Page last updated: 2024-09-04

cariporide and pd 98059

cariporide has been researched along with pd 98059 in 3 studies

Compound Research Comparison

Studies
(cariporide)
Trials
(cariporide)
Recent Studies (post-2010)
(cariporide)
Studies
(pd 98059)
Trials
(pd 98059)
Recent Studies (post-2010) (pd 98059)
40910794,93931,001

Protein Interaction Comparison

ProteinTaxonomycariporide (IC50)pd 98059 (IC50)
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)2.8
Luciferin 4-monooxygenasePhotinus pyralis (common eastern firefly)6.3
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)2.8
Prostaglandin G/H synthase 1Homo sapiens (human)1
Mitogen-activated protein kinase 1Homo sapiens (human)2.8
Dual specificity mitogen-activated protein kinase kinase 2 Rattus norvegicus (Norway rat)4.2
Dual specificity mitogen-activated protein kinase kinase 1 Rattus norvegicus (Norway rat)4.2
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)2.4

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bantekas, C; Kaloyianni, M; Koliakos, G; Konstantinidis, D; Liakos, P; Trachana, V; Vafia, K1
Ajiro, Y; Giles, WR; Saegusa, N; Spitzer, KW; Stafforini, DM1
Chang, G; Li, Q; Lin, Y; Ma, L; Pang, T; Wang, C; Wang, J; Xu, H; Zhang, H; Zhang, Y1

Other Studies

3 other study(ies) available for cariporide and pd 98059

ArticleYear
Inhibition of the Na+-H+ exchanger isoform-1 and the extracellular signal-regulated kinase induces apoptosis: a time course of events.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2006, Volume: 18, Issue:4-5

    Topics: Annexin A5; Apoptosis; Caspase 3; Cation Transport Proteins; Cells, Cultured; DNA Fragmentation; DNA Replication; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Guanidines; Humans; Hydrogen-Ion Concentration; Protein Isoforms; Protein Kinase Inhibitors; Reactive Oxygen Species; Sodium; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Sulfones; Thymidine; Time Factors

2006
Platelet-activating factor stimulates sodium-hydrogen exchange in ventricular myocytes.
    American journal of physiology. Heart and circulatory physiology, 2011, Volume: 301, Issue:6

    Topics: Acidosis; Alkalosis; Animals; Azepines; Benzophenanthridines; Dose-Response Relationship, Drug; Flavonoids; Guanidines; Guinea Pigs; Heart Ventricles; Hydrogen-Ion Concentration; Indoles; Ion Transport; Maleimides; Mitogen-Activated Protein Kinase Kinases; Myocytes, Cardiac; Phospholipid Ethers; Platelet Activating Factor; Platelet Membrane Glycoproteins; Protein Kinase C; Protein Kinase Inhibitors; Receptors, G-Protein-Coupled; Signal Transduction; Sodium; Sodium-Hydrogen Exchangers; Spectrometry, Fluorescence; Sulfones; Time Factors; Triazoles

2011
CD44 targets Na(+)/H(+) exchanger 1 to mediate MDA-MB-231 cells' metastasis via the regulation of ERK1/2.
    British journal of cancer, 2014, Feb-18, Volume: 110, Issue:4

    Topics: Animals; Anti-Arrhythmia Agents; Breast Neoplasms; Calcium-Calmodulin-Dependent Protein Kinases; Cation Transport Proteins; Cell Line, Tumor; Cell Movement; Down-Regulation; Extracellular Signal-Regulated MAP Kinases; Female; Flavonoids; Gene Expression Regulation, Neoplastic; Guanidines; HL-60 Cells; Humans; Hyaluronan Receptors; Jurkat Cells; Lung Neoplasms; MAP Kinase Kinase 1; MAP Kinase Signaling System; MCF-7 Cells; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplasm Invasiveness; Protein Kinase Inhibitors; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Sulfones; Wound Healing

2014