cariporide has been researched along with carbachol in 6 studies
Studies (cariporide) | Trials (cariporide) | Recent Studies (post-2010) (cariporide) | Studies (carbachol) | Trials (carbachol) | Recent Studies (post-2010) (carbachol) |
---|---|---|---|---|---|
409 | 10 | 79 | 13,918 | 81 | 968 |
Protein | Taxonomy | cariporide (IC50) | carbachol (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | 0.7849 | |
Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | 2.0626 | |
Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | 3.4134 | |
Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | 2.9961 | |
Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | 2.535 | |
Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | 2.9961 | |
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 2.6638 | |
Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | 4.849 | |
Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | 4.99 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (16.67) | 18.2507 |
2000's | 3 (50.00) | 29.6817 |
2010's | 2 (33.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
Bachmann, O; Gregor, M; Lamprecht, G; Seidler, U; Siegel, WK; Sonnentag, T; Weichert, A | 1 |
Bachmann, O; Heinzmann, A; Mack, A; Manns, MP; Seidler, U | 1 |
Couturier, K; Demaison, L; Dubouchaud, H; Lanson, M; Leverve, X; Vial, G | 1 |
Foskett, JK; Harlow, JM; Lee, RJ; Limberis, MP; Wilson, JM | 1 |
Biczó, G; Czepán, M; Dimaline, R; Geisz, A; Hegyi, P; Lázár, G; Lertkowit, N; Lonovics, J; Rakonczay, Z; Schnúr, A; Simonka, Z; Steele, I; Varró, A; Venglovecz, V; Wittmann, T | 1 |
6 other study(ies) available for cariporide and carbachol
Article | Year |
---|---|
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Different acid secretagogues activate different Na+/H+ exchanger isoforms in rabbit parietal cells.
Topics: Aminopyrine; Animals; Biological Transport; Carbachol; Cells, Cultured; Colforsin; Cytochalasin D; Gastric Acid; Guanidines; Histamine; Imidazoles; Kinetics; Omeprazole; Parietal Cells, Gastric; Rabbits; Sodium-Hydrogen Exchangers; Sulfones; Time Factors | 1998 |
Mechanisms of secretion-associated shrinkage and volume recovery in cultured rabbit parietal cells.
Topics: Adenosine Triphosphatases; Amiloride; Animals; Carbachol; Cell Size; Cells, Cultured; Charybdotoxin; Chloride Channels; Chromans; Colforsin; Enzyme Inhibitors; Guanidines; Hydrogen-Ion Concentration; Imidazoles; Ion Channels; KCNQ1 Potassium Channel; Nitrobenzoates; Parietal Cells, Gastric; Potassium Channel Blockers; Rabbits; Sodium-Calcium Exchanger; Sodium-Hydrogen Exchangers; Sulfonamides; Sulfones | 2007 |
Na+/H+ exchange inhibition with cariporide prevents alterations of coronary endothelial function in streptozotocin-induced diabetes.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Blood Glucose; Carbachol; Diabetes Mellitus, Experimental; Dilatation; Endothelium, Vascular; Glucose; Guanidines; Heart; Heart Function Tests; In Vitro Techniques; Lactic Acid; Male; Monocarboxylic Acid Transporters; Nitroprusside; Rats; Rats, Wistar; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Streptozocin; Sulfones; Symporters | 2008 |
HCO3(-) secretion by murine nasal submucosal gland serous acinar cells during Ca2+-stimulated fluid secretion.
Topics: Amiloride; Animals; Bicarbonates; Calcium Signaling; Carbachol; Cation Transport Proteins; Cell Size; Cells, Cultured; Chloride Channels; Chlorides; Cystic Fibrosis Transmembrane Conductance Regulator; Cytoplasm; Epithelial Cells; Exocrine Glands; Guanidines; Hydrogen-Ion Concentration; Mice; Mice, Inbred C57BL; Mice, Knockout; Nasal Mucosa; Niflumic Acid; Protein Isoforms; Sodium; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2; Sulfones | 2008 |
NHE1 activity contributes to migration and is necessary for proliferation of human gastric myofibroblasts.
Topics: Adult; Aged; Antiporters; Carbachol; Cation Transport Proteins; Cell Movement; Cell Proliferation; Female; Guanidines; Humans; Hydrogen-Ion Concentration; Insulin-Like Growth Factor II; Male; Myofibroblasts; Sodium-Bicarbonate Symporters; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchanger 3; Sodium-Hydrogen Exchangers; Stomach; Sulfones | 2012 |