Page last updated: 2024-09-04

cariporide and tetrodotoxin

cariporide has been researched along with tetrodotoxin in 3 studies

Compound Research Comparison

Studies
(cariporide)
Trials
(cariporide)
Recent Studies (post-2010)
(cariporide)
Studies
(tetrodotoxin)
Trials
(tetrodotoxin)
Recent Studies (post-2010) (tetrodotoxin)
409107912,992111,477
409107920015

Protein Interaction Comparison

ProteinTaxonomycariporide (IC50)tetrodotoxin (IC50)
Sodium channel protein type 9 subunit alphaHomo sapiens (human)0.0203
Sodium channel protein type 11 subunit alphaRattus norvegicus (Norway rat)1
Sodium channel protein type 1 subunit alphaRattus norvegicus (Norway rat)0.01
Sodium channel protein type 2 subunit alphaRattus norvegicus (Norway rat)0.0093
Sodium channel protein type 3 subunit alphaRattus norvegicus (Norway rat)0.015
Sodium channel protein type 5 subunit alphaRattus norvegicus (Norway rat)2
Sodium channel protein type 1 subunit alphaHomo sapiens (human)0.017
Sodium channel protein type 4 subunit alphaHomo sapiens (human)0.0209
Sodium channel protein type 7 subunit alphaHomo sapiens (human)0.036
Sodium channel protein type 5 subunit alphaHomo sapiens (human)1
Sodium channel protein type 2 subunit alphaHomo sapiens (human)0.022
Sodium channel protein type 3 subunit alphaHomo sapiens (human)0.0176
Sodium channel protein type 11 subunit alphaHomo sapiens (human)0.03
Sodium channel protein type 8 subunit alphaHomo sapiens (human)0.0161
Sodium channel protein type 8 subunit alphaMus musculus (house mouse)0.006

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Eng, S; Kardami, E; Maddaford, TG; Pierce, GN1
Chattou, S; Coulombe, A; Diacono, J; Feuvray, D; John, G; Le Grand, B1
Borras, M; Colpaert, F; Cuisiat, F; Le Grand, B; Létienne, R; Mas, A; Pignier, C; Rolland, F; Vacher, B1

Other Studies

3 other study(ies) available for cariporide and tetrodotoxin

ArticleYear
Protection against myocardial ischemic/reperfusion injury by inhibitors of two separate pathways of Na+ entry.
    Journal of molecular and cellular cardiology, 1998, Volume: 30, Issue:4

    Topics: Animals; Drug Interactions; Guanidines; Heart; Male; Myocardial Ischemia; Myocardial Reperfusion Injury; Rats; Rats, Sprague-Dawley; Sodium; Sodium Channel Blockers; Sodium-Hydrogen Exchangers; Sulfones; Tetrodotoxin

1998
Slowly inactivating component of sodium current in ventricular myocytes is decreased by diabetes and partially inhibited by known Na(+)-H(+)Exchange blockers.
    Journal of molecular and cellular cardiology, 2000, Volume: 32, Issue:7

    Topics: Amiloride; Animals; Anti-Arrhythmia Agents; Cells, Cultured; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Guanidines; Heart Ventricles; Lysophosphatidylcholines; Male; Myocardium; Patch-Clamp Techniques; Rats; Rats, Wistar; Sodium Channels; Sodium-Hydrogen Exchangers; Streptozocin; Sulfones; Tetrodotoxin; Veratrine

2000
Na+ currents in cardioprotection: better to be late.
    Journal of medicinal chemistry, 2009, Jul-23, Volume: 52, Issue:14

    Topics: Animals; Benzothiepins; Benzoxazoles; Cardiotonic Agents; Cell Line; Electric Conductivity; Female; Guinea Pigs; Humans; Male; Myocardial Infarction; Rats; Sodium Channel Blockers; Sodium Channels; Structure-Activity Relationship; Swine; Time Factors

2009