Page last updated: 2024-09-03

celastrol and axitinib

celastrol has been researched along with axitinib in 1 studies

Compound Research Comparison

Studies
(celastrol)
Trials
(celastrol)
Recent Studies (post-2010)
(celastrol)
Studies
(axitinib)
Trials
(axitinib)
Recent Studies (post-2010) (axitinib)
8851741765145683

Protein Interaction Comparison

ProteinTaxonomycelastrol (IC50)axitinib (IC50)
Serine/threonine-protein kinase PLK4Homo sapiens (human)0.045
Tyrosine-protein kinase ABL1Homo sapiens (human)0.0658
Cytochrome P450 3A4Homo sapiens (human)0.046
Vascular endothelial growth factor receptor 1 Homo sapiens (human)0.0001
Vascular endothelial growth factor receptor 3Homo sapiens (human)0.0001
Vascular endothelial growth factor receptor 2Homo sapiens (human)0.0079
Serine/threonine-protein kinase TBK1Homo sapiens (human)0.47

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Choi, HG; Choi, JY; Jeong, JH; Kim, J; Kim, JO; Kim, JR; Kim, SY; Ku, SK; Ramasamy, T; Yong, CS; Youn, YS1

Other Studies

1 other study(ies) available for celastrol and axitinib

ArticleYear
PEGylated lipid bilayer-supported mesoporous silica nanoparticle composite for synergistic co-delivery of axitinib and celastrol in multi-targeted cancer therapy.
    Acta biomaterialia, 2016, 07-15, Volume: 39

    Topics: Animals; Axitinib; Cell Line, Tumor; Drug Delivery Systems; Drug Screening Assays, Antitumor; Female; Imidazoles; Indazoles; Lipid Bilayers; Mice; Mice, Inbred BALB C; Mice, Nude; Nanoparticles; Neoplasms, Experimental; Pentacyclic Triterpenes; Porosity; Silicon Dioxide; Triterpenes

2016