Page last updated: 2024-09-03

celastrol and epoxomicin

celastrol has been researched along with epoxomicin in 2 studies

Compound Research Comparison

Studies
(celastrol)
Trials
(celastrol)
Recent Studies (post-2010)
(celastrol)
Studies
(epoxomicin)
Trials
(epoxomicin)
Recent Studies (post-2010) (epoxomicin)
88517412510111

Protein Interaction Comparison

ProteinTaxonomycelastrol (IC50)epoxomicin (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.98
Proteasome subunit beta type-1Homo sapiens (human)1.25
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.98
Proteasome subunit beta type-5Homo sapiens (human)0.0256
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.98
Proteasome subunit beta type-2Homo sapiens (human)0.57
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.98
GABA theta subunitRattus norvegicus (Norway rat)0.98
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.98

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Leibel, R; Tortoriello, DV; Weisberg, S1

Other Studies

2 other study(ies) available for celastrol and epoxomicin

ArticleYear
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Proteasome inhibitors, including curcumin, improve pancreatic β-cell function and insulin sensitivity in diabetic mice.
    Nutrition & diabetes, 2016, Apr-25, Volume: 6

    Topics: 3T3-L1 Cells; Animals; Body Composition; Cell Survival; Curcumin; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Dietary Supplements; Glycated Hemoglobin; Homeostasis; Hyperglycemia; Insulin; Insulin Resistance; Insulin Secretion; Insulin-Secreting Cells; Male; Mice; Mice, Inbred C57BL; Obesity; Oligopeptides; Pentacyclic Triterpenes; Polyphenols; Proteasome Inhibitors; Receptors, Leptin; Triterpenes

2016