney Diseases; Metabolic Clearance Rate; Probenecid | 1992 |
The carbacephems: a new beta-lactam antibiotic class.
Topics: Ambulatory Care; Animals; Anti-Bacterial Agents; Biological Availability; Cephalosporins; Clinical Trials as Topic; Dogs; Drug Evaluation, Preclinical; Drug Stability; Esters; Haplorhini; Humans; Mice; Microbial Sensitivity Tests | 1992 |
The safety profile of loracarbef: clinical trials in respiratory, skin, and urinary tract infections.
Topics: Adult; Adverse Drug Reaction Reporting Systems; Aged; Cephalosporins; Child; Diarrhea; Headache; Humans; Incidence; Intestines; Respiratory Tract Infections; Skin Diseases, Infectious; Urinary Tract Infections | 1992 |
Acute bronchitis: results of U.S. and European trials of antibiotic therapy.
Topics: Acute Disease; Bronchitis; Cephalosporins; Clinical Trials as Topic; Drug Resistance, Microbial; Europe; Gastrointestinal Diseases; Humans; Respiratory Tract Infections; United States | 1992 |
Loracarbef (LY163892) in the treatment of acute exacerbations of chronic bronchitis: results of U.S. and European comparative clinical trials.
Topics: Acute Disease; Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Bronchitis; Cephalosporins; Chronic Disease; Clavulanic Acids; Diarrhea; Drug Therapy, Combination; Europe; Female; Headache; Humans; Incidence; Male; Middle Aged; Treatment Outcome; United States | 1992 |
Efficacy and safety of loracarbef in the treatment of pneumonia.
Topics: Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Bacterial Infections; Cephalosporins; Clavulanic Acids; Drug Therapy, Combination; Humans; Nausea; Pneumonia; Randomized Controlled Trials as Topic; Vomiting | 1992 |
In vitro activity of loracarbef and effects of susceptibility test methods.
Topics: Cephalosporins; Clinical Protocols; Clinical Trials as Topic; Drug Evaluation, Preclinical; Drug Resistance, Microbial; Humans; Microbial Sensitivity Tests; Treatment Outcome | 1992 |
Acute bacterial maxillary sinusitis: results of U.S. and European comparative therapy trials.
Topics: Adolescent; Adult; Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Cephalosporins; Clavulanic Acids; Double-Blind Method; Doxycycline; Drug Therapy, Combination; Female; Finland; Humans; Iceland; Male; Maxillary Sinusitis; Middle Aged; Single-Blind Method; Sweden; Treatment Outcome; United States | 1992 |
Antibiotic therapy for urinary tract infections.
Topics: Cefaclor; Cephalosporins; Clinical Trials as Topic; Europe; Female; Humans; Male; Norfloxacin; United States; Urinary Tract Infections | 1992 |
Loracarbef. A review of its antimicrobial activity, pharmacokinetic properties and therapeutic efficacy.
Topics: Adolescent; Adult; Aged; Cephalosporins; Child; Humans; Microbial Sensitivity Tests; Middle Aged; Randomized Controlled Trials as Topic | 1993 |
A critical review of the new oral cephalosporins. Considerations and place in therapy.
Topics: Administration, Oral; Anti-Infective Agents; Cefixime; Cefotaxime; Cefpodoxime; Cefprozil; Ceftizoxime; Cephalosporins; Humans | 1994 |
The role of newer oral cephalosporins, fluoroquinolones, and macrolides in the treatment of pediatric infections.
Topics: Administration, Oral; Anti-Bacterial Agents; Anti-Infective Agents; Azithromycin; Bacterial Infections; Cefixime; Cefotaxime; Cefpodoxime Proxetil; Cefprozil; Ceftibuten; Ceftizoxime; Cefuroxime; Cephalosporins; Child; Clarithromycin; Fluoroquinolones; Humans | 1994 |
Symposium on antimicrobial therapy. V. The carbapenems and monobactams.
Topics: Aztreonam; Bacterial Infections; Cephalosporins; Humans; Imipenem; Microbial Sensitivity Tests | 1993 |
Loracarbef: a new orally administered carbacephem antibiotic.
Topics: Administration, Oral; Bacterial Infections; Cephalosporins; Drug Interactions; Humans; Microbial Sensitivity Tests | 1993 |
Pharmacokinetics of new oral cephalosporins, including a new carbacephem.
Topics: Administration, Oral; Aged; Biological Availability; Cephalosporins; Child; Drug Administration Schedule; Drug Interactions; Food; Humans; Infant | 1993 |
Comparison of cefprozil, cefpodoxime proxetil, loracarbef, cefixime, and ceftibuten.
Topics: Bacterial Infections; Cefixime; Cefotaxime; Cefpodoxime Proxetil; Cefprozil; Ceftibuten; Ceftizoxime; Cephalosporins; Humans; Microbial Sensitivity Tests; Prodrugs; Randomized Controlled Trials as Topic | 1996 |
A systematic review of randomised clinical trials for oral antibiotic treatment of acute pyelonephritis.
Topics: Acute Disease; Administration, Oral; Anti-Bacterial Agents; Cephalosporins; Ciprofloxacin; Drug Combinations; Humans; Norfloxacin; Pyelonephritis; Randomized Controlled Trials as Topic; Sulfamethizole; Trimethoprim | 2018 |
25 trial(s) available for cephalosporin c and ly 163892
Article | Year |
---|---|
Pharmacokinetics of loracarbef and interaction with acetylcysteine.
Topics: Acetylcysteine; Administration, Oral; Adult; Cephalosporins; Drug Combinations; Drug Interactions; Eating; Fasting; Humans; Male | 1992 |
Loracarbef (LY 163892) vs amoxicillin/clavulanate in bacterial maxillary sinusitis.
Topics: Adolescent; Adult; Aged; Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Bacterial Infections; Cephalosporins; Clavulanic Acids; Decision Trees; Drug Therapy, Combination; Female; Humans; Male; Maxillary Sinusitis; Middle Aged; Severity of Illness Index | 1992 |
Comparative United States and European trials of loracarbef in the treatment of acute otitis media.
Topics: Acute Disease; Amoxicillin; Cephalosporins; Clinical Trials as Topic; Europe; Humans; Otitis Media; United States | 1992 |
Loracarbef (LY163892) vs. penicillin VK in the treatment of streptococcal pharyngitis and tonsillitis.
Topics: Cephalosporins; Child; Child, Preschool; Double-Blind Method; Female; Humans; Infant; Male; Penicillin V; Pharyngitis; Streptococcal Infections; Streptococcus pyogenes; Tonsillitis | 1992 |
Loracarbef vs. cefaclor in pediatric skin and skin structure infections.
Topics: Cefaclor; Cephalosporins; Child; Child, Preschool; Double-Blind Method; Female; Haemophilus Infections; Haemophilus influenzae; Humans; Infant; Male; Skin Diseases, Infectious; Staphylococcal Skin Infections; Staphylococcus aureus; Streptococcal Infections; Streptococcus pyogenes | 1992 |
Loracarbef (LY163892) versus amoxicillin-clavulanate in the treatment of bacterial acute otitis media with effusion.
Topics: Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Bacterial Infections; Cephalosporins; Clavulanic Acids; Double-Blind Method; Drug Evaluation; Drug Therapy, Combination; Female; Haemophilus influenzae; Humans; Infant; Male; Moraxella catarrhalis; Otitis Media with Effusion; Streptococcus pneumoniae | 1992 |
Loracarbef (LY163892) in the treatment of acute exacerbations of chronic bronchitis: results of U.S. and European comparative clinical trials.
Topics: Acute Disease; Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Bronchitis; Cephalosporins; Chronic Disease; Clavulanic Acids; Diarrhea; Drug Therapy, Combination; Europe; Female; Headache; Humans; Incidence; Male; Middle Aged; Treatment Outcome; United States | 1992 |
Acute bacterial maxillary sinusitis: results of U.S. and European comparative therapy trials.
Topics: Adolescent; Adult; Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Cephalosporins; Clavulanic Acids; Double-Blind Method; Doxycycline; Drug Therapy, Combination; Female; Finland; Humans; Iceland; Male; Maxillary Sinusitis; Middle Aged; Single-Blind Method; Sweden; Treatment Outcome; United States | 1992 |
Loracarbef versus penicillin VK in the treatment of streptococcal pharyngitis and tonsillitis in an adult population.
Topics: Adult; Cephalosporins; Cough; Diarrhea; Double-Blind Method; Headache; Humans; North America; Penicillin V; Pharyngitis; Streptococcal Infections; Streptococcus pyogenes; Tonsillitis | 1992 |
Loracarbef (LY163892) versus cefaclor in the treatment of bacterial skin and skin-structure infections in an adult population.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Bacterial Infections; Cefaclor; Cephalosporins; Child; Double-Blind Method; Gastrointestinal Diseases; Headache; Humans; Incidence; Middle Aged; Skin Diseases, Infectious; Treatment Outcome | 1992 |
Loracarbef (LY163892) versus cefaclor and norfloxacin in the treatment of uncomplicated pyelonephritis.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Cefaclor; Cephalosporins; Diarrhea; Double-Blind Method; Europe; Female; Headache; Humans; Male; Middle Aged; Nausea; Norfloxacin; Pyelonephritis; Treatment Outcome; United States | 1992 |
Bactericidal titers of loracarbef (LY 163892) in serum and killing rates in volunteers receiving 400 versus 200 milligrams.
Topics: Administration, Oral; Adult; Cephalosporins; Dose-Response Relationship, Drug; Female; Humans; Male; Microbial Sensitivity Tests; Middle Aged; Random Allocation | 1992 |
Comparative evaluation of loracarbef and amoxicillin-clavulanate for acute otitis media.
Topics: Acute Disease; Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Bacteria; Cephalosporins; Child, Preschool; Clavulanic Acids; Drug Therapy, Combination; Female; Follow-Up Studies; Humans; Infant; Male; Microbial Sensitivity Tests; Otitis Media; Random Allocation; Recurrence | 1991 |
Loracarbef versus cefaclor in the treatment of urinary tract infections in women.
Topics: Cefaclor; Cephalosporins; Double-Blind Method; Female; Humans; Urinary Tract Infections | 1991 |
Pharmacokinetic disposition of loracarbef in healthy young men and women at steady state.
Topics: Adult; Cephalosporins; Drug Administration Schedule; Female; Humans; Male; Metabolic Clearance Rate; Specimen Handling; Time Factors | 1994 |
Antimicrobial drug suspensions: a blinded comparison of taste of twelve common pediatric drugs including cefixime, cefpodoxime, cefprozil and loracarbef.
Topics: Analysis of Variance; Anti-Bacterial Agents; Anti-Infective Agents; Cefixime; Cefotaxime; Cefpodoxime; Cefprozil; Ceftizoxime; Cephalosporins; Child; Child, Preschool; Drug Combinations; Humans; Infant; Single-Blind Method; Smell; Suspensions; Taste | 1994 |
Loracarbef versus doxycycline in the treatment of acute bacterial maxillary sinusitis. Scandinavian Study Group.
Topics: Acute Disease; Bacteria; Cephalosporins; Double-Blind Method; Doxycycline; Humans; Maxillary Sinusitis; Microbial Sensitivity Tests | 1993 |
Factors influencing outcome in children treated with antibiotics for acute otitis media.
Topics: Acute Disease; Amoxicillin; Anti-Bacterial Agents; Cefaclor; Cefixime; Cefotaxime; Cephalosporins; Child; Child, Preschool; Clinical Trials as Topic; Female; Follow-Up Studies; Humans; Infant; Male; Otitis Media; Regression Analysis; Risk Factors; Treatment Outcome | 1993 |
A national collaborative study of the in vitro activity of oral cephalosporins and loracarbef (LY 163892). Australian Group for the Study of Antimicrobial Resistance (AGAR).
Topics: Administration, Oral; Australia; Cephalosporins; Drug Resistance, Microbial; Enterobacteriaceae; Gram-Positive Bacteria; Laboratories, Hospital; Microbial Sensitivity Tests; Streptococcus pneumoniae | 1997 |
Loracarbef versus phenoxymethylpenicillin in the treatment of recurrent streptococcal pharyngotonsillitis.
Topics: Cephalosporins; Double-Blind Method; Humans; Penicillin V; Penicillins; Pharyngeal Diseases; Streptococcal Infections; Tonsillitis | 1997 |
Comparative bioavailability of loracarbef chewable tablet vs. oral suspension in children.
Topics: Administration, Oral; Analysis of Variance; Area Under Curve; Bacterial Infections; Biological Availability; Cephalosporins; Child; Child, Preschool; Female; Humans; Male; Suspensions; Tablets | 1998 |
Loracarbef versus clarithromycin in children with acute otitis media with effusion.
Topics: Acute Disease; Anti-Bacterial Agents; Cephalosporins; Child, Preschool; Clarithromycin; Humans; Infant; Otitis Media with Effusion; Single-Blind Method; Treatment Outcome | 1999 |
A comparison of a five-day regimen of cefdinir with a seven-day regimen of loracarbef for the treatment of acute exacerbations of chronic bronchitis.
Topics: Adolescent; Adult; Aged; Anti-Infective Agents; Bacterial Infections; Bronchitis; Cefdinir; Cephalosporins; Chronic Disease; Double-Blind Method; Drug Administration Schedule; Female; Humans; Male; Middle Aged; Prospective Studies; Sputum; Treatment Outcome | 2000 |
Penicillin V, loracarbef and clindamycin in tonsillar surface fluid during acute group A streptococcal pharyngotonsillitis.
Topics: Adult; Aged; Anti-Bacterial Agents; C-Reactive Protein; Cephalosporins; Clindamycin; Female; Humans; Male; Middle Aged; Orosomucoid; Palatine Tonsil; Penicillin V; Streptococcal Infections; Streptococcus pyogenes; Tissue Distribution; Tonsillitis | 2005 |
Twice-daily dosing of loracarbef 15 mg/kg versus 30 mg/kg in the treatment of children with acute sinusitis.
Topics: Acute Disease; Anti-Bacterial Agents; Cephalosporins; Child; Child, Preschool; Dose-Response Relationship, Drug; Drug Administration Schedule; Humans; Sinusitis | 2005 |
63 other study(ies) available for cephalosporin c and ly 163892
Article | Year |
---|---|
Advances in outpatient antimicrobial therapy: loracarbef.
Topics: Ambulatory Care; Cephalosporins; Humans; Randomized Controlled Trials as Topic | 1992 |
Antibiotic susceptibility of upper respiratory tract pathogens in Sweden: a seven year follow-up study including loracarbef. Swedish Respiratory Tract Study Group.
Topics: Cephalosporins; Drug Resistance, Microbial; Follow-Up Studies; Haemophilus influenzae; Humans; Moraxella catarrhalis; Respiratory Tract Infections; Streptococcus pneumoniae; Streptococcus pyogenes; Sweden | 1992 |
In vitro susceptibility of Haemophilus influenzae to cefaclor, cefixime, cefetamet and loracarbef.
Topics: Ampicillin Resistance; Cefaclor; Cefixime; Cefotaxime; Ceftizoxime; Cephalosporins; Haemophilus influenzae; Microbial Sensitivity Tests; Regression Analysis | 1992 |
Development of revised quality control limits for disk diffusion susceptibility tests of selected cephem antibiotics with Haemophilus influenzae and description of a new control strain.
Topics: Ampicillin; Cefaclor; Cefamandole; Cefonicid; Cefuroxime; Cephalosporins; Evaluation Studies as Topic; Haemophilus influenzae; Humans; Microbial Sensitivity Tests; Quality Control; Reference Standards | 1992 |
Iron transport-mediated antibacterial activity of and development of resistance to hydroxamate and catechol siderophore-carbacephalosporin conjugates.
Topics: Catechols; Cell Division; Cephalosporins; Drug Resistance, Microbial; Escherichia coli; Ferric Compounds; Hydroxamic Acids; Microbial Sensitivity Tests | 1992 |
Loracarbef.
Topics: Adult; Cephalosporins; Child; Clinical Trials as Topic; Costs and Cost Analysis; Humans; Microbial Sensitivity Tests; Respiratory Tract Infections; Skin Diseases, Infectious; Urinary Tract Infections | 1992 |
Pharmaceutical properties of loracarbef: the remarkable solution stability of an oral 1-carba-1-dethiacephalosporin antibiotic.
Topics: Cefaclor; Cephalexin; Cephalosporins; Chromatography, High Pressure Liquid; Colorimetry; Crystallization; Drug Stability; Hydrogen-Ion Concentration; Isoelectric Focusing; Kinetics; Solubility; Solutions; Thermodynamics; X-Ray Diffraction | 1992 |
New antibiotics for skin and skin structure infections.
Topics: Cefprozil; Cephalosporins; Humans; Skin Diseases, Infectious | 1992 |
Advances in outpatient antimicrobial therapy: loracarbef. June 12-15, 1991, San Francisco, California. Proceedings.
Topics: Ambulatory Care; Cephalosporins; Humans | 1992 |
Comparative in vitro activity of cefixime, cefaclor and loracarbef against urinary pathogens.
Topics: Anti-Infective Agents, Urinary; Bacteria; Cefaclor; Cefixime; Cefotaxime; Cephalosporins; Humans; Microbial Sensitivity Tests; Urinary Tract Infections | 1991 |
Effect of loracarbef on the normal oropharyngeal and intestinal microflora.
Topics: Administration, Oral; Adult; Bacteria; Cephalosporins; Feces; Female; Humans; Intestines; Male; Oropharynx | 1991 |
In-vitro activity of cefprozil (BMY 28100) and loracarbef (LY 163892) against pathogens obtained from middle ear fluid.
Topics: Acute Disease; Cefprozil; Cephalosporins; Ear, Middle; Haemophilus influenzae; Moraxella catarrhalis; Otitis Media; Streptococcus pneumoniae | 1991 |
High-performance liquid chromatographic determination of loracarbef, a potential metabolite, cefaclor and cephalexin in human plasma, serum and urine.
Topics: Cefaclor; Cephalexin; Cephalosporins; Chromatography, High Pressure Liquid; Humans; Molecular Structure; Spectrophotometry, Ultraviolet | 1991 |
In vitro activity of loracarbef (LY163892), a new oral carbacephem antimicrobial agent, against respiratory isolates of Haemophilus influenzae and Moraxella catarrhalis.
Topics: Anti-Bacterial Agents; Bacterial Infections; beta-Lactamases; Cephalosporins; Haemophilus Infections; Haemophilus influenzae; Humans; Microbial Sensitivity Tests; Moraxella catarrhalis; Respiratory Tract Infections | 1991 |
Influence of subinhibitory concentrations of loracarbef (LY 163892) and daptomycin (LY 146032) on bacterial phagocytosis, killing and serum sensitivity.
Topics: Bacteria; Blood Bactericidal Activity; Cephalosporins; Daptomycin; Drug Resistance, Microbial; Humans; Immune Sera; Macrophages; Neutrophils; Peptides; Phagocytosis | 1990 |
Loracarbef concentrations in middle ear fluid.
Topics: Body Fluids; Cephalosporins; Child; Child, Preschool; Ear, Middle; Female; Humans; Infant; Male; Otitis Media; Tympanoplasty | 1990 |
In vitro and in vivo antibacterial activity of KT3777, a new orally active carbacephem.
Topics: Administration, Oral; Animals; Bacterial Infections; Cefaclor; Cephalexin; Cephalosporins; Female; Gram-Negative Bacteria; Gram-Positive Bacteria; Male; Mice; Microbial Sensitivity Tests | 1989 |
Comparative in-vitro activity of a new oral carbacephem, LY163892.
Topics: Bacteria; Cephalosporins; Escherichia coli; Haemophilus influenzae; Microbial Sensitivity Tests; Penicillins; Staphylococcus aureus | 1988 |
In vitro susceptibilities of common pediatric pathogens to LY163892.
Topics: Anti-Bacterial Agents; Bacteria; Cephalosporins; Child; Escherichia coli; Haemophilus influenzae; Humans; Microbial Sensitivity Tests; Moraxella catarrhalis; Staphylococcus aureus; Streptococcus pneumoniae; Streptococcus pyogenes | 1988 |
In vitro activity of LY163892 against pathogens isolated from pediatric patients.
Topics: Bacteria; Cephalosporins; Drug Resistance, Microbial; Haemophilus influenzae; Humans; Moraxella catarrhalis; Streptococcus pneumoniae | 1988 |
In vitro activity and beta-lactamase stability of LY163892.
Topics: Administration, Oral; Bacteria; beta-Lactamases; Cefaclor; Cefotaxime; Cephalexin; Cephalosporins; Enzyme Stability | 1988 |
Antimicrobial activity of LY163892, an orally administered 1-carbacephem.
Topics: Bacteria; Cefaclor; Cephalexin; Cephalosporins; Microbial Sensitivity Tests | 1988 |
Influence of storage and susceptibility test conditions on stability and activity of LY163892 and four other cephalosporins.
Topics: Bacteria; Cephalosporins; Culture Media; Drug Stability; Drug Storage; Humans; Hydrogen-Ion Concentration; Microbial Sensitivity Tests | 1988 |
Pharmacokinetics of LY163892 in infants and children.
Topics: Adolescent; Cephalosporins; Child; Child, Preschool; Female; Half-Life; Humans; Infant; Male; Metabolic Clearance Rate | 1988 |
Disk diffusion susceptibility testing for LY163892 (KT-3777), a new orally administered 1-carbacephem.
Topics: Bacteria; Cefaclor; Cephalexin; Cephalosporins; Enterobacter; Haemophilus influenzae; Microbial Sensitivity Tests; Predictive Value of Tests; Providencia | 1988 |
In-vitro activity and beta-lactamase stability of LY163892.
Topics: Amoxicillin; Bacteria; beta-Lactamases; Cell Wall; Cephalosporins; Clavulanic Acids; Enzyme Stability; Microbial Sensitivity Tests | 1988 |
In vitro activities of LY163892, cefaclor, and cefuroxime.
Topics: Anti-Bacterial Agents; Bacteria; Cefaclor; Cefuroxime; Cephalexin; Cephalosporins; Drug Stability; Temperature | 1988 |
Beta-lactamase hydrolysis and inhibition studies of the new 1-carbacephem LY163892.
Topics: beta-Lactamase Inhibitors; beta-Lactamases; Cefaclor; Cefotaxime; Cephaloridine; Cephalosporins; Hydrolysis | 1987 |
Formation of fluorescent pyrazine derivatives via a novel degradation pathway of the carbacephalosporin loracarbef.
Topics: Cephalosporins; Chromatography, High Pressure Liquid; Magnetic Resonance Spectroscopy; Pyrazines; Spectrometry, Fluorescence; Spectrometry, Mass, Fast Atom Bombardment; Spectrophotometry, Ultraviolet | 1995 |
Mechanism and kinetics of transcellular transport of a new beta-lactam antibiotic loracarbef across an intestinal epithelial membrane model system (Caco-2).
Topics: Amino Acid Sequence; Biological Transport; Cells, Cultured; Cephalosporins; Culture Media; Dipeptides; Epithelial Cells; Epithelium; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Intestinal Mucosa; Mannitol; Models, Biological; Molecular Sequence Data | 1994 |
Revised disk diffusion interpretive criteria for cefaclor, loracarbef, cefprozil and cefixime when testing Haemophilus influenzae on haemophilus test medium.
Topics: Cefaclor; Cefixime; Cefotaxime; Cefprozil; Cephalosporins; Culture Media; Haemophilus Infections; Haemophilus influenzae; Humans; Microbial Sensitivity Tests; Quality Control | 1994 |
FDA announces recall of liquid antibiotics.
Topics: Cefaclor; Cephalexin; Cephalosporins; Drug and Narcotic Control; United States; United States Food and Drug Administration | 1994 |
Effect of loracarbef and amoxicillin on the oropharyngeal and intestinal microflora of patients with bronchitis.
Topics: Acute Disease; Adolescent; Adult; Amoxicillin; Bacteria, Anaerobic; Bronchitis; Cephalosporins; Enterococcus faecalis; Female; Gram-Negative Aerobic Bacteria; Humans; Intestines; Male; Microbial Sensitivity Tests; Oropharynx; Yeasts | 1994 |
The pharmacokinetics, tissue penetration and in-vitro activity of loracarbef, a beta-lactam antibiotic of the carbacephem class.
Topics: Adult; Amoxicillin; Amoxicillin-Potassium Clavulanate Combination; Cefaclor; Cephalosporins; Clavulanic Acids; Drug Therapy, Combination; Enterobacteriaceae; Exudates and Transudates; Haemophilus influenzae; Half-Life; Humans; Male; Microbial Sensitivity Tests; Moraxella catarrhalis; Staphylococcus aureus; Streptococcus pneumoniae | 1993 |
Predictive accuracy of disk diffusion test for Proteus vulgaris and Providencia species against five newer orally administered cephalosporins, cefdinir, cefetamet, cefprozil, cefuroxime, and loracarbef.
Topics: Administration, Oral; Cefdinir; Cefprozil; Ceftizoxime; Cefuroxime; Cephalosporins; Drug Resistance, Microbial; Evaluation Studies as Topic; False Positive Reactions; Humans; Microbial Sensitivity Tests; Proteus vulgaris; Providencia | 1994 |
Transport mechanisms responsible for the absorption of loracarbef, cefixime, and cefuroxime axetil into human intestinal Caco-2 cells.
Topics: Adenocarcinoma; Amino Acids; Biological Transport; Cefixime; Cefotaxime; Cefuroxime; Cephalosporins; Colonic Neoplasms; Dipeptides; Drug Antagonism; Energy Metabolism; Humans; Intestinal Absorption; Tumor Cells, Cultured | 1994 |
Sputum and serum pharmacokinetics of loracarbef (LY163892) in patients with chronic bronchial sepsis.
Topics: Adult; Aged; Albumins; Anti-Bacterial Agents; beta-Lactamases; Bronchiectasis; Cephalosporins; Chronic Disease; Female; Humans; Lung; Male; Middle Aged; Serum Albumin; Sputum | 1994 |
Aqueous acidic degradation of the carbacephalosporin loracarbef.
Topics: Cefaclor; Cephalosporins; Chromatography, High Pressure Liquid; Drug Stability; Hydrogen-Ion Concentration; Magnetic Resonance Spectroscopy; Mass Spectrometry; Molecular Structure; Solutions | 1993 |
Haemophilus influenzae infection of human respiratory mucosa in low concentrations of antibiotics.
Topics: Adenoids; Amoxicillin; Anti-Bacterial Agents; Cephalosporins; Child, Preschool; Ciprofloxacin; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Haemophilus Infections; Haemophilus influenzae; Humans; Microbial Sensitivity Tests; Microscopy, Electron; Mucociliary Clearance; Mucous Membrane; Organ Culture Techniques; Respiratory Tract Infections | 1993 |
Effects of renal dysfunction on the pharmacokinetics of loracarbef.
Topics: Adult; Cephalosporins; Female; Humans; Kidney Failure, Chronic; Kidney Function Tests; Male; Middle Aged; Renal Dialysis | 1993 |
New antibacterial agents.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Cephalosporins; Fluoroquinolones; Humans; Macrolides | 1993 |
General pharmacology of loracarbef in animals.
Topics: Anesthetics, Local; Animals; Anti-Bacterial Agents; Blood Coagulation; Blood Glucose; Central Nervous System; Cephalosporins; Digestive System; Dogs; Guinea Pigs; Hemodynamics; Hemolysis; Immune System; Inflammation; Irritants; Kidney; Male; Mice; Platelet Aggregation; Rabbits; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Rats, Wistar | 1993 |
In vitro effect on group A streptococci of loracarbef versus cefadroxil, cefaclor and penicillin V.
Topics: Anti-Bacterial Agents; Cefaclor; Cefadroxil; Cephalosporins; Humans; In Vitro Techniques; Microbial Sensitivity Tests; Penicillin V; Pharyngitis; Streptococcal Infections; Streptococcus pyogenes | 1993 |
Sputum and serum pharmacokinetics of loracarbef (LY163892) in patients with bronchial sepsis.
Topics: beta-Lactamases; Bronchial Diseases; Cephalosporins; Humans; Sepsis; Sputum | 1995 |
Acute interstitial nephritis associated with loracarbef therapy.
Topics: Acute Disease; Anti-Bacterial Agents; Biopsy; Cephalosporins; Humans; Infant; Kidney; Male; Necrosis; Nephritis, Interstitial; Otitis Media | 1995 |
Cephalosporin and carbacephem nephrotoxicity. Roles of tubular cell uptake and acylating potential.
Topics: Acylation; Ampicillin; Animals; Anti-Bacterial Agents; Biological Transport; Cephaloglycin; Cephalosporins; Half-Life; Infusions, Intravenous; Kidney; Kidney Cortex; Penicillins; Rabbits; Structure-Activity Relationship; Tissue Distribution | 1996 |
Stereoselective uptake of beta-lactam antibiotics by the intestinal peptide transporter.
Topics: Animals; Anti-Bacterial Agents; Cadherins; Carrier Proteins; Cell Line; Cephalexin; Cephalosporins; Hydrolysis; Intestinal Mucosa; Membrane Transport Proteins; Microinjections; Oocytes; Peptides; Stereoisomerism; Xenopus laevis | 1995 |
Bactericidal activities of cefprozil, penicillin, cefaclor, cefixime, and loracarbef against penicillin-susceptible and -resistant Streptococcus pneumoniae in an in vitro pharmacodynamic infection model.
Topics: Cefaclor; Cefixime; Cefotaxime; Cefprozil; Cephalosporins; Colony-Forming Units Assay; Humans; Microbial Sensitivity Tests; Models, Theoretical; Penicillin Resistance; Penicillins; Streptococcus pneumoniae | 1996 |
Uptake characteristics of loracarbef and cephalexin in the Caco-2 cell culture model: effects of the proton gradient and possible presence of a distinctive second component.
Topics: Caco-2 Cells; Cephalexin; Cephalosporins; Humans; Peptides; Protons | 1996 |
Peptide transporter function and prolidase activities in Caco-2 cells: a lack of coordinated expression.
Topics: Basement Membrane; Biological Transport; Caco-2 Cells; Cell Division; Cephalosporins; Dipeptidases; Dipeptides; Humans; Kinetics; Peptides; Protons | 1995 |
Recurrence of pneumococcal sepsis caused by an intermediately penicillin-resistant organism treated with loracarbef.
Topics: Bacteremia; Cephalosporins; Drug Resistance, Microbial; Humans; Infant; Male; Pneumococcal Infections; Recurrence | 1996 |
Acute liver injury due to loracarbef.
Topics: Acute Disease; Aged; Biopsy; Cephalosporins; Chemical and Drug Induced Liver Injury; Cholestasis, Extrahepatic; Follow-Up Studies; Humans; Liver Diseases; Male | 1997 |
Structure-activity relationship of carbacephalosporins and cephalosporins: antibacterial activity and interaction with the intestinal proton-dependent dipeptide transport carrier of Caco-2 cells.
Topics: Caco-2 Cells; Cadherins; Carrier Proteins; Cephalexin; Cephalosporins; Humans; Lactams; Membrane Transport Proteins; Microbial Sensitivity Tests; Stereoisomerism; Structure-Activity Relationship | 1997 |
Cefaclor: a contemporary look at susceptibility of key pathogens from around the globe.
Topics: Anti-Infective Agents; Cefaclor; Cephalosporins; Ciprofloxacin; Escherichia coli; Haemophilus influenzae; Methicillin Resistance; Microbial Sensitivity Tests; Moraxella catarrhalis; Penicillin Resistance; Staphylococcus aureus | 1998 |
The effects of the morphological response of Enterobacteriaceae to cephalosporins on PAE and CERT.
Topics: Cefaclor; Cefuroxime; Cephalosporins; Colony Count, Microbial; Culture Media; Electric Impedance; Enterobacteriaceae; Luminescent Measurements; Microbial Sensitivity Tests | 1998 |
Determination of the antimicrobial susceptibilities of Canadian isolates of Haemophilus influenzae, Streptococcus pneumoniae and Moraxella catarrhalis. Canadian Antimicrobial Study Group.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Cephalosporins; Ciprofloxacin; Haemophilus influenzae; Microbial Sensitivity Tests; Moraxella catarrhalis; Penicillin Resistance; Respiratory Tract Infections; Streptococcus pneumoniae | 1999 |
Assessment of the susceptibility of Streptococcus pneumoniae to cefaclor and loracarbef in 13 countries.
Topics: Cefaclor; Cephalosporins; Europe; Humans; Microbial Sensitivity Tests; North America; Penicillin Resistance; Russia; Streptococcus pneumoniae | 2000 |
Effect of step-down therapy of ceftriaxone plus loracarbef versus parenteral therapy of ceftriaxone on the intestinal microflora in patients with community-acquired pneumonia.
Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Ceftriaxone; Cephalosporins; Community-Acquired Infections; Drug Therapy, Combination; Feces; Female; Hospitalization; Humans; Infusions, Intravenous; Intestines; Male; Middle Aged; Pneumonia; Treatment Outcome | 2001 |
In-vitro susceptibility of Haemophilus influenzae to loracarbef (LY 163892) and other oral antibiotics. Collaborative Study Group on Pediatric Infectious Disease in Lombardy.
Topics: Adult; Ampicillin; Anti-Bacterial Agents; Cephalosporins; Child; Dose-Response Relationship, Drug; Drug Resistance, Bacterial; Erythromycin; Haemophilus Infections; Haemophilus influenzae; Humans; Microbial Sensitivity Tests; Penicillins | 1991 |
Serologically documented loracarbef (Lorabid)-induced immune thrombocytopenia.
Topics: Autoantibodies; Blood Platelets; Cephalosporins; Female; Flow Cytometry; Humans; Methylprednisolone; Middle Aged; Purpura, Thrombocytopenic, Idiopathic; Respiratory Tract Infections | 2003 |
In vitro evaluation of Ly 163892, a new oral cephalosporin.
Topics: Anti-Bacterial Agents; Bacteria; Cefaclor; Cephalosporins; Microbial Sensitivity Tests | 1989 |
Differentiation of cefaclor and its delta-3 isomer by electrospray mass spectrometry, infrared multiple photon dissociation spectroscopy and theoretical calculations.
Topics: Cefaclor; Cephalosporins; Isomerism; Quantum Theory; Spectrometry, Mass, Electrospray Ionization; Spectrophotometry, Infrared; Tandem Mass Spectrometry | 2015 |
Kinetic Study of Laboratory Mutants of NDM-1 Metallo-β-Lactamase and the Importance of an Isoleucine at Position 35.
Topics: Amino Acid Substitution; Anti-Bacterial Agents; beta-Lactam Resistance; beta-Lactamases; Biocatalysis; Catalytic Domain; Cephalosporins; Cloning, Molecular; Escherichia coli; Gene Expression; Isoleucine; Kinetics; Models, Molecular; Mutation; Protein Structure, Secondary; Recombinant Proteins; Serine; Threonine | 2016 |