Page last updated: 2024-09-03

celastrol and acetyl isogambogic acid

celastrol has been researched along with acetyl isogambogic acid in 2 studies

Compound Research Comparison

Studies
(celastrol)
Trials
(celastrol)
Recent Studies (post-2010)
(celastrol)
Studies
(acetyl isogambogic acid)
Trials
(acetyl isogambogic acid)
Recent Studies (post-2010) (acetyl isogambogic acid)
8851741504

Protein Interaction Comparison

ProteinTaxonomycelastrol (IC50)acetyl isogambogic acid (IC50)
Ubiquitin carboxyl-terminal hydrolase 2Homo sapiens (human)5.4
Ubiquitin carboxyl-terminal hydrolase isozyme L1Homo sapiens (human)5.4
Ubiquitin carboxyl-terminal hydrolase isozyme L3Homo sapiens (human)5.4
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)5.3703
Ubiquitin carboxyl-terminal hydrolase 15Homo sapiens (human)5.4
Ubiquitin carboxyl-terminal hydrolase isozyme L5Homo sapiens (human)5.4
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)4.0738

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baljinnyam, B; Jadhav, A; Ott, CA; Simeonov, A; Zakharov, AV; Zhuang, Z1
Abbas, S; Bhoumik, A; Cosford, ND; Dahl, R; Krajewski, S; Ronai, ZA; Vasile, S1

Other Studies

2 other study(ies) available for celastrol and acetyl isogambogic acid

ArticleYear
Cell Lysate-Based AlphaLISA Deubiquitinase Assay Platform for Identification of Small Molecule Inhibitors.
    ACS chemical biology, 2017, 09-15, Volume: 12, Issue:9

    Topics: Drug Evaluation, Preclinical; Enzyme Assays; Enzyme Inhibitors; HEK293 Cells; High-Throughput Screening Assays; Humans; Small Molecule Libraries; Ubiquitin Thiolesterase

2017
Preclinical studies of celastrol and acetyl isogambogic acid in melanoma.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2007, Nov-15, Volume: 13, Issue:22 Pt 1

    Topics: Activating Transcription Factor 2; Animals; Cell Line, Tumor; Chromones; Drug Evaluation, Preclinical; Drug Screening Assays, Antitumor; Humans; MAP Kinase Kinase 4; Melanoma; Mice; Pentacyclic Triterpenes; Proto-Oncogene Proteins c-jun; Skin Neoplasms; Small Molecule Libraries; Transcription, Genetic; Triterpenes

2007