Page last updated: 2024-09-04

cdri 85-287 and diethylstilbestrol

cdri 85-287 has been researched along with diethylstilbestrol in 2 studies

Compound Research Comparison

Studies
(cdri 85-287)
Trials
(cdri 85-287)
Recent Studies (post-2010)
(cdri 85-287)
Studies
(diethylstilbestrol)
Trials
(diethylstilbestrol)
Recent Studies (post-2010) (diethylstilbestrol)
22038,585322491

Protein Interaction Comparison

ProteinTaxonomycdri 85-287 (IC50)diethylstilbestrol (IC50)
high affinity choline transporter 1 isoform aHomo sapiens (human)12.5893
Estrogen receptorHomo sapiens (human)0.1312
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)3.67
Adenosine receptor A3Homo sapiens (human)2.208
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)2.963
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)2.208
Substance-K receptorHomo sapiens (human)9.553
D(1A) dopamine receptorHomo sapiens (human)7.763
Prostaglandin G/H synthase 1Homo sapiens (human)5.6
Sodium-dependent noradrenaline transporter Homo sapiens (human)3.67
Thromboxane-A synthase Homo sapiens (human)4.359
5-hydroxytryptamine receptor 2AHomo sapiens (human)4.79
Adenosine receptor A2aHomo sapiens (human)9.013
Adenosine receptor A1Homo sapiens (human)2.856
Mu-type opioid receptorHomo sapiens (human)5.778
D(3) dopamine receptorHomo sapiens (human)8.796
Delta-type opioid receptorHomo sapiens (human)2.718
Kappa-type opioid receptorHomo sapiens (human)4.563
5-hydroxytryptamine receptor 2BHomo sapiens (human)3.14
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)2.208
Sodium-dependent dopamine transporter Homo sapiens (human)1.071
Aldehyde oxidaseHomo sapiens (human)0.46
Estrogen receptor betaHomo sapiens (human)0.1588
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)0.5

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kon, OL; Ng, SC; Sim, KY; Teo, CC1
Dwivedi, A; Kamboj, VP; Setty, BS; Singh, MM; Sreenivasulu, S1

Other Studies

2 other study(ies) available for cdri 85-287 and diethylstilbestrol

ArticleYear
Synthesis of 2-(p-chlorobenzyl)-3-aryl-6-methoxybenzofurans as selective ligands for antiestrogen-binding sites. Effects on cell proliferation and cholesterol synthesis.
    Journal of medicinal chemistry, 1992, Apr-17, Volume: 35, Issue:8

    Topics: Benzofurans; Binding Sites; Binding, Competitive; Cell Division; Cell Line; Cholesterol; Estrogen Antagonists; Humans; Ligands; Receptors, Estrogen; Thymidine

1992
CDRI-85/287, a novel antiestrogen and antiimplantation agent: biological profile and interaction with the estrogen receptors in immature rat uterus.
    Contraception, 1992, Volume: 45, Issue:1

    Topics: Animals; Benzopyrans; Cell Nucleus; Corpus Luteum; Cytosol; Diethylstilbestrol; Embryo Implantation; Estradiol; Estrogen Antagonists; Female; Organ Size; Ovariectomy; Piperidines; Pregnancy; Rats; Rats, Inbred Strains; Receptors, Estrogen; Sexual Maturation; Uterus

1992