celecoxib and piperidines

celecoxib has been researched along with piperidines in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's8 (40.00)29.6817
2010's8 (40.00)24.3611
2020's4 (20.00)2.80

Authors

AuthorsStudies
Cassels, A; Cole, C; Hughes, MA; Lexchin, J; McCormack, JP; Mintzes, B1
O'Brien, LA; Sutherland, JJ; Weaver, DF1
Chichorro, JG; Rae, GA; Souza, GE; Zampronio, AR1
Ballabh, P; Braun, A; Csiszar, A; Goldman, SA; Hu, F; Lou, N; Nedergaard, M; Rivera, A; Smith, K; Ungvari, Z; Xu, H1
Sharma, B; Singh, M; Singh, N1
Jaggi, AS; Sharma, B; Singh, M; Singh, N1
Bosetti, F; Tomita, YA; Toscano, CD; Ueda, Y; Vicini, S1
Antunes, E; Desouza, IA; Ferreira, T; Macedo, ML; Mariano, NS; Mello, GC1
Abdellatif, KR; Chowdhury, MA; Das, D; Dong, Y; Huang, Z; Knaus, EE; Rahman, M; Suresh, MR; Velázquez, CA; Yu, G1
Bakhle, YS; Camêlo, VM; Dos Reis, WG; Faraco, A; Francischi, JN; Paiva-Lima, P; Rezende, RM1
Bastos-Pereira, AL; Fraga, D; Leite, MC; Zampronio, AR1
Adinolfi, B; Breschi, MC; Carpi, S; Costa, B; Da Pozzo, E; Fogli, S; Martini, C; Nieri, P; Pellegrino, M; Podestà, A; Romanini, A1
Chen, JM; Chen, S; Du, W; Huang, W; Liu, J; Liu, RY; Pan, C; Shen, J; Wu, J; Zhou, L; Zhou, Y; Zhu, X1
Baset, MA; El-Eraky, WI; Fahmy, HH; Khalifa, NM; Nossier, ES1
Bastos-Pereira, AL; Dreifuss, AA; Fraga, D; Zampronio, AR1
Hammock, BD; Harris, TR; Hwang, SH; Imai, DM; Kodani, S; Rand, AA; Yang, J1
Bortolanza, M; Crivelaro do Nascimento, G; Del Bel, EA; Ferrari, DP; Ferreira-Junior, NC; Guimaraes, FS1
McDougall, JJ; Philpott, HT1
Jaisin, Y; Malaniyom, K; Natewong, S; Ratanachamnong, P; Watthammawut, A; Wongsawatkul, O1
Chaturvedi, S; Dewangan, J; Divakar, A; Kumar, S; Mishra, S; Rath, SK; Srivastava, S; Wahajuddin, M1

Other Studies

20 other study(ies) available for celecoxib and piperidines

ArticleYear
Drugs in the news: an analysis of Canadian newspaper coverage of new prescription drugs.
    CMAJ : Canadian Medical Association journal = journal de l'Association medicale canadienne, 2003, Apr-29, Volume: 168, Issue:9

    Topics: Acetamides; Advertising; Anti-Inflammatory Agents, Non-Steroidal; Anticholesteremic Agents; Antiviral Agents; Atorvastatin; Bibliometrics; Canada; Celecoxib; Cholinesterase Inhibitors; Consumer Product Safety; Disclosure; Donepezil; Drug Industry; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Estrogen Antagonists; Heptanoic Acids; Humans; Indans; Newspapers as Topic; Oseltamivir; Patient Education as Topic; Piperidines; Pyrazoles; Pyrroles; Raloxifene Hydrochloride; Sulfonamides

2003
Pruned receptor surface models and pharmacophores for three-dimensional database searching.
    Journal of medicinal chemistry, 2004, Jul-15, Volume: 47, Issue:15

    Topics: Amidines; Angiotensin-Converting Enzyme Inhibitors; Benzodiazepines; Celecoxib; Cholinesterase Inhibitors; Cyclooxygenase 2; Databases, Factual; Donepezil; Enalapril; Enzymes; Estradiol; Imidazoles; Indans; Isoenzymes; Ligands; Models, Molecular; Molecular Structure; Naphthalenes; Piperidines; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Quantitative Structure-Activity Relationship; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Estrogen; Receptors, GABA-A; Sulfonamides; Thrombin

2004
Orofacial cold hyperalgesia due to infraorbital nerve constriction injury in rats: reversal by endothelin receptor antagonists but not non-steroidal anti-inflammatory drugs.
    Pain, 2006, Volume: 123, Issue:1-2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Atrasentan; Bosentan; Carrageenan; Celecoxib; Cold Temperature; Dexamethasone; Disease Models, Animal; Drug Evaluation, Preclinical; Endothelin-1; Endothelins; Grooming; Hyperalgesia; Indomethacin; Male; Maxillary Nerve; Nerve Compression Syndromes; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Piperidines; Pyrazoles; Pyrrolidines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B; Sulfonamides; Trigeminal Neuralgia

2006
Angiogenic inhibition reduces germinal matrix hemorrhage.
    Nature medicine, 2007, Volume: 13, Issue:4

    Topics: Aborted Fetus; Angiopoietin-2; Animals; Blotting, Western; Brain; Celecoxib; Cell Proliferation; Cyclooxygenase 2 Inhibitors; Endothelial Cells; Humans; Immunohistochemistry; Infant, Newborn; Infant, Premature; Intracranial Hemorrhages; Neovascularization, Physiologic; Piperidines; Pyrazoles; Quinazolines; Rabbits; Sulfonamides; Vascular Endothelial Growth Factor Receptor-2

2007
Modulation of celecoxib- and streptozotocin-induced experimental dementia of Alzheimer's disease by pitavastatin and donepezil.
    Journal of psychopharmacology (Oxford, England), 2008, Volume: 22, Issue:2

    Topics: Acetylcholinesterase; Administration, Oral; Alzheimer Disease; Animals; Brain; Celecoxib; Disease Models, Animal; Donepezil; Dose-Response Relationship, Drug; Drug Therapy, Combination; Escape Reaction; Female; Glutathione; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Indans; Injections, Intraventricular; Male; Maze Learning; Mental Recall; Mice; Nootropic Agents; Piperidines; Pyrazoles; Quinolines; Streptozocin; Sulfonamides; Thiobarbituric Acid Reactive Substances

2008
Exploitation of HIV protease inhibitor Indinavir as a memory restorative agent in experimental dementia.
    Pharmacology, biochemistry, and behavior, 2008, Volume: 89, Issue:4

    Topics: Acetylcholinesterase; Animals; Antibiotics, Antineoplastic; Brain; Celecoxib; Cyclooxygenase Inhibitors; Dementia; Donepezil; Female; Glutathione; HIV Protease Inhibitors; Indans; Indinavir; Male; Maze Learning; Memory; Memory Disorders; Mice; Nootropic Agents; Oxidative Stress; Piperidines; Pyrazoles; Streptozocin; Sulfonamides; Thiobarbituric Acid Reactive Substances

2008
Altered GABAergic neurotransmission is associated with increased kainate-induced seizure in prostaglandin-endoperoxide synthase-2 deficient mice.
    Brain research bulletin, 2008, Mar-28, Volume: 75, Issue:5

    Topics: Analysis of Variance; Animals; Autoradiography; Celecoxib; Chromatography, High Pressure Liquid; Cyclooxygenase 1; Cyclooxygenase 2; Enzyme-Linked Immunosorbent Assay; gamma-Aminobutyric Acid; Hippocampus; Kainic Acid; Male; Membrane Potentials; Membrane Proteins; Mice; Mice, Knockout; Neurons; Patch-Clamp Techniques; Piperidines; Pyrazoles; Seizures; Statistics, Nonparametric; Sulfonamides; Synaptic Transmission

2008
Mechanisms involved in the rat peritoneal leukocyte migration induced by a Kunitz-type inhibitor isolated from Dimorphandra mollis seeds.
    Toxicon : official journal of the International Society on Toxinology, 2009, Mar-01, Volume: 53, Issue:3

    Topics: Analysis of Variance; Animals; Benzoquinones; Celecoxib; Cell Movement; Dexamethasone; Fabaceae; Indomethacin; Inflammation; Leukocytes; Male; NG-Nitroarginine Methyl Ester; Peptides; Peritoneal Lavage; Piperidines; Plant Proteins; Pyrazoles; Quinuclidines; Rats; Rats, Wistar; Seeds; Sulfonamides

2009
Celecoxib analogs possessing a N-(4-nitrooxybutyl)piperidin-4-yl or N-(4-nitrooxybutyl)-1,2,3,6-tetrahydropyridin-4-yl nitric oxide donor moiety: synthesis, biological evaluation and nitric oxide release studies.
    Bioorganic & medicinal chemistry letters, 2010, Feb-15, Volume: 20, Issue:4

    Topics: Animals; Anti-Inflammatory Agents; Aspirin; Celecoxib; Crystallography, X-Ray; Cyclooxygenase 2 Inhibitors; Humans; Hydrogen-Ion Concentration; Ibuprofen; Inhibitory Concentration 50; Molecular Structure; Nitric Oxide; Nitric Oxide Donors; Piperidines; Prodrugs; Pyrazoles; Rats; Sheep; Structure-Activity Relationship; Sulfonamides

2010
Endogenous opioid and cannabinoid mechanisms are involved in the analgesic effects of celecoxib in the central nervous system.
    Pharmacology, 2012, Volume: 89, Issue:3-4

    Topics: Analgesics; Animals; Carrageenan; Celecoxib; Central Nervous System; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Inflammation; Male; Naltrexone; Pain; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Opioid, delta; Receptors, Opioid, mu; Sulfonamides

2012
Central mediators involved in the febrile response induced by polyinosinic-polycytidylic acid: lack of involvement of endothelins and substance P.
    Journal of neuroimmunology, 2015, Jan-15, Volume: 278

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antibodies; Body Temperature; Celecoxib; Central Nervous System; Cytokines; Dinoprostone; Endothelin B Receptor Antagonists; Fever; Indomethacin; Interferon Inducers; Male; Oligopeptides; Peptides; Piperidines; Poly I-C; Pyrazoles; Rats; Rats, Wistar; Sulfonamides; Tropanes

2015
AM251 induces apoptosis and G2/M cell cycle arrest in A375 human melanoma cells.
    Anti-cancer drugs, 2015, Volume: 26, Issue:7

    Topics: Antineoplastic Agents; Apoptosis; Calcium Channels; Celecoxib; Cell Line, Tumor; Cell Survival; Cyclic AMP; Cyclooxygenase 2; Drug Inverse Agonism; Drug Synergism; G2 Phase Cell Cycle Checkpoints; Humans; Melanoma; Mutation; Nerve Tissue Proteins; Piperidines; Proto-Oncogene Proteins B-raf; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Cannabinoid; Receptors, G-Protein-Coupled; Skin Neoplasms; Sulfonamides; Transient Receptor Potential Channels; TRPA1 Cation Channel

2015
ZD6474, a new treatment strategy for human osteosarcoma, and its potential synergistic effect with celecoxib.
    Oncotarget, 2015, Aug-28, Volume: 6, Issue:25

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Bone Neoplasms; Celecoxib; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Dose-Response Relationship, Drug; Down-Regulation; Drug Synergism; ErbB Receptors; Female; G1 Phase; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Humans; Mice; Mice, Inbred BALB C; Mice, Nude; Osteosarcoma; Phosphorylation; Piperidines; Quinazolines; Xenograft Model Antitumor Assays

2015
Design and Synthesis of Novel Pyrazole-Substituted Different Nitrogenous Heterocyclic Ring Systems as Potential Anti-Inflammatory Agents.
    Molecules (Basel, Switzerland), 2017, Mar-24, Volume: 22, Issue:4

    Topics: Animals; Anti-Inflammatory Agents; Carrageenan; Celecoxib; Cyclooxygenase Inhibitors; Drug Design; Edema; Heterocyclic Compounds; Injections; Male; Molecular Docking Simulation; Piperidines; Pyrazoles; Rats; Rimonabant

2017
Central mediators of the zymosan-induced febrile response.
    Journal of basic and clinical physiology and pharmacology, 2017, Nov-27, Volume: 28, Issue:6

    Topics: Animals; Body Temperature; Celecoxib; Dinoprostone; Fever; Indomethacin; Infusions, Intraventricular; Injections, Intra-Articular; Injections, Intraperitoneal; Male; Oligopeptides; Peptide Fragments; Piperidines; Rats; Somatostatin; Tropanes; Zymosan

2017
Celecoxib Does Not Protect against Fibrosis and Inflammation in a Carbon Tetrachloride-Induced Model of Liver Injury.
    Molecular pharmacology, 2018, Volume: 94, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carbon Tetrachloride; Celecoxib; Collagen; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Dinoprostone; Disease Models, Animal; Enzyme Inhibitors; Epoxide Hydrolases; Liver Cirrhosis; Male; Mice; Phenylurea Compounds; Piperidines

2018
Cannabidiol increases the nociceptive threshold in a preclinical model of Parkinson's disease.
    Neuropharmacology, 2020, Volume: 163

    Topics: Amidohydrolases; Analgesics; Animals; Benzamides; Brain; Cannabidiol; Capsaicin; Carbamates; Celecoxib; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Morphine; Nociception; Oxidopamine; Pain; Parkinson Disease; Piperidines; Pyrazoles; Thienamycins

2020
Combatting joint pain and inflammation by dual inhibition of monoacylglycerol lipase and cyclooxygenase-2 in a rat model of osteoarthritis.
    Arthritis research & therapy, 2020, 01-14, Volume: 22, Issue:1

    Topics: Animals; Anti-Inflammatory Agents; Arthralgia; Benzodioxoles; Celecoxib; Cyclooxygenase 2 Inhibitors; Disease Models, Animal; Drug Therapy, Combination; Enzyme Inhibitors; Inflammation; Knee Joint; Male; Monoacylglycerol Lipases; Osteoarthritis, Knee; Piperidines; Rats; Rats, Wistar

2020
Antioxidant and anti-inflammatory effects of piperine on UV-B-irradiated human HaCaT keratinocyte cells.
    Life sciences, 2020, Dec-15, Volume: 263

    Topics: Alkaloids; Anti-Inflammatory Agents; Antioxidants; Apoptosis; Benzodioxoles; Celecoxib; Cell Line; Dose-Response Relationship, Drug; Humans; Inflammation; Keratinocytes; Piperidines; Polyunsaturated Alkamides; Skin; Ultraviolet Rays

2020
Piperine and Celecoxib synergistically inhibit colon cancer cell proliferation via modulating Wnt/β-catenin signaling pathway.
    Phytomedicine : international journal of phytotherapy and phytopharmacology, 2021, Volume: 84

    Topics: Alkaloids; Animals; Antineoplastic Agents; Apoptosis; Benzodioxoles; beta Catenin; Celecoxib; Cell Line, Tumor; Cell Proliferation; Cell Survival; Colonic Neoplasms; Cyclooxygenase 2 Inhibitors; Drug Synergism; Humans; Mice; Piperidines; Polyunsaturated Alkamides; Rats; Wnt Signaling Pathway

2021