Page last updated: 2024-09-04

cariporide and imatinib mesylate

cariporide has been researched along with imatinib mesylate in 3 studies

Compound Research Comparison

Studies
(cariporide)
Trials
(cariporide)
Recent Studies (post-2010)
(cariporide)
Studies
(imatinib mesylate)
Trials
(imatinib mesylate)
Recent Studies (post-2010) (imatinib mesylate)
409107911,4779605,773

Protein Interaction Comparison

ProteinTaxonomycariporide (IC50)imatinib mesylate (IC50)
Tyrosine-protein kinase ABL1Homo sapiens (human)0.31
Mast/stem cell growth factor receptor KitHomo sapiens (human)0.1

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Hu, R; Jin, W; Li, H; Li, Q; Lin, Y; Lu, Y; Ma, L; Pang, T; Wang, J; Wang, L1
Mihaila, RG1

Reviews

1 review(s) available for cariporide and imatinib mesylate

ArticleYear
A minireview on NHE1 inhibitors. A rediscovered hope in oncohematology.
    Biomedical papers of the Medical Faculty of the University Palacky, Olomouc, Czechoslovakia, 2015, Volume: 159, Issue:4

    Topics: Amiloride; Antineoplastic Agents; Apoptosis; Cation Transport Proteins; Cell Line, Tumor; DNA Damage; Drug Interactions; fms-Like Tyrosine Kinase 3; Genes, abl; Guanidines; Heme Oxygenase-1; Humans; Hydrogen-Ion Concentration; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Mutation; Niacinamide; Osmolar Concentration; Patents as Topic; Phenylurea Compounds; Protein Kinase Inhibitors; Signal Transduction; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Sorafenib; Sulfones; Tumor Hypoxia; Up-Regulation

2015

Other Studies

2 other study(ies) available for cariporide and imatinib mesylate

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Reversal of Imatinib resistance in BCR-ABL-positive leukemia after inhibition of the Na+/H+ exchanger.
    Cancer letters, 2011, Sep-01, Volume: 308, Issue:1

    Topics: Adolescent; Adult; Aged; Benzamides; Cell Line, Tumor; Child; Child, Preschool; Doxorubicin; Drug Resistance, Neoplasm; Drug Synergism; Female; Guanidines; Humans; Imatinib Mesylate; K562 Cells; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Male; Middle Aged; Mitogen-Activated Protein Kinases; Piperazines; Pyrimidines; Sodium-Hydrogen Exchangers; Sulfones; Young Adult

2011