Page last updated: 2024-09-04

caseins and elacridar

caseins has been researched along with elacridar in 2 studies

Compound Research Comparison

Studies
(caseins)
Trials
(caseins)
Recent Studies (post-2010)
(caseins)
Studies
(elacridar)
Trials
(elacridar)
Recent Studies (post-2010) (elacridar)
16,8635614,1702848119

Protein Interaction Comparison

ProteinTaxonomycaseins (IC50)elacridar (IC50)
ATP-dependent translocase ABCB1Homo sapiens (human)0.4427
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)0.2852

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Danielsson, L; Oskarsson, A; Tallkvist, J; Yagdiran, Y1
Assaraf, YG; Bar-Zeev, M; Kelmansky, D; Livney, YD1

Other Studies

2 other study(ies) available for caseins and elacridar

ArticleYear
A model of secreting murine mammary epithelial HC11 cells comprising endogenous Bcrp/Abcg2 expression and function.
    Cell biology and toxicology, 2015, Volume: 31, Issue:2

    Topics: Acridines; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Caseins; Cell Differentiation; Cell Line; Epithelial Cells; Female; Gene Expression Regulation; Hydrocortisone; Mammary Glands, Animal; Mice; Mitoxantrone; Models, Biological; Prolactin; RNA, Small Interfering; Signal Transduction; Tetrahydroisoquinolines

2015
β-Casein micelles for oral delivery of SN-38 and elacridar to overcome BCRP-mediated multidrug resistance in gastric cancer.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 2018, Volume: 133

    Topics: Acridines; Administration, Oral; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; Caseins; Cell Line, Tumor; Drug Delivery Systems; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Irinotecan; Micelles; Nanoparticles; Neoplasm Proteins; Stomach Neoplasms; Tetrahydroisoquinolines

2018