Page last updated: 2024-09-03

celastrol and tacrolimus

celastrol has been researched along with tacrolimus in 3 studies

Compound Research Comparison

Studies
(celastrol)
Trials
(celastrol)
Recent Studies (post-2010)
(celastrol)
Studies
(tacrolimus)
Trials
(tacrolimus)
Recent Studies (post-2010) (tacrolimus)
885174117,7572,3196,661

Protein Interaction Comparison

ProteinTaxonomycelastrol (IC50)tacrolimus (IC50)
Bile salt export pumpHomo sapiens (human)7.18
Cytochrome P450 3A4Homo sapiens (human)0.58
Cytochrome P450 3A5Homo sapiens (human)0.385
Serine/threonine-protein kinase mTORHomo sapiens (human)0.0021
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)0.2547
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoformHomo sapiens (human)0.0148
Splicing factor 3B subunit 3Homo sapiens (human)0.0123
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)3.3
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)3.7

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's1 (33.33)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Dong, G; Liu, N; Sheng, C; Tu, J; Wang, Y1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Fukazawa, T; Kubo, T; Kunieda, T; Naora, Y1

Reviews

1 review(s) available for celastrol and tacrolimus

ArticleYear
Emerging New Targets for the Treatment of Resistant Fungal Infections.
    Journal of medicinal chemistry, 2018, 07-12, Volume: 61, Issue:13

    Topics: Antifungal Agents; Drug Resistance, Fungal; Humans; Molecular Targeted Therapy; Mycoses

2018

Other Studies

2 other study(ies) available for celastrol and tacrolimus

ArticleYear
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Suppression of the immune response potentiates tadpole tail regeneration during the refractory period.
    Development (Cambridge, England), 2009, Volume: 136, Issue:14

    Topics: Animals; Base Sequence; Chemokines; Cyclosporine; Gene Expression Profiling; Immunosuppressive Agents; Larva; Oligodeoxyribonucleotides, Antisense; Pentacyclic Triterpenes; Proto-Oncogene Proteins; Regeneration; T-Lymphocytes, Regulatory; Tacrolimus; Tail; Time Factors; Trans-Activators; Triterpenes; Xenopus laevis; Xenopus Proteins

2009