Page last updated: 2024-09-03

cd 349 and nicardipine

cd 349 has been researched along with nicardipine in 4 studies

Compound Research Comparison

Studies
(cd 349)
Trials
(cd 349)
Recent Studies (post-2010)
(cd 349)
Studies
(nicardipine)
Trials
(nicardipine)
Recent Studies (post-2010) (nicardipine)
23002,646444312

Protein Interaction Comparison

ProteinTaxonomycd 349 (IC50)nicardipine (IC50)
Bile salt export pumpHomo sapiens (human)8.314
ATP-dependent translocase ABCB1Mus musculus (house mouse)8
ATP-dependent translocase ABCB1Homo sapiens (human)4.2992
Cytochrome P450 3A4Homo sapiens (human)0.42
Cytochrome P450 2C9 Homo sapiens (human)1.69
ATP-dependent translocase ABCB1Mus musculus (house mouse)2.5
Cytochrome P450 2J2Homo sapiens (human)1.69
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)4.925
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)4.8

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19902 (50.00)18.7374
1990's2 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kamata, K; Kasuya, Y; Miyata, N; Nishiyama, H2
Hidaka, H; Matsushima, S; Saitoh, M; Tanaka, T; Watanabe, M1
Aihara, H; Kaneko, K; Tsuchida, K; Yamazaki, R1

Other Studies

4 other study(ies) available for cd 349 and nicardipine

ArticleYear
Effects of CD-349, a dihydropyridine derivative, on contraction induced by vasoactive agents in canine basilar artery after subarachnoid hemorrhage.
    Research communications in chemical pathology and pharmacology, 1991, Volume: 72, Issue:2

    Topics: Animals; Basilar Artery; Calcium; Dihydropyridines; Dogs; Endothelium, Vascular; In Vitro Techniques; Male; Methylene Blue; Nicardipine; Potassium; Serotonin; Subarachnoid Hemorrhage; Tetradecanoylphorbol Acetate; Vasoconstriction

1991
Changes in responsiveness of the canine basilar artery to endothelin-1 after subarachnoid hemorrhage.
    Life sciences, 1991, Volume: 49, Issue:3

    Topics: Animals; Basilar Artery; Calcium; Calcium Channel Blockers; Dihydropyridines; Dogs; Endothelins; In Vitro Techniques; Male; Muscle Contraction; Nicardipine; Subarachnoid Hemorrhage; Tetradecanoylphorbol Acetate

1991
Different sensitivities of Ca2+, calmodulin-dependent cyclic nucleotide phosphodiesterases from rabbit aorta and brain to dihydropyridine calcium channel blockers.
    Biochemical and biophysical research communications, 1987, Nov-13, Volume: 148, Issue:3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Aorta; Brain; Calcium Channel Blockers; Cyclic Nucleotide Phosphodiesterases, Type 1; Dihydropyridines; Enzyme Activation; In Vitro Techniques; Kinetics; Nicardipine; Nimodipine; Nucleotides, Cyclic; Phosphodiesterase Inhibitors; Rabbits

1987
Effects of the new calcium antagonist 2-nitratopropyl-3-nitratopropyl-2,6-dimethyl-4-(3-nitrophe nyl)- 1,4-dihydropyridine-3,5-dicarboxylate on cerebral circulation in dogs.
    Arzneimittel-Forschung, 1987, Volume: 37, Issue:11

    Topics: Animals; Basilar Artery; Calcium Channel Blockers; Cerebrovascular Circulation; Dihydropyridines; Dinoprost; Dogs; Female; Heart Rate; Hemodynamics; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Nimodipine; Potassium Chloride; Prostaglandins F; Serotonin

1987