Page last updated: 2024-08-24

carfentanil and naltrexone

carfentanil has been researched along with naltrexone in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-19901 (3.33)18.7374
1990's10 (33.33)18.2507
2000's10 (33.33)29.6817
2010's8 (26.67)24.3611
2020's1 (3.33)2.80

Authors

AuthorsStudies
Galzi, JL; Goeldner, M; Hirth, C; Ilien, B; Mejean, A; Meunier, JC; Mollereau, C1
Malan, JH; Quandt, SK; Raath, JP1
Bice, AN; Dannals, RF; Frost, JJ; Lee, MC; Tanada, S; Wagner, HN1
Gates, CC; Haigh, JC1
Carpenter, JW; Leith, DE; Shaw, ML1
Clyde, VL; Ramsay, EC; Sleeman, JM1
Lance, WR; Miller, MW; Wild, MA1
Carter, W; Ramsay, EC; Sleeman, JM; Tobin, T1
Citino, SB; Heard, DJ; Schumacher, J; Young, L1
Civelek, AC; Dannals, RF; Dixon, RB; Joh, T; Kao, PF; Kim, S; Ravert, HT; Villemagne, VL; Wagner, HN1
Braselton, WE; Cook, RA; Dierenfeld, ES; House, C; Karesh, WB; Puche, H; Torres, A; Uhart, MM1
Mama, KR; Steffey, EP; Withrow, SJ1
Kearns, KS; Ramsay, EC; Swenson, B1
Cebra, CK; Larsen, RS; Wild, MA1
Hunter, RP; Isaza, R; Koch, DE; Mutlow, A1
Adams, KA; Miller, BF; Miller, KV; Muller, LI; Osborn, DA; Ramsay, EC; Storms, TN; Warren, RJ1
Bares, R; Braus, DF; Braus, DH; Croissant, B; Dohmen, BM; Heinz, A; Hermann, D; Machulla, HJ; Mann, K; Mundle, G; Reimold, M; Schumann, G; Wrase, J1
Carpenter, JW; Hunter, RP; Isaza, R; Koch, DE; Mutlow, A1
Aalto, S; Hagelberg, N; Hietala, J; Ingman, K; Juhakoski, A; Kallio, A; Karhuvaara, S; Någren, K; Oikonen, V; Scheinin, H1
Carpenter, JW; Cole, A; Dresser, BL; Hunter, RP; Isaza, R; Koch, DE; Mutlow, A1
Dannals, RF; Frost, JJ; Kim, YK; Lee, JS; McCaul, ME; Wand, GS; Weerts, EM1
Erickson, TB; George, AV; Lu, JJ; Metz, J; Pisano, MV1
Caulkett, NA; Shury, TK; Woodbury, MR1
Beaver, J; Bullmore, ET; Bush, MA; Gunn, RN; Hill, S; Howard, J; Long, C; Makwana, A; Matthews, PM; Miller, SR; Nathan, PJ; Newbould, RD; Passchier, J; Rabiner, EA; Reiley, R; Searle, G1
Kellie, KA; Kreeger, TJ1
Kalk, P; Moore, RP; Rainwater, KL; Sykes, JM; Valitutto, MT1
Dong, H; Gao, X; Gong, Z; Ma, W; Su, R; Yong, Z1
Batra, A; Hansson, AC; Hermann, D; Hirth, N; Hoffmann, S; Kiefer, F; la Fougère, C; Mann, K; Noori, HR; Reimold, M; Reischl, G; Smolka, MN; Sommer, WH; Spanagel, R1
McCranor, BJ; Pierce, SA; Racine, MC; Sciuto, AM; Tressler, J; Tuet, WY; Wong, B1
Flynn, SM; France, CP1

Trials

5 trial(s) available for carfentanil and naltrexone

ArticleYear
Efficacy and safety of naltrexone hydrochloride for antagonizing carfentanil citrate immobilization in captive Rocky Mountain elk (Cervus elaphus nelsoni).
    Journal of wildlife diseases, 1996, Volume: 32, Issue:2

    Topics: Analgesics, Opioid; Animals; Deer; Female; Fentanyl; Immobilization; Male; Naltrexone; Narcotic Antagonists

1996
Longer occupancy of opioid receptors by nalmefene compared to naloxone as measured in vivo by a dual-detector system.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1997, Volume: 38, Issue:11

    Topics: Adult; Analgesics, Opioid; Brain; Carbon Radioisotopes; Cross-Over Studies; Female; Fentanyl; Humans; Male; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Time Factors; Tomography, Emission-Computed

1997
Prolonged central mu-opioid receptor occupancy after single and repeated nalmefene dosing.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:12

    Topics: Adolescent; Adult; Analgesics, Opioid; Area Under Curve; Caudate Nucleus; Electrocardiography; Fentanyl; Glucuronides; Humans; Male; Naltrexone; Narcotic Antagonists; Positron-Emission Tomography; Prefrontal Cortex; Receptors, Opioid, mu; Thalamus

2005
Pharmacological differentiation of opioid receptor antagonists by molecular and functional imaging of target occupancy and food reward-related brain activation in humans.
    Molecular psychiatry, 2011, Volume: 16, Issue:8

    Topics: Adult; Amygdala; Brain; Brain Mapping; Corpus Striatum; Dose-Response Relationship, Drug; Fentanyl; Food; Humans; Indans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Radioligand Assay; Radionuclide Imaging; Reward; Triazoles

2011
Low μ-Opioid Receptor Status in Alcohol Dependence Identified by Combined Positron Emission Tomography and Post-Mortem Brain Analysis.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2017, Volume: 42, Issue:3

    Topics: Adult; Aged; Alcoholism; Analgesics, Opioid; Fentanyl; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Positron-Emission Tomography; Receptors, Opioid, mu; Tissue Banks; Ventral Striatum

2017

Other Studies

25 other study(ies) available for carfentanil and naltrexone

ArticleYear
Photoactivatable opiate derivatives as irreversible probes of the mu-opioid receptor.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:9

    Topics: Affinity Labels; Animals; Azides; Azo Compounds; Binding Sites; Brain; Chemical Phenomena; Chemistry; Guinea Pigs; Narcotics; Rats; Receptors, Opioid; Receptors, Opioid, mu; Structure-Activity Relationship

1990
Ostrich (Struthio camelus) immobilisation using carfentanil and xylazine and reversal with yohimbine and naltrexone.
    Journal of the South African Veterinary Association, 1992, Volume: 63, Issue:4

    Topics: Animals; Birds; Fentanyl; Immobilization; Naltrexone; Xylazine; Yohimbine

1992
Duration of occupancy of opiate receptors by naltrexone.
    Journal of nuclear medicine : official publication, Society of Nuclear Medicine, 1988, Volume: 29, Issue:7

    Topics: Administration, Oral; Adult; Brain; Carbon Radioisotopes; Female; Fentanyl; Humans; Male; Naltrexone; Radionuclide Imaging; Receptors, Opioid; Receptors, Opioid, mu; Time Factors

1988
Capture of wood bison (Bison bison athabascae) using carfentanil-based mixtures.
    Journal of wildlife diseases, 1995, Volume: 31, Issue:1

    Topics: Analgesics, Opioid; Animals; Bison; Diprenorphine; Drug Combinations; Female; Fentanyl; Hypnotics and Sedatives; Immobilization; Injections, Intramuscular; Injections, Intravenous; Injections, Subcutaneous; Male; Naloxone; Naltrexone; Narcotic Antagonists; Northwest Territories; Piperidines; Tranquilizing Agents; Xylazine

1995
Complications with the use of carfentanil citrate and xylazine hydrochloride to immobilize domestic horses.
    Journal of the American Veterinary Medical Association, 1995, Mar-15, Volume: 206, Issue:6

    Topics: Analgesics, Opioid; Animals; Animals, Domestic; Fentanyl; Horse Diseases; Horses; Hypertension; Immobilization; Naloxone; Naltrexone; Pulmonary Edema; Tachycardia; Xylazine

1995
Immobilization of black bears (Ursus americanus) with orally administered carfentanil citrate.
    Journal of wildlife diseases, 1995, Volume: 31, Issue:3

    Topics: Administration, Oral; Analgesics, Opioid; Animals; Diazepam; Female; Fentanyl; Immobilization; Male; Muscle Relaxants, Central; Muscle, Skeletal; Naltrexone; Narcotic Antagonists; Oxygen; Respiration; Ursidae

1995
Immobilization of domestic goats (Capra hircus) using orally administered carfentanil citrate and detomidine hydrochloride.
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 1997, Volume: 28, Issue:2

    Topics: Absorption; Administration, Oral; Adrenergic alpha-Antagonists; Analgesics; Analgesics, Opioid; Animals; Blood Pressure; Body Temperature; Drug Interactions; Enzyme-Linked Immunosorbent Assay; Female; Fentanyl; Goats; Heart Rate; Hypnotics and Sedatives; Imidazoles; Immobilization; Naltrexone; Narcotic Antagonists; Respiration; Saponins; Yohimbine

1997
Cardiopulmonary effects of carfentanil in dama gazelles (Gazella dama).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 1997, Volume: 28, Issue:2

    Topics: Analgesics, Opioid; Animals; Animals, Zoo; Antelopes; Blood Gas Analysis; Blood Pressure; Carbon Dioxide; Female; Fentanyl; Heart Rate; Immobilization; Male; Naltrexone; Narcotic Antagonists; Oximetry; Oxygen; Pregnancy; Reproducibility of Results; Respiration

1997
Health evaluation of free-ranging guanaco (Lama guanicoe).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 1998, Volume: 29, Issue:2

    Topics: Analgesics, Opioid; Anesthetics; Animals; Animals, Domestic; Animals, Wild; Antibodies; Antidotes; Blood Chemical Analysis; Camelids, New World; Communicable Diseases; Drug Combinations; Enzymes; Female; Fentanyl; Flumazenil; Health Status; Immobilization; Male; Minerals; Naltrexone; Narcotic Antagonists; Physical Examination; Reference Values; Sheep; Tiletamine; Vitamins; Zolazepam

1998
Use of orally administered carfentanil prior to isoflurane-induced anesthesia in a Kodiak brown bear.
    Journal of the American Veterinary Medical Association, 2000, Aug-15, Volume: 217, Issue:4

    Topics: Acid-Base Equilibrium; Administration, Oral; Analgesics, Opioid; Anesthetics, Inhalation; Animals; Blood Gas Analysis; Blood Pressure; Fentanyl; Fibrosarcoma; Forelimb; Heart Rate; Isoflurane; Male; Naltrexone; Narcotic Antagonists; Preanesthetic Medication; Respiration; Soft Tissue Neoplasms; Ursidae

2000
Oral induction of anesthesia with droperidol and transmucosal carfentanil citrate in chimpanzees (Pan troglodytes).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2000, Volume: 31, Issue:2

    Topics: Administration, Oral; Analgesics, Opioid; Anesthetics, Combined; Anesthetics, Dissociative; Animals; Anti-Anxiety Agents; Antipsychotic Agents; Benzodiazepines; Blood Gas Analysis; Body Temperature; Droperidol; Female; Fentanyl; Heart Rate; Least-Squares Analysis; Male; Mouth Mucosa; Naltrexone; Oximetry; Pan troglodytes; Tiletamine; Zolazepam

2000
Diagnosis and treatment of obstructive urolithiasis in a captive Rocky Mountain wapiti (Cervus elaphus nelsoni).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2000, Volume: 31, Issue:2

    Topics: Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Deer; Fentanyl; Hematuria; Hydrogen-Ion Concentration; Male; Naltrexone; Penis; Phenylbutazone; Specific Gravity; Urethra; Urethral Obstruction; Urinary Bladder; Urinary Calculi

2000
Extraction and quantitation of carfentanil and naltrexone in goat plasma with liquid chromatography-mass spectrometry.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2003, Aug-15, Volume: 793, Issue:2

    Topics: Analgesics, Opioid; Animals; Chromatography, Liquid; Fentanyl; Goats; Naltrexone; Reproducibility of Results; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization

2003
A comparison of carfentanil/xylazine and Telazol/xylazine for immobilization of white-tailed deer.
    Journal of wildlife diseases, 2003, Volume: 39, Issue:4

    Topics: Adrenergic alpha-Agonists; Anesthetics; Animals; Deer; Dose-Response Relationship, Drug; Drug Combinations; Female; Fentanyl; Heart Rate; Immobilization; Injections, Intramuscular; Male; Naltrexone; Random Allocation; Respiration; Safety; Tiletamine; Time Factors; Xylazine; Yohimbine; Zolazepam

2003
Correlation of stable elevations in striatal mu-opioid receptor availability in detoxified alcoholic patients with alcohol craving: a positron emission tomography study using carbon 11-labeled carfentanil.
    Archives of general psychiatry, 2005, Volume: 62, Issue:1

    Topics: Adult; Alcohol Drinking; Alcoholism; Basal Ganglia; Behavior, Addictive; Carbon Radioisotopes; Fentanyl; Hospitalization; Humans; Male; Naltrexone; Narcotic Antagonists; Positron-Emission Tomography; Psychiatric Status Rating Scales; Receptors, Opioid, mu; Severity of Illness Index; Temperance

2005
Pharmacokinetics of carfentanil and naltrexone in domestic goats (Capra hircus).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2004, Volume: 35, Issue:4

    Topics: Absorption; Analgesics, Opioid; Animals; Cross-Over Studies; Female; Fentanyl; Gas Chromatography-Mass Spectrometry; Goats; Half-Life; Immobilization; Injections, Intramuscular; Injections, Intravenous; Injections, Subcutaneous; Male; Metabolic Clearance Rate; Naltrexone; Narcotic Antagonists; Random Allocation

2004
Pharmacokinetics and pharmacodynamics of carfentanil and naltrexone in female common eland (Taurotragus oryx).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2006, Volume: 37, Issue:3

    Topics: Analgesics, Opioid; Animals; Antelopes; Area Under Curve; Body Temperature; Female; Fentanyl; Gas Chromatography-Mass Spectrometry; Half-Life; Heart Rate; Immobilization; Injections, Intramuscular; Metabolic Clearance Rate; Naltrexone; Narcotic Antagonists; Random Allocation; Respiration

2006
Differences in delta- and mu-opioid receptor blockade measured by positron emission tomography in naltrexone-treated recently abstinent alcohol-dependent subjects.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2008, Volume: 33, Issue:3

    Topics: Adult; Alcoholism; Analgesics, Opioid; Data Interpretation, Statistical; Female; Fentanyl; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Positron-Emission Tomography; Radiopharmaceuticals; Receptors, Opioid, delta; Receptors, Opioid, mu; Substance Withdrawal Syndrome; Temperance

2008
Carfentanil--an ultra potent opioid.
    The American journal of emergency medicine, 2010, Volume: 28, Issue:4

    Topics: Accidents, Occupational; Adult; Analgesics, Opioid; Fentanyl; Humans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Veterinarians

2010
Intranasal naltrexone and atipamezole for reversal of white-tailed deer immobilized with carfentanil and medetomidine.
    The Canadian veterinary journal = La revue veterinaire canadienne, 2010, Volume: 51, Issue:5

    Topics: Administration, Intranasal; Adrenergic alpha-Antagonists; Animals; Cross-Over Studies; Deer; Dose-Response Relationship, Drug; Drug Combinations; Female; Fentanyl; Imidazoles; Immobilization; Injections, Intramuscular; Medetomidine; Naltrexone; Narcotic Antagonists; Random Allocation

2010
Sufentanil citrate immobilization of Alaskan moose calves.
    Journal of wildlife diseases, 2012, Volume: 48, Issue:4

    Topics: Alaska; Anesthesia Recovery Period; Animals; Animals, Newborn; Animals, Wild; Deer; Dose-Response Relationship, Drug; Female; Fentanyl; Immobilization; Male; Naltrexone; Narcotics; Oxygen; Respiration; Sufentanil; Time Factors; Tolazoline; Xylazine

2012
Comparison of two injectable immobilization combinations in Himalayan tahr (Hemitragus jemlahicus): medetomidine, ketamine, and atipamezole versus carfentanil, xylazine, naltrexone, and atipamezole.
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2013, Volume: 44, Issue:3

    Topics: Animals; Fentanyl; Hypnotics and Sedatives; Imidazoles; Ketamine; Medetomidine; Naltrexone; Ruminants; Xylazine

2013
Nalmefene reverses carfentanil-induced loss of righting reflex and respiratory depression in rats.
    European journal of pharmacology, 2014, Sep-05, Volume: 738

    Topics: Analgesics, Opioid; Animals; Blood Gas Analysis; Dose-Response Relationship, Drug; Fentanyl; Male; Naltrexone; Rats; Rats, Sprague-Dawley; Reflex, Righting; Respiratory Insufficiency; Time Factors

2014
Changes in murine respiratory dynamics induced by aerosolized carfentanil inhalation: Efficacy of naloxone and naltrexone.
    Toxicology letters, 2019, Volume: 316

    Topics: Administration, Inhalation; Aerosols; Analgesics, Opioid; Animals; Computer Simulation; Dose-Response Relationship, Drug; Fentanyl; Humans; Lung; Male; Mice; Models, Biological; Naloxone; Naltrexone; Narcotic Antagonists; Plethysmography, Whole Body; Respiration; Respiratory Insufficiency; Risk Assessment

2019
Discriminative stimulus effects of carfentanil in rats discriminating fentanyl: Differential antagonism by naltrexone.
    Drug and alcohol dependence, 2021, 04-01, Volume: 221

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Fentanyl; Heroin; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu

2021