Page last updated: 2024-09-04

cariporide and carbachol

cariporide has been researched along with carbachol in 6 studies

Compound Research Comparison

Studies
(cariporide)
Trials
(cariporide)
Recent Studies (post-2010)
(cariporide)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
409107913,91881968

Protein Interaction Comparison

ProteinTaxonomycariporide (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (16.67)18.2507
2000's3 (50.00)29.6817
2010's2 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Bachmann, O; Gregor, M; Lamprecht, G; Seidler, U; Siegel, WK; Sonnentag, T; Weichert, A1
Bachmann, O; Heinzmann, A; Mack, A; Manns, MP; Seidler, U1
Couturier, K; Demaison, L; Dubouchaud, H; Lanson, M; Leverve, X; Vial, G1
Foskett, JK; Harlow, JM; Lee, RJ; Limberis, MP; Wilson, JM1
Biczó, G; Czepán, M; Dimaline, R; Geisz, A; Hegyi, P; Lázár, G; Lertkowit, N; Lonovics, J; Rakonczay, Z; Schnúr, A; Simonka, Z; Steele, I; Varró, A; Venglovecz, V; Wittmann, T1

Other Studies

6 other study(ies) available for cariporide and carbachol

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Different acid secretagogues activate different Na+/H+ exchanger isoforms in rabbit parietal cells.
    The American journal of physiology, 1998, Volume: 275, Issue:5

    Topics: Aminopyrine; Animals; Biological Transport; Carbachol; Cells, Cultured; Colforsin; Cytochalasin D; Gastric Acid; Guanidines; Histamine; Imidazoles; Kinetics; Omeprazole; Parietal Cells, Gastric; Rabbits; Sodium-Hydrogen Exchangers; Sulfones; Time Factors

1998
Mechanisms of secretion-associated shrinkage and volume recovery in cultured rabbit parietal cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2007, Volume: 292, Issue:3

    Topics: Adenosine Triphosphatases; Amiloride; Animals; Carbachol; Cell Size; Cells, Cultured; Charybdotoxin; Chloride Channels; Chromans; Colforsin; Enzyme Inhibitors; Guanidines; Hydrogen-Ion Concentration; Imidazoles; Ion Channels; KCNQ1 Potassium Channel; Nitrobenzoates; Parietal Cells, Gastric; Potassium Channel Blockers; Rabbits; Sodium-Calcium Exchanger; Sodium-Hydrogen Exchangers; Sulfonamides; Sulfones

2007
Na+/H+ exchange inhibition with cariporide prevents alterations of coronary endothelial function in streptozotocin-induced diabetes.
    Molecular and cellular biochemistry, 2008, Volume: 310, Issue:1-2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Blood Glucose; Carbachol; Diabetes Mellitus, Experimental; Dilatation; Endothelium, Vascular; Glucose; Guanidines; Heart; Heart Function Tests; In Vitro Techniques; Lactic Acid; Male; Monocarboxylic Acid Transporters; Nitroprusside; Rats; Rats, Wistar; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Streptozocin; Sulfones; Symporters

2008
HCO3(-) secretion by murine nasal submucosal gland serous acinar cells during Ca2+-stimulated fluid secretion.
    The Journal of general physiology, 2008, Volume: 132, Issue:1

    Topics: Amiloride; Animals; Bicarbonates; Calcium Signaling; Carbachol; Cation Transport Proteins; Cell Size; Cells, Cultured; Chloride Channels; Chlorides; Cystic Fibrosis Transmembrane Conductance Regulator; Cytoplasm; Epithelial Cells; Exocrine Glands; Guanidines; Hydrogen-Ion Concentration; Mice; Mice, Inbred C57BL; Mice, Knockout; Nasal Mucosa; Niflumic Acid; Protein Isoforms; Sodium; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchangers; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2; Sulfones

2008
NHE1 activity contributes to migration and is necessary for proliferation of human gastric myofibroblasts.
    Pflugers Archiv : European journal of physiology, 2012, Volume: 463, Issue:3

    Topics: Adult; Aged; Antiporters; Carbachol; Cation Transport Proteins; Cell Movement; Cell Proliferation; Female; Guanidines; Humans; Hydrogen-Ion Concentration; Insulin-Like Growth Factor II; Male; Myofibroblasts; Sodium-Bicarbonate Symporters; Sodium-Hydrogen Exchanger 1; Sodium-Hydrogen Exchanger 3; Sodium-Hydrogen Exchangers; Stomach; Sulfones

2012