Page last updated: 2024-09-03

celastrol and gedunin

celastrol has been researched along with gedunin in 5 studies

Compound Research Comparison

Studies
(celastrol)
Trials
(celastrol)
Recent Studies (post-2010)
(celastrol)
Studies
(gedunin)
Trials
(gedunin)
Recent Studies (post-2010) (gedunin)
885174161045
88517411906

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (40.00)29.6817
2010's3 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chiosis, G; Clardy, J; Clement, C; Du, J; Golub, TR; Hahn, WC; Hieronymus, H; Lamb, J; Maloney, KN; Nieto, M; Peng, XP; Raj, SM; Rodina, A; Ross, KN; Stegmaier, K1
Ansar, S; Blagg, BS; Lu, Y; Michaelis, ML1
Blagg, BS; Brandt, GE; Dixit, A; Donnelly, AC; Lu, Y; Matts, RL; Mollapour, M; Neckers, L; Verkhivker, G; Wang, S1
Blagg, BS; Halaweish, F; Hall, JA; Kopel, L; Rice, N; Seedarala, S1
Abdeen, S; Chapman, E; Chitre, S; Hoang, QQ; Johnson, SM; Park, Y; Ray, AM; Salim, N; Sivinski, J; Stevens, M; Washburn, A1

Other Studies

5 other study(ies) available for celastrol and gedunin

ArticleYear
Gene expression signature-based chemical genomic prediction identifies a novel class of HSP90 pathway modulators.
    Cancer cell, 2006, Volume: 10, Issue:4

    Topics: Antibiotics, Antineoplastic; Benzoquinones; Biomarkers, Tumor; Cell Culture Techniques; Cell Line; Cell Line, Tumor; Cell Survival; ErbB Receptors; fms-Like Tyrosine Kinase 3; Fusion Proteins, bcr-abl; Gene Expression; Gene Expression Profiling; Genome, Human; HSP90 Heat-Shock Proteins; Humans; Inhibitory Concentration 50; Lactams, Macrocyclic; Limonins; Male; Metribolone; Pentacyclic Triterpenes; Prostatic Neoplasms; Receptors, Androgen; Reproducibility of Results; RNA, Messenger; Triterpenes

2006
Neuroprotective activity and evaluation of Hsp90 inhibitors in an immortalized neuronal cell line.
    Bioorganic & medicinal chemistry, 2009, Feb-15, Volume: 17, Issue:4

    Topics: Cell Death; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; HSP90 Heat-Shock Proteins; Humans; Models, Neurological; Neurons; Neuroprotective Agents; Novobiocin

2009
A systematic protocol for the characterization of Hsp90 modulators.
    Bioorganic & medicinal chemistry, 2011, Jan-01, Volume: 19, Issue:1

    Topics: Benzoquinones; Cell Line, Tumor; Chromatography, Affinity; HSP90 Heat-Shock Proteins; Humans; Hydrolysis; Immunoprecipitation; Lactams, Macrocyclic; Models, Molecular; Novobiocin; Pentacyclic Triterpenes; Triterpenes

2011
Cucurbitacin D Is a Disruptor of the HSP90 Chaperone Machinery.
    Journal of natural products, 2015, Apr-24, Volume: 78, Issue:4

    Topics: Benzoquinones; Cucurbitaceae; DNA-Binding Proteins; Heat Shock Transcription Factors; HSP90 Heat-Shock Proteins; Humans; Lactams, Macrocyclic; MCF-7 Cells; Molecular Chaperones; Molecular Structure; Neoplasms; Transcription Factors; Triterpenes

2015
HSP60/10 chaperonin systems are inhibited by a variety of approved drugs, natural products, and known bioactive molecules.
    Bioorganic & medicinal chemistry letters, 2019, 05-01, Volume: 29, Issue:9

    Topics: Biological Products; Chaperonin 10; Chaperonin 60; Escherichia coli; Humans; Inhibitory Concentration 50; Protein Folding; Rafoxanide; Salicylanilides; Suramin

2019