Page last updated: 2024-09-04

cariporide and glyburide

cariporide has been researched along with glyburide in 5 studies

Compound Research Comparison

Studies
(cariporide)
Trials
(cariporide)
Recent Studies (post-2010)
(cariporide)
Studies
(glyburide)
Trials
(glyburide)
Recent Studies (post-2010) (glyburide)
40910796,5546201,344

Protein Interaction Comparison

ProteinTaxonomycariporide (IC50)glyburide (IC50)
ATP-binding cassette sub-family C member 9Homo sapiens (human)0.22
Bile salt export pumpRattus norvegicus (Norway rat)5.7
Bile salt export pumpHomo sapiens (human)5.5333
Cytochrome P450 2C9 Homo sapiens (human)1.602
ATP-binding cassette sub-family C member 8Homo sapiens (human)0.0043
ATP-sensitive inward rectifier potassium channel 11Homo sapiens (human)0.1121
NACHT, LRR and PYD domains-containing protein 3 Mus musculus (house mouse)10
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.8

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (20.00)18.2507
2000's3 (60.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Farhangkhgoee, P; Karmazyn, M; Mathur, S1
Jayachandran, JV; Olgin, JE; Weksler, J; Zipes, DP1
Athanatou, E; Hanrath, P; Robert, J; Schotten, U; Stellbrink, C; Zarse, M1
Eguchi, Y; Higashijima, N; Hoshiai, M; Ishida, H; Kadono, T; Nakazawa, H; Nakazawa, S; Toda, T1

Other Studies

5 other study(ies) available for cariporide and glyburide

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Cardioprotective effects of propofol and sevoflurane in ischemic and reperfused rat hearts: role of K(ATP) channels and interaction with the sodium-hydrogen exchange inhibitor HOE 642 (cariporide).
    Anesthesiology, 1999, Volume: 91, Issue:5

    Topics: Adenosine Triphosphate; Anesthetics, Inhalation; Anesthetics, Intravenous; Animals; Biotransformation; Drug Interactions; Energy Metabolism; Glyburide; Guanidines; Hemodynamics; In Vitro Techniques; Male; Methyl Ethers; Myocardial Reperfusion Injury; Potassium Channels; Propofol; Rats; Rats, Sprague-Dawley; Sevoflurane; Sodium-Hydrogen Exchangers; Sulfones; Ventricular Function, Left

1999
Role of the Na(+)/H(+) exchanger in short-term atrial electrophysiological remodeling.
    Circulation, 2000, Apr-18, Volume: 101, Issue:15

    Topics: Analysis of Variance; Animals; Anti-Arrhythmia Agents; Atrial Fibrillation; Dogs; Electrophysiology; Glyburide; Guanidines; Myocardial Ischemia; Sodium-Hydrogen Exchangers; Sulfones; Time Factors

2000
Verapamil prevents stretch-induced shortening of atrial effective refractory period in langendorff-perfused rabbit heart.
    Journal of cardiovascular electrophysiology, 2001, Volume: 12, Issue:1

    Topics: Animals; Anti-Arrhythmia Agents; Atrial Fibrillation; Atrial Function; Calcium Channel Blockers; Cardiac Pacing, Artificial; Glyburide; Guanidines; In Vitro Techniques; Myocardial Contraction; Rabbits; Refractory Period, Electrophysiological; Sulfones; Time Factors; Verapamil

2001
Na+/H+ exchanger inhibitor cariporide attenuates the mitochondrial Ca2+ overload and PTP opening.
    American journal of physiology. Heart and circulatory physiology, 2007, Volume: 293, Issue:6

    Topics: Animals; Anti-Arrhythmia Agents; Arsenicals; Calcium; Cardiotonic Agents; Decanoic Acids; Glyburide; Guanidines; Heart Ventricles; Hydroxy Acids; In Vitro Techniques; Male; Membrane Potential, Mitochondrial; Mitochondria, Heart; Mitochondrial Membrane Transport Proteins; Mitochondrial Permeability Transition Pore; Myocardial Contraction; Myocytes, Cardiac; Ouabain; Oxidative Stress; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Sodium; Sodium-Hydrogen Exchangers; Sulfones; Time Factors

2007